BE864809A - Derives de benzodiazepine - Google Patents

Derives de benzodiazepine

Info

Publication number: BE864809A
Authority: BE; Belgium
Prior art keywords: benzodiazepine derivatives; benzodiazepine; derivatives
Prior art date: 1977-03-11

Application number

BE185863A

Other languages

English (en)

Original Assignee

Hoffmann La Roche

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1977-03-11

Filing date

1978-03-13

Publication date

1978-09-13

1978-03-13 Application filed by Hoffmann La Roche filed Critical Hoffmann La Roche

1978-09-13 Publication of BE864809A publication Critical patent/BE864809A/fr

Links

229940053197 benzodiazepine derivative antiepileptics Drugs 0.000 title 1
150000001557 benzodiazepines Chemical class 0.000 title 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P21/00—Drugs for disorders of the muscular or neuromuscular system
- A61P21/02—Muscle relaxants, e.g. for tetanus or cramps
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/20—Hypnotics; Sedatives
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/26—Psychostimulants, e.g. nicotine, cocaine
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D243/00—Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms
- C07D243/06—Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4
- C07D243/10—Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4 condensed with carbocyclic rings or ring systems
- C07D243/14—1,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines
- C07D243/16—1,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines substituted in position 5 by aryl radicals

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
Veterinary Medicine (AREA)
Life Sciences & Earth Sciences (AREA)
Neurology (AREA)
Public Health (AREA)
Bioinformatics & Cheminformatics (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Engineering & Computer Science (AREA)
Pharmacology & Pharmacy (AREA)
General Health & Medical Sciences (AREA)
Animal Behavior & Ethology (AREA)
Biomedical Technology (AREA)
Neurosurgery (AREA)
Psychiatry (AREA)
Anesthesiology (AREA)
Pain & Pain Management (AREA)
Orthopedic Medicine & Surgery (AREA)
Physical Education & Sports Medicine (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)

BE185863A 1977-03-11 1978-03-13 Derives de benzodiazepine BE864809A (fr)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
US05/776,820 US4125726A (en)	1977-03-11	1977-03-11	Imidazo[1,5-a][1,4]benzodiazepines

Publications (1)

Publication Number	Publication Date
BE864809A true BE864809A (fr)	1978-09-13

Family

ID=25108467

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
BE185863A BE864809A (fr)	1977-03-11	1978-03-13	Derives de benzodiazepine

Country Status (13)

Country	Link
US (3)	US4125726A (fr)
JP (1)	JPS53112897A (fr)
AU (1)	AU516873B2 (fr)
BE (1)	BE864809A (fr)
CA (1)	CA1093073A (fr)
CH (1)	CH638208A5 (fr)
DE (1)	DE2810476A1 (fr)
DK (1)	DK108078A (fr)
FR (1)	FR2383183A1 (fr)
GB (1)	GB1594867A (fr)
NL (1)	NL7802675A (fr)
SE (1)	SE437029B (fr)
ZA (1)	ZA781384B (fr)

Families Citing this family (16)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US4280957A (en) *	1974-09-11	1981-07-28	Hoffmann-La Roche Inc.	Imidazodiazepines and processes therefor
DE2754112A1 (de) *	1977-12-05	1979-06-13	Kali Chemie Pharma Gmbh	1,4-benzodiazepinderivate, ihre salze und diese verbindungen enthaltende arzneipraeparate
US4226768A (en) *	1979-05-29	1980-10-07	Hoffmann-La Roche Inc.	Process for the preparation of imidazobenzodiazepines
US4259241A (en) *	1979-05-29	1981-03-31	Hoffmann-La Roche Inc.	Process for the preparation of imidazobenzodiazepines
US4250095A (en) *	1979-07-25	1981-02-10	Hoffmann-La Roche Inc.	Imidazobenzodiazepines
US4226771A (en) *	1979-07-25	1980-10-07	Hoffmann-La Roche Inc.	1,2,5-Oxadiazino[5,4-a][1,4]benzodiazepine derivatives
US4238610A (en) *	1979-12-20	1980-12-09	Hoffmann-La Roche Inc.	Intermediates for the production of imidazobenzodiazepines
US4247463A (en) *	1980-04-11	1981-01-27	Hoffmann-La Roche Inc.	Process for the preparation of imidazobenzodiazepines
ZA845757B (en) *	1983-08-25	1985-04-24	Hoffmann La Roche	Benzodiazepine derivatives
DE102007035350A1 (de) *	2007-07-27	2009-01-29	Dr. Ing. H.C. F. Porsche Aktiengesellschaft	Förderleitung für ein Hydrauliksystem und Hydrauliksystem
AU2017313753B2 (en)	2016-08-16	2022-01-27	The Trustees Of Columbia University In The City Of New York	GABA(A) receptor modulators and methods to control airway hyperresponsiveness and inflammation in asthma
TW201837026A (zh)	2017-01-10	2018-10-16	德商拜耳廠股份有限公司	作為除害劑之雜環衍生物（二）
KR102515694B1 (ko)	2017-01-10	2023-03-29	바이엘 악티엔게젤샤프트	해충 방제제로서의 헤테로사이클 유도체
TWI820231B (zh)	2018-10-11	2023-11-01	德商拜耳廠股份有限公司	用於製備經取代咪唑衍生物之方法
BR112022026904A2 (pt)	2020-07-02	2023-01-24	Bayer Ag	Derivados de heterocicleno como agentes de controle de pragas
WO2025026738A1 (fr)	2023-07-31	2025-02-06	Bayer Aktiengesellschaft	Dérivés de 6-[5-(éthylsulfonyl)-1-méthyl-1h-imidazol-4-yl]-7-méthyl-3-(pentafluoroéthyl)-7h-imidazo [4,5-c]pyridazine en tant que pesticides

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US3852461A (en) *	1971-08-04	1974-12-03	Upjohn Co	Benzodiapines used as minor tranquilizers
US3763179A (en) *	1972-05-05	1973-10-02	Upjohn Co	2-imidazol-1-yl benzophenones
ZA755418B (en)	1974-09-11	1977-06-29	Hoffmann La Roche	Diazepine derivatives
US3910946A (en) *	1974-09-12	1975-10-07	Upjohn Co	4H-Imidazo{8 1,2-a{9 {8 1,4{9 benzodiazepines
AT361486B (de) *	1975-08-07	1981-03-10	Hoffmann La Roche	Verfahren zur herstellung von neuen imidazo(1,5 -a) (1,4)diazepinverbindungen, ihren salzen und optisch aktiven formen
US4005099A (en) *	1975-11-21	1977-01-25	The Upjohn Company	1-[(Dimethylamino)-methyl]-6-aryl-4H-imidazo[1,5-a][1,4]benzodiazepines

1977
- 1977-03-11 US US05/776,820 patent/US4125726A/en not_active Expired - Lifetime
1978
- 1978-03-09 ZA ZA00781384A patent/ZA781384B/xx unknown
- 1978-03-09 CH CH257578A patent/CH638208A5/de not_active IP Right Cessation
- 1978-03-10 DE DE19782810476 patent/DE2810476A1/de not_active Ceased
- 1978-03-10 DK DK108078A patent/DK108078A/da not_active Application Discontinuation
- 1978-03-10 GB GB9577/78A patent/GB1594867A/en not_active Expired
- 1978-03-10 FR FR7806983A patent/FR2383183A1/fr active Granted
- 1978-03-10 CA CA298,645A patent/CA1093073A/fr not_active Expired
- 1978-03-10 NL NL7802675A patent/NL7802675A/xx not_active Application Discontinuation
- 1978-03-10 JP JP2675478A patent/JPS53112897A/ja active Pending
- 1978-03-10 AU AU34056/78A patent/AU516873B2/en not_active Expired
- 1978-03-10 SE SE7802787A patent/SE437029B/sv not_active IP Right Cessation
- 1978-03-13 BE BE185863A patent/BE864809A/fr not_active IP Right Cessation
- 1978-07-27 US US05/928,479 patent/US4146722A/en not_active Expired - Lifetime
- 1978-07-27 US US05/928,765 patent/US4147875A/en not_active Expired - Lifetime

Also Published As

Publication number	Publication date
NL7802675A (nl)	1978-09-13
AU3405678A (en)	1979-09-13
US4147875A (en)	1979-04-03
CH638208A5 (de)	1983-09-15
ZA781384B (en)	1979-02-28
FR2383183A1 (fr)	1978-10-06
DK108078A (da)	1978-09-12
US4125726A (en)	1978-11-14
CA1093073A (fr)	1981-01-06
FR2383183B1 (fr)	1980-06-06
US4146722A (en)	1979-03-27
SE7802787L (sv)	1978-09-12
SE437029B (sv)	1985-02-04
AU516873B2 (en)	1981-06-25
DE2810476A1 (de)	1978-09-14
GB1594867A (en)	1981-08-05
JPS53112897A (en)	1978-10-02

Legal Events

Date

Code

Title

Description

1988-09-30

RE

Patent lapsed

Owner name: F. HOFFMANN-LA ROCHE & CIE S.A.

Effective date: 19880331

Publication	Publication Date	Title
BE867269A (fr)	1978-11-20	Derives de thiopropanoylamino-acides
SE7805879L (sv)	1978-11-25	Mevalonolaktonderivat
DK370778A (da)	1979-02-23	Triphenylakenderivater
LU80925A1 (fr)	1979-06-18	Derives de dehydrocyclicimino-acides
SE7811194L (sv)	1979-04-29	Imidazolidinderivat
BE866156A (fr)	1978-10-19	Derives de la guanidine
SE7803057L (sv)	1978-10-01	Bensimidazolderivat
SE7803328L (sv)	1978-09-24	Morfinderivat
DK543178A (da)	1979-06-02	Thiodydantoinderivater
BE839364A (fr)	1976-09-09	Derives de diazepine
SE7804446L (sv)	1978-11-06	Tienamycinderivat
SE7801997L (sv)	1978-08-27	Dipeptidderivat
SE7805260L (sv)	1978-11-17	Alkylendiaminderivat
BE862939A (fr)	1978-07-17	Derives de cyclohexene
ZA781384B (en)	1979-02-28	Benzodiazepine derivatives
BE851846A (fr)	1977-06-16	Derives de 1-nitro-9-amonoacridine
SE7805140L (sv)	1978-11-04	Bensimidazolderivat
FI783393A7 (fi)	1979-05-08	2-imino-imidazolidinderivat
FI780344A7 (fi)	1978-08-05	Oxadiazolopyrimidinderivat
BE866492A (fr)	1978-10-27	Derives de pyridazinone
FI780343A7 (fi)	1978-08-05	Oxadiazolopyrimidinderivat
FR2350345A1 (fr)	1977-12-02	Derives de la benzodiazepine
BR7808456A (pt)	1979-08-07	Novos derivados de pirazina
SE7803419L (sv)	1978-09-25	Kinazolinderivat
BE869866A (fr)	1979-02-21	Derives de thiazine