EE9900135A - N-(2-bensotiasolüül)-1-piperidiinetaanamiini derivaadid, nende valmistamine ja kasutamine raviks - Google Patents

N-(2-bensotiasolüül)-1-piperidiinetaanamiini derivaadid, nende valmistamine ja kasutamine raviks

Info

Publication number
EE9900135A
EE9900135A EEP199900135A EE9900135A EE9900135A EE 9900135 A EE9900135 A EE 9900135A EE P199900135 A EEP199900135 A EE P199900135A EE 9900135 A EE9900135 A EE 9900135A EE 9900135 A EE9900135 A EE 9900135A
Authority
EE
Estonia
Prior art keywords
piperidinethanamine
benzothiazolyl
therapy
derivatives
preparation
Prior art date
Application number
EEP199900135A
Other languages
English (en)
Estonian (et)
Inventor
Dargazanli Gihad
George Pascal
Lardenois Patrick
Frost Jonathan
Schoemaker Johannes
Renones Maria-Carmen
Magat Pascale
Original Assignee
Synthlabo
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Synthlabo filed Critical Synthlabo
Publication of EE9900135A publication Critical patent/EE9900135A/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/425—Thiazoles
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • Neurosurgery (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Hydrogenated Pyridines (AREA)
EEP199900135A 1996-10-01 1997-09-26 N-(2-bensotiasolüül)-1-piperidiinetaanamiini derivaadid, nende valmistamine ja kasutamine raviks EE9900135A (et)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR9611925A FR2753970B1 (fr) 1996-10-01 1996-10-01 Derives de n-(benzothiazol-2-yl) piperidine-1-ethanamine, leur preparation et leur application en therapeutique
PCT/FR1997/001692 WO1998014444A1 (fr) 1996-10-01 1997-09-26 Derives de n-(benzothiazol-2-yl)piperidine-1-ethanamine, leur preparation et leur application en therapeutique

Publications (1)

Publication Number Publication Date
EE9900135A true EE9900135A (et) 1999-12-15

Family

ID=9496217

Family Applications (1)

Application Number Title Priority Date Filing Date
EEP199900135A EE9900135A (et) 1996-10-01 1997-09-26 N-(2-bensotiasolüül)-1-piperidiinetaanamiini derivaadid, nende valmistamine ja kasutamine raviks

Country Status (23)

Country Link
EP (1) EP0929550A1 (cs)
JP (1) JP2001501217A (cs)
KR (1) KR20000048767A (cs)
CN (1) CN1230959A (cs)
AR (1) AR009105A1 (cs)
AU (1) AU722147B2 (cs)
BG (1) BG103271A (cs)
BR (1) BR9711842A (cs)
CA (1) CA2266510A1 (cs)
CO (1) CO4650030A1 (cs)
CZ (1) CZ112699A3 (cs)
EE (1) EE9900135A (cs)
FR (1) FR2753970B1 (cs)
HU (1) HUP9904091A3 (cs)
IL (1) IL128902A (cs)
NO (1) NO991581L (cs)
NZ (1) NZ334553A (cs)
PL (1) PL332648A1 (cs)
SK (1) SK42299A3 (cs)
TR (1) TR199900634T2 (cs)
TW (1) TW438800B (cs)
WO (1) WO1998014444A1 (cs)
ZA (1) ZA978772B (cs)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB9725541D0 (en) * 1997-12-02 1998-02-04 Pharmacia & Upjohn Spa Amino-benzothiazole derivatives
US6107313A (en) * 1998-10-02 2000-08-22 Combichem, Inc. Dopamine receptor antagonists
RU2251419C2 (ru) 2000-06-21 2005-05-10 Ф. Хоффманн-Ля Рош Аг Производные бензотиазола
US7087761B2 (en) 2003-01-07 2006-08-08 Hoffmann-La Roche Inc. Cyclization process for substituted benzothiazole derivatives
EP1680408A2 (en) * 2003-10-24 2006-07-19 F. Hoffmann-La Roche Ag Ccr3 receptor antagonists
AU2005247567B2 (en) 2004-05-24 2010-09-02 F. Hoffmann-La Roche Ag 4-hydroxy-4-methyl-piperidine-1-carboxylic acid (4-methoxy-7-morpholin-4-yl-benzothiazol-2-yl)-amide
EP1812392B1 (en) 2004-11-05 2008-07-09 F.Hoffmann-La Roche Ag Process for preparation of isonicotinic acid derivatives
PT1863818E (pt) 2005-03-23 2010-04-09 Hoffmann La Roche Derivados de acetilenil-pirazolo-pirimidina como antagonistas de mglur2
ATE463495T1 (de) 2005-09-27 2010-04-15 Hoffmann La Roche Oxadiazolylpyrazolopyrimidine als mglur2- antagonisten

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA1260474A (en) * 1984-12-03 1989-09-26 Raymond A. Stokbroekx Benzoxazol- and benzothiazolamine derivatives
KR930005004B1 (ko) * 1985-04-15 1993-06-11 쟈안센 파아마슈우티카 엔. 부이. 치환된 n-[(4-피페리디닐)알킬]이환 축합 옥사졸아민 및 티아졸아민의 제조방법

Also Published As

Publication number Publication date
BG103271A (en) 2000-05-31
SK42299A3 (en) 1999-12-10
JP2001501217A (ja) 2001-01-30
TR199900634T2 (xx) 1999-06-21
PL332648A1 (en) 1999-09-27
AU722147B2 (en) 2000-07-20
KR20000048767A (ko) 2000-07-25
NZ334553A (en) 2000-11-24
CN1230959A (zh) 1999-10-06
IL128902A0 (en) 2000-02-17
TW438800B (en) 2001-06-07
FR2753970B1 (fr) 1998-10-30
CZ112699A3 (cs) 1999-06-16
IL128902A (en) 2001-07-24
BR9711842A (pt) 1999-08-24
CO4650030A1 (es) 1998-09-03
HUP9904091A2 (hu) 2000-05-28
WO1998014444A1 (fr) 1998-04-09
NO991581L (no) 1999-06-01
NO991581D0 (no) 1999-03-30
AR009105A1 (es) 2000-03-08
FR2753970A1 (fr) 1998-04-03
HUP9904091A3 (en) 2000-07-28
EP0929550A1 (fr) 1999-07-21
AU4463897A (en) 1998-04-24
ZA978772B (en) 1998-03-27
CA2266510A1 (en) 1998-04-09

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