BG103271A - Derivatives of n-(benzothiazol-2-yl) piperidine-1-ethaneamines, method for their preparation and application as therapeutical means - Google Patents

Derivatives of n-(benzothiazol-2-yl) piperidine-1-ethaneamines, method for their preparation and application as therapeutical means

Info

Publication number
BG103271A
BG103271A BG103271A BG10327199A BG103271A BG 103271 A BG103271 A BG 103271A BG 103271 A BG103271 A BG 103271A BG 10327199 A BG10327199 A BG 10327199A BG 103271 A BG103271 A BG 103271A
Authority
BG
Bulgaria
Prior art keywords
ethaneamines
benzothiazol
piperidine
derivatives
preparation
Prior art date
Application number
BG103271A
Other languages
Bulgarian (bg)
English (en)
Inventor
Gihad Dargazanli
Pascal George
Patrick Lardenois
Jonathan Frost
Johannes Schoemaker
Maria-Carmen Renones
Pascale Magat
Original Assignee
Sanofi-Synthelabo
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sanofi-Synthelabo filed Critical Sanofi-Synthelabo
Publication of BG103271A publication Critical patent/BG103271A/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/425—Thiazoles
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • Neurosurgery (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Hydrogenated Pyridines (AREA)
BG103271A 1996-10-01 1999-03-22 Derivatives of n-(benzothiazol-2-yl) piperidine-1-ethaneamines, method for their preparation and application as therapeutical means BG103271A (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR9611925A FR2753970B1 (fr) 1996-10-01 1996-10-01 Derives de n-(benzothiazol-2-yl) piperidine-1-ethanamine, leur preparation et leur application en therapeutique
PCT/FR1997/001692 WO1998014444A1 (fr) 1996-10-01 1997-09-26 Derives de n-(benzothiazol-2-yl)piperidine-1-ethanamine, leur preparation et leur application en therapeutique

Publications (1)

Publication Number Publication Date
BG103271A true BG103271A (en) 2000-05-31

Family

ID=9496217

Family Applications (1)

Application Number Title Priority Date Filing Date
BG103271A BG103271A (en) 1996-10-01 1999-03-22 Derivatives of n-(benzothiazol-2-yl) piperidine-1-ethaneamines, method for their preparation and application as therapeutical means

Country Status (23)

Country Link
EP (1) EP0929550A1 (cs)
JP (1) JP2001501217A (cs)
KR (1) KR20000048767A (cs)
CN (1) CN1230959A (cs)
AR (1) AR009105A1 (cs)
AU (1) AU722147B2 (cs)
BG (1) BG103271A (cs)
BR (1) BR9711842A (cs)
CA (1) CA2266510A1 (cs)
CO (1) CO4650030A1 (cs)
CZ (1) CZ112699A3 (cs)
EE (1) EE9900135A (cs)
FR (1) FR2753970B1 (cs)
HU (1) HUP9904091A3 (cs)
IL (1) IL128902A (cs)
NO (1) NO991581L (cs)
NZ (1) NZ334553A (cs)
PL (1) PL332648A1 (cs)
SK (1) SK42299A3 (cs)
TR (1) TR199900634T2 (cs)
TW (1) TW438800B (cs)
WO (1) WO1998014444A1 (cs)
ZA (1) ZA978772B (cs)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB9725541D0 (en) * 1997-12-02 1998-02-04 Pharmacia & Upjohn Spa Amino-benzothiazole derivatives
US6107313A (en) * 1998-10-02 2000-08-22 Combichem, Inc. Dopamine receptor antagonists
RU2251419C2 (ru) 2000-06-21 2005-05-10 Ф. Хоффманн-Ля Рош Аг Производные бензотиазола
US7087761B2 (en) 2003-01-07 2006-08-08 Hoffmann-La Roche Inc. Cyclization process for substituted benzothiazole derivatives
EP1680408A2 (en) * 2003-10-24 2006-07-19 F. Hoffmann-La Roche Ag Ccr3 receptor antagonists
AU2005247567B2 (en) 2004-05-24 2010-09-02 F. Hoffmann-La Roche Ag 4-hydroxy-4-methyl-piperidine-1-carboxylic acid (4-methoxy-7-morpholin-4-yl-benzothiazol-2-yl)-amide
EP1812392B1 (en) 2004-11-05 2008-07-09 F.Hoffmann-La Roche Ag Process for preparation of isonicotinic acid derivatives
PT1863818E (pt) 2005-03-23 2010-04-09 Hoffmann La Roche Derivados de acetilenil-pirazolo-pirimidina como antagonistas de mglur2
ATE463495T1 (de) 2005-09-27 2010-04-15 Hoffmann La Roche Oxadiazolylpyrazolopyrimidine als mglur2- antagonisten

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA1260474A (en) * 1984-12-03 1989-09-26 Raymond A. Stokbroekx Benzoxazol- and benzothiazolamine derivatives
KR930005004B1 (ko) * 1985-04-15 1993-06-11 쟈안센 파아마슈우티카 엔. 부이. 치환된 n-[(4-피페리디닐)알킬]이환 축합 옥사졸아민 및 티아졸아민의 제조방법

Also Published As

Publication number Publication date
SK42299A3 (en) 1999-12-10
JP2001501217A (ja) 2001-01-30
TR199900634T2 (xx) 1999-06-21
PL332648A1 (en) 1999-09-27
AU722147B2 (en) 2000-07-20
KR20000048767A (ko) 2000-07-25
EE9900135A (et) 1999-12-15
NZ334553A (en) 2000-11-24
CN1230959A (zh) 1999-10-06
IL128902A0 (en) 2000-02-17
TW438800B (en) 2001-06-07
FR2753970B1 (fr) 1998-10-30
CZ112699A3 (cs) 1999-06-16
IL128902A (en) 2001-07-24
BR9711842A (pt) 1999-08-24
CO4650030A1 (es) 1998-09-03
HUP9904091A2 (hu) 2000-05-28
WO1998014444A1 (fr) 1998-04-09
NO991581L (no) 1999-06-01
NO991581D0 (no) 1999-03-30
AR009105A1 (es) 2000-03-08
FR2753970A1 (fr) 1998-04-03
HUP9904091A3 (en) 2000-07-28
EP0929550A1 (fr) 1999-07-21
AU4463897A (en) 1998-04-24
ZA978772B (en) 1998-03-27
CA2266510A1 (en) 1998-04-09

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