BG17800A3 - Метод за получаване на 2-(5-нитро-2-фурил)-тиено (3,2-d)пиримидини - Google Patents

Метод за получаване на 2-(5-нитро-2-фурил)-тиено (3,2-d)пиримидини

Info

Publication number
BG17800A3
BG17800A3 BG017732A BG1773270A BG17800A3 BG 17800 A3 BG17800 A3 BG 17800A3 BG 017732 A BG017732 A BG 017732A BG 1773270 A BG1773270 A BG 1773270A BG 17800 A3 BG17800 A3 BG 17800A3
Authority
BG
Bulgaria
Prior art keywords
thieno
pyrimidines
furyl
nitro
preparation
Prior art date
Application number
BG017732A
Other languages
Bulgarian (bg)
English (en)
Inventor
Eberhard Woitun
Wolfgang Reuter
Original Assignee
Dr. Karl Thomae Gmbh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from DE19691959403 external-priority patent/DE1959403A1/de
Priority claimed from DE19702050814 external-priority patent/DE2050814A1/de
Priority claimed from DE19702050816 external-priority patent/DE2050816A1/de
Priority claimed from DE19702050815 external-priority patent/DE2050815A1/de
Application filed by Dr. Karl Thomae Gmbh filed Critical Dr. Karl Thomae Gmbh
Publication of BG17800A3 publication Critical patent/BG17800A3/xx

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D495/00Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
    • C07D495/02Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D495/04Ortho-condensed systems
    • YGENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02PCLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00Technologies relating to chemical industry
    • Y02P20/50Improvements relating to the production of bulk chemicals
    • Y02P20/55Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
BG017732A 1969-11-26 1970-11-17 Метод за получаване на 2-(5-нитро-2-фурил)-тиено (3,2-d)пиримидини BG17800A3 (bg)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
DE19691959403 DE1959403A1 (de) 1969-11-26 1969-11-26 Neue 2-(5-Nitro-2-furyl)-thieno[3,2-d]pyrimidine und Verfahren zu ihrer Herstellung
DE19702050814 DE2050814A1 (de) 1970-10-16 1970-10-16 Neue Verfahren zur Herstellung von 2-(5-Nitro-2-furyl)-thieno eckige Klammer auf 3,2-d eckige Klammer zu pyrimidinen
DE19702050816 DE2050816A1 (de) 1970-10-16 1970-10-16 Neue 2-(Nitro-2-furyl>thieno eckige Klammer auf 3,2-d eckige Klammer zu pyrimidine
DE19702050815 DE2050815A1 (de) 1970-10-16 1970-10-16 Neue 2-(5-Nitro-2-furyl)-thieno eckige Klammer auf 3,2-d eckige Klammer zu pyrimidine

Publications (1)

Publication Number Publication Date
BG17800A3 true BG17800A3 (bg) 1973-12-25

Family

ID=27430978

Family Applications (2)

Application Number Title Priority Date Filing Date
BG017732A BG17800A3 (bg) 1969-11-26 1970-11-17 Метод за получаване на 2-(5-нитро-2-фурил)-тиено (3,2-d)пиримидини
BG016080A BG17799A3 (bg) 1969-11-26 1970-11-17 Метод за получаване на 2-/5-нитро-2-фурил/-тиено/3,2-d/ пиримидини

Family Applications After (1)

Application Number Title Priority Date Filing Date
BG016080A BG17799A3 (bg) 1969-11-26 1970-11-17 Метод за получаване на 2-/5-нитро-2-фурил/-тиено/3,2-d/ пиримидини

Country Status (13)

Country Link
US (1) US3661908A (mo)
BE (1) BE759493A (mo)
BG (2) BG17800A3 (mo)
CA (1) CA926865A (mo)
CH (3) CH568324A5 (mo)
DK (1) DK128781B (mo)
FR (1) FR2073416B1 (mo)
GB (1) GB1321316A (mo)
IE (1) IE34765B1 (mo)
IL (1) IL35729A (mo)
NL (1) NL7017210A (mo)
NO (1) NO129954B (mo)
SE (1) SE377938B (mo)

Families Citing this family (21)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3932642A (en) * 1971-04-10 1976-01-13 Boehringer Ingelheim Gmbh Biocidal compositions containing a 2- (5'-nitro-2'-furyl)-thieno(2,3-d) pyrimidine and methods of use
US6187777B1 (en) 1998-02-06 2001-02-13 Amgen Inc. Compounds and methods which modulate feeding behavior and related diseases
US6608053B2 (en) * 2000-04-27 2003-08-19 Yamanouchi Pharmaceutical Co., Ltd. Fused heteroaryl derivatives
US20040138238A1 (en) * 2002-08-08 2004-07-15 Dhanoa Dale S. Substituted aminopyrimidine compounds as neurokinin antagonists
GB0423653D0 (en) * 2004-10-25 2004-11-24 Piramed Ltd Pharmaceutical compounds
JP5148597B2 (ja) 2006-04-26 2013-02-20 エフ.ホフマン−ラ ロシュ アーゲー 医薬化合物
CL2007001167A1 (es) 2006-04-26 2008-01-25 Genentech Inc Compuestos derivados de pirimidina condensada, inhibidores de p13-quinasa; procesos para preparar los compuestos; composicion farmaceutica que los comprende; uso de los compuestos en la preparacion de medicamentos; proceso para preparar la composicion farmaceutica; y kit que incluye a la composicionfarmaceutica.
KR101402474B1 (ko) * 2006-04-26 2014-06-19 제넨테크, 인크. 포스포이노시티드 3-키나제 억제제 화합물 및 이를 포함하는 약학적 조성물
ES2571028T3 (es) * 2006-12-07 2016-05-23 Genentech Inc Compuestos inhibidores de fosfoinositida 3-cinasa y métodos de uso
JP5284977B2 (ja) 2006-12-07 2013-09-11 エフ・ホフマン−ラ・ロシュ・アクチェンゲゼルシャフト ホスホイノシチド3−キナーゼ阻害剤化合物及び使用方法
ATE510841T1 (de) * 2007-06-12 2011-06-15 Hoffmann La Roche Thiazoliopyrimidine und ihre verwendung als hemmer der phosphatidylinositol-3 kinase
ES2399774T3 (es) * 2007-09-24 2013-04-03 Genentech, Inc. Compuestos de tiazolopirimidina inhibidores de PI3K y métodos de uso
CN101909631B (zh) * 2007-10-25 2012-09-12 健泰科生物技术公司 制备噻吩并嘧啶化合物的方法
GB0721095D0 (en) * 2007-10-26 2007-12-05 Piramed Ltd Pharmaceutical compounds
EP2405916B1 (en) 2009-03-12 2018-02-07 Genentech, Inc. Combinations of phosphoinositide 3-kinase inhibitor compounds and chemotherapeutic agents for the treatment of hematopoietic malignancies
EP2435438A1 (en) 2009-05-27 2012-04-04 Genentech, Inc. Bicyclic pyrimidine pi3k inhibitor compounds selective for p110 delta, and methods of use
CA2772371A1 (en) * 2009-05-27 2010-12-02 F. Hoffmann-La Roche Ag Bicyclic indole-pyrimidine pi3k inhibitor compounds selective for p110 delta, and methods of use
ES2609767T3 (es) * 2009-10-12 2017-04-24 F. Hoffmann-La Roche Ag Combinaciones de un inhibidor de PI3K y un inhibidor de MEK
JP2013528787A (ja) 2010-04-16 2013-07-11 ジェネンテック, インコーポレイテッド Pi3k/aktキナーゼ経路インヒビターの効果の予測バイオマーカーとしてのfox03a
WO2012088254A1 (en) 2010-12-22 2012-06-28 Genentech, Inc. Autophagy inducer and inhibitor combination therapy for the treatment of neoplasms
CA2901126C (en) 2013-02-25 2022-01-25 Genentech, Inc. Methods and compositions for detecting and treating drug resistant akt mutant

Also Published As

Publication number Publication date
NL7017210A (mo) 1971-05-28
IE34765L (en) 1971-05-26
CA926865A (en) 1973-05-22
CH567029A5 (mo) 1975-09-30
DK128781B (da) 1974-07-01
BE759493A (fr) 1971-05-25
IL35729A (en) 1974-01-14
FR2073416A1 (mo) 1971-10-01
BG17799A3 (bg) 1973-12-25
IL35729A0 (en) 1971-01-28
SE377938B (mo) 1975-08-04
NO129954B (mo) 1974-06-17
IE34765B1 (en) 1975-08-06
US3661908A (en) 1972-05-09
CH568324A5 (mo) 1975-10-31
GB1321316A (en) 1973-06-27
FR2073416B1 (mo) 1975-04-18
CH559210A5 (mo) 1975-02-28

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