BG107135A - Съединения, съдържащи бензоамидпиперидин и сроднисъединения - Google Patents
Съединения, съдържащи бензоамидпиперидин и сроднисъединения Download PDFInfo
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- BG107135A BG107135A BG107135A BG10713502A BG107135A BG 107135 A BG107135 A BG 107135A BG 107135 A BG107135 A BG 107135A BG 10713502 A BG10713502 A BG 10713502A BG 107135 A BG107135 A BG 107135A
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- Bulgaria
- Prior art keywords
- methyl
- phenyl
- methoxy
- piperidin
- ylamino
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Classifications
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- C07—ORGANIC CHEMISTRY
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- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
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- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/16—Drugs for disorders of the alimentary tract or the digestive system for liver or gallbladder disorders, e.g. hepatoprotective agents, cholagogues, litholytics
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- A—HUMAN NECESSITIES
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- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/06—Antiasthmatics
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- A—HUMAN NECESSITIES
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| EP2593452B1 (de) | 2010-07-14 | 2017-01-18 | Novartis AG | Heterocyclische verbindungen als ip-rezeptoragonisten |
| ES2376564B1 (es) | 2010-08-12 | 2013-01-24 | Manuel Vicente Salinas Martín | Utilización de anticuerpos contra los receptores nk1, nk2 y/o nk3, para producir apoptosis en las células tumorales y modificar el estroma, la inmunidad y la vascularización intra y peritumorales, como tratamiento del cáncer. |
| US8664247B2 (en) | 2011-08-26 | 2014-03-04 | Radiorx, Inc. | Acyclic organonitro compounds for use in treating cancer |
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| EP2837381A4 (de) | 2011-12-13 | 2015-12-09 | Servicio Andaluz De Salud | Verwendung von mitteln zur behandlung von krebs, die die peritumoralumgebung verändern |
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| US9987270B1 (en) | 2015-10-29 | 2018-06-05 | Epicentrix, Inc. | Treatment of gliomas using organonitro compound combination therapy |
| CN109069420A (zh) | 2016-01-11 | 2018-12-21 | 埃皮辛特瑞柯斯公司 | 2-溴-1-(3,3-二硝基氮杂环丁烷-1-基)乙酮静脉施用的组合物和方法 |
| RU2643091C2 (ru) * | 2016-04-08 | 2018-01-31 | Федеральное государственное бюджетное научное учреждение "Научно-исследовательский институт фармакологии имени В.В. Закусова" | Производные оксимов 4-бензоилпиридина, обладающие противосудорожной активностью, как средства лечения эпилепсии и пароксизмальных состояний |
| SG11201903312VA (en) | 2016-10-14 | 2019-05-30 | Epicentrix Inc | Sulfoxyalkyl organonitro and related compounds and pharmaceutical compositions for use in medicine |
| EP3648740A1 (de) | 2017-07-07 | 2020-05-13 | EpicentRx, Inc. | Zusammensetzungen zur parenteralen verabreichung von therapeutika |
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| US3539584A (en) * | 1967-11-14 | 1970-11-10 | Colgate Palmolive Co | 5-substituted-2,1-benzisothiazolines |
| US4581356A (en) * | 1983-03-22 | 1986-04-08 | Fujisawa Pharmaceutical Co., Ltd. | Triazine derivatives, and pharmaceutical compositions comprising the same |
| DE69109125T2 (de) * | 1990-09-28 | 1995-09-28 | Pfizer | Ringverknüpfte analoge von stickstoffenthaltenden nichtaromatischen heterocyclen. |
| TW202432B (de) * | 1991-06-21 | 1993-03-21 | Pfizer | |
| US6180647B1 (en) * | 1995-07-07 | 2001-01-30 | Pfizer Inc. | Substituted benzolactam compounds as substance P antagonists |
| TWI220143B (en) * | 1998-05-13 | 2004-08-11 | Solvay Pharm Gmbh | Method for stereochemically controlled production of isomerically pure highly substituted azacyclic compounds and novel cyclic compounds, and intermediate products |
| WO2000073312A1 (en) * | 1999-05-26 | 2000-12-07 | Astrazeneca Ab | Compounds |
| SE9901901D0 (sv) * | 1999-05-26 | 1999-05-26 | Astra Ab | Compounds |
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2001
- 2001-04-06 PL PL01358623A patent/PL358623A1/xx not_active Application Discontinuation
- 2001-04-06 BR BR0109936-1A patent/BR0109936A/pt not_active IP Right Cessation
- 2001-04-06 DE DE60112064T patent/DE60112064T2/de not_active Expired - Fee Related
- 2001-04-06 ES ES01919702T patent/ES2244599T3/es not_active Expired - Lifetime
- 2001-04-06 MX MXPA02010029A patent/MXPA02010029A/es active IP Right Grant
- 2001-04-06 EA EA200200963A patent/EA005409B1/ru not_active IP Right Cessation
- 2001-04-06 CA CA002405089A patent/CA2405089A1/en not_active Abandoned
- 2001-04-06 CN CN01807882A patent/CN1432011A/zh active Pending
- 2001-04-06 AU AU2001246761A patent/AU2001246761A1/en not_active Abandoned
- 2001-04-06 HR HRP20020808 patent/HRP20020808A2/hr not_active Application Discontinuation
- 2001-04-06 AP APAP/P/2002/002647A patent/AP2002002647A0/en unknown
- 2001-04-06 YU YU73902A patent/YU73902A/sh unknown
- 2001-04-06 HU HU0300413A patent/HUP0300413A2/hu unknown
- 2001-04-06 NZ NZ521346A patent/NZ521346A/en unknown
- 2001-04-06 OA OA1200200312A patent/OA12245A/en unknown
- 2001-04-06 KR KR1020027013582A patent/KR20020087134A/ko not_active Ceased
- 2001-04-06 JP JP2001575573A patent/JP4001486B2/ja not_active Expired - Fee Related
- 2001-04-06 WO PCT/IB2001/000629 patent/WO2001077100A2/en not_active Ceased
- 2001-04-06 EE EEP200200588A patent/EE200200588A/xx unknown
- 2001-04-06 EP EP01919702A patent/EP1272484B1/de not_active Expired - Lifetime
- 2001-04-06 SK SK1394-2002A patent/SK13942002A3/sk not_active Application Discontinuation
- 2001-04-06 IL IL15220901A patent/IL152209A0/xx unknown
- 2001-04-06 CZ CZ20023213A patent/CZ20023213A3/cs unknown
- 2001-04-06 AT AT01919702T patent/ATE299875T1/de not_active IP Right Cessation
- 2001-04-09 AR ARP010101678A patent/AR033976A1/es unknown
- 2001-04-10 UY UY26662A patent/UY26662A1/es not_active Application Discontinuation
- 2001-04-10 PA PA20018515101A patent/PA8515101A1/es unknown
- 2001-04-10 PE PE2001000329A patent/PE20011311A1/es not_active Application Discontinuation
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2002
- 2002-09-20 IS IS6561A patent/IS6561A/is unknown
- 2002-09-23 BG BG107135A patent/BG107135A/bg unknown
- 2002-10-02 MA MA26848A patent/MA26891A1/fr unknown
- 2002-10-09 NO NO20024874A patent/NO20024874L/no not_active Application Discontinuation
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2003
- 2003-06-26 AR ARP030102296A patent/AR040346A2/es unknown
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