ATE87926T1 - Ethylierte avermectine. - Google Patents

Ethylierte avermectine.

Info

Publication number
ATE87926T1
ATE87926T1 AT88310457T AT88310457T ATE87926T1 AT E87926 T1 ATE87926 T1 AT E87926T1 AT 88310457 T AT88310457 T AT 88310457T AT 88310457 T AT88310457 T AT 88310457T AT E87926 T1 ATE87926 T1 AT E87926T1
Authority
AT
Austria
Prior art keywords
avermectins
ethylated
cleandrose
ethoxy
sec
Prior art date
Application number
AT88310457T
Other languages
English (en)
Inventor
Steven Joseph Hawrylik
Shih-Jen Edward Lee
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Application granted granted Critical
Publication of ATE87926T1 publication Critical patent/ATE87926T1/de

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H19/00—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
    • C07H19/01—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing oxygen
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/90—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having two or more relevant hetero rings, condensed among themselves or with a common carbocyclic ring system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A61P33/10—Anthelmintics
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y10—TECHNICAL SUBJECTS COVERED BY FORMER USPC
    • Y10S—TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y10S435/00—Chemistry: molecular biology and microbiology
    • Y10S435/8215—Microorganisms
    • Y10S435/822—Microorganisms using bacteria or actinomycetales
    • Y10S435/886—Streptomyces

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Veterinary Medicine (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Molecular Biology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Biochemistry (AREA)
  • Biotechnology (AREA)
  • Genetics & Genomics (AREA)
  • Medicinal Chemistry (AREA)
  • Agronomy & Crop Science (AREA)
  • Pest Control & Pesticides (AREA)
  • Plant Pathology (AREA)
  • Dentistry (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Saccharide Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Fodder In General (AREA)
AT88310457T 1987-11-09 1988-11-07 Ethylierte avermectine. ATE87926T1 (de)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US11868487A 1987-11-09 1987-11-09
EP88310457A EP0316124B1 (de) 1987-11-09 1988-11-07 Ethylierte Avermectine

Publications (1)

Publication Number Publication Date
ATE87926T1 true ATE87926T1 (de) 1993-04-15

Family

ID=22380121

Family Applications (1)

Application Number Title Priority Date Filing Date
AT88310457T ATE87926T1 (de) 1987-11-09 1988-11-07 Ethylierte avermectine.

Country Status (10)

Country Link
US (1) US5387509A (de)
EP (1) EP0316124B1 (de)
JP (1) JPH0695947B2 (de)
AT (1) ATE87926T1 (de)
CA (1) CA1340771C (de)
DE (1) DE3880088T2 (de)
DK (1) DK621688A (de)
ES (1) ES2045146T3 (de)
IE (1) IE62446B1 (de)
PT (1) PT88952B (de)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6426333B1 (en) 1996-09-19 2002-07-30 Merial Spot-on formulations for combating parasites
GB8726730D0 (en) * 1987-11-14 1987-12-16 Pfizer Ltd Antiparasitic agents
EP0393890B1 (de) * 1989-04-11 1992-08-12 Pfizer Limited Injizierbare Arzneizubereitungen, die 25-Cyclohexylavermectin B1 enthalten
US6998131B2 (en) * 1996-09-19 2006-02-14 Merial Limited Spot-on formulations for combating parasites

Family Cites Families (19)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
SE434277B (sv) * 1976-04-19 1984-07-16 Merck & Co Inc Sett att framstella nya antihelmintiskt verkande foreningar genom odling av streptomyces avermitilis
PH15982A (en) * 1977-10-03 1983-05-18 Merck & Co Inc Selective hydrogenation producta of c-076 compounds and derivatives thereof
US4199569A (en) * 1977-10-03 1980-04-22 Merck & Co., Inc. Selective hydrogenation products of C-076 compounds and derivatives thereof
IL56149A (en) * 1977-12-19 1989-09-28 Merck & Co Inc 13-halo and 13-deoxy derivatives of c-076 compounds,their preparation and method for the treatment of parasitic infections in animals therewith
US4203976A (en) * 1978-08-02 1980-05-20 Merck & Co., Inc. Sugar derivatives of C-076 compounds
US4200581A (en) * 1978-08-04 1980-04-29 Merck & Co., Inc. Alkyl derivatives of C-076 compounds
US4429042A (en) * 1978-09-08 1984-01-31 Merck & Co., Inc. Strain of Streptomyces for producing antiparasitic compounds
US4328335A (en) * 1979-08-13 1982-05-04 Merck & Co., Inc. Process for the interconversion of C-076 compounds
US4285963A (en) * 1980-08-07 1981-08-25 Merck & Co., Inc. Novel derivatives of C-076 compounds
US4378353A (en) * 1981-02-17 1983-03-29 Merck & Co., Inc. Novel C-076 compounds
US4333925A (en) * 1981-05-11 1982-06-08 Merck & Co., Inc. Derivatives of C-076 compounds
US4423209A (en) * 1982-02-26 1983-12-27 Merck & Co., Inc. Processes for the interconversion of avermectin compounds
CH666690A5 (de) * 1984-09-14 1988-08-15 Glaxo Group Ltd Antibiotisch wirkende verbindungen der makrolidgruppe aus streptomyces-mikroorganismen, ihre herstellung und verwendung.
HUT39739A (en) * 1984-12-04 1986-10-29 Ciba Geigy Ag Process for production of derivatives of 13,3-milbemycin and medical preparatives containing thereof
IL78621A (en) * 1985-04-30 1991-06-30 American Cyanamid Co Mylbemycin analogs,their preparation and pesticidal compositions containing them
ES8800986A1 (es) * 1985-07-27 1987-12-01 Pfizer Un procedimiento para la produccion de un nuevo derivado de avermectina
EP0215654B1 (de) * 1985-09-13 1995-03-15 American Cyanamid Company Makrolide Antibiotika und Verfahren zu deren Herstellung
GB8606120D0 (en) * 1986-03-12 1986-04-16 Glaxo Group Ltd Process
US4831016A (en) * 1986-10-31 1989-05-16 Merck & Co., Inc. Reduced avermectin derivatives

Also Published As

Publication number Publication date
ES2045146T3 (es) 1994-01-16
CA1340771C (en) 1999-09-28
JPH0695947B2 (ja) 1994-11-30
PT88952B (pt) 1993-02-26
JPH01157986A (ja) 1989-06-21
IE62446B1 (en) 1995-02-08
DK621688A (da) 1989-07-06
EP0316124B1 (de) 1993-04-07
US5387509A (en) 1995-02-07
IE883358L (en) 1989-05-09
EP0316124A2 (de) 1989-05-17
DE3880088T2 (de) 1993-07-22
PT88952A (pt) 1988-12-01
EP0316124A3 (en) 1989-10-18
DE3880088D1 (de) 1993-05-13
DK621688D0 (da) 1988-11-08

Similar Documents

Publication Publication Date Title
DE3785198D1 (de) Liposomes praeparat und antibiotikum.
FI884341L (fi) Foerfarande och apparat foer belaeggning av glas med metalloxid.
FI884947A0 (fi) Tetrahydro-furo- och tieno/2,3-c/ pyridiner, deras anvaendning saosom laekemedel och foerfarande foer deras framstaellning.
FI860473L (fi) Nya -(2-okso-2,4,5,6,7,7a -hexahydro-tieno(3,2-c)-5-pyridyl)fenylaettiksyraderivat, foerfarande foer deras framstaellning och deras terapeutiska anvaendning.
FI891338A0 (fi) Parannus menetelmään 2',3'-dideoksi-2',3'-didehydronukleosidien valmistamiseksi
ATE162796T1 (de) 4-a-substutierte avermectinderivate
PT86800A (pt) Process for the preparation of erythromycin derivatives
FI903752A7 (fi) Menetelmä 1,2,3,4-tetrahydro-9-akridiiniamiinin johdannaisten valmistamiseksi
ES2086065T3 (es) Preparacion de tetrahidropiridinas sustituidas.
NO883447L (no) Stabilisert antracyklinpreparat.
FR2616429B1 (fr) Procede de preparation du 1,2,5,6,9,10-hexabromocyclododecane
DE3880088D1 (de) Ethylierte avermectine.
PT88493A (pt) Process for preparing milbemycin derivatives useful as antiparasitic agents
FI890612L (fi) Menetelmä 4-demetoksidaunomysinonin, joka on 4-demetoksidaunorubisiinin aglykoni, valmistamiseksi
DK360888D0 (da) 3',4'-dinitrogen-substituerede epipodophyllotoxinglucosidderivater
PT92270A (pt) Processo para a preparacao de solvatos de um antibiotico beta-lactamico
FI883812A0 (fi) 4'-deshydroxiepipodofyllotoxin -glukosider, syntes och anvaendning.
FI884461A7 (fi) Menetelmä trans-1,1,2-trifenyylibut-1-eenijohdannaisten valmistamiseksi
ATE18233T1 (de) De-(mycinosyloxy)-tylosin-derivate.
FI882465A7 (fi) Benzofuro (3,2-c) kinolinfoereningar.
ES551678A0 (es) Un procedimiento para la preparacion de un nuevo compuesto denominado sustancia n. 51262 por cultivo de un microorganismo del genero streptomyces
PT86624A (pt) Process for the preparation of cycloalkane-]1,2-c[4,3-c:" dipyrazoles
DE3588208D1 (de) Cephalosporinderivative
FI800410A7 (fi) Menetelmä alempi alkyyli 4,10-dihydro-10-oksotieno /3,2-c/ /l/- bentsoksepiini-8-asetaatin valmistamiseksi.
PT86745A (pt) Process for preparing oxime ethers of 2,6-dioxabicyclo ]3.3.o" octanones

Legal Events

Date Code Title Description
UEP Publication of translation of european patent specification
REN Ceased due to non-payment of the annual fee