OA12245A - Benzoamide piperidine compounds as substance P antagonists. - Google Patents
Benzoamide piperidine compounds as substance P antagonists. Download PDFInfo
- Publication number
- OA12245A OA12245A OA1200200312A OA1200200312A OA12245A OA 12245 A OA12245 A OA 12245A OA 1200200312 A OA1200200312 A OA 1200200312A OA 1200200312 A OA1200200312 A OA 1200200312A OA 12245 A OA12245 A OA 12245A
- Authority
- OA
- OAPI
- Prior art keywords
- methyl
- phenyl
- methoxy
- piperidin
- ylamino
- Prior art date
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- NXUSCSCBRVCRCN-UHFFFAOYSA-N benzamide;piperidine Chemical class C1CCNCC1.NC(=O)C1=CC=CC=C1 NXUSCSCBRVCRCN-UHFFFAOYSA-N 0.000 title abstract description 3
- 239000003890 substance P antagonist Substances 0.000 title description 3
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| AU2003902882A0 (en) * | 2003-06-10 | 2003-06-26 | Fujisawa Pharmaceutical Co., Ltd. | Piperidyl derivatives |
| ES2246687B2 (es) | 2004-02-11 | 2006-11-16 | Miguel Muñoz Saez | Utilizacion de antagonistas no peptidicos de receptores nk1 para la produccion de apoptosis en celulas tumorales. |
| WO2006023630A2 (en) * | 2004-08-20 | 2006-03-02 | Targacept, Inc. | The use of n-aryl diazaspiracyclic compounds in the treatment of addiction |
| TW200800959A (en) | 2005-06-10 | 2008-01-01 | Wyeth Corp | Piperazine-piperidine antagonists and agonists of the 5-HT1a receptor |
| US20060281670A1 (en) * | 2005-06-10 | 2006-12-14 | Wisconsin Alumni Research Foundation (Warf) | Compositions and methods for modulating angiogenesis |
| US7507842B2 (en) | 2005-08-12 | 2009-03-24 | Radiorx, Inc. | Cyclic nitro compounds, pharmaceutical compositions thereof and uses thereof |
| US20070135380A1 (en) | 2005-08-12 | 2007-06-14 | Radiorx, Inc. | O-nitro compounds, pharmaceutical compositions thereof and uses thereof |
| DE102006033114A1 (de) | 2006-07-18 | 2008-01-24 | Grünenthal GmbH | Spirocyclische Azaindol-Derivate |
| CL2008000119A1 (es) | 2007-01-16 | 2008-05-16 | Wyeth Corp | Compuestos derivados de pirazol, antagonistas del receptor nicotinico de acetilcolina; composicion farmaceutica; y uso en el tratamiento de enfermedades tales como demencia senil, alzheimer y esquizofrenia. |
| JP2010516734A (ja) | 2007-01-24 | 2010-05-20 | グラクソ グループ リミテッド | 3,5−ジアミノ−6−(2,3−ジクロロフェニル)−1,2,4−トリアジンまたはr(−)−2,4−ジアミノ−5−(2,3−ジクロロフェニル)−6−フルオロメチルピリミジンを含む医薬組成物 |
| US8471041B2 (en) | 2010-02-09 | 2013-06-25 | Alliant Techsystems Inc. | Methods of synthesizing and isolating N-(bromoacetyl)-3,3-dinitroazetidine and a composition including the same |
| MA34373B1 (fr) * | 2010-07-14 | 2013-07-03 | Novartis Ag | Composés hétérocycliques agonistes du récepteur ip |
| ES2376564B1 (es) | 2010-08-12 | 2013-01-24 | Manuel Vicente Salinas Martín | Utilización de anticuerpos contra los receptores nk1, nk2 y/o nk3, para producir apoptosis en las células tumorales y modificar el estroma, la inmunidad y la vascularización intra y peritumorales, como tratamiento del cáncer. |
| US8664247B2 (en) | 2011-08-26 | 2014-03-04 | Radiorx, Inc. | Acyclic organonitro compounds for use in treating cancer |
| CA2850723C (en) | 2011-10-07 | 2019-07-09 | Radiorx, Inc. | Organonitro thioether compounds and medical uses thereof |
| US20140308260A1 (en) | 2011-10-07 | 2014-10-16 | Radiorx, Inc. | Methods and compositions comprising a nitrite-reductase promoter for treatment of medical disorders and preservation of blood products |
| WO2013087964A1 (es) | 2011-12-13 | 2013-06-20 | Servicio Andaluz De Salud | Uso de agentes modificadores del ambiente peritumoral para el tratamiento del cáncer |
| JP6440625B2 (ja) | 2012-11-14 | 2018-12-19 | ザ・ジョンズ・ホプキンス・ユニバーシティー | 精神分裂病を処置するための方法および組成物 |
| RU2506077C1 (ru) * | 2013-01-25 | 2014-02-10 | Общество С Ограниченной Ответственностью "Валента-Интеллект" | Комбинация для профилактики, коррекции и терапии боли, связанной с нейродегенерацией или ассоциированной с соматоформными расстройствами |
| ES2493693B1 (es) | 2013-02-11 | 2015-07-07 | Servicio Andaluz De Salud | Método para predecir o pronosticar la respuesta de un sujeto humano que padece un cáncer al tratamiento con un antagonista del receptor NK1 |
| US9604981B2 (en) | 2013-02-13 | 2017-03-28 | Novartis Ag | IP receptor agonist heterocyclic compounds |
| ES2541870B1 (es) | 2013-12-27 | 2016-05-12 | Servicio Andaluz De Salud | Uso de antagonistas no peptídicos de NK1 en una determinada dosis para el tratamiento del cáncer |
| WO2016105448A1 (en) * | 2014-12-22 | 2016-06-30 | Darryl Rideout | Imidazoline receptor type 1 ligands for use as therapeutics |
| US10342778B1 (en) | 2015-10-20 | 2019-07-09 | Epicentrx, Inc. | Treatment of brain metastases using organonitro compound combination therapy |
| US9987270B1 (en) | 2015-10-29 | 2018-06-05 | Epicentrix, Inc. | Treatment of gliomas using organonitro compound combination therapy |
| SG11201805942UA (en) | 2016-01-11 | 2018-08-30 | Epicentrx Inc | Compositions and methods for intravenous administration of 2-bromo-1-(3,3-dinitroazetidin-1-yl)ethanone |
| RU2643091C2 (ru) * | 2016-04-08 | 2018-01-31 | Федеральное государственное бюджетное научное учреждение "Научно-исследовательский институт фармакологии имени В.В. Закусова" | Производные оксимов 4-бензоилпиридина, обладающие противосудорожной активностью, как средства лечения эпилепсии и пароксизмальных состояний |
| EA201990949A1 (ru) | 2016-10-14 | 2019-10-31 | Сульфоксиалкильные органические нитросоединения и родственные соединения и фармацевтические композиции для применения в медицине | |
| IL311727A (en) | 2017-07-07 | 2024-05-01 | Epicentrx Inc | Preparations for intravenous administration of medical substances |
| WO2019164593A2 (en) | 2018-01-08 | 2019-08-29 | Epicentrx, Inc. | Methods and compositions utilizing rrx-001 combination therapy for radioprotection |
| US12497362B2 (en) | 2020-08-18 | 2025-12-16 | Merck Sharp & Dohme Llc | Cyclopentapyrrole orexin receptor agonists |
| IL312896A (en) * | 2021-11-18 | 2024-07-01 | Wuhan Humanwell Innovative Drug Res And Development Center Limited Company | 15-PGDH inhibitor and its use |
| US20250214980A1 (en) | 2022-03-14 | 2025-07-03 | Slap Pharmaceuticals Llc | Multicyclic compounds |
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| US3539584A (en) * | 1967-11-14 | 1970-11-10 | Colgate Palmolive Co | 5-substituted-2,1-benzisothiazolines |
| US4581356A (en) * | 1983-03-22 | 1986-04-08 | Fujisawa Pharmaceutical Co., Ltd. | Triazine derivatives, and pharmaceutical compositions comprising the same |
| AU651145B2 (en) * | 1990-09-28 | 1994-07-14 | Pfizer Inc. | Fused ring analogs of nitrogen containing nonaromatic heterocycles |
| TW202432B (de) * | 1991-06-21 | 1993-03-21 | Pfizer | |
| ATE199552T1 (de) * | 1995-07-07 | 2001-03-15 | Pfizer | Substituierte benzolaktamverbindungen als substanz-p-antagonisten |
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- 2001-04-06 PL PL01358623A patent/PL358623A1/xx not_active Application Discontinuation
- 2001-04-06 KR KR1020027013582A patent/KR20020087134A/ko not_active Ceased
- 2001-04-06 YU YU73902A patent/YU73902A/sh unknown
- 2001-04-06 CN CN01807882A patent/CN1432011A/zh active Pending
- 2001-04-06 OA OA1200200312A patent/OA12245A/en unknown
- 2001-04-06 WO PCT/IB2001/000629 patent/WO2001077100A2/en not_active Ceased
- 2001-04-06 EE EEP200200588A patent/EE200200588A/xx unknown
- 2001-04-06 JP JP2001575573A patent/JP4001486B2/ja not_active Expired - Fee Related
- 2001-04-06 HR HRP20020808 patent/HRP20020808A2/hr not_active Application Discontinuation
- 2001-04-06 ES ES01919702T patent/ES2244599T3/es not_active Expired - Lifetime
- 2001-04-06 BR BR0109936-1A patent/BR0109936A/pt not_active IP Right Cessation
- 2001-04-06 SK SK1394-2002A patent/SK13942002A3/sk not_active Application Discontinuation
- 2001-04-06 HU HU0300413A patent/HUP0300413A2/hu unknown
- 2001-04-06 EP EP01919702A patent/EP1272484B1/de not_active Expired - Lifetime
- 2001-04-06 AT AT01919702T patent/ATE299875T1/de not_active IP Right Cessation
- 2001-04-06 AU AU2001246761A patent/AU2001246761A1/en not_active Abandoned
- 2001-04-09 AR ARP010101678A patent/AR033976A1/es unknown
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- 2001-04-10 PE PE2001000329A patent/PE20011311A1/es not_active Application Discontinuation
- 2001-04-10 UY UY26662A patent/UY26662A1/es not_active Application Discontinuation
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2002
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- 2002-09-23 BG BG107135A patent/BG107135A/bg unknown
- 2002-10-02 MA MA26848A patent/MA26891A1/fr unknown
- 2002-10-09 NO NO20024874A patent/NO20024874L/no not_active Application Discontinuation
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2003
- 2003-06-26 AR ARP030102296A patent/AR040346A2/es unknown
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