BE783044A - Nouvelles thieno(3,2-d) pyrimidines - Google Patents

Nouvelles thieno(3,2-d) pyrimidines

Info

Publication number
BE783044A
BE783044A BE783044A BE783044A BE783044A BE 783044 A BE783044 A BE 783044A BE 783044 A BE783044 A BE 783044A BE 783044 A BE783044 A BE 783044A BE 783044 A BE783044 A BE 783044A
Authority
BE
Belgium
Prior art keywords
thieno
pyrimidines
news
news thieno
Prior art date
Application number
BE783044A
Other languages
English (en)
Original Assignee
Thomae Gmbh Dr K
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from DE19712121950 external-priority patent/DE2121950A1/de
Priority claimed from DE19712137341 external-priority patent/DE2137341A1/de
Priority claimed from DE19722215299 external-priority patent/DE2215299A1/de
Application filed by Thomae Gmbh Dr K filed Critical Thomae Gmbh Dr K
Publication of BE783044A publication Critical patent/BE783044A/fr

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D495/00Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
    • C07D495/02Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D495/04Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
BE783044A 1971-05-04 1972-05-04 Nouvelles thieno(3,2-d) pyrimidines BE783044A (fr)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
DE19712121950 DE2121950A1 (en) 1971-05-04 1971-05-04 Thieno(3,2-d)pyrimidine derivs - with thrombocyte aggregation inhibiting activity
DE19712137341 DE2137341A1 (de) 1971-07-26 1971-07-26 Neue thieno eckige klammer auf 3,2-d eckige klammer zu pyrimidine
DE19722215299 DE2215299A1 (de) 1972-03-29 1972-03-29 Neue thieno eckige klammer auf 3,2-d eckige klammer zu pyrimidine

Publications (1)

Publication Number Publication Date
BE783044A true BE783044A (fr) 1972-11-06

Family

ID=27183398

Family Applications (1)

Application Number Title Priority Date Filing Date
BE783044A BE783044A (fr) 1971-05-04 1972-05-04 Nouvelles thieno(3,2-d) pyrimidines

Country Status (15)

Country Link
US (1) US3888851A (fr)
AT (1) AT318619B (fr)
AU (1) AU4181572A (fr)
BE (1) BE783044A (fr)
BG (1) BG20593A3 (fr)
DD (1) DD97656A5 (fr)
DK (1) DK129844B (fr)
ES (1) ES402302A1 (fr)
FR (1) FR2135294B1 (fr)
GB (1) GB1393161A (fr)
HU (1) HU163960B (fr)
IL (1) IL39341A (fr)
NL (1) NL7206041A (fr)
PL (1) PL82381B1 (fr)
RO (1) RO62428A (fr)

Families Citing this family (23)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4054656A (en) * 1975-09-10 1977-10-18 Mead Johnson & Company Thieno[2,3-d]pyrimidine antiallergic agents
US5098902A (en) * 1991-03-18 1992-03-24 Warner-Lambert Company Method of treating neurodegenerative diseases
EP0626964A1 (fr) * 1992-02-19 1994-12-07 Pfizer Inc. Composes heterocycliques ameliorant l'activite antitumorale
AU745579B2 (en) 1997-10-20 2002-03-21 F. Hoffmann-La Roche Ag Bicyclic kinase inhibitors
US6187777B1 (en) 1998-02-06 2001-02-13 Amgen Inc. Compounds and methods which modulate feeding behavior and related diseases
GB0423653D0 (en) 2004-10-25 2004-11-24 Piramed Ltd Pharmaceutical compounds
EP2060575A1 (fr) * 2006-04-19 2009-05-20 Boehringer Ingelheim International GmbH Dihydrothienopyrimidines et leur utilisation pour traiter des maladies inflammatoires
KR101402474B1 (ko) 2006-04-26 2014-06-19 제넨테크, 인크. 포스포이노시티드 3-키나제 억제제 화합물 및 이를 포함하는 약학적 조성물
JP5148597B2 (ja) 2006-04-26 2013-02-20 エフ.ホフマン−ラ ロシュ アーゲー 医薬化合物
CL2007001167A1 (es) 2006-04-26 2008-01-25 Genentech Inc Compuestos derivados de pirimidina condensada, inhibidores de p13-quinasa; procesos para preparar los compuestos; composicion farmaceutica que los comprende; uso de los compuestos en la preparacion de medicamentos; proceso para preparar la composicion farmaceutica; y kit que incluye a la composicionfarmaceutica.
ES2571028T3 (es) 2006-12-07 2016-05-23 Genentech Inc Compuestos inhibidores de fosfoinositida 3-cinasa y métodos de uso
JP5284977B2 (ja) 2006-12-07 2013-09-11 エフ・ホフマン−ラ・ロシュ・アクチェンゲゼルシャフト ホスホイノシチド3−キナーゼ阻害剤化合物及び使用方法
ES2399774T3 (es) 2007-09-24 2013-04-03 Genentech, Inc. Compuestos de tiazolopirimidina inhibidores de PI3K y métodos de uso
BRPI0817781A2 (pt) * 2007-10-19 2019-09-24 Boehringer Ingelheim Int piperazino-diidroteinopirimidinas substituídas com heterociclo
CN101909631B (zh) * 2007-10-25 2012-09-12 健泰科生物技术公司 制备噻吩并嘧啶化合物的方法
GB0721095D0 (en) 2007-10-26 2007-12-05 Piramed Ltd Pharmaceutical compounds
EP2405916B1 (fr) 2009-03-12 2018-02-07 Genentech, Inc. Combinaison de composés inhibiteurs de la phosphoinositide 3-kinase et d'agents chimiothérapeutiques pour le traitement de tumeurs malignes hématopoïétiques
CA2772371A1 (fr) * 2009-05-27 2010-12-02 F. Hoffmann-La Roche Ag Composes bicycliques indole-pyrimidine inhibiteurs de pi3k selectifs pour p110 delta et leurs procedes d'utilisation
EP2435438A1 (fr) 2009-05-27 2012-04-04 Genentech, Inc. Composés pyrimidines bicycliques inhibiteurs de pi3k sélectifs pour p110 delta, et procédés d'utilisation
JP2013528787A (ja) 2010-04-16 2013-07-11 ジェネンテック, インコーポレイテッド Pi3k/aktキナーゼ経路インヒビターの効果の予測バイオマーカーとしてのfox03a
WO2012088254A1 (fr) 2010-12-22 2012-06-28 Genentech, Inc. Polythérapie par inducteur et inhibiteur d'autophagie pour le traitement de néoplasmes
CA2901126C (fr) 2013-02-25 2022-01-25 Genentech, Inc. Procedes et compositions pour detecter et traiter un mutant d'akt resistant aux medicaments
GB201410816D0 (en) * 2014-06-17 2014-07-30 Ucb Biopharma Sprl And Katholieke Universiteit Leuven Therapeutic agents

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3259623A (en) * 1963-06-14 1966-07-05 Olin Mathieson Process for preparing 2-(secondary amino)-halogenopyrimidines
DE1470356A1 (de) * 1964-01-15 1970-04-30 Thomae Gmbh Dr K Neue Thieno[3,2-d]pyrimidine und Verfahren zu ihrer Herstellung
US3210368A (en) * 1964-09-29 1965-10-05 Ciba Geigy Corp Certain 2-amino-4-aryl-5-n, n-disubstituted amino-lower alkyl-thiazole compounds

Also Published As

Publication number Publication date
IL39341A (en) 1975-08-31
AT318619B (de) 1974-11-11
FR2135294A1 (fr) 1972-12-15
DD97656A5 (fr) 1973-05-12
PL82381B1 (fr) 1975-10-31
NL7206041A (fr) 1972-11-07
AU4181572A (en) 1973-11-08
HU163960B (fr) 1973-11-28
FR2135294B1 (fr) 1975-10-17
ES402302A1 (es) 1975-04-01
DK129844C (fr) 1975-05-12
US3888851A (en) 1975-06-10
GB1393161A (en) 1975-05-07
DK129844B (da) 1974-11-25
IL39341A0 (en) 1972-07-26
RO62428A (fr) 1978-01-15
BG20593A3 (bg) 1975-12-05

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