ATE63556T1 - Makrolid-derivate, verfahren zu ihrer herstellung und ihre verwendung. - Google Patents

Makrolid-derivate, verfahren zu ihrer herstellung und ihre verwendung.

Info

Publication number: ATE63556T1
Authority: AT; Austria
Prior art keywords: processes; production; macrolide derivatives; milbemycins; avermectins
Prior art date: 1986-01-07

Application number

AT87300108T

Other languages

English (en)

Inventor

Toshiaki Yanai

Kazuo Sato

Akira Nishida

Keiji Tanaka

Yasu-Cho Yasu

Original Assignee

Sankyo Co

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1986-01-07

Filing date

1987-01-07

Publication date

1991-06-15

1987-01-07 Application filed by Sankyo Co filed Critical Sankyo Co

1991-06-15 Application granted granted Critical

1991-06-15 Publication of ATE63556T1 publication Critical patent/ATE63556T1/de

Links

239000003120 macrolide antibiotic agent Substances 0.000 title 1
239000005660 Abamectin Substances 0.000 abstract 2
ZLBGSRMUSVULIE-GSMJGMFJSA-N milbemycin A3 Chemical class O1[C@H](C)[C@@H](C)CC[C@@]11O[C@H](C\C=C(C)\C[C@@H](C)\C=C\C=C/2[C@]3([C@H](C(=O)O4)C=C(C)[C@@H](O)[C@H]3OC\2)O)C[C@H]4C1 ZLBGSRMUSVULIE-GSMJGMFJSA-N 0.000 abstract 2
230000000895 acaricidal effect Effects 0.000 abstract 1
230000010933 acylation Effects 0.000 abstract 1
238000005917 acylation reaction Methods 0.000 abstract 1
230000000507 anthelmentic effect Effects 0.000 abstract 1
238000006735 epoxidation reaction Methods 0.000 abstract 1
230000000749 insecticidal effect Effects 0.000 abstract 1
FXWHFKOXMBTCMP-WMEDONTMSA-N milbemycin Natural products COC1C2OCC3=C/C=C/C(C)CC(=CCC4CC(CC5(O4)OC(C)C(C)C(OC(=O)C(C)CC(C)C)C5O)OC(=O)C(C=C1C)C23O)C FXWHFKOXMBTCMP-WMEDONTMSA-N 0.000 abstract 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H19/00—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
- C07H19/01—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing oxygen
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D493/00—Heterocyclic compounds containing oxygen atoms as the only ring hetero atoms in the condensed system
- C07D493/22—Heterocyclic compounds containing oxygen atoms as the only ring hetero atoms in the condensed system in which the condensed system contains four or more hetero rings
- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
- A01N43/90—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having two or more relevant hetero rings, condensed among themselves or with a common carbocyclic ring system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
- A61P33/10—Anthelmintics

Landscapes

Chemical & Material Sciences (AREA)
Health & Medical Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
Organic Chemistry (AREA)
General Health & Medical Sciences (AREA)
Engineering & Computer Science (AREA)
Veterinary Medicine (AREA)
Agronomy & Crop Science (AREA)
Dentistry (AREA)
Pharmacology & Pharmacy (AREA)
Medicinal Chemistry (AREA)
Animal Behavior & Ethology (AREA)
General Chemical & Material Sciences (AREA)
Public Health (AREA)
Chemical Kinetics & Catalysis (AREA)
Pest Control & Pesticides (AREA)
Plant Pathology (AREA)
Tropical Medicine & Parasitology (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Wood Science & Technology (AREA)
Zoology (AREA)
Environmental Sciences (AREA)
Biochemistry (AREA)
Biotechnology (AREA)
Genetics & Genomics (AREA)
Molecular Biology (AREA)
Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
Saccharide Compounds (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Agricultural Chemicals And Associated Chemicals (AREA)

AT87300108T 1986-01-07 1987-01-07 Makrolid-derivate, verfahren zu ihrer herstellung und ihre verwendung. ATE63556T1 (de)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
JP61001190A JPH0678342B2 (ja)	1986-01-07	1986-01-07	新規マクロライド化合物
EP87300108A EP0230347B1 (de)	1986-01-07	1987-01-07	Makrolid-Derivate, Verfahren zu ihrer Herstellung und ihre Verwendung

Publications (1)

Publication Number	Publication Date
ATE63556T1 true ATE63556T1 (de)	1991-06-15

Family

ID=11494531

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
AT87300108T ATE63556T1 (de)	1986-01-07	1987-01-07	Makrolid-derivate, verfahren zu ihrer herstellung und ihre verwendung.

Country Status (7)

Country	Link
US (1)	US4912090A (de)
EP (1)	EP0230347B1 (de)
JP (1)	JPH0678342B2 (de)
KR (1)	KR940006632B1 (de)
AT (1)	ATE63556T1 (de)
DE (1)	DE3770000D1 (de)
ES (1)	ES2033819T3 (de)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
GB8811036D0 (en) *	1988-05-10	1988-06-15	Glaxo Group Ltd	Chemical compounds
GB8813150D0 (en) *	1988-06-03	1988-07-06	American Cyanamid Co	Chemical compounds
FR2665898B1 (fr) *	1990-08-20	1994-03-11	Sanofi	Derives d'amido-3 pyrazole, procede pour leur preparation et compositions pharmaceutiques les contenant.
US5461168A (en) *	1992-09-01	1995-10-24	Sankyo Company, Limited	Processes for the production of 13-ether derivatives of milbemycins, and intermediates therefor
US6562588B2 (en)	1993-05-17	2003-05-13	Genentech, Inc.	Sialidase and recombinant cell lines
WO1996019920A1 (en) *	1994-12-27	1996-07-04	Pfizer Pharmaceuticals Inc.	Compositions for treating nematode infections in trees
US5773422A (en) *	1996-01-29	1998-06-30	Komer; Gene	Avermectin formulation
CN1441790A (zh) *	2000-01-28	2003-09-10	罗姆和哈斯公司	增强性质的药物
US6376548B1 (en)	2000-01-28	2002-04-23	Rohm And Haas Company	Enhanced propertied pesticides
JP4373080B2 (ja) *	2002-12-24	2009-11-25	三井化学アグロ株式会社	ミルベマイシン類の精製法
GB0501220D0 (en) *	2005-01-21	2005-03-02	Norbrook Lab Ltd	Anthelmintic composition

Family Cites Families (10)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US4201861A (en) *	1977-10-03	1980-05-06	Merck & Co., Inc.	Acyl derivatives of C-076 compounds
IL56149A (en) *	1977-12-19	1989-09-28	Merck & Co Inc	13-halo and 13-deoxy derivatives of c-076 compounds,their preparation and method for the treatment of parasitic infections in animals therewith
US4200581A (en) *	1978-08-04	1980-04-29	Merck & Co., Inc.	Alkyl derivatives of C-076 compounds
JPS5936681A (ja) *	1982-08-23	1984-02-28	Sankyo Co Ltd	ミルペマイシンｄのエポキシ誘導体
US4469682A (en) *	1983-01-28	1984-09-04	Merck & Co., Inc.	Avermectin and milbemycin phosphate esters, pharmaceutical compositions, and method of use
US4530921A (en) *	1983-10-03	1985-07-23	Merck & Co., Inc.	Avermectin epoxide derivatives and method of use
JPS60126289A (ja) *	1983-11-14	1985-07-05	Sankyo Co Ltd	ミルベマイシン類の５−カ−ボネ−ト誘導体
JPS60158191A (ja) *	1983-12-30	1985-08-19	チバ‐ガイギー　アクチエンゲゼルシヤフト	ミルベマイシン誘導体、その製法、及び有害生物防除剤組成物
DK614084A (da) *	1983-12-30	1985-07-01	Ciba Geigy Ag	Milbemycim-derivater samt deres fremstilling og anvendelse
US4696922A (en) *	1984-11-26	1987-09-29	Ciba-Geigy Corporation	5-azolylacetoxymilbemycins as ecto- and endoparasites

1986
- 1986-01-07 JP JP61001190A patent/JPH0678342B2/ja not_active Expired - Fee Related
- 1986-12-30 US US06/947,615 patent/US4912090A/en not_active Expired - Fee Related
1987
- 1987-01-07 KR KR1019870000057A patent/KR940006632B1/ko not_active Expired - Fee Related
- 1987-01-07 AT AT87300108T patent/ATE63556T1/de not_active IP Right Cessation
- 1987-01-07 EP EP87300108A patent/EP0230347B1/de not_active Expired - Lifetime
- 1987-01-07 DE DE8787300108T patent/DE3770000D1/de not_active Expired - Fee Related
- 1987-01-07 ES ES198787300108T patent/ES2033819T3/es not_active Expired - Lifetime

Also Published As

Publication number	Publication date
KR870007150A (ko)	1987-08-17
EP0230347B1 (de)	1991-05-15
DE3770000D1 (de)	1991-06-20
ES2033819T3 (es)	1993-04-01
KR940006632B1 (ko)	1994-07-23
JPS62161788A (ja)	1987-07-17
JPH0678342B2 (ja)	1994-10-05
US4912090A (en)	1990-03-27
EP0230347A1 (de)	1987-07-29

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Legal Events

Date	Code	Title	Description
1992-03-15	UEP	Publication of translation of european patent specification
2002-10-15	REN	Ceased due to non-payment of the annual fee