ATE97128T1 - Sparsomycinderivate. - Google Patents

Sparsomycinderivate.

Info

Publication number: ATE97128T1
Authority: AT; Austria
Prior art keywords: carbon; group; alkyl; alkoxy; carbon alkyl
Prior art date: 1984-07-18

Application number

AT85108888T

Other languages

English (en)

Inventor

Douglas W Beight

Gary A Flynn

Original Assignee

Merrell Dow Pharma

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1984-07-18

Filing date

1985-07-16

Publication date

1993-11-15

1985-07-16 Application filed by Merrell Dow Pharma filed Critical Merrell Dow Pharma

1993-11-15 Application granted granted Critical

1993-11-15 Publication of ATE97128T1 publication Critical patent/ATE97128T1/de

Links

XKLZIVIOZDNKEQ-CLQLPEFOSA-N sparsomycin Chemical class CSC[S@](=O)C[C@H](CO)NC(=O)\C=C\C1=C(C)NC(=O)NC1=O XKLZIVIOZDNKEQ-CLQLPEFOSA-N 0.000 title abstract 2
229910052799 carbon Inorganic materials 0.000 abstract 10
-1 cyanomethyl carboxymethyl Chemical group 0.000 abstract 3
229910052739 hydrogen Inorganic materials 0.000 abstract 2
239000001257 hydrogen Substances 0.000 abstract 2
239000002253 acid Substances 0.000 abstract 1
125000003545 alkoxy group Chemical group 0.000 abstract 1
125000000217 alkyl group Chemical group 0.000 abstract 1
230000000844 anti-bacterial effect Effects 0.000 abstract 1
230000000842 anti-protozoal effect Effects 0.000 abstract 1
229940088710 antibiotic agent Drugs 0.000 abstract 1
229940036589 antiprotozoals Drugs 0.000 abstract 1
125000003236 benzoyl group Chemical group [H]C1=C([H])C([H])=C(C([H])=C1[H])C(*)=O 0.000 abstract 1
125000001797 benzyl group Chemical group [H]C1=C([H])C([H])=C(C([H])=C1[H])C([H])([H])* 0.000 abstract 1
125000004093 cyano group Chemical group *C#N 0.000 abstract 1
125000002425 furfuryl group Chemical group C(C1=CC=CO1)* 0.000 abstract 1
125000002541 furyl group Chemical group 0.000 abstract 1
229910052736 halogen Inorganic materials 0.000 abstract 1
150000002367 halogens Chemical class 0.000 abstract 1
150000002431 hydrogen Chemical group 0.000 abstract 1
125000004435 hydrogen atom Chemical group [H]* 0.000 abstract 1
125000004356 hydroxy functional group Chemical group O* 0.000 abstract 1
125000001841 imino group Chemical group [H]N=* 0.000 abstract 1
125000000449 nitro group Chemical group [O-][N+](*)=O 0.000 abstract 1
125000001997 phenyl group Chemical group [H]C1=C([H])C([H])=C(*)C([H])=C1[H] 0.000 abstract 1
125000004076 pyridyl group Chemical group 0.000 abstract 1
150000003839 salts Chemical class 0.000 abstract 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
- C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
- C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
- C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
- C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
- C07D239/52—Two oxygen atoms
- C07D239/54—Two oxygen atoms as doubly bound oxygen atoms or as unsubstituted hydroxy radicals
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents

Landscapes

Organic Chemistry (AREA)
Chemical & Material Sciences (AREA)
Health & Medical Sciences (AREA)
Veterinary Medicine (AREA)
Life Sciences & Earth Sciences (AREA)
Animal Behavior & Ethology (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Pharmacology & Pharmacy (AREA)
Public Health (AREA)
Chemical Kinetics & Catalysis (AREA)
General Health & Medical Sciences (AREA)
Tropical Medicine & Parasitology (AREA)
Communicable Diseases (AREA)
Oncology (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Saccharide Compounds (AREA)
Preparation Of Compounds By Using Micro-Organisms (AREA)
Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)

AT85108888T 1984-07-18 1985-07-16 Sparsomycinderivate. ATE97128T1 (de)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
US06/632,133 US4595687A (en)	1984-07-18	1984-07-18	Sparsomycin derivatives
EP85108888A EP0168813B1 (de)	1984-07-18	1985-07-16	Sparsomycinderivate

Publications (1)

Publication Number	Publication Date
ATE97128T1 true ATE97128T1 (de)	1993-11-15

Family

ID=24534214

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
AT85108888T ATE97128T1 (de)	1984-07-18	1985-07-16	Sparsomycinderivate.

Country Status (6)

Country	Link
US (2)	US4595687A (de)
EP (1)	EP0168813B1 (de)
JP (1)	JPS6140274A (de)
AT (1)	ATE97128T1 (de)
CA (1)	CA1250577A (de)
DE (1)	DE3587653T2 (de)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US4595687A (en) *	1984-07-18	1986-06-17	Merrell Dow Pharmaceuticals Inc.	Sparsomycin derivatives
US4808590A (en) *	1987-07-17	1989-02-28	Harbor Branch Oceanographic Institution, Inc.	Antiviral, antitumor and antifungal compositions and their methods of use
DE3903404A1 (de) *	1989-02-06	1990-08-09	Hoechst Ag	Pyrimidintrionderivate, verfahren zu ihrer herstellung, sie enthaltende mittel und ihre verwendung als schaedlingsbekaempfungsmittel
DE4401101A1 (de) *	1994-01-17	1995-07-20	Bayer Ag	Phenylthio-oxazolin-Derivate
CN100451006C (zh) *	2005-12-08	2009-01-14	南开大学	一种羧酰胺类化合物及其制备方法和用途

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
AU565425B2 (en) *	1982-11-01	1987-09-17	Stichting Katholieke Universiteit	Sparsomycin (sc-rs) derivative
US4595687A (en) *	1984-07-18	1986-06-17	Merrell Dow Pharmaceuticals Inc.	Sparsomycin derivatives

1984
- 1984-07-18 US US06/632,133 patent/US4595687A/en not_active Expired - Lifetime
1985
- 1985-07-15 CA CA000486836A patent/CA1250577A/en not_active Expired
- 1985-07-16 EP EP85108888A patent/EP0168813B1/de not_active Expired - Lifetime
- 1985-07-16 AT AT85108888T patent/ATE97128T1/de not_active IP Right Cessation
- 1985-07-16 DE DE85108888T patent/DE3587653T2/de not_active Expired - Fee Related
- 1985-07-17 JP JP15617785A patent/JPS6140274A/ja active Pending
1987
- 1987-02-24 US US07/018,765 patent/US4730044A/en not_active Expired - Lifetime

Also Published As

Publication number	Publication date
EP0168813B1 (de)	1993-11-10
DE3587653D1 (de)	1993-12-16
JPS6140274A (ja)	1986-02-26
EP0168813A1 (de)	1986-01-22
DE3587653T2 (de)	1994-04-07
US4595687A (en)	1986-06-17
CA1250577A (en)	1989-02-28
US4730044A (en)	1988-03-08

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Legal Events

Date	Code	Title	Description
1994-05-15	RER	Ceased as to paragraph 5 lit. 3 law introducing patent treaties