PT84561B - Processo aperfeicoado para a preparacao de derivados macrolidos - Google Patents

Processo aperfeicoado para a preparacao de derivados macrolidos

Info

Publication number
PT84561B
PT84561B PT84561A PT8456187A PT84561B PT 84561 B PT84561 B PT 84561B PT 84561 A PT84561 A PT 84561A PT 8456187 A PT8456187 A PT 8456187A PT 84561 B PT84561 B PT 84561B
Authority
PT
Portugal
Prior art keywords
macrolidary
derivatives
preparation
appropriate process
appropriate
Prior art date
Application number
PT84561A
Other languages
English (en)
Other versions
PT84561A (en
Inventor
Eddie Vi-Ping Tao
Jeffrey Thomas Vicenzi
Original Assignee
Lilly Co Eli
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Lilly Co Eli filed Critical Lilly Co Eli
Publication of PT84561A publication Critical patent/PT84561A/pt
Publication of PT84561B publication Critical patent/PT84561B/pt

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H5/00Compounds containing saccharide radicals in which the hetero bonds to oxygen have been replaced by the same number of hetero bonds to halogen, nitrogen, sulfur, selenium, or tellurium
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/04Heterocyclic radicals containing only oxygen as ring hetero atoms
    • C07H17/08Hetero rings containing eight or more ring members, e.g. erythromycins
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H15/00Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Molecular Biology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Biochemistry (AREA)
  • Biotechnology (AREA)
  • General Health & Medical Sciences (AREA)
  • Genetics & Genomics (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Saccharide Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
PT84561A 1986-03-31 1987-03-26 Processo aperfeicoado para a preparacao de derivados macrolidos PT84561B (pt)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US06/846,446 US4921947A (en) 1986-03-31 1986-03-31 Process for preparing macrolide derivatives

Publications (2)

Publication Number Publication Date
PT84561A PT84561A (en) 1987-04-01
PT84561B true PT84561B (pt) 1989-11-10

Family

ID=25297965

Family Applications (1)

Application Number Title Priority Date Filing Date
PT84561A PT84561B (pt) 1986-03-31 1987-03-26 Processo aperfeicoado para a preparacao de derivados macrolidos

Country Status (21)

Country Link
US (1) US4921947A (pt)
EP (1) EP0240264B1 (pt)
JP (1) JPH0710876B2 (pt)
KR (1) KR900001166B1 (pt)
CN (1) CN1018647B (pt)
AR (1) AR247402A1 (pt)
AT (1) ATE66678T1 (pt)
AU (1) AU593894B2 (pt)
CA (1) CA1292737C (pt)
DE (1) DE3772423D1 (pt)
DK (1) DK172935B1 (pt)
EG (1) EG18550A (pt)
ES (1) ES2028865T3 (pt)
GR (1) GR3002764T3 (pt)
HK (1) HK82492A (pt)
HU (1) HU199864B (pt)
IE (1) IE61018B1 (pt)
IL (1) IL82005A (pt)
NZ (1) NZ219784A (pt)
PT (1) PT84561B (pt)
ZA (1) ZA872201B (pt)

Families Citing this family (24)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2638458A1 (fr) * 1988-10-27 1990-05-04 Adir Nouveaux derives de la tylosine, leur procede de preparation et les compositions pharmaceutiques qui les contiennent
US5354708A (en) * 1992-06-04 1994-10-11 Taskar Nikhil R Method of nitrogen doping of II-VI semiconductor compounds during epitaxial growth using an amine
TW226373B (pt) * 1992-07-15 1994-07-11 Pfizer
US5677287A (en) * 1993-03-18 1997-10-14 Pfizer Inc. Antibacterial 16-membered ring macrolides containing olefins at C-20
EP0708770B1 (en) * 1993-07-15 1997-04-16 Pfizer Inc. Amide derivatives of 16-membered ring antibiotic macrolides
ES2076107B1 (es) * 1993-09-20 1996-04-01 Pfizer Derivados de antibioticos macrolidos de anillos de 16 miembros.
EP0778283A3 (en) * 1995-12-05 1998-01-28 Pfizer Inc. Antibiotic macrolides
DE102004027417A1 (de) * 2004-06-04 2005-12-22 Basf Ag Verbundelement
CN103214484B (zh) 2005-12-13 2016-07-06 因塞特控股公司 作为两面神激酶抑制剂的杂芳基取代的吡咯并[2,3-b]吡啶和吡咯并[2,3-b]嘧啶
EP2077271A4 (en) * 2006-05-01 2010-09-15 Taisho Pharmaceutical Co Ltd Macrolide derivative
NZ574193A (en) * 2006-07-28 2011-09-30 Intervet Int Bv Macrolide synthesis process
AU2007278195B2 (en) * 2006-07-28 2012-09-13 Intervet International B.V. Macrolide synthesis process
EP2019112A1 (en) * 2007-07-26 2009-01-28 Intervet International BV Macrolide solid-state forms
WO2012068440A1 (en) 2010-11-19 2012-05-24 Incyte Corporation Heterocyclic-substituted pyrrolopyridines and pyrrolopyrimidines as jak inhibitors
CA2818542A1 (en) 2010-11-19 2012-05-24 Incyte Corporation Cyclobutyl substituted pyrrolopyridine and pyrrolopyrimidine derivatives as jak inhibitors
MY165963A (en) 2011-06-20 2018-05-18 Incyte Holdings Corp Azetidinyl phenyl, pyridyl or pyrazinyl carboxamide derivatives as jak inhibitors
CN104302653B (zh) 2011-11-25 2017-02-22 拜耳知识产权有限责任公司 抗菌的泰乐菌素衍生物及其制备方法
CN102382159B (zh) * 2011-12-07 2013-11-13 齐鲁动物保健品有限公司 一种替米考星的制备方法
MX384910B (es) 2013-03-06 2025-03-14 Incyte Holdings Corp Procesos e intermedios para hacer un inhibidor de jak.
HUE037868T2 (hu) * 2013-05-23 2018-09-28 Bayer Animal Health Gmbh Tilozin-származékok és eljárás elõállításukra
CN105837648B (zh) * 2015-11-02 2018-07-06 湖北龙翔药业科技股份有限公司 一种磷酸替米考星的制备方法
CN108299531B (zh) * 2018-01-23 2021-02-05 郑州大学 甲哌泰万菌素可药用盐及其制备方法
CN111269275A (zh) * 2020-03-09 2020-06-12 浙江康牧药业有限公司 一种替米考星的制备方法
CN117304241B (zh) * 2023-11-30 2024-03-01 中国农业科学院饲料研究所 一种大环内酯类化合物及其制备方法与应用

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
SI8110592A8 (en) * 1981-03-06 1996-06-30 Pliva Pharm & Chem Works Process for preparing of n-methyl-11-aza-10-deoxo-10-dihydroerythromycine a and derivatives thereof
JPS58146595A (ja) * 1982-02-25 1983-09-01 Satoshi Omura マクロライド系抗生物質
US4454314A (en) * 1982-08-02 1984-06-12 Pfizer Inc. Antibacterial mycaminosyl tylonolide and related macrolide derivatives
US4443436A (en) * 1982-09-13 1984-04-17 Eli Lilly And Company C-20-Modified macrolide derivatives of the macrolide antibiotics tylosin, desmycosin, macrocin, and lactenocin
IL69666A (en) * 1982-09-13 1987-10-20 Lilly Co Eli 20-amino-20-deoxo-5-o-mycaminosyl-23-o-mycinosyltylonolide derivatives,their preparation and veterinary antibiotic use
US4468511A (en) * 1983-02-28 1984-08-28 Eli Lilly And Company C-20- And C-23-Modified macrolide derivatives

Also Published As

Publication number Publication date
PT84561A (en) 1987-04-01
DK154087D0 (da) 1987-03-26
ZA872201B (en) 1988-10-26
CN1018647B (zh) 1992-10-14
NZ219784A (en) 1989-01-27
KR900001166B1 (ko) 1990-02-27
JPH0710876B2 (ja) 1995-02-08
DE3772423D1 (de) 1991-10-02
HK82492A (en) 1992-10-30
HUT43087A (en) 1987-09-28
IE870796L (en) 1987-09-30
US4921947A (en) 1990-05-01
AU593894B2 (en) 1990-02-22
EG18550A (en) 1993-10-30
HU199864B (en) 1990-03-28
EP0240264A2 (en) 1987-10-07
JPS62240681A (ja) 1987-10-21
IL82005A0 (en) 1987-10-20
AR247402A1 (es) 1994-12-29
CN87102397A (zh) 1987-10-07
EP0240264B1 (en) 1991-08-28
CA1292737C (en) 1991-12-03
EP0240264A3 (en) 1987-11-19
KR870008906A (ko) 1987-10-21
AU7067087A (en) 1987-10-08
ES2028865T3 (es) 1992-07-16
DK154087A (da) 1987-10-01
GR3002764T3 (en) 1993-01-25
IE61018B1 (en) 1994-09-07
ATE66678T1 (de) 1991-09-15
IL82005A (en) 1991-08-16
DK172935B1 (da) 1999-10-11

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