BG104451A - Antiestrogen and progestin-containing peroral contraceptives - Google Patents

Antiestrogen and progestin-containing peroral contraceptives

Info

Publication number: BG104451A
Authority: BG; Bulgaria
Prior art keywords: antiestrogen; progestin; peroral; contraceptives; neuterotrophic
Prior art date: 1997-11-06

Application number

BG104451A

Other languages

Bulgarian (bg)

English (en)

Inventor

Michael Gast

Christopher Miller

Original Assignee

Wyeth

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1997-11-06

Filing date

2000-05-17

Publication date

2000-12-29

2000-05-17 Application filed by Wyeth filed Critical Wyeth

2000-12-29 Publication of BG104451A publication Critical patent/BG104451A/xx

Links

RJKFOVLPORLFTN-LEKSSAKUSA-N Progesterone Chemical class C1CC2=CC(=O)CC[C@]2(C)[C@@H]2[C@@H]1[C@@H]1CC[C@H](C(=O)C)[C@@]1(C)CC2 RJKFOVLPORLFTN-LEKSSAKUSA-N 0.000 title abstract 2
229940046836 anti-estrogen Drugs 0.000 title abstract 2
230000001833 anti-estrogenic effect Effects 0.000 title abstract 2
239000000328 estrogen antagonist Substances 0.000 title abstract 2
239000000583 progesterone congener Substances 0.000 title abstract 2
229940124558 contraceptive agent Drugs 0.000 title 1
239000003433 contraceptive agent Substances 0.000 title 1
230000027758 ovulation cycle Effects 0.000 abstract 1
230000001850 reproductive effect Effects 0.000 abstract 1

Classifications

- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
- A61K31/565—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
- A61K31/57—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane or progesterone
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A61P15/18—Feminine contraceptives

Landscapes

Health & Medical Sciences (AREA)
Pharmacology & Pharmacy (AREA)
Veterinary Medicine (AREA)
Public Health (AREA)
General Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Animal Behavior & Ethology (AREA)
Life Sciences & Earth Sciences (AREA)
Medicinal Chemistry (AREA)
Epidemiology (AREA)
Reproductive Health (AREA)
Organic Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
General Chemical & Material Sciences (AREA)
Chemical Kinetics & Catalysis (AREA)
Endocrinology (AREA)
Bioinformatics & Cheminformatics (AREA)
Engineering & Computer Science (AREA)
Gynecology & Obstetrics (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Steroid Compounds (AREA)
Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)

BG104451A 1997-11-06 2000-05-17 Antiestrogen and progestin-containing peroral contraceptives BG104451A (en)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
US96508397A	1997-11-06	1997-11-06
PCT/US1998/023427 WO1999024027A2 (fr)	1997-11-06	1998-11-04	Contraceptifs oraux a base d'anti-oestrogenes associes a un progestatif

Publications (1)

Publication Number	Publication Date
BG104451A true BG104451A (en)	2000-12-29

Family

ID=25509417

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
BG104451A BG104451A (en)	1997-11-06	2000-05-17	Antiestrogen and progestin-containing peroral contraceptives

Country Status (28)

Country	Link
EP (1)	EP1051179B1 (fr)
JP (1)	JP2001522798A (fr)
CN (1)	CN1278732A (fr)
AR (1)	AR016667A1 (fr)
AT (1)	ATE304359T1 (fr)
AU (2)	AU760540B2 (fr)
BG (1)	BG104451A (fr)
BR (1)	BR9813982A (fr)
CA (1)	CA2307210A1 (fr)
CZ (1)	CZ294155B6 (fr)
DE (1)	DE69831605T2 (fr)
DK (1)	DK1051179T3 (fr)
EA (1)	EA200000492A1 (fr)
EE (1)	EE04092B1 (fr)
ES (1)	ES2246541T3 (fr)
GE (1)	GEP20043290B (fr)
HR (1)	HRP20000269A2 (fr)
HU (1)	HUP0100293A3 (fr)
ID (1)	ID24568A (fr)
IL (1)	IL135621A0 (fr)
NO (1)	NO20002167L (fr)
NZ (1)	NZ503890A (fr)
PL (1)	PL340623A1 (fr)
SK (1)	SK6482000A3 (fr)
TR (1)	TR200001268T2 (fr)
UA (1)	UA68365C2 (fr)
WO (1)	WO1999024027A2 (fr)
ZA (1)	ZA9810136B (fr)

Families Citing this family (35)

* Cited by examiner, † Cited by third party
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IL120263A0 (en) *	1996-02-28	1997-06-10	Pfizer	Combination therapy to prevent bone loss-progesterone and estrogen agonists
US6479535B1 (en)	1998-05-15	2002-11-12	Wyeth	2-phenyl-1-[4-(2-aminoethoxy)-benzyl]-indole and estrogen formulations
EA005932B1 (ru) *	1998-05-15	2005-08-25	Уайт	2-фенил-1-[4-(2-аминоэтокси)бензил]индол в комбинации с эстрогенами
US6380166B1 (en)	1999-09-13	2002-04-30	American Home Products Corporation	Glucopyranosides conjugates of 2-(4-hydroxy-phenyl)-3-methyl-1-[4-(2-amin-1-yl-ethoxy)-benzyl]-1H-indol-5-ols
CA2382683A1 (fr) *	1999-09-13	2001-03-22	American Home Products Corporation	Conjugues glucopyranosides de 2-(4-hydroxy-phenyl)-1-{4-(2-amin-1-yl-ethoxy)-benzyl\|-1h-indol-5-ols
US6376486B1 (en)	2000-07-06	2002-04-23	American Home Products Corporation	Methods of inhibiting sphincter incontinence
JP2005504032A (ja)	2001-07-31	2005-02-10	ファイザー・プロダクツ・インク	エストロゲン・アゴニスト／アンタゴニスト、エストロゲン及びプロゲスチンの組み合わせを含む医薬組成物、キット及び方法
SI1809602T1 (sl)	2004-10-27	2009-04-30	Janssen Pharmaceutica Nv	Indolni derivati, uporabni kot modulatorji progesteronskega receptorja
FR2880625B1 (fr) *	2005-01-07	2007-03-09	Sanofi Aventis Sa	Derives de n-(heteroaryl)-1h-indole-2-carboxamides, leur preparation et leur application en therapeutique
UY29527A1 (es)	2005-05-13	2006-12-29	Schering Ag	Composicinn farmaccutica que contienen gestrgenos y/o estrngenos y 5-metil - (6s) - tetrhidrofolato.
DE102008057230A1 (de) *	2008-11-11	2010-05-12	Bayer Schering Pharma Aktiengesellschaft	Synergistische pharmazeutische Kombination mit einem Estrogenrezeptorantagonisten und einem Progestin
RS56042B1 (sr)	2010-06-10	2017-09-29	Seragon Pharmaceuticals Inc	Modulatori estrogenih receptora i njihove upotrebe
WO2013090829A1 (fr)	2011-12-14	2013-06-20	Aragon Pharmaceuticals, Inc.	Modulateurs des récepteurs des œstrogènes et ses utilisations
KR20240142622A (ko)	2015-10-01	2024-09-30	올레마 파마슈티컬스 인코포레이티드	테트라히드로-1H-피리도[3,4-b]인돌 항에스트로겐 약물
LT3386500T (lt)	2015-12-09	2022-12-27	The Board Of Trustees Of The University Of Illinois	Selektyvūs estrogenų receptorių slopintojai benzotiofeno pagrindu
ES2990061T3 (es)	2016-05-10	2024-11-28	C4 Therapeutics Inc	Degronímeros espirocíclicos para la degradación de proteínas diana
CN109641874A (zh)	2016-05-10	2019-04-16	C4医药公司	用于靶蛋白降解的c3-碳连接的戊二酰亚胺降解决定子体
EP3454856B1 (fr)	2016-05-10	2024-09-11	C4 Therapeutics, Inc.	Dégronimères hétérocycliques pour la dégradation de protéines cibles
CN109790143A (zh)	2016-05-10	2019-05-21	C4医药公司	用于靶蛋白降解的胺连接的c3-戊二酰亚胺降解决定子体
RU2019102647A (ru)	2016-07-01	2020-08-03	Г1 Терапьютикс, Инк.	Антипролиферационные средства на основе пиримидина
WO2018081168A2 (fr)	2016-10-24	2018-05-03	The Board Of Trustees Of The University Of Illinois	Répresseurs du récepteur oestrogénique sélectifs mixtes à base de benzothiophène
MX2019008158A (es)	2017-01-06	2019-12-09	G1 Therapeutics Inc	Terapia de combinacion para el tratamiento del cancer.
KR20190117582A (ko)	2017-02-10	2019-10-16	쥐원 쎄라퓨틱스, 인크.	벤조티오펜 에스트로겐 수용체 조정제
CN110769822A (zh)	2017-06-20	2020-02-07	C4医药公司	用于蛋白降解的n/o-连接的降解决定子和降解决定子体
WO2019006393A1 (fr)	2017-06-29	2019-01-03	G1 Therapeutics, Inc.	Formes morphiques de git38 et leurs procédés de fabrication
CN120698983A (zh)	2018-12-20	2025-09-26	C4医药公司	靶向蛋白降解
KR20220034129A (ko)	2019-07-07	2022-03-17	올레마 파마슈티컬스 인코포레이티드	에스트로겐 수용체 길항제 요법
KR20220119415A (ko)	2019-12-20	2022-08-29	씨4 테라퓨틱스, 인코포레이티드	Egfr 분해를 위한 이소인돌리논 및 인다졸 화합물
TW202146412A (zh)	2020-03-05	2021-12-16	美商Ｃ４醫藥公司	用於標靶降解brd9之化合物
IL300397A (en)	2020-08-05	2023-04-01	C4 Therapeutics Inc	Compounds for targeted knockdown of RET
MX2023014059A (es)	2021-06-08	2024-03-12	C4 Therapeutics Inc	Terapeuticos para la degradacion de una proteina quiinasa de serina/ treonina mutante.
WO2024030968A1 (fr)	2022-08-03	2024-02-08	Brystol-Myers Squibb Company	Composés pour moduler la protéine ret
EP4611901A1 (fr)	2022-11-04	2025-09-10	Bristol-Myers Squibb Company	Agents de dégradation de protéine ret-ldd
WO2024097980A1 (fr)	2022-11-04	2024-05-10	Bristol-Myers Squibb Company	Inhibiteurs de protéines ret-ldd
EP4735452A2 (fr)	2023-06-30	2026-05-06	Merck Patent GmbH	Composés hétérobifonctionnels pour la dégradation de la protéine kras

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
ZA716118B (en) *	1970-10-05	1972-05-31	Richardson Merrell Inc	Contraception
ZA9510926B (en) *	1994-12-23	1996-07-03	Schering Ag	Compounds with progesterone-antagonistic and antiestrogenic action to be used together for female contraception
IL120263A0 (en) *	1996-02-28	1997-06-10	Pfizer	Combination therapy to prevent bone loss-progesterone and estrogen agonists
IL120266A (en) *	1996-02-28	2005-05-17	Pfizer	Use of estrogen antagonists and estrogen agonists in the preparation of medicaments for inhibiting pathological conditions
PT802183E (pt) *	1996-04-19	2002-03-28	American Home Prod	Agentes estrogenicos
US5747480A (en) *	1996-05-08	1998-05-05	American Home Products Corporation	Oral contraceptive

1998
- 1998-04-11 ID IDW20000811A patent/ID24568A/id unknown
- 1998-04-11 UA UA2000063196A patent/UA68365C2/uk unknown
- 1998-11-04 GE GEAP19985364A patent/GEP20043290B/en unknown
- 1998-11-04 SK SK648-2000A patent/SK6482000A3/sk unknown
- 1998-11-04 EP EP98956525A patent/EP1051179B1/fr not_active Expired - Lifetime
- 1998-11-04 BR BR9813982-7A patent/BR9813982A/pt not_active Application Discontinuation
- 1998-11-04 EA EA200000492A patent/EA200000492A1/ru unknown
- 1998-11-04 PL PL98340623A patent/PL340623A1/xx unknown
- 1998-11-04 CN CN98810911A patent/CN1278732A/zh active Pending
- 1998-11-04 WO PCT/US1998/023427 patent/WO1999024027A2/fr not_active Ceased
- 1998-11-04 HR HR20000269A patent/HRP20000269A2/hr not_active Application Discontinuation
- 1998-11-04 CZ CZ20001661A patent/CZ294155B6/cs not_active IP Right Cessation
- 1998-11-04 JP JP2000520119A patent/JP2001522798A/ja not_active Ceased
- 1998-11-04 ES ES98956525T patent/ES2246541T3/es not_active Expired - Lifetime
- 1998-11-04 DE DE69831605T patent/DE69831605T2/de not_active Expired - Lifetime
- 1998-11-04 NZ NZ503890A patent/NZ503890A/xx unknown
- 1998-11-04 CA CA002307210A patent/CA2307210A1/fr not_active Abandoned
- 1998-11-04 AU AU13031/99A patent/AU760540B2/en not_active Ceased
- 1998-11-04 HU HU0100293A patent/HUP0100293A3/hu unknown
- 1998-11-04 AT AT98956525T patent/ATE304359T1/de not_active IP Right Cessation
- 1998-11-04 TR TR2000/01268T patent/TR200001268T2/xx unknown
- 1998-11-04 DK DK98956525T patent/DK1051179T3/da active
- 1998-11-04 IL IL13562198A patent/IL135621A0/xx unknown
- 1998-11-04 EE EEP200000211A patent/EE04092B1/xx not_active IP Right Cessation
- 1998-11-05 AR ARP980105591A patent/AR016667A1/es not_active Application Discontinuation
- 1998-11-05 ZA ZA9810136A patent/ZA9810136B/xx unknown
2000
- 2000-04-27 NO NO20002167A patent/NO20002167L/no not_active Application Discontinuation
- 2000-05-17 BG BG104451A patent/BG104451A/xx unknown
2003
- 2003-06-23 AU AU2003204896A patent/AU2003204896B2/en not_active Ceased

Also Published As

Publication number	Publication date
CZ294155B6 (cs)	2004-10-13
NZ503890A (en)	2002-08-28
CN1278732A (zh)	2001-01-03
SK6482000A3 (en)	2000-11-07
AU760540B2 (en)	2003-05-15
DK1051179T3 (da)	2005-10-31
EE200000211A (et)	2001-04-16
WO1999024027A2 (fr)	1999-05-20
WO1999024027A3 (fr)	1999-07-15
ES2246541T3 (es)	2006-02-16
ID24568A (id)	2000-07-27
EA200000492A1 (ru)	2000-10-30
GEP20043290B (en)	2004-07-26
EP1051179A2 (fr)	2000-11-15
HRP20000269A2 (en)	2000-12-31
AR016667A1 (es)	2001-07-25
ATE304359T1 (de)	2005-09-15
IL135621A0 (en)	2001-05-20
AU1303199A (en)	1999-05-31
AU2003204896B2 (en)	2006-06-15
DE69831605T2 (de)	2006-06-14
EE04092B1 (et)	2003-08-15
HUP0100293A3 (en)	2002-12-28
JP2001522798A (ja)	2001-11-20
ZA9810136B (en)	2000-05-05
NO20002167L (no)	2000-06-28
HUP0100293A2 (hu)	2001-10-28
TR200001268T2 (tr)	2001-01-22
EP1051179B1 (fr)	2005-09-14
DE69831605D1 (de)	2005-10-20
CA2307210A1 (fr)	1999-05-20
UA68365C2 (en)	2004-08-16
BR9813982A (pt)	2000-09-26
NO20002167D0 (no)	2000-04-27
PL340623A1 (en)	2001-02-12
CZ20001661A3 (cs)	2000-12-13

Publication	Publication Date	Title
BG104451A (en)	2000-12-29	Antiestrogen and progestin-containing peroral contraceptives
NZ330741A (en)	2000-03-27	Contraceptive process and kit for female mammals, comprising a combination of gestagen and oestrogen
AU560487B2 (en)	1987-04-09	Contraceptive comprising gestodene and ethinylestradiol
DK0491415T3 (da)	1996-07-08	Orale svangerskabsforebyggende midler med lavt østrogen
DE69118494D1 (de)	1996-05-09	Kontrazeptionsverfahren und Schema
FI922206A0 (fi)	1992-05-14	Osmotisk, oral doseringsform foer fertilitets kontroll.
DE69710896D1 (en)	2002-04-11	Progestogen-anti-progestogen therapien
LU90341I2 (fr)	1999-03-29	75 Ug de désogestrel en l'absence éthinyl oestradiol (cerazette)
NZ333750A (en)	2000-09-29	Monophasic contraceptive method and kit comprising a combination of a progestin and estrogen
ATE91410T1 (de)	1993-07-15	Osmotische dosierungsform.
MX9707009A (es)	1997-11-29	Inyeccion de una vez al mes como un contraceptivo de base y para terapia de reemplazamiento hormonal para mujeres perimenopausicas y premenopausicas.
KR950024496U (ko)	1995-09-13	여성용 콘돔(女性用 condom)