ATE550323T1 - Piperidinyl-prostaglandinanaloga als den augeninnendruck senkende mittel - Google Patents
Piperidinyl-prostaglandinanaloga als den augeninnendruck senkende mittelInfo
- Publication number
- ATE550323T1 ATE550323T1 AT05749871T AT05749871T ATE550323T1 AT E550323 T1 ATE550323 T1 AT E550323T1 AT 05749871 T AT05749871 T AT 05749871T AT 05749871 T AT05749871 T AT 05749871T AT E550323 T1 ATE550323 T1 AT E550323T1
- Authority
- AT
- Austria
- Prior art keywords
- piperidinyl
- intra
- lowering agents
- prostaglandin analogs
- eye pressure
- Prior art date
Links
- 239000000651 prodrug Substances 0.000 abstract 3
- 229940002612 prodrug Drugs 0.000 abstract 3
- 150000003839 salts Chemical class 0.000 abstract 3
- 150000001875 compounds Chemical class 0.000 abstract 2
- 201000010099 disease Diseases 0.000 abstract 1
- 208000037265 diseases, disorders, signs and symptoms Diseases 0.000 abstract 1
- 239000003814 drug Substances 0.000 abstract 1
- 239000000203 mixture Substances 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
- C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D211/68—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member
- C07D211/72—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen, directly attached to ring carbon atoms
- C07D211/74—Oxygen atoms
- C07D211/76—Oxygen atoms attached in position 2 or 6
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
- C07F9/02—Phosphorus compounds
- C07F9/547—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
- C07F9/553—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom having one nitrogen atom as the only ring hetero atom
- C07F9/576—Six-membered rings
- C07F9/59—Hydrogenated pyridine rings
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Biochemistry (AREA)
- General Health & Medical Sciences (AREA)
- Molecular Biology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Hydrogenated Pyridines (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US57736104P | 2004-06-04 | 2004-06-04 | |
| PCT/US2005/017167 WO2005121086A2 (en) | 2004-06-04 | 2005-05-16 | Piperidinyl prostaglandin analogs as ocular hypotensive agents |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ATE550323T1 true ATE550323T1 (de) | 2012-04-15 |
Family
ID=35431920
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| AT05749871T ATE550323T1 (de) | 2004-06-04 | 2005-05-16 | Piperidinyl-prostaglandinanaloga als den augeninnendruck senkende mittel |
Country Status (9)
| Country | Link |
|---|---|
| US (1) | US7435746B2 (de) |
| EP (1) | EP1761495B1 (de) |
| AT (1) | ATE550323T1 (de) |
| AU (1) | AU2005252171A1 (de) |
| CA (1) | CA2569464C (de) |
| DK (1) | DK1761495T3 (de) |
| ES (1) | ES2381377T3 (de) |
| PL (1) | PL1761495T3 (de) |
| WO (1) | WO2005121086A2 (de) |
Families Citing this family (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US7326716B2 (en) * | 2003-06-06 | 2008-02-05 | Allergan, Inc. | Treatment of inflammatory bowel disease |
Family Cites Families (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| RU2296122C2 (ru) * | 2001-07-16 | 2007-03-27 | Ф.Хоффманн-Ля Рош Аг | Производные 2-пирролидона в качестве простаноидных агонистов и фармацевтическая композиция |
| WO2003047513A2 (en) * | 2001-12-03 | 2003-06-12 | Merck & Co., Inc. | Method for treating ocular hypertension |
| AU2003207900A1 (en) * | 2002-03-18 | 2003-09-29 | Pfizer Products Inc. | Methods of treatment with selective ep4 receptor agonists |
| US6573294B1 (en) * | 2002-05-14 | 2003-06-03 | Allergan, Inc. | 8-azaprostaglandin analogs as agents for lowering intraocular pressure |
| CN1735597A (zh) * | 2003-01-10 | 2006-02-15 | 霍夫曼-拉罗奇有限公司 | 作为前列腺素激动剂的2-哌啶酮衍生物 |
| CA2528179C (en) * | 2003-06-06 | 2013-10-22 | Allergan, Inc. | Piperidinyl prostaglandin e analogs |
-
2005
- 2005-05-16 AU AU2005252171A patent/AU2005252171A1/en not_active Abandoned
- 2005-05-16 PL PL05749871T patent/PL1761495T3/pl unknown
- 2005-05-16 EP EP05749871A patent/EP1761495B1/de not_active Expired - Lifetime
- 2005-05-16 ES ES05749871T patent/ES2381377T3/es not_active Expired - Lifetime
- 2005-05-16 CA CA2569464A patent/CA2569464C/en not_active Expired - Fee Related
- 2005-05-16 WO PCT/US2005/017167 patent/WO2005121086A2/en not_active Ceased
- 2005-05-16 AT AT05749871T patent/ATE550323T1/de active
- 2005-05-16 DK DK05749871.9T patent/DK1761495T3/da active
- 2005-05-16 US US10/564,829 patent/US7435746B2/en not_active Expired - Lifetime
Also Published As
| Publication number | Publication date |
|---|---|
| EP1761495B1 (de) | 2012-03-21 |
| WO2005121086A3 (en) | 2006-04-27 |
| US20060281713A1 (en) | 2006-12-14 |
| CA2569464A1 (en) | 2005-12-22 |
| AU2005252171A1 (en) | 2005-12-22 |
| EP1761495A2 (de) | 2007-03-14 |
| WO2005121086A2 (en) | 2005-12-22 |
| PL1761495T3 (pl) | 2012-07-31 |
| CA2569464C (en) | 2012-10-23 |
| ES2381377T3 (es) | 2012-05-25 |
| US7435746B2 (en) | 2008-10-14 |
| DK1761495T3 (da) | 2012-06-18 |
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