BG102759A - Therapeutical form for diabetes - Google Patents

Therapeutical form for diabetes

Info

Publication number
BG102759A
BG102759A BG102759A BG10275998A BG102759A BG 102759 A BG102759 A BG 102759A BG 102759 A BG102759 A BG 102759A BG 10275998 A BG10275998 A BG 10275998A BG 102759 A BG102759 A BG 102759A
Authority
BG
Bulgaria
Prior art keywords
carbon atoms
substituted alkyl
formulawhere
carbonatoms
therapeutical
Prior art date
Application number
BG102759A
Other languages
Bulgarian (bg)
English (en)
Inventor
Hisashi Shinkai
Hidekazu Ozeki
Noboru Furukawa
Original Assignee
Japan Tobacco Inc.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Japan Tobacco Inc. filed Critical Japan Tobacco Inc.
Publication of BG102759A publication Critical patent/BG102759A/xx

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    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/12—Ketones
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    • C07D207/00—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D207/18—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member
    • C07D207/22—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D207/24—Oxygen or sulfur atoms
    • C07D207/26—2-Pyrrolidones
    • C07D207/263—2-Pyrrolidones with only hydrogen atoms or radicals containing only hydrogen and carbon atoms directly attached to other ring carbon atoms
    • C07D207/27—2-Pyrrolidones with only hydrogen atoms or radicals containing only hydrogen and carbon atoms directly attached to other ring carbon atoms with substituted hydrocarbon radicals directly attached to the ring nitrogen atom
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    • C07C233/00—Carboxylic acid amides
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    • C07C233/30—Carboxylic acid amides having carbon atoms of carboxamide groups bound to hydrogen atoms or to acyclic carbon atoms having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a hydrocarbon radical substituted by doubly-bound oxygen atoms
    • C07C233/31—Carboxylic acid amides having carbon atoms of carboxamide groups bound to hydrogen atoms or to acyclic carbon atoms having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a hydrocarbon radical substituted by doubly-bound oxygen atoms with the substituted hydrocarbon radical bound to the nitrogen atom of the carboxamide group by an acyclic carbon atom
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    • C07C49/76—Ketones containing a keto group bound to a six-membered aromatic ring
    • C07C49/794—Ketones containing a keto group bound to a six-membered aromatic ring having unsaturation outside an aromatic ring
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    • C07C49/80—Ketones containing a keto group bound to a six-membered aromatic ring containing halogen
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    • C07C49/84—Ketones containing a keto group bound to a six-membered aromatic ring containing ether groups, groups, groups, or groups
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    • C07C59/40—Unsaturated compounds
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    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

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BG102759A 1996-02-19 1998-09-09 Therapeutical form for diabetes BG102759A (en)

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JP5688396 1996-02-19
PCT/JP1997/000422 WO1997030017A1 (en) 1996-02-19 1997-02-17 Therapeutic agent for diabetes

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FR2849599B1 (fr) * 2003-01-07 2006-12-29 Merck Sante Sas Utilisation d'inhibiteurs de la kynurenine-3-hydroxylase pour le traitement du diabete
FR2849598B1 (fr) 2003-01-07 2006-09-22 Merck Sante Sas Utilisation d'inhibiteurs de la kynurenine-3-hydroxylase pour le traitement du diabete, par augmentation du nombre de cellules des ilots de langerhans
FR2880885B1 (fr) * 2005-01-14 2009-01-30 Merck Sante Soc Par Actions Si Derives d'acide phenylbenzoique, procedes pour leur preparation, compositions pharmaceutiques les contenant et applications en therapeutique
DE102006031813B4 (de) * 2006-07-07 2011-04-28 Christian-Albrechts-Universität Zu Kiel Verwendung basischer Acetophenone als Hemmstoffe von NO-Synthasen
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CN102344369A (zh) * 2010-07-30 2012-02-08 华东师范大学 侧链含芴单元的高取向发光聚乙炔单体及其制备方法
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DK3206686T3 (da) 2014-08-20 2019-12-16 Samumed Llc Gamma-diketoner til behandling og forebyggelse af ældning af huden og rynker
CN109420175A (zh) * 2017-09-01 2019-03-05 任洁 基于cox的血糖调节机制
CN109419790A (zh) * 2017-09-04 2019-03-05 任洁 芬布芬的新用途
CN109419791A (zh) * 2017-09-04 2019-03-05 任洁 芬布芬作为糖尿病相关靶点调节剂的新用途
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IL125820A0 (en) 1999-04-11
CN1216522A (zh) 1999-05-12
NO983770L (no) 1998-10-19
ID15967A (id) 1997-08-21
WO1997030017A1 (en) 1997-08-21
PL328519A1 (en) 1999-02-01
BR9707588A (pt) 1999-07-27
CA2246725A1 (en) 1997-08-21
AU719396B2 (en) 2000-05-11
NO983770D0 (no) 1998-08-18
AU1673297A (en) 1997-09-02
HUP9900715A3 (en) 2000-11-28
HUP9900715A2 (hu) 1999-06-28
CZ256198A3 (cs) 1998-12-16
NZ331801A (en) 2001-01-26
KR19990082639A (ko) 1999-11-25
EP0885869A1 (en) 1998-12-23

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