BE768137A - Derives de piperazinyl-alcoyl-quinazolone-(4), leur procede de preparation et medicaments en contenant - Google Patents

Derives de piperazinyl-alcoyl-quinazolone-(4), leur procede de preparation et medicaments en contenant

Info

Publication number
BE768137A
BE768137A BE768137A BE768137A BE768137A BE 768137 A BE768137 A BE 768137A BE 768137 A BE768137 A BE 768137A BE 768137 A BE768137 A BE 768137A BE 768137 A BE768137 A BE 768137A
Authority
BE
Belgium
Prior art keywords
alcoyl
quinazolone
piperazinyl
derivatives
preparation process
Prior art date
Application number
BE768137A
Other languages
English (en)
Inventor
H Amschler
W Schoetensack
K Klemm
Original Assignee
Byk Gulden Lomberg Chem Fab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Byk Gulden Lomberg Chem Fab filed Critical Byk Gulden Lomberg Chem Fab
Publication of BE768137A publication Critical patent/BE768137A/fr

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
BE768137A 1970-06-05 1971-06-04 Derives de piperazinyl-alcoyl-quinazolone-(4), leur procede de preparation et medicaments en contenant BE768137A (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE19702027645 DE2027645A1 (de) 1970-06-05 1970-06-05 Piperazinylalkyl chinazolon (4) den vate, Verfahren zu deren Herstellung und sie enthaltende Arzneimittel

Publications (1)

Publication Number Publication Date
BE768137A true BE768137A (fr) 1971-12-06

Family

ID=5773104

Family Applications (1)

Application Number Title Priority Date Filing Date
BE768137A BE768137A (fr) 1970-06-05 1971-06-04 Derives de piperazinyl-alcoyl-quinazolone-(4), leur procede de preparation et medicaments en contenant

Country Status (10)

Country Link
US (1) US3984555A (fr)
AT (3) AT318628B (fr)
BE (1) BE768137A (fr)
CA (1) CA951319A (fr)
CH (3) CH569732A5 (fr)
DE (1) DE2027645A1 (fr)
FR (1) FR2100726B1 (fr)
GB (1) GB1331522A (fr)
LU (1) LU63267A1 (fr)
NL (1) NL7107695A (fr)

Families Citing this family (32)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4287341A (en) * 1979-11-01 1981-09-01 Pfizer Inc. Alkoxy-substituted-6-chloro-quinazoline-2,4-diones
US6723727B1 (en) * 1996-12-20 2004-04-20 Hoechst Aktiengesellschaft Substituted purine derivatives, processes for their preparation, their use, and compositions comprising them
US5972929A (en) * 1997-08-21 1999-10-26 Shiseido Co., Ltd. Quinazolinone derivative, hair growth promoter and external composition for skin using the same
EP1216243A1 (fr) * 1999-10-01 2002-06-26 Advanced Medicine, Inc. Quinazolinones et analogues et leur utilisation comme anesthesiques locaux
US6667300B2 (en) 2000-04-25 2003-12-23 Icos Corporation Inhibitors of human phosphatidylinositol 3-kinase delta
ES2788383T3 (es) * 2000-04-25 2020-10-21 Icos Corp Inhibidores de delta fosfatidilo-inositol 3-quinasa humana
AUPR201600A0 (en) * 2000-12-11 2001-01-11 Fujisawa Pharmaceutical Co., Ltd. Quinazolinone derivative
JP2005507876A (ja) 2001-09-05 2005-03-24 ミナーバ バイオテクノロジーズ コーポレイション 癌を治療する組成物および方法
EP1434584A2 (fr) * 2001-09-05 2004-07-07 Minerva Biotechnologies Corporation Compositions et methodes de traitement du cancer
CA2465491A1 (fr) * 2001-11-07 2003-05-15 Merck & Co., Inc. Inhibiteurs de la kinesine mitotique
AUPS019702A0 (en) * 2002-01-29 2002-02-21 Fujisawa Pharmaceutical Co., Ltd. Condensed heterocyclic compounds
US20040048853A1 (en) * 2002-08-21 2004-03-11 Gustave Bergnes Compounds, compositions, and methods
CA2502302A1 (fr) * 2002-11-04 2004-05-21 Nps Pharmaceuticals, Inc. Composes de quinazolinone utilises comme calcilytiques
DE602004022819D1 (de) * 2003-06-06 2009-10-08 Vertex Pharma Von atp-bindende kassette transportern
WO2005016348A1 (fr) * 2003-08-14 2005-02-24 Icos Corporation Methodes d'inhibition de reponses immunes stimulees par un facteur endogene
US20050054614A1 (en) * 2003-08-14 2005-03-10 Diacovo Thomas G. Methods of inhibiting leukocyte accumulation
SI2612862T1 (sl) 2004-05-13 2017-04-26 Icos Corporation Kinazolini kot inhibitorji humane fosfatidilinozitol 3-kinaze delta
JP2008500338A (ja) * 2004-05-25 2008-01-10 イコス・コーポレイション 造血細胞の異常増殖を治療及び／又は予防する方法
WO2006089106A2 (fr) * 2005-02-17 2006-08-24 Icos Corporation Procede d'inhibition d'accumulation de leucocytes
EP2010505B1 (fr) * 2006-03-28 2012-12-05 Atir Holding S.A. Composés hétérocycliques et leurs utilisations dans le traitement de troubles sexuels
CN102271683B (zh) 2008-11-13 2014-07-09 吉里德卡利斯托加公司 恶性血液病的治疗
US9492449B2 (en) 2008-11-13 2016-11-15 Gilead Calistoga Llc Therapies for hematologic malignancies
CA2756347A1 (fr) 2009-03-24 2010-09-30 Gilead Calistoga Llc Atropisomeres de derives de 2-purinyl-3-tolyl-quinazolinone et procedes d'utilisation
CN102458410A (zh) * 2009-04-20 2012-05-16 吉联亚·卡利斯托加有限责任公司 治疗实体瘤的方法
EA201270184A1 (ru) 2009-07-21 2012-08-30 ГИЛИЭД КАЛИСТОГА ЭлЭлСи Лечение расстройств печени ингибиторами pi3k
BRPI1003506B1 (pt) 2010-09-24 2019-12-03 Ache Int Bvi Ltd composto alquil-piperazino-fenil-4(3h)quinazolinonas e uso do composto alquil-piperazino-fenil-4(3h)quinazolinonas associado aos receptores serotoninérgicos 5-ht1a e 5-ht2a
WO2012140642A1 (fr) * 2011-04-10 2012-10-18 Atir Holding S.A. Composés hétérocycliques et leurs utilisations dans le traitement de troubles sexuels
SI2834241T1 (sl) 2012-03-05 2021-06-30 Gilead Calistoga Llc Polimorfne oblike (S)-2-(1-(9H-purin-6-ilamino)propil)-5-fluoro-3-fenilkinazolin-4(3H)-ONA
ES2595240T3 (es) 2012-07-09 2016-12-28 Lupin Limited Derivados de tetrahidroquinazolinona como inhibidores de PARP
WO2015095601A1 (fr) 2013-12-20 2015-06-25 Gilead Calistoga Llc Procédés de synthèse d'inhibiteurs de la phosphatidylinositol 3-kinase
US9708327B2 (en) 2013-12-20 2017-07-18 Gilead Calistoga Llc Polymorphic forms of a hydrochloride salt of (S)-2-(1-(9H-purin-6-ylamino)propyl)-5-fluoro-3-phenylquinazolin-4(3H)-one
EP3154960A1 (fr) 2014-06-13 2017-04-19 Gilead Sciences, Inc. Inhibiteurs de la phosphatidylinositol 3-kinase

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1053063A (fr) * 1963-05-18

Also Published As

Publication number Publication date
FR2100726A1 (fr) 1972-03-24
CH557829A (de) 1975-01-15
GB1331522A (en) 1973-09-26
CH569732A5 (fr) 1975-11-28
FR2100726B1 (fr) 1975-10-10
CH558374A (de) 1975-01-31
DE2027645A1 (de) 1971-12-09
US3984555A (en) 1976-10-05
AT317899B (de) 1974-09-25
LU63267A1 (fr) 1972-08-23
CA951319A (en) 1974-07-16
AT318628B (de) 1974-11-11
NL7107695A (fr) 1971-12-07
AT318615B (de) 1974-11-11

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