BE2018C028I2 - - Google Patents
Info
- Publication number
- BE2018C028I2 BE2018C028I2 BE2018C028C BE2018C028C BE2018C028I2 BE 2018C028 I2 BE2018C028 I2 BE 2018C028I2 BE 2018C028 C BE2018C028 C BE 2018C028C BE 2018C028 C BE2018C028 C BE 2018C028C BE 2018C028 I2 BE2018C028 I2 BE 2018C028I2
- Authority
- BE
- Belgium
Links
Classifications
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/4353—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
- A61K31/437—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems the heterocyclic ring system containing a five-membered ring having nitrogen as a ring hetero atom, e.g. indolizine, beta-carboline
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- A—HUMAN NECESSITIES
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/02—Stomatological preparations, e.g. drugs for caries, aphtae, periodontitis
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
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- A—HUMAN NECESSITIES
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- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/16—Drugs for disorders of the alimentary tract or the digestive system for liver or gallbladder disorders, e.g. hepatoprotective agents, cholagogues, litholytics
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- A—HUMAN NECESSITIES
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- A61P1/18—Drugs for disorders of the alimentary tract or the digestive system for pancreatic disorders, e.g. pancreatic enzymes
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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- A—HUMAN NECESSITIES
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- A—HUMAN NECESSITIES
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- A—HUMAN NECESSITIES
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- A—HUMAN NECESSITIES
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- A—HUMAN NECESSITIES
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- A—HUMAN NECESSITIES
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- A61P7/04—Antihaemorrhagics; Procoagulants; Haemostatic agents; Antifibrinolytic agents
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Organic Chemistry (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- Veterinary Medicine (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Biomedical Technology (AREA)
- Virology (AREA)
- Diabetes (AREA)
- Immunology (AREA)
- Endocrinology (AREA)
- Physical Education & Sports Medicine (AREA)
- Oncology (AREA)
- Pulmonology (AREA)
- Communicable Diseases (AREA)
- Urology & Nephrology (AREA)
- Reproductive Health (AREA)
- Hematology (AREA)
- Rheumatology (AREA)
- Pain & Pain Management (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Ophthalmology & Optometry (AREA)
- Molecular Biology (AREA)
- Pregnancy & Childbirth (AREA)
- Psychiatry (AREA)
- Nutrition Science (AREA)
- Addiction (AREA)
- Obesity (AREA)
- Gynecology & Obstetrics (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US66059205P | 2005-03-11 | 2005-03-11 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| BE2018C028I2 true BE2018C028I2 (es) | 2025-09-05 |
Family
ID=36649530
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| BE2018C028C BE2018C028I2 (es) | 2005-03-11 | 2018-07-05 |
Country Status (23)
| Country | Link |
|---|---|
| US (1) | US7960407B2 (es) |
| EP (1) | EP1861400B1 (es) |
| JP (1) | JP5069415B2 (es) |
| KR (1) | KR100911073B1 (es) |
| CN (1) | CN101137656B (es) |
| AR (1) | AR055567A1 (es) |
| AT (1) | ATE469150T1 (es) |
| AU (1) | AU2006221699A1 (es) |
| BE (1) | BE2018C028I2 (es) |
| BR (1) | BRPI0608819B8 (es) |
| CA (1) | CA2600510C (es) |
| DE (1) | DE602006014516D1 (es) |
| ES (1) | ES2344310T3 (es) |
| FR (1) | FR18C1028I2 (es) |
| IL (1) | IL185145A0 (es) |
| IN (1) | IN2014DN09939A (es) |
| MX (1) | MX2007011110A (es) |
| NL (1) | NL300944I2 (es) |
| PL (1) | PL1861400T3 (es) |
| RU (1) | RU2357968C1 (es) |
| TW (1) | TW200643021A (es) |
| WO (1) | WO2006095268A1 (es) |
| ZA (1) | ZA200707568B (es) |
Families Citing this family (22)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| MX2011003166A (es) | 2008-09-25 | 2011-04-27 | Merck Frosst Canada Ltd | Derivados de sulfonilurea beta-carbolina como antagonistas del receptor ep4. |
| CA2754702C (en) * | 2009-04-22 | 2016-06-07 | Yukinori Take | Selective ep4 antagonistic substance for treatment of cancer |
| CA2789665C (en) * | 2010-02-22 | 2020-06-16 | Askat Inc. | Use of ep4 receptor antagonists in the treatment of il-23 mediated diseases |
| RU2451680C1 (ru) | 2011-02-21 | 2012-05-27 | Общество С Ограниченной Ответственностью "Научно-Исследовательская Компания "Медбиофарм" | Клатратный комплекс циклодекстрина или арабиногалактана с 9-фенил-симм-октагидроселеноксантеном, способ его получения (варианты), фармацевтическая композиция и лекарственное средство |
| RU2464042C1 (ru) * | 2011-03-31 | 2012-10-20 | Общество С Ограниченной Ответственностью "Научно-Исследовательская Компания "Медбиофарм" | КЛАТРАТНЫЙ КОМПЛЕКС β-ЦИКЛОДЕКСТРИНА С ПРОИЗВОДНЫМ 5-ГИДРОКСИ-4-АМИНОМЕТИЛ-1-ЦИКЛОГЕКСИЛ(ИЛИ ЦИКЛОГЕПТИЛ)-3-АЛКОКСИКАРБОНИЛИНДОЛА, СПОСОБ ЕГО ПОЛУЧЕНИЯ (ВАРИАНТЫ), ФАРМАЦЕВТИЧЕСКАЯ КОМПОЗИЦИЯ И ЛЕКАРСТВЕННОЕ СРЕДСТВО |
| US10391086B2 (en) | 2013-03-19 | 2019-08-27 | Askat Inc. | Use of EP4 receptor antagonists in the treatment of cartilage disease |
| KR20150130404A (ko) * | 2013-03-19 | 2015-11-23 | 에스크엣 인크. | 연골질환 치료에서의 ep4 수용체 길항제의 용도 |
| US12109218B2 (en) | 2014-12-09 | 2024-10-08 | Aratana Therapeutics, Inc. | Compositions of grapiprant and methods for using the same |
| TWI664969B (zh) | 2014-03-06 | 2019-07-11 | 雅瑞塔那醫療公司 | 格拉匹綸(ｇｒａｐｉｐｒａｎｔ)組合物及其使用方法 |
| CA2997692A1 (en) * | 2014-03-06 | 2015-09-11 | Aratana Therapeutics, Inc. | Crystalline forms of grapiprant |
| US10342785B2 (en) | 2016-11-04 | 2019-07-09 | Askat Inc. | Use of EP4 receptor antagonists for the treatment of NASH-associated liver cancer |
| CN112292128A (zh) | 2018-04-16 | 2021-01-29 | 阿瑞斯医疗有限公司 | Ep4抑制剂和其用途 |
| WO2019245590A1 (en) | 2018-06-18 | 2019-12-26 | Avista Pharma Solutions, Inc. | Chemical compounds |
| US20210315909A1 (en) * | 2018-07-11 | 2021-10-14 | Arrys Therapeutics, Inc. | Polymorphic compounds and uses thereof |
| IL280051B2 (en) * | 2018-07-11 | 2024-03-01 | Arrys Therapeutics Inc | EP4 inhibitors and their synthesis |
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| US11512088B2 (en) | 2019-01-30 | 2022-11-29 | Avista Pharma Solutions, Inc. | Synthetic process and intermediates |
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| WO2021226162A1 (en) | 2020-05-05 | 2021-11-11 | Arrys Therapeutics, Inc. | Ep4 antagonists and their use in the treatment of proliferative diseases |
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| CN116478155B (zh) * | 2022-01-17 | 2025-06-13 | 洛阳惠中兽药有限公司 | 一种格拉匹伦及其中间体的制备方法 |
| CN117800905A (zh) * | 2022-09-26 | 2024-04-02 | 洛阳惠中兽药有限公司 | 4-(2,6-二甲基-3-硝基吡啶-4-基氨基)苯乙基氨基甲酸苄基酯的制备方法 |
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| IL110296A (en) * | 1993-07-16 | 1999-12-31 | Smithkline Beecham Corp | Imidazole compounds process for their preparation and pharmaceutical compositions containing them |
| HN2001000224A (es) | 2000-10-19 | 2002-06-13 | Pfizer | Compuestos de imidazol condensado con arilo o heteroarilo como agentes anti - inflamatorios y analgesicos. |
| BR0309200A (pt) * | 2002-04-12 | 2005-02-22 | Pfizer | Uso de ligandos receptores ep4 no tratamento de doenças envolvidas com a il-6 |
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- 2006-03-01 PL PL06710609T patent/PL1861400T3/pl unknown
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- 2007-09-03 ZA ZA200707568A patent/ZA200707568B/xx unknown
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2018
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| BRPI0608819B1 (pt) | 2019-11-12 |
| IN2014DN09939A (es) | 2015-08-14 |
| WO2006095268A1 (en) | 2006-09-14 |
| DE602006014516D1 (es) | 2010-07-08 |
| CN101137656B (zh) | 2010-12-22 |
| PL1861400T3 (pl) | 2010-09-30 |
| BRPI0608819A2 (pt) | 2010-01-26 |
| FR18C1028I2 (fr) | 2019-07-19 |
| ES2344310T3 (es) | 2010-08-24 |
| CA2600510A1 (en) | 2006-09-14 |
| ZA200707568B (en) | 2009-09-30 |
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| AR055567A1 (es) | 2007-08-22 |
| KR20070103484A (ko) | 2007-10-23 |
| JP2006249089A (ja) | 2006-09-21 |
| TW200643021A (en) | 2006-12-16 |
| RU2007133802A (ru) | 2009-03-20 |
| ATE469150T1 (de) | 2010-06-15 |
| BRPI0608819B8 (pt) | 2021-05-25 |
| RU2357968C1 (ru) | 2009-06-10 |
| CN101137656A (zh) | 2008-03-05 |
| NL300944I2 (nl) | 2018-08-07 |
| EP1861400B1 (en) | 2010-05-26 |
| US20090018158A1 (en) | 2009-01-15 |
| KR100911073B1 (ko) | 2009-08-06 |
| AU2006221699A1 (en) | 2006-09-14 |
| BRPI0608819A8 (pt) | 2017-10-10 |
| US7960407B2 (en) | 2011-06-14 |
| IL185145A0 (en) | 2007-12-03 |
| CA2600510C (en) | 2010-11-02 |
| EP1861400A1 (en) | 2007-12-05 |
| MX2007011110A (es) | 2008-02-21 |