|
FI824314L
(fi)
*
|
1981-12-16 |
1983-06-17 |
Sankyo Co |
Thienopyrimidin-derivater, deras framstaellning och deras medicinska anvaendning
|
|
JPS60146891A
(ja)
*
|
1984-01-05 |
1985-08-02 |
Mitsubishi Chem Ind Ltd |
〔2,3−d〕チエノピリミジン誘導体およびその塩
|
|
WO1986006721A1
(fr)
*
|
1985-05-07 |
1986-11-20 |
Alkaloida Vegyészeti Gyár |
Derives de triazolyl-quinoline
|
|
US4670560A
(en)
*
|
1986-04-28 |
1987-06-02 |
Ortho Pharmaceutical Corporation |
Thienopyrimidine-2,4-dione derivatives and intermediates thereof
|
|
WO1989008113A1
(fr)
*
|
1988-03-02 |
1989-09-08 |
Yoshitomi Pharmaceutical Industries, Ltd. |
COMPOSES DE 3,4-DIHYDROTHIENO[2,3-d]PYRIMIDINE ET LEURS APPLICATIONS PHARMACOLOGIQUES
|
|
US5280026A
(en)
*
|
1989-05-30 |
1994-01-18 |
Smithkline Beecham Intercredit B.V. |
Thienopyrimidines
|
|
GB8912335D0
(en)
*
|
1989-05-30 |
1989-07-12 |
Smithkline Beckman Intercredit |
Compounds
|
|
DE4008726A1
(de)
*
|
1990-03-19 |
1991-09-26 |
Basf Ag |
Thieno(2,3-d)pyrimidinderivate
|
|
AU651337B2
(en)
*
|
1990-03-30 |
1994-07-21 |
Dowelanco |
Thienopyrimidine derivatives
|
|
US5869486A
(en)
*
|
1995-02-24 |
1999-02-09 |
Ono Pharmaceutical Co., Ltd. |
Fused pyrimidines and pyriazines as pharmaceutical compounds
|
|
PT757984E
(pt)
*
|
1995-08-08 |
2003-02-28 |
Ono Pharmaceutical Co |
Derivados de acido hidroxamico uteis para inibir a gelatinase
|
|
DE19632423A1
(de)
*
|
1996-08-12 |
1998-02-19 |
Merck Patent Gmbh |
Thienopyrimidine
|
|
DE19650378A1
(de)
*
|
1996-12-05 |
1998-06-10 |
Basf Ag |
Neue Pyrimidylverbindungen als Pflanzenschutzmittel
|
|
AU5698398A
(en)
*
|
1996-12-18 |
1998-07-15 |
Eli Lilly And Company |
Combinatorial process for preparing fused pyrimidine libraries
|
|
US20030162795A1
(en)
*
|
1998-10-22 |
2003-08-28 |
Pfizer Inc. |
Thienopyrimidine and thienopyridine derivatives useful as anticancer agents
|
|
US6133271A
(en)
*
|
1998-11-19 |
2000-10-17 |
Cell Pathways, Inc. |
Method for inhibiting neoplastic cells and related conditions by exposure thienopyrimidine derivatives
|
|
US6608053B2
(en)
*
|
2000-04-27 |
2003-08-19 |
Yamanouchi Pharmaceutical Co., Ltd. |
Fused heteroaryl derivatives
|
|
US6503914B1
(en)
*
|
2000-10-23 |
2003-01-07 |
Board Of Regents, The University Of Texas System |
Thienopyrimidine-based inhibitors of the Src family
|
|
MXPA03009925A
(es)
*
|
2001-04-30 |
2004-06-30 |
Bayer Pharmaceuticals Corp |
Nuevas tiofeno [2,3-d]pirimidinas 4-amino-5,6-sustituidas.
|
|
US6805491B2
(en)
*
|
2002-05-20 |
2004-10-19 |
Stratos International, Inc. |
Stub having an optical fiber
|
|
AR044743A1
(es)
*
|
2002-09-26 |
2005-10-05 |
Nihon Nohyaku Co Ltd |
Herbicida, metodo de emplearlo, derivados de tienopirimidina sustituida,compuestos intermediarios, y procedimientos que se utilizan para producirlos,
|
|
US20050222175A1
(en)
*
|
2004-03-31 |
2005-10-06 |
Dhanoa Dale S |
New piperidinylamino-thieno[2,3-D] pyrimidine compounds
|
|
US7612078B2
(en)
*
|
2003-03-31 |
2009-11-03 |
Epix Delaware, Inc. |
Piperidinylamino-thieno[2,3-D] pyrimidine compounds
|
|
NZ542236A
(en)
*
|
2003-03-31 |
2008-05-30 |
Predix Pharmaceuticals Holding |
New piperidinylamino-thieno[2,3-d]pyrimidine compounds
|
|
GB0315950D0
(en)
|
2003-06-11 |
2003-08-13 |
Xention Discovery Ltd |
Compounds
|
|
US7488736B2
(en)
*
|
2004-05-17 |
2009-02-10 |
Epix Delaware, Inc. |
Thienopyridinone compounds and methods of treatment
|
|
GB0412467D0
(en)
*
|
2004-06-04 |
2004-07-07 |
Astrazeneca Ab |
Chemical compounds
|
|
GB0412986D0
(en)
|
2004-06-10 |
2004-07-14 |
Xention Discovery Ltd |
Compounds
|
|
MX2007000631A
(es)
*
|
2004-07-16 |
2007-03-30 |
Sunesis Pharmaceuticals Inc |
Tienopirimidinas utiles como inhibidores de aurora cinasa.
|
|
GB0420719D0
(en)
*
|
2004-09-17 |
2004-10-20 |
Addex Pharmaceuticals Sa |
Novel allosteric modulators
|
|
US7407966B2
(en)
*
|
2004-10-07 |
2008-08-05 |
Epix Delaware, Inc. |
Thienopyridinone compounds and methods of treatment
|
|
US7598265B2
(en)
*
|
2004-09-30 |
2009-10-06 |
Epix Delaware, Inc. |
Compositions and methods for treating CNS disorders
|
|
US7576211B2
(en)
*
|
2004-09-30 |
2009-08-18 |
Epix Delaware, Inc. |
Synthesis of thienopyridinone compounds and related intermediates
|
|
US7557112B2
(en)
*
|
2004-10-08 |
2009-07-07 |
Astellas Pharma Inc. |
Aromatic-ring-fused pyrimidine derivative
|
|
US8008487B2
(en)
*
|
2004-10-21 |
2011-08-30 |
Dow Agrosciences Llc |
Substituted thieno[2,3-D]pyrimidines as fungicides
|
|
GB0423653D0
(en)
|
2004-10-25 |
2004-11-24 |
Piramed Ltd |
Pharmaceutical compounds
|
|
US7576212B2
(en)
|
2004-12-09 |
2009-08-18 |
Xention Limited |
Thieno[2,3-B] pyridines as potassium channel inhibitors
|
|
US7576080B2
(en)
*
|
2004-12-23 |
2009-08-18 |
Memory Pharmaceuticals Corporation |
Certain thienopyrimidine derivatives as phosphodiesterase 10 inhibitors
|
|
US7816351B2
(en)
*
|
2005-09-23 |
2010-10-19 |
Equispharm Co., Ltd |
5,6-dimethylthieno[2,3-di] pyrimidine derivatives, the preparation method thereof and the pharmaceutical composition comprising the same for anti-virus
|
|
EP1937691A1
(fr)
|
2005-10-21 |
2008-07-02 |
Dow Agrosciences LLC |
Composes de thieno-pyrimidine a activite fongicide
|
|
US7531482B2
(en)
*
|
2005-10-21 |
2009-05-12 |
Dow Agrosciences Llc |
Thieno-pyrimidine compounds having fungicidal activity
|
|
WO2007056214A2
(fr)
*
|
2005-11-02 |
2007-05-18 |
Cytovia, Inc |
N-alkyl-n-aryl-thienopyrimidin-4-amines et analogues en tant qu'activateurs de caspases et inducteurs d'apoptose et utilisation associee
|
|
US20070099877A1
(en)
*
|
2005-11-02 |
2007-05-03 |
Cytovia, Inc. |
N-aryl-thienopyrimidin-4-amines and analogs as activators of caspases and inducers of apoptosis and the use thereof
|
|
WO2007056208A2
(fr)
*
|
2005-11-02 |
2007-05-18 |
Cytovia, Inc. |
N-arylalkyl-thienopyrimidin-4-amines et analogues en tant qu'activateurs de caspases et inducteurs d'apoptose et utilisation de ceux-ci
|
|
GB0525164D0
(en)
|
2005-12-09 |
2006-01-18 |
Xention Discovery Ltd |
Compounds
|
|
AR059898A1
(es)
|
2006-03-15 |
2008-05-07 |
Janssen Pharmaceutica Nv |
Derivados de 3-ciano-piridona 1,4-disustituida y su uso como moduladores alostericos de los receptores mglur2
|
|
WO2007129161A2
(fr)
*
|
2006-04-26 |
2007-11-15 |
F. Hoffmann-La Roche Ag |
Composés pharmaceutiques
|
|
TWI498332B
(zh)
*
|
2006-04-26 |
2015-09-01 |
Hoffmann La Roche |
作為pi3k抑制劑之嘧啶衍生物及相關製備方法、醫藥組合物、用途、套組及產物
|
|
TW200801012A
(en)
|
2006-04-26 |
2008-01-01 |
Piramed Ltd |
Phosphoinositide 3-kinase inhibitor compounds and methods of use
|
|
AP2008004687A0
(en)
|
2006-05-22 |
2008-12-31 |
Basf Se |
Insecticidal methods using 4-amino-5-chloro-thieno(2,3-d)-pyrimidine compounds
|
|
MX2009005950A
(es)
*
|
2006-12-07 |
2009-10-12 |
Genentech Inc |
Compuestos inhibidores de fosfoinositido 3-quinasas y metodos de uso.
|
|
RU2470936C2
(ru)
*
|
2006-12-07 |
2012-12-27 |
Дженентек, Инк. |
Соединения-ингибиторы фосфоинозитид 3-киназы и способы применения
|
|
TW200900065A
(en)
|
2007-03-07 |
2009-01-01 |
Janssen Pharmaceutica Nv |
3-cyano-4-(4-pyridinyloxy-phenyl)-pyridin-2-one derivatives
|
|
TW200845978A
(en)
*
|
2007-03-07 |
2008-12-01 |
Janssen Pharmaceutica Nv |
3-cyano-4-(4-tetrahydropyran-phenyl)-pyridin-2-one derivatives
|
|
US9603848B2
(en)
*
|
2007-06-08 |
2017-03-28 |
Senomyx, Inc. |
Modulation of chemosensory receptors and ligands associated therewith
|
|
US8633186B2
(en)
|
2007-06-08 |
2014-01-21 |
Senomyx Inc. |
Modulation of chemosensory receptors and ligands associated therewith
|
|
US7928111B2
(en)
*
|
2007-06-08 |
2011-04-19 |
Senomyx, Inc. |
Compounds including substituted thienopyrimidinone derivatives as ligands for modulating chemosensory receptors
|
|
SI2203439T1
(sl)
|
2007-09-14 |
2011-05-31 |
Ortho Mcneil Janssen Pharm |
1',3'-disubstituirani 4-fenil-3,4,5,6-tetrahidro-2H-1'H-(1,4')bipiridinil-2'-oni
|
|
CN101801930B
(zh)
*
|
2007-09-14 |
2013-01-30 |
奥梅-杨森制药有限公司 |
1,3-二取代的-4-苯基-1h-吡啶-2-酮
|
|
PL2200985T3
(pl)
|
2007-09-14 |
2011-12-30 |
Ortho Mcneil Janssen Pharmaceuticals Inc |
1,3-Dipodstawione-4-(arylo-X-fenylo)-1H-pirydyn-2-ony
|
|
JP5348725B2
(ja)
*
|
2007-10-25 |
2013-11-20 |
ジェネンテック, インコーポレイテッド |
チエノピリミジン化合物の製造方法
|
|
GB0721095D0
(en)
*
|
2007-10-26 |
2007-12-05 |
Piramed Ltd |
Pharmaceutical compounds
|
|
CN101861316B
(zh)
*
|
2007-11-14 |
2013-08-21 |
奥梅-杨森制药有限公司 |
咪唑并[1,2-a]吡啶衍生物及其作为MGLUR2受体的正变构调节剂的用途
|
|
WO2010014813A2
(fr)
|
2008-07-31 |
2010-02-04 |
Senomyx, Inc. |
Compositions comprenant des édulcorants et leurs procédés de préparation
|
|
ES2915065T3
(es)
|
2008-07-31 |
2022-06-20 |
Firmenich Incorporated |
Procedimientos para hacer potenciadores del sabor dulce
|
|
EP2344470B1
(fr)
|
2008-09-02 |
2013-11-06 |
Janssen Pharmaceuticals, Inc. |
Dérivés de 3-azabicyclo[3.1.0]hexyle comme modulateurs des récepteurs métabotropiques du glutamate
|
|
WO2010043396A1
(fr)
|
2008-10-16 |
2010-04-22 |
Ortho-Mcneil-Janssen Pharmaceuticals, Inc. |
Dérivés d’indole et de benzomorpholine en tant que modulateurs des récepteurs métabotropiques du glutamate
|
|
JP5690277B2
(ja)
|
2008-11-28 |
2015-03-25 |
ジャンセン ファーマシューティカルズ, インコーポレイテッド. |
代謝型グルタミン酸受容体の調節因子としてのインドールおよびベンゾオキサジン誘導体
|
|
US8114894B2
(en)
*
|
2008-12-03 |
2012-02-14 |
Nanotherapeutics, Inc. |
Bicyclic compounds and methods of making and using same
|
|
BRPI1010831A2
(pt)
|
2009-05-12 |
2016-04-05 |
Addex Pharmaceuticals Sa |
derivados de 1,2,4-triazolo[4,3-a]piridina e seu como moduladores alostéricos positivos de receptores de mglur2
|
|
MY153913A
(en)
|
2009-05-12 |
2015-04-15 |
Janssen Pharmaceuticals Inc |
7-aryl-1,2,4-triazolo[4,3-a]pyridine derivatives and their use as positive allosteric modulators of mglur2 receptors
|
|
CN102439008B
(zh)
|
2009-05-12 |
2015-04-29 |
杨森制药有限公司 |
1,2,4-三唑并[4,3-a]吡啶衍生物及其用于治疗或预防神经和精神病症的用途
|
|
US8158625B2
(en)
*
|
2009-05-27 |
2012-04-17 |
Genentech, Inc. |
Bicyclic indole-pyrimidine PI3K inhibitor compounds selective for P110 delta, and methods of use
|
|
BRPI1009022A2
(pt)
*
|
2009-05-27 |
2016-03-08 |
Hoffmann La Roche |
"composto, composição farmacêutica, processo para produzir uma composição farmacêutica, uso de um composto, método para tratamento de uma doença ou transtorno e kit"
|
|
PL2455371T3
(pl)
*
|
2009-07-16 |
2014-05-30 |
Sds Biotech Corp |
Pochodne 4-(3-butynylo)aminopirymidyny jako środki do zwalczania szkodników do stosowania w rolnictwie i ogrodnictwie
|
|
BR112012002164B1
(pt)
|
2009-07-30 |
2021-04-20 |
Merial, Inc |
compostos inseticidas de 4-amino-tieno[2,3-d]-pirimidina e métodos para seu uso
|
|
CA2776944A1
(fr)
*
|
2009-10-12 |
2011-05-12 |
F. Hoffmann-La Roche Ag |
Combinaisons d'un inhibiteur de pi3k et d'un inhibiteur de mek
|
|
EP2595993B1
(fr)
*
|
2010-07-23 |
2018-04-18 |
President and Fellows of Harvard College |
Composés renforçant l'activité protéasome tricyclique
|
|
WO2012021837A2
(fr)
|
2010-08-12 |
2012-02-16 |
Senomyx, Inc. |
Méthode pour améliorer la stabilité d'un exhausteur de goût sucré, et composition contenant un exhausteur de goût sucré stabilisé
|
|
US9271967B2
(en)
|
2010-11-08 |
2016-03-01 |
Janssen Pharmaceuticals, Inc. |
1,2,4-triazolo[4,3-a]pyridine derivatives and their use as positive allosteric modulators of mGluR2 receptors
|
|
ES2536433T3
(es)
|
2010-11-08 |
2015-05-25 |
Janssen Pharmaceuticals, Inc. |
Derivados de 1,2,4-triazolo[4,3-a]piridina y su uso como moduladores alostéricos positivos de receptores mGluR2
|
|
AU2011328203B2
(en)
|
2010-11-08 |
2015-03-19 |
Janssen Pharmaceuticals, Inc. |
1,2,4-triazolo[4,3-a]pyridine derivatives and their use as positive allosteric modulators of mGluR2 receptors
|
|
TW201500358A
(zh)
|
2010-12-16 |
2015-01-01 |
赫夫門羅氏藥廠股份有限公司 |
三環pi3k抑制劑化合物及其使用方法
|
|
AU2011354895B2
(en)
*
|
2011-01-14 |
2016-05-05 |
Sds Biotech K. K. |
Agri-horticultural pest control compositions comprising 4- (3-butynyl)aminopyrimidine derivatives
|
|
RU2013138835A
(ru)
|
2011-02-09 |
2015-03-20 |
Ф. Хоффманн-Ля Рош Аг |
Гетероциклические соединения в качестве ингибиторов pi3 киназы
|
|
AR088218A1
(es)
|
2011-07-19 |
2014-05-21 |
Infinity Pharmaceuticals Inc |
Compuestos heterociclicos utiles como inhibidores de pi3k
|
|
BR112015002380B1
(pt)
|
2012-08-06 |
2021-09-28 |
Firmenich Incorporated |
Composto, composições ingeríveis, processos para aumentar o sabor doce de composição e formulação flavorizante concentrada
|
|
JO3155B1
(ar)
|
2013-02-19 |
2017-09-20 |
Senomyx Inc |
معدِّل نكهة حلوة
|
|
JO3368B1
(ar)
|
2013-06-04 |
2019-03-13 |
Janssen Pharmaceutica Nv |
مركبات 6، 7- ثاني هيدرو بيرازولو [5،1-a] بيرازين- 4 (5 يد)- اون واستخدامها بصفة منظمات تفارغية سلبية لمستقبلات ميجلور 2
|
|
JO3367B1
(ar)
|
2013-09-06 |
2019-03-13 |
Janssen Pharmaceutica Nv |
مركبات 2،1، 4- ثلاثي زولو [3،4-a] بيريدين واستخدامها بصفة منظمات تفارغية موجبة لمستقبلات ميجلور 2
|
|
MX386697B
(es)
|
2014-01-21 |
2025-03-19 |
Janssen Pharmaceutica Nv |
Combinaciones que comprenden agonistas ortostericos o moduladores alostericos positivos del receptor glutamatergico metabotropico de subtipo 2 y su uso
|
|
ME03518B
(fr)
|
2014-01-21 |
2020-04-20 |
Janssen Pharmaceutica Nv |
Combinaisons comprenant des modulateurs allostériques positifs de sous-type 2 de récepteurs glutamatergiques métabotropes et leur utilisation
|
|
CN104725398B
(zh)
*
|
2015-01-29 |
2017-01-18 |
杨威 |
一种jak/stat3磷酸化抑制剂及其制备方法与用途
|
|
EP3324974B1
(fr)
*
|
2015-07-24 |
2022-06-08 |
University Of Louisville Research Foundation, Inc. |
Composés, compositions, procédés pour le traitement de maladies et procédés pour la préparation de composés
|
|
US20220117968A1
(en)
*
|
2017-07-17 |
2022-04-21 |
Saint Louis University |
Thieno[2,3-d)pyrimidines and benzofuro(3,2-d)pyrimidines as antimicrobial agents
|
|
BR112021002261A2
(pt)
|
2018-08-07 |
2021-05-04 |
Firmenich Incorporated |
2,2-dióxidos de 4-amino-1h-benzo[c][1,2,6]tiadiazina 5-substituídos e formulações e usos dos mesmos
|