BE861451A - Phenyl-5 oxazolidines et thiazolidines, et medicaments qui en contiennent - Google Patents

Phenyl-5 oxazolidines et thiazolidines, et medicaments qui en contiennent

Info

Publication number: BE861451A
Authority: BE; Belgium
Prior art keywords: thiazolidines; oxazolidines; phenyl; products containing; medicinal products
Prior art date: 1976-12-03

Application number

BE183130A

Other languages

English (en)

Original Assignee

Schering Ag

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1976-12-03

Filing date

1977-12-02

Publication date

1978-06-02

1977-12-02 Application filed by Schering Ag filed Critical Schering Ag

1978-06-02 Publication of BE861451A publication Critical patent/BE861451A/fr

Links

OGYGFUAIIOPWQD-UHFFFAOYSA-N 1,3-thiazolidine Chemical compound C1CSCN1 OGYGFUAIIOPWQD-UHFFFAOYSA-N 0.000 title 1
229940126601 medicinal product Drugs 0.000 title 1
150000002917 oxazolidines Chemical class 0.000 title 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D263/00—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings
- C07D263/02—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings
- C07D263/08—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
- C07D263/16—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D263/00—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings
- C07D263/02—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings
- C07D263/08—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
- C07D263/16—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D263/18—Oxygen atoms
- C07D263/20—Oxygen atoms attached in position 2
- C07D263/24—Oxygen atoms attached in position 2 with hydrocarbon radicals, substituted by oxygen atoms, attached to other ring carbon atoms
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
- C07D277/08—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
- C07D277/12—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D277/14—Oxygen atoms
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
- C07D277/08—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
- C07D277/12—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D277/16—Sulfur atoms

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)

BE183130A 1976-12-03 1977-12-02 Phenyl-5 oxazolidines et thiazolidines, et medicaments qui en contiennent BE861451A (fr)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
DE19762655369 DE2655369A1 (de)	1976-12-03	1976-12-03	5-(subst. phenyl)-oxazolidinone und deren schwefelanaloga sowie verfahren zu deren herstellung

Publications (1)

Publication Number	Publication Date
BE861451A true BE861451A (fr)	1978-06-02

Family

ID=5994882

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
BE183130A BE861451A (fr)	1976-12-03	1977-12-02	Phenyl-5 oxazolidines et thiazolidines, et medicaments qui en contiennent

Country Status (3)

Country	Link
US (1)	US4186129A (fr)
BE (1)	BE861451A (fr)
DE (1)	DE2655369A1 (fr)

Families Citing this family (32)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US4754047A (en) *	1979-08-16	1988-06-28	American Cyanamid Company	Phenylethanolamine derivatives and acid addition salts thereof for enhancing the growth rate of meat-producing animals and/or improving the efficiency of feed utilization thereby
IL61016A (en) *	1979-10-03	1984-02-29	Nippon Soda Co	3-carboxamide(or carbothiamide)derivatives of oxazolidine and thiazolidine-2-one(or 2-thione),their preparation and acaricidal compositions containing them
AU6610081A (en) *	1980-01-24	1981-07-30	Senju Pharmaceutical Co., Ltd.	Thiazolidine derivatives
US4522822A (en) *	1980-12-22	1985-06-11	American Cyanamid Company	Phenylethane derivatives and acid addition salts thereof for increasing lean meat deposition and/or improving lean meat to fat ratio in warm blooded animals
US4501751A (en) *	1980-12-22	1985-02-26	American Cyanamid Company	Phenylethanolamine derivatives and acid addition salts thereof for enhancing the growth rate of meat-producing animals and improving the efficiency of feed utilization thereby
US4416818A (en) *	1981-10-09	1983-11-22	The Dow Chemical Company	Preparation of N-alkoxycarbonyl-substituted cyclic lactams and ketones
US5243056A (en) *	1983-06-02	1993-09-07	Zambon S.P.A.	Intermediates for the preparation of 1-(phenyl)-1-hydroxy-2-amino-3-fluoro propane derivatives
HU191408B (en) *	1984-04-25	1987-02-27	Egis Gyogyszergyar,Hu	Process for preparing new imino-thiazolidine derivatives
US5783591A (en) *	1984-10-19	1998-07-21	Schering Aktiengesellschaft	Administration of oxazolidinone and pyrolidinone compounds for the treatment of inflammation
DE3438839A1 (de) *	1984-10-19	1986-04-24	Schering AG, 1000 Berlin und 4709 Bergkamen	Pharmazeutische praeparate
US4870169A (en) *	1985-07-17	1989-09-26	President And Fellows Of Harvard College	Intermediates for beta-lactam antibiotics
US4681940A (en) *	1985-11-19	1987-07-21	American Home Products Corporation	5-[3-[[2-quinolyl]methoxy]phenyl]-1,3-oxazoles
JPH0755937B2 (ja) *	1986-07-29	1995-06-14	日本曹達株式会社	オキサ（チア）ゾリジン誘導体その製造方法及び殺ダニ剤
DE3639225A1 (de) *	1986-11-14	1988-05-19	Schering Ag	Verwendung von 5-(subst. phenyl)-oxazolidinonderiaten als psychopharmaka
US5274002A (en) *	1987-04-14	1993-12-28	Warner-Lambert Company	Trisubstituted phenyl analogs having activity for congestive heart failure
US4971959A (en) *	1987-04-14	1990-11-20	Warner-Lambert Company	Trisubstituted phenyl analogs having activity for congestive heart failure
JPH03504499A (ja) *	1988-05-27	1991-10-03	セントカー・インコーポレーテツド	抗体試薬のための配合物
DE3823299A1 (de) *	1988-07-07	1990-01-11	Schering Ag	Substituierte phenyl-pyrrolidin-2-one, -oxazolidin-2-one und -imidazolidin-2-one, ihre herstellung sowie verwendung in arzneimitteln
US5344936A (en) *	1989-10-06	1994-09-06	University Of South Carolina	Chalcogen-based chiral reagents for nuclear magnetic resonance detection of stereochemical assignments and enantiomeric ratios
DK0542795T5 (da) *	1990-08-03	1998-09-07	Smithkline Beecham Corp	TNF-inhibitorer
US5124455A (en) *	1990-08-08	1992-06-23	American Home Products Corporation	Oxime-carbamates and oxime-carbonates as bronchodilators and anti-inflammatory agents
US5547979A (en) *	1992-03-30	1996-08-20	Smithkline Beecham	TNF inhibition
IL117090A (en) *	1995-02-10	2000-07-26	Schering Ag	Pharmaceutical compositions containing oxazolidinone derivatives
DE19540475A1 (de) *	1995-10-20	1997-04-24	Schering Ag	Chirale Methylphenyloxazolidinone
DE19617864A1 (de) *	1996-04-23	1997-10-30	Schering Ag	Neue chirale Phenyldihydrofuranone
FR2753449B1 (fr) *	1996-09-13	1998-12-04	Union Pharma Scient Appl	Nouveaux derives 3,4-diaryloxazolone, leurs procedes de preparation, et leurs utilisations en therapeutique
US6414160B1 (en) *	1997-07-10	2002-07-02	Ube Industries, Ltd.	Process for producing 4-alkoxycarbonyl-2-oxazolidinone compound
NZ530385A (en) *	1999-04-30	2004-05-28	Lilly Co Eli	Monofluoroalkyl derivatives
US7125568B2 (en)	2001-08-23	2006-10-24	Sung Michael T	Lipophilic drug compositions
DOP2005000123A (es) *	2004-07-02	2011-07-15	Merck Sharp & Dohme	Inhibidores de cetp
US20150218145A1 (en) *	2012-09-26	2015-08-06	Ranbaxy Laboratories Limited	Process for the preparation of rivaroxaban
US11141410B2 (en)	2015-12-16	2021-10-12	Merck Sharp & Dohme Corp	Oxazolidinones as taro inhibitors

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
DE1109691B (de) *	1957-06-11	1961-06-29	Om Lab Sa	Verfahren zur Herstellung von 5-[(o-Methoxy)-phenoxymethyl]-oxazolidon-(2)
BE763964A (fr) *	1970-03-24	1971-09-08	Delalande Sa	Nouveaux derives de l'aminocarbonyl-3 oxazolidinone-2, leur procede de preparation et leur application en therapeutique
IT995110B (it) *	1973-08-01	1975-11-10	Snam Progetti	Procedimento per la produzione di composti eterociclici e prodotti ottenuti
FR2281114A1 (fr) *	1974-08-09	1976-03-05	Inst Nat Sante Rech Med	Oxazolidinones, leur preparation et leurs applications

1976
- 1976-12-03 DE DE19762655369 patent/DE2655369A1/de not_active Withdrawn
1977
- 1977-11-30 US US05/855,867 patent/US4186129A/en not_active Expired - Lifetime
- 1977-12-02 BE BE183130A patent/BE861451A/fr not_active IP Right Cessation

Also Published As

Publication number	Publication date
US4186129A (en)	1980-01-29
DE2655369A1 (de)	1978-06-08

Legal Events

Date

Code

Title

Description

1993-06-30

RE

Patent lapsed

Owner name: SCHERING A.G.

Effective date: 19921231

Publication	Publication Date	Title
BE861451A (fr)	1978-06-02	Phenyl-5 oxazolidines et thiazolidines, et medicaments qui en contiennent
BE860877A (fr)	1978-05-16	Spirolactones steroidiques et medicaments qui en contiennent
BE846335R (fr)	1977-03-17	(polyalcoxy-phenyl)-4-pyrrolidinones-2 et medicaments qui en contiennent
BE865870A (fr)	1978-10-11	Derives du benzimidazole et medicaments qui en contiennent
FR2295739A1 (fr)	1976-07-23	Oxo-20 homopregnanes et medicaments qui en contiennent
BE853558A (fr)	1977-10-13	Nouvelles fluoroacylresorcines substituees et medicaments, cosmetiques et pesticides les renfermant.
FR2312240A1 (fr)	1976-12-24	Derives du prostane et medicaments qui en contiennent
FR2281123A1 (fr)	1976-03-05	Oxo-20 pregnanes et medicaments qui en contiennent
FR2336129A1 (fr)	1977-07-22	Ethers d'imidazolyl-oximes et medicaments qui en contiennent
BE843505A (fr)	1976-12-28	Pyrrolidones et medicaments qui en contiennent
FR2342990A1 (fr)	1977-09-30	Androstenones et medicaments qui en contiennent
BE869166A (fr)	1979-01-22	Nouvelles 4-pyrones substituees en positions 2, 3 et 6 et medicament les contenant
FR2287224A1 (fr)	1976-05-07	Derives de la pyridine et medicaments qui en contiennent
DK513575A (da)	1976-05-17	Aminopropanolderivater, fremgangsmade til fremstilling heraf og legemidler indeholdende disse
FR2287908A1 (fr)	1976-05-14	Hydroxy-7 oestradiols et medicaments qui en contiennent
FR2342973A1 (fr)	1977-09-30	Azapurines et medicaments contenant ces substances
FR2350099A1 (fr)	1977-12-02	2-imino-thiazolidines et thiazolines utiles comme medicaments
FR2307526A1 (fr)	1976-11-12	Oxo-11 prostaglandines et medicaments qui en contiennent
BE788322A (fr)	1973-03-01	3,4-dihydro-2h-isoquinoleine-1-ones et medicaments qui en contiennent
BE849346R (fr)	1977-06-13	Pyrrolidones et medicaments qui en contiennent
FR2347925A1 (fr)	1977-11-10	Medicaments, cosmetiques et pesticides renfermant des fluoroacyl-resorcines
FR2316941A1 (fr)	1977-02-04	Pyrrolidones et medicaments qui en contiennent
FR2343482A1 (fr)	1977-10-07	La 2- (2-acetamido-2-deoxy-3-o-d-glucopyranosyl) -d-propionyl-l-seryl-d-isoglutamine et medicaments la contenant
BE848385A (fr)	1977-05-16	Nouvelles phenylpyridylhydantoines substituees et medicament les contenant,
FR2283674A1 (fr)	1976-04-02	Homo-steroides et medicaments qui en renferment