DK108078A - Benzodiazepinderivater deres fremstilling og anvendelse - Google Patents

Benzodiazepinderivater deres fremstilling og anvendelse

Info

Publication number
DK108078A
DK108078A DK108078A DK108078A DK108078A DK 108078 A DK108078 A DK 108078A DK 108078 A DK108078 A DK 108078A DK 108078 A DK108078 A DK 108078A DK 108078 A DK108078 A DK 108078A
Authority
DK
Denmark
Prior art keywords
manufacture
benzodiazepin
derivatives
benzodiazepin derivatives
Prior art date
Application number
DK108078A
Other languages
English (en)
Inventor
A Walser
R I Fryer
L Benjamin
Original Assignee
Hoffmann La Roche
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoffmann La Roche filed Critical Hoffmann La Roche
Publication of DK108078A publication Critical patent/DK108078A/da

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P21/00—Drugs for disorders of the muscular or neuromuscular system
    • A61P21/02—Muscle relaxants, e.g. for tetanus or cramps
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/20—Hypnotics; Sedatives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/26—Psychostimulants, e.g. nicotine, cocaine
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D243/00—Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms
    • C07D243/06—Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4
    • C07D243/10—Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4 condensed with carbocyclic rings or ring systems
    • C07D243/14—1,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines
    • C07D243/16—1,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines substituted in position 5 by aryl radicals

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Neurology (AREA)
  • Public Health (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • Psychiatry (AREA)
  • Anesthesiology (AREA)
  • Pain & Pain Management (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
DK108078A 1977-03-11 1978-03-10 Benzodiazepinderivater deres fremstilling og anvendelse DK108078A (da)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US05/776,820 US4125726A (en) 1977-03-11 1977-03-11 Imidazo[1,5-a][1,4]benzodiazepines

Publications (1)

Publication Number Publication Date
DK108078A true DK108078A (da) 1978-09-12

Family

ID=25108467

Family Applications (1)

Application Number Title Priority Date Filing Date
DK108078A DK108078A (da) 1977-03-11 1978-03-10 Benzodiazepinderivater deres fremstilling og anvendelse

Country Status (13)

Country Link
US (3) US4125726A (da)
JP (1) JPS53112897A (da)
AU (1) AU516873B2 (da)
BE (1) BE864809A (da)
CA (1) CA1093073A (da)
CH (1) CH638208A5 (da)
DE (1) DE2810476A1 (da)
DK (1) DK108078A (da)
FR (1) FR2383183A1 (da)
GB (1) GB1594867A (da)
NL (1) NL7802675A (da)
SE (1) SE437029B (da)
ZA (1) ZA781384B (da)

Families Citing this family (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4280957A (en) * 1974-09-11 1981-07-28 Hoffmann-La Roche Inc. Imidazodiazepines and processes therefor
DE2754112A1 (de) * 1977-12-05 1979-06-13 Kali Chemie Pharma Gmbh 1,4-benzodiazepinderivate, ihre salze und diese verbindungen enthaltende arzneipraeparate
US4226768A (en) * 1979-05-29 1980-10-07 Hoffmann-La Roche Inc. Process for the preparation of imidazobenzodiazepines
US4259241A (en) * 1979-05-29 1981-03-31 Hoffmann-La Roche Inc. Process for the preparation of imidazobenzodiazepines
US4250095A (en) * 1979-07-25 1981-02-10 Hoffmann-La Roche Inc. Imidazobenzodiazepines
US4226771A (en) * 1979-07-25 1980-10-07 Hoffmann-La Roche Inc. 1,2,5-Oxadiazino[5,4-a][1,4]benzodiazepine derivatives
US4238610A (en) * 1979-12-20 1980-12-09 Hoffmann-La Roche Inc. Intermediates for the production of imidazobenzodiazepines
US4247463A (en) * 1980-04-11 1981-01-27 Hoffmann-La Roche Inc. Process for the preparation of imidazobenzodiazepines
ZA845757B (en) * 1983-08-25 1985-04-24 Hoffmann La Roche Benzodiazepine derivatives
DE102007035350A1 (de) * 2007-07-27 2009-01-29 Dr. Ing. H.C. F. Porsche Aktiengesellschaft Förderleitung für ein Hydrauliksystem und Hydrauliksystem
AU2017313753B2 (en) 2016-08-16 2022-01-27 The Trustees Of Columbia University In The City Of New York GABA(A) receptor modulators and methods to control airway hyperresponsiveness and inflammation in asthma
TW201837026A (zh) 2017-01-10 2018-10-16 德商拜耳廠股份有限公司 作為除害劑之雜環衍生物(二)
KR102515694B1 (ko) 2017-01-10 2023-03-29 바이엘 악티엔게젤샤프트 해충 방제제로서의 헤테로사이클 유도체
TWI820231B (zh) 2018-10-11 2023-11-01 德商拜耳廠股份有限公司 用於製備經取代咪唑衍生物之方法
BR112022026904A2 (pt) 2020-07-02 2023-01-24 Bayer Ag Derivados de heterocicleno como agentes de controle de pragas
WO2025026738A1 (en) 2023-07-31 2025-02-06 Bayer Aktiengesellschaft 6-[5-(ethylsulfonyl)-1-methyl-1h-imidazol-4-yl]-7-methyl-3-(pentafluoroethyl)-7h-imidazo[4,5-c]pyridazine derivatives as pesticides

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3852461A (en) * 1971-08-04 1974-12-03 Upjohn Co Benzodiapines used as minor tranquilizers
US3763179A (en) * 1972-05-05 1973-10-02 Upjohn Co 2-imidazol-1-yl benzophenones
ZA755418B (en) 1974-09-11 1977-06-29 Hoffmann La Roche Diazepine derivatives
US3910946A (en) * 1974-09-12 1975-10-07 Upjohn Co 4H-Imidazo{8 1,2-a{9 {8 1,4{9 benzodiazepines
AT361486B (de) * 1975-08-07 1981-03-10 Hoffmann La Roche Verfahren zur herstellung von neuen imidazo(1,5 -a) (1,4)diazepinverbindungen, ihren salzen und optisch aktiven formen
US4005099A (en) * 1975-11-21 1977-01-25 The Upjohn Company 1-[(Dimethylamino)-methyl]-6-aryl-4H-imidazo[1,5-a][1,4]benzodiazepines

Also Published As

Publication number Publication date
NL7802675A (nl) 1978-09-13
AU3405678A (en) 1979-09-13
US4147875A (en) 1979-04-03
CH638208A5 (de) 1983-09-15
ZA781384B (en) 1979-02-28
FR2383183A1 (fr) 1978-10-06
US4125726A (en) 1978-11-14
CA1093073A (en) 1981-01-06
FR2383183B1 (da) 1980-06-06
US4146722A (en) 1979-03-27
SE7802787L (sv) 1978-09-12
SE437029B (sv) 1985-02-04
AU516873B2 (en) 1981-06-25
DE2810476A1 (de) 1978-09-14
BE864809A (fr) 1978-09-13
GB1594867A (en) 1981-08-05
JPS53112897A (en) 1978-10-02

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Legal Events

Date Code Title Description
AHS Application shelved for other reasons than non-payment