ATE66678T1 - Verfahren zur herstellung von makrolidderivaten. - Google Patents

Verfahren zur herstellung von makrolidderivaten.

Info

Publication number: ATE66678T1
Authority: AT; Austria
Prior art keywords: macrolid; derivatives; production; macrolid derivatives
Prior art date: 1986-03-31

Application number

AT87302663T

Other languages

English (en)

Inventor

Eddie Vi-Ping Tao

Jeffrey Thomas Vicenzi

Original Assignee

Lilly Co Eli

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1986-03-31

Filing date

1987-03-27

Publication date

1991-09-15

1987-03-27 Application filed by Lilly Co Eli filed Critical Lilly Co Eli

1991-09-15 Application granted granted Critical

1991-09-15 Publication of ATE66678T1 publication Critical patent/ATE66678T1/de

Links

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
- C07H17/04—Heterocyclic radicals containing only oxygen as ring hetero atoms
- C07H17/08—Hetero rings containing eight or more ring members, e.g. erythromycins
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H5/00—Compounds containing saccharide radicals in which the hetero bonds to oxygen have been replaced by the same number of hetero bonds to halogen, nitrogen, sulfur, selenium, or tellurium
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H15/00—Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Molecular Biology (AREA)
Life Sciences & Earth Sciences (AREA)
Biochemistry (AREA)
Biotechnology (AREA)
General Health & Medical Sciences (AREA)
Genetics & Genomics (AREA)
Health & Medical Sciences (AREA)
Engineering & Computer Science (AREA)
Saccharide Compounds (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Plural Heterocyclic Compounds (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)

AT87302663T 1986-03-31 1987-03-27 Verfahren zur herstellung von makrolidderivaten. ATE66678T1 (de)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
US06/846,446 US4921947A (en)	1986-03-31	1986-03-31	Process for preparing macrolide derivatives
EP87302663A EP0240264B1 (de)	1986-03-31	1987-03-27	Verfahren zur Herstellung von Makrolidderivaten

Publications (1)

Publication Number	Publication Date
ATE66678T1 true ATE66678T1 (de)	1991-09-15

Family

ID=25297965

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
AT87302663T ATE66678T1 (de)	1986-03-31	1987-03-27	Verfahren zur herstellung von makrolidderivaten.

Country Status (21)

Country	Link
US (1)	US4921947A (de)
EP (1)	EP0240264B1 (de)
JP (1)	JPH0710876B2 (de)
KR (1)	KR900001166B1 (de)
CN (1)	CN1018647B (de)
AR (1)	AR247402A1 (de)
AT (1)	ATE66678T1 (de)
AU (1)	AU593894B2 (de)
CA (1)	CA1292737C (de)
DE (1)	DE3772423D1 (de)
DK (1)	DK172935B1 (de)
EG (1)	EG18550A (de)
ES (1)	ES2028865T3 (de)
GR (1)	GR3002764T3 (de)
HK (1)	HK82492A (de)
HU (1)	HU199864B (de)
IE (1)	IE61018B1 (de)
IL (1)	IL82005A (de)
NZ (1)	NZ219784A (de)
PT (1)	PT84561B (de)
ZA (1)	ZA872201B (de)

Families Citing this family (24)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
FR2638458A1 (fr) *	1988-10-27	1990-05-04	Adir	Nouveaux derives de la tylosine, leur procede de preparation et les compositions pharmaceutiques qui les contiennent
US5354708A (en) *	1992-06-04	1994-10-11	Taskar Nikhil R	Method of nitrogen doping of II-VI semiconductor compounds during epitaxial growth using an amine
TW226373B (de) *	1992-07-15	1994-07-11	Pfizer
US5677287A (en) *	1993-03-18	1997-10-14	Pfizer Inc.	Antibacterial 16-membered ring macrolides containing olefins at C-20
AU6980094A (en) *	1993-07-15	1995-02-13	Pfizer Inc.	Amide derivatives of 16-membered ring antibiotic macrolides
ES2076107B1 (es) *	1993-09-20	1996-04-01	Pfizer	Derivados de antibioticos macrolidos de anillos de 16 miembros.
EP0778283A3 (de) *	1995-12-05	1998-01-28	Pfizer Inc.	Antibiotische Makrolide
DE102004027417A1 (de) *	2004-06-04	2005-12-22	Basf Ag	Verbundelement
HUE028588T2 (hu)	2005-12-13	2016-12-28	Incyte Holdings Corp	Heteroaril-szubsztituált pirrolo[2,3-b]piridinek és pirrolo[2,3-b]pirimidinek mint Janus-kináz inhibitorok
JP5126685B2 (ja) *	2006-05-01	2013-01-23	大正製薬株式会社	マクロライド誘導体
JP5323696B2 (ja) *	2006-07-28	2013-10-23	インターベツト・インターナシヨナル・ベー・ベー	マクロライド合成方法
EP2019112A1 (de) *	2007-07-26	2009-01-28	Intervet International BV	Festkörper-Makrolidformen
CN102875622B (zh) *	2006-07-28	2016-12-07	英特威国际有限公司	大环内酯合成方法
CA2818542A1 (en)	2010-11-19	2012-05-24	Incyte Corporation	Cyclobutyl substituted pyrrolopyridine and pyrrolopyrimidine derivatives as jak inhibitors
ES2536415T3 (es)	2010-11-19	2015-05-25	Incyte Corporation	Pirrolopiridinas y pirrolopirimidinas sustituidas heterocíclicas como inhibidores de JAK
US8691807B2 (en)	2011-06-20	2014-04-08	Incyte Corporation	Azetidinyl phenyl, pyridyl or pyrazinyl carboxamide derivatives as JAK inhibitors
CA2856708C (en)	2011-11-25	2022-01-11	Bayer Intellectual Property Gmbh	Antibacterial tylosin derivatives and methods for their preparation
CN102382159B (zh) *	2011-12-07	2013-11-13	齐鲁动物保健品有限公司	一种替米考星的制备方法
EP3489239B1 (de)	2013-03-06	2021-09-15	Incyte Holdings Corporation	Verfahren und zwischenprodukte zur herstellung eines jak-hemmers
TR201809189T4 (tr)	2013-05-23	2018-07-23	Bayer Animal Health Gmbh	Tylosin türevleri̇ ve bunlarin hazirlanmasina yöneli̇k yöntem.
CN105837648B (zh) *	2015-11-02	2018-07-06	湖北龙翔药业科技股份有限公司	一种磷酸替米考星的制备方法
CN108299531B (zh) *	2018-01-23	2021-02-05	郑州大学	甲哌泰万菌素可药用盐及其制备方法
CN111269275A (zh) *	2020-03-09	2020-06-12	浙江康牧药业有限公司	一种替米考星的制备方法
CN117304241B (zh) *	2023-11-30	2024-03-01	中国农业科学院饲料研究所	一种大环内酯类化合物及其制备方法与应用

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
YU43006B (en) *	1981-03-06	1989-02-28	Pliva Pharm & Chem Works	Process for preparing n-methyl-11-aza-10-deoxo-10-dihydro erythromycin and derivatives thereof
JPS58146595A (ja) *	1982-02-25	1983-09-01	Satoshi Omura	マクロライド系抗生物質
US4454314A (en) *	1982-08-02	1984-06-12	Pfizer Inc.	Antibacterial mycaminosyl tylonolide and related macrolide derivatives
AU561147B2 (en) *	1982-09-13	1987-04-30	Eli Lilly And Company	20-amino macrolide antibiotics
US4443436A (en) *	1982-09-13	1984-04-17	Eli Lilly And Company	C-20-Modified macrolide derivatives of the macrolide antibiotics tylosin, desmycosin, macrocin, and lactenocin
US4468511A (en) *	1983-02-28	1984-08-28	Eli Lilly And Company	C-20- And C-23-Modified macrolide derivatives

1986
- 1986-03-31 US US06/846,446 patent/US4921947A/en not_active Expired - Lifetime
1987
- 1987-03-25 ZA ZA872201A patent/ZA872201B/xx unknown
- 1987-03-25 CA CA000532905A patent/CA1292737C/en not_active Expired - Lifetime
- 1987-03-25 IL IL82005A patent/IL82005A/xx not_active IP Right Cessation
- 1987-03-26 DK DK198701540A patent/DK172935B1/da not_active IP Right Cessation
- 1987-03-26 AR AR87307119A patent/AR247402A1/es active
- 1987-03-26 EG EG182/87A patent/EG18550A/xx active
- 1987-03-26 PT PT84561A patent/PT84561B/pt unknown
- 1987-03-26 JP JP62075752A patent/JPH0710876B2/ja not_active Expired - Lifetime
- 1987-03-26 NZ NZ219784A patent/NZ219784A/xx unknown
- 1987-03-26 AU AU70670/87A patent/AU593894B2/en not_active Expired
- 1987-03-26 HU HU871328A patent/HU199864B/hu unknown
- 1987-03-27 CN CN87102397A patent/CN1018647B/zh not_active Expired
- 1987-03-27 ES ES198787302663T patent/ES2028865T3/es not_active Expired - Lifetime
- 1987-03-27 EP EP87302663A patent/EP0240264B1/de not_active Expired - Lifetime
- 1987-03-27 AT AT87302663T patent/ATE66678T1/de not_active IP Right Cessation
- 1987-03-27 IE IE79687A patent/IE61018B1/en not_active IP Right Cessation
- 1987-03-27 KR KR1019870002839A patent/KR900001166B1/ko not_active Expired
- 1987-03-27 DE DE8787302663T patent/DE3772423D1/de not_active Expired - Lifetime
1991
- 1991-09-19 GR GR91401376T patent/GR3002764T3/el unknown
1992
- 1992-10-22 HK HK824/92A patent/HK82492A/en not_active IP Right Cessation

Also Published As

Publication number	Publication date
HU199864B (en)	1990-03-28
EP0240264A3 (en)	1987-11-19
US4921947A (en)	1990-05-01
KR900001166B1 (ko)	1990-02-27
HUT43087A (en)	1987-09-28
CA1292737C (en)	1991-12-03
EP0240264B1 (de)	1991-08-28
AU7067087A (en)	1987-10-08
IL82005A0 (en)	1987-10-20
AR247402A1 (es)	1994-12-29
JPH0710876B2 (ja)	1995-02-08
CN87102397A (zh)	1987-10-07
AU593894B2 (en)	1990-02-22
HK82492A (en)	1992-10-30
GR3002764T3 (en)	1993-01-25
NZ219784A (en)	1989-01-27
PT84561B (pt)	1989-11-10
KR870008906A (ko)	1987-10-21
JPS62240681A (ja)	1987-10-21
IL82005A (en)	1991-08-16
ES2028865T3 (es)	1992-07-16
CN1018647B (zh)	1992-10-14
EP0240264A2 (de)	1987-10-07
EG18550A (en)	1993-10-30
DE3772423D1 (de)	1991-10-02
ZA872201B (en)	1988-10-26
PT84561A (en)	1987-04-01
DK154087A (da)	1987-10-01
DK172935B1 (da)	1999-10-11
DK154087D0 (da)	1987-03-26
IE61018B1 (en)	1994-09-07
IE870796L (en)	1987-09-30

Legal Events

Date	Code	Title	Description
2007-06-15	EELA	Cancelled due to lapse of time

Publication	Publication Date	Title
DE3789746D1 (de)	1994-06-09	Verfahren zur Herstellung von Zink-Nickel-Phosphatüberzügen.
DE3689259D1 (de)	1993-12-09	Verfahren zur Herstellung von Polyolefinen.
DE3787307D1 (de)	1993-10-14	Verfahren zur Herstellung von Reibungselementen.
DE58908451D1 (de)	1994-11-03	Verfahren zur Herstellung von Organochlorsilanen.
DE3750318D1 (de)	1994-09-08	Verfahren zur Herstellung von Halosilanen.
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DE69022631D1 (de)	1995-11-02	Verfahren zur Herstellung von L-Tryptophan.
DE3789557D1 (de)	1994-05-11	Verfahren zur Herstellung von Maleimid.
DE68923643D1 (de)	1995-09-07	Verfahren zur Herstellung von L-Tryptophan.
DE59001820D1 (de)	1993-07-29	Verfahren zur herstellung von indolcarbonsaeurederivaten.
DE3789680D1 (de)	1994-06-01	Verfahren zur Herstellung von Halbleiterbauelementen.
DE68918050D1 (de)	1994-10-13	Verfahren zur Herstellung von Windschutzscheiben.
DE58907777D1 (de)	1994-07-07	Verfahren zur Herstellung von Caprolactam.
DE3881091D1 (de)	1993-06-24	Verfahren zur herstellung von phosphatidsaeurederivaten.
DE68920351D1 (de)	1995-02-16	Verfahren zur Herstellung von Indigoverbindungen.
DE68916760D1 (de)	1994-08-18	Verfahren zur Herstellung von Gamma-Lactonen.
DE58907409D1 (de)	1994-05-11	Verfahren zur Herstellung von Caprolactam.
ATE86619T1 (de)	1993-03-15	Verfahren zur herstellung von nitroethenderivaten.
DE68920087D1 (de)	1995-02-02	Verfahren zur Herstellung von Neuraminidase.
DE58906122D1 (de)	1993-12-16	Verfahren zur Herstellung von Phenylethanolen.
DE68910919D1 (de)	1994-01-05	Verfahren zur Herstellung von Pigment.
ATE94538T1 (de)	1993-10-15	Verfahren zur herstellung von harnstoffen.
DE3788412D1 (de)	1994-01-20	Verfahren zur Herstellung synthetischen Mazzits.
DE3862774D1 (de)	1991-06-20	Verfahren zur herstellung von vinylphosphonsaeuredialkylestern.
DE68924502D1 (de)	1995-11-16	Verfahren zur Herstellung von Einzelsubstraten.