AU734734B2 - Local administration of phosphodiesterase inhibitors for the treatment of erectile dysfunction - Google Patents

Local administration of phosphodiesterase inhibitors for the treatment of erectile dysfunction Download PDF

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Publication number
AU734734B2
AU734734B2 AU11254/99A AU1125499A AU734734B2 AU 734734 B2 AU734734 B2 AU 734734B2 AU 11254/99 A AU11254/99 A AU 11254/99A AU 1125499 A AU1125499 A AU 1125499A AU 734734 B2 AU734734 B2 AU 734734B2
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AU
Australia
Prior art keywords
phosphodiesterase inhibitor
phosphodiesterase
type
formulation
drug
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Ceased
Application number
AU11254/99A
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English (en)
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AU1125499A (en
Inventor
Paul C. Doherty Jr.
Virgil A. Place
William L. Smith
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Vivus LLC
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Vivus LLC
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Filing date
Publication date
Priority claimed from US09/181,070 external-priority patent/US6037346A/en
Application filed by Vivus LLC filed Critical Vivus LLC
Publication of AU1125499A publication Critical patent/AU1125499A/en
Application granted granted Critical
Publication of AU734734B2 publication Critical patent/AU734734B2/en
Anticipated expiration legal-status Critical
Ceased legal-status Critical Current

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    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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    • A61K31/33—Heterocyclic compounds
    • A61K31/335—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
    • A61K31/34—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having five-membered rings with one oxygen as the only ring hetero atom, e.g. isosorbide
    • A61K31/343—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having five-membered rings with one oxygen as the only ring hetero atom, e.g. isosorbide condensed with a carbocyclic ring, e.g. coumaran, bufuralol, befunolol, clobenfurol, amiodarone
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    • A61K31/4015—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil having oxo groups directly attached to the heterocyclic ring, e.g. piracetam, ethosuximide
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  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Urology & Nephrology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
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AU11254/99A 1997-10-28 1998-10-28 Local administration of phosphodiesterase inhibitors for the treatment of erectile dysfunction Ceased AU734734B2 (en)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US95881697A 1997-10-28 1997-10-28
US08/958816 1997-10-28
US09/181,070 US6037346A (en) 1997-10-28 1998-10-27 Local administration of phosphodiesterase inhibitors for the treatment of erectile dysfunction
US09/181070 1998-10-27
PCT/US1998/022928 WO1999021558A2 (fr) 1997-10-28 1998-10-28 Apport local d'inhibiteurs de phosphodiesterases, dans le traitement du dysfonctionnement erectile

Publications (2)

Publication Number Publication Date
AU1125499A AU1125499A (en) 1999-05-17
AU734734B2 true AU734734B2 (en) 2001-06-21

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AU11254/99A Ceased AU734734B2 (en) 1997-10-28 1998-10-28 Local administration of phosphodiesterase inhibitors for the treatment of erectile dysfunction

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EP (1) EP1027054A4 (fr)
JP (1) JP2003525845A (fr)
AU (1) AU734734B2 (fr)
CA (1) CA2305394C (fr)
WO (1) WO1999021558A2 (fr)

Families Citing this family (30)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6331543B1 (en) 1996-11-01 2001-12-18 Nitromed, Inc. Nitrosated and nitrosylated phosphodiesterase inhibitors, compositions and methods of use
AU742787B2 (en) 1997-07-09 2002-01-10 Androsolutions, Inc. Improved methods and compositions for treating male erectile dysfunction
US6103765A (en) 1997-07-09 2000-08-15 Androsolutions, Inc. Methods for treating male erectile dysfunction
US6548490B1 (en) 1997-10-28 2003-04-15 Vivus, Inc. Transmucosal administration of phosphodiesterase inhibitors for the treatment of erectile dysfunction
US6403597B1 (en) 1997-10-28 2002-06-11 Vivus, Inc. Administration of phosphodiesterase inhibitors for the treatment of premature ejaculation
US6472425B1 (en) 1997-10-31 2002-10-29 Nitromed, Inc. Methods for treating female sexual dysfunctions
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CA2305394C (fr) 2006-12-12
AU1125499A (en) 1999-05-17
JP2003525845A (ja) 2003-09-02
EP1027054A4 (fr) 2002-11-04
EP1027054A1 (fr) 2000-08-16
WO1999021558A3 (fr) 2000-10-26
CA2305394A1 (fr) 1999-05-06
WO1999021558A2 (fr) 1999-05-06

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