BG20593A3 - Метод за получаване на тиено<3,2-д>пиримидини - Google Patents
Метод за получаване на тиено<3,2-д>пиримидиниInfo
- Publication number
- BG20593A3 BG20593A3 BG020371A BG2037172A BG20593A3 BG 20593 A3 BG20593 A3 BG 20593A3 BG 020371 A BG020371 A BG 020371A BG 2037172 A BG2037172 A BG 2037172A BG 20593 A3 BG20593 A3 BG 20593A3
- Authority
- BG
- Bulgaria
- Prior art keywords
- pyrimidines
- thieno
- obtaining
- obtaining thieno
- Prior art date
Links
- 150000003230 pyrimidines Chemical class 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
- C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
- C07D495/04—Ortho-condensed systems
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DE19712121950 DE2121950A1 (en) | 1971-05-04 | 1971-05-04 | Thieno(3,2-d)pyrimidine derivs - with thrombocyte aggregation inhibiting activity |
| DE19712137341 DE2137341A1 (de) | 1971-07-26 | 1971-07-26 | Neue thieno eckige klammer auf 3,2-d eckige klammer zu pyrimidine |
| DE19722215299 DE2215299A1 (de) | 1972-03-29 | 1972-03-29 | Neue thieno eckige klammer auf 3,2-d eckige klammer zu pyrimidine |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| BG20593A3 true BG20593A3 (bg) | 1975-12-05 |
Family
ID=27183398
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| BG020371A BG20593A3 (bg) | 1971-05-04 | 1972-05-03 | Метод за получаване на тиено<3,2-д>пиримидини |
Country Status (15)
| Country | Link |
|---|---|
| US (1) | US3888851A (fr) |
| AT (1) | AT318619B (fr) |
| AU (1) | AU4181572A (fr) |
| BE (1) | BE783044A (fr) |
| BG (1) | BG20593A3 (fr) |
| DD (1) | DD97656A5 (fr) |
| DK (1) | DK129844B (fr) |
| ES (1) | ES402302A1 (fr) |
| FR (1) | FR2135294B1 (fr) |
| GB (1) | GB1393161A (fr) |
| HU (1) | HU163960B (fr) |
| IL (1) | IL39341A (fr) |
| NL (1) | NL7206041A (fr) |
| PL (1) | PL82381B1 (fr) |
| RO (1) | RO62428A (fr) |
Families Citing this family (23)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4054656A (en) * | 1975-09-10 | 1977-10-18 | Mead Johnson & Company | Thieno[2,3-d]pyrimidine antiallergic agents |
| US5098902A (en) * | 1991-03-18 | 1992-03-24 | Warner-Lambert Company | Method of treating neurodegenerative diseases |
| CA2129337A1 (fr) * | 1992-02-19 | 1993-09-02 | Jotham W. Coe | Composes heterocycliques pour ameliorer l'activite antitumorale |
| PL340412A1 (en) | 1997-10-20 | 2001-01-29 | Hoffmann La Roche | Bicyclic kinase inhibitors |
| US6187777B1 (en) | 1998-02-06 | 2001-02-13 | Amgen Inc. | Compounds and methods which modulate feeding behavior and related diseases |
| GB0423653D0 (en) | 2004-10-25 | 2004-11-24 | Piramed Ltd | Pharmaceutical compounds |
| CN101163706A (zh) * | 2005-04-21 | 2008-04-16 | 贝林格尔·英格海姆国际有限公司 | 用于治疗炎性疾病的二氢噻吩并嘧啶 |
| PL2041139T3 (pl) | 2006-04-26 | 2012-05-31 | Hoffmann La Roche | Związki farmaceutyczne |
| MX2008013583A (es) | 2006-04-26 | 2008-10-31 | Genentech Inc | Compuestos del inhibidor de fosfoinositido 3-cinasa y composiciones farmaceuticas que los contienen. |
| KR101533461B1 (ko) | 2006-04-26 | 2015-07-02 | 에프. 호프만-라 로슈 아게 | Pi3k저해제로 유용한 티에노[3,2-d]피리미딘 유도체 |
| AR064154A1 (es) * | 2006-12-07 | 2009-03-18 | Piramed Ltd | Compuestos inhibidores de fodfoinostida 3- quinasas y composiciones farmaceuticas |
| PE20081679A1 (es) | 2006-12-07 | 2008-12-18 | Hoffmann La Roche | Compuestos del inhibidor de fosfoinositida 3-cinasa y metodos de uso |
| JP5736171B2 (ja) | 2007-09-24 | 2015-06-17 | ジェネンテック, インコーポレイテッド | チアゾロピリミジンpi3k阻害剤化合物および使用方法 |
| JP5341899B2 (ja) * | 2007-10-19 | 2013-11-13 | ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング | ヘテロ環置換ピペラジノ−ジヒドロチエノピリミジン |
| EP2214675B1 (fr) | 2007-10-25 | 2013-11-20 | Genentech, Inc. | Procédé de préparation de composés de thiénopyrimidine |
| GB0721095D0 (en) | 2007-10-26 | 2007-12-05 | Piramed Ltd | Pharmaceutical compounds |
| BRPI1006189A2 (pt) | 2009-03-12 | 2020-08-18 | Genentech Inc | uso de uma combinação terapêutica, formulação farmacêutica, artigo de manufatura, produto, método para determinar compostos a serem utilizados em combinação para o tratamento de uma malignidade hematopoiética e método para selecionar compostos a serem utilizados em combinação para o tratamento de câncer |
| US8173650B2 (en) | 2009-05-27 | 2012-05-08 | Genentech, Inc. | Bicyclic pyrimidine PI3K inhibitor compounds selective for P110 delta, and methods of use |
| WO2010136491A1 (fr) * | 2009-05-27 | 2010-12-02 | F. Hoffmann-La Roche Ag | Composés bicycliques indole-pyrimidine inhibiteurs de pi3k sélectifs pour p110 delta et leurs procédés d'utilisation |
| CN103038643A (zh) | 2010-04-16 | 2013-04-10 | 基因泰克公司 | 作为pi3k/akt激酶途径抑制剂效能的预测性生物标记的foxo3a |
| WO2012088254A1 (fr) | 2010-12-22 | 2012-06-28 | Genentech, Inc. | Polythérapie par inducteur et inhibiteur d'autophagie pour le traitement de néoplasmes |
| WO2014130923A2 (fr) | 2013-02-25 | 2014-08-28 | Genentech, Inc. | Procédés et compositions pour détecter et traiter un mutant d'akt résistant aux médicaments |
| GB201410816D0 (en) * | 2014-06-17 | 2014-07-30 | Ucb Biopharma Sprl And Katholieke Universiteit Leuven | Therapeutic agents |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3259623A (en) * | 1963-06-14 | 1966-07-05 | Olin Mathieson | Process for preparing 2-(secondary amino)-halogenopyrimidines |
| DE1470356A1 (de) * | 1964-01-15 | 1970-04-30 | Thomae Gmbh Dr K | Neue Thieno[3,2-d]pyrimidine und Verfahren zu ihrer Herstellung |
| US3210368A (en) * | 1964-09-29 | 1965-10-05 | Ciba Geigy Corp | Certain 2-amino-4-aryl-5-n, n-disubstituted amino-lower alkyl-thiazole compounds |
-
1972
- 1972-04-28 RO RO7200070735A patent/RO62428A/fr unknown
- 1972-05-02 ES ES402302A patent/ES402302A1/es not_active Expired
- 1972-05-02 HU HUTO875A patent/HU163960B/hu unknown
- 1972-05-03 BG BG020371A patent/BG20593A3/xx unknown
- 1972-05-03 DK DK219672AA patent/DK129844B/da unknown
- 1972-05-03 DD DD162711A patent/DD97656A5/xx unknown
- 1972-05-03 PL PL1972155128A patent/PL82381B1/pl unknown
- 1972-05-03 AU AU41815/72A patent/AU4181572A/en not_active Expired
- 1972-05-03 IL IL39341A patent/IL39341A/xx unknown
- 1972-05-03 GB GB2058472A patent/GB1393161A/en not_active Expired
- 1972-05-03 AT AT382972A patent/AT318619B/de not_active IP Right Cessation
- 1972-05-03 US US249782A patent/US3888851A/en not_active Expired - Lifetime
- 1972-05-04 FR FR7215929A patent/FR2135294B1/fr not_active Expired
- 1972-05-04 BE BE783044A patent/BE783044A/fr unknown
- 1972-05-04 NL NL7206041A patent/NL7206041A/xx unknown
Also Published As
| Publication number | Publication date |
|---|---|
| AU4181572A (en) | 1973-11-08 |
| ES402302A1 (es) | 1975-04-01 |
| GB1393161A (en) | 1975-05-07 |
| HU163960B (fr) | 1973-11-28 |
| PL82381B1 (fr) | 1975-10-31 |
| IL39341A (en) | 1975-08-31 |
| DK129844C (fr) | 1975-05-12 |
| NL7206041A (fr) | 1972-11-07 |
| AT318619B (de) | 1974-11-11 |
| RO62428A (fr) | 1978-01-15 |
| DD97656A5 (fr) | 1973-05-12 |
| US3888851A (en) | 1975-06-10 |
| IL39341A0 (en) | 1972-07-26 |
| FR2135294B1 (fr) | 1975-10-17 |
| BE783044A (fr) | 1972-11-06 |
| DK129844B (da) | 1974-11-25 |
| FR2135294A1 (fr) | 1972-12-15 |
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