BE783044A - Nouvelles thieno(3,2-d) pyrimidines - Google Patents
Nouvelles thieno(3,2-d) pyrimidinesInfo
- Publication number
- BE783044A BE783044A BE783044A BE783044A BE783044A BE 783044 A BE783044 A BE 783044A BE 783044 A BE783044 A BE 783044A BE 783044 A BE783044 A BE 783044A BE 783044 A BE783044 A BE 783044A
- Authority
- BE
- Belgium
- Prior art keywords
- thieno
- pyrimidines
- news
- news thieno
- Prior art date
Links
- 150000003230 pyrimidines Chemical class 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
- C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
- C07D495/04—Ortho-condensed systems
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DE19712121950 DE2121950A1 (en) | 1971-05-04 | 1971-05-04 | Thieno(3,2-d)pyrimidine derivs - with thrombocyte aggregation inhibiting activity |
| DE19712137341 DE2137341A1 (de) | 1971-07-26 | 1971-07-26 | Neue thieno eckige klammer auf 3,2-d eckige klammer zu pyrimidine |
| DE19722215299 DE2215299A1 (de) | 1972-03-29 | 1972-03-29 | Neue thieno eckige klammer auf 3,2-d eckige klammer zu pyrimidine |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| BE783044A true BE783044A (fr) | 1972-11-06 |
Family
ID=27183398
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| BE783044A BE783044A (fr) | 1971-05-04 | 1972-05-04 | Nouvelles thieno(3,2-d) pyrimidines |
Country Status (15)
| Country | Link |
|---|---|
| US (1) | US3888851A (fr) |
| AT (1) | AT318619B (fr) |
| AU (1) | AU4181572A (fr) |
| BE (1) | BE783044A (fr) |
| BG (1) | BG20593A3 (fr) |
| DD (1) | DD97656A5 (fr) |
| DK (1) | DK129844B (fr) |
| ES (1) | ES402302A1 (fr) |
| FR (1) | FR2135294B1 (fr) |
| GB (1) | GB1393161A (fr) |
| HU (1) | HU163960B (fr) |
| IL (1) | IL39341A (fr) |
| NL (1) | NL7206041A (fr) |
| PL (1) | PL82381B1 (fr) |
| RO (1) | RO62428A (fr) |
Families Citing this family (23)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4054656A (en) * | 1975-09-10 | 1977-10-18 | Mead Johnson & Company | Thieno[2,3-d]pyrimidine antiallergic agents |
| US5098902A (en) * | 1991-03-18 | 1992-03-24 | Warner-Lambert Company | Method of treating neurodegenerative diseases |
| EP0626964A1 (fr) * | 1992-02-19 | 1994-12-07 | Pfizer Inc. | Composes heterocycliques ameliorant l'activite antitumorale |
| AU745579B2 (en) | 1997-10-20 | 2002-03-21 | F. Hoffmann-La Roche Ag | Bicyclic kinase inhibitors |
| US6187777B1 (en) | 1998-02-06 | 2001-02-13 | Amgen Inc. | Compounds and methods which modulate feeding behavior and related diseases |
| GB0423653D0 (en) | 2004-10-25 | 2004-11-24 | Piramed Ltd | Pharmaceutical compounds |
| EP2060575A1 (fr) * | 2006-04-19 | 2009-05-20 | Boehringer Ingelheim International GmbH | Dihydrothienopyrimidines et leur utilisation pour traiter des maladies inflammatoires |
| KR101402474B1 (ko) | 2006-04-26 | 2014-06-19 | 제넨테크, 인크. | 포스포이노시티드 3-키나제 억제제 화합물 및 이를 포함하는 약학적 조성물 |
| JP5148597B2 (ja) | 2006-04-26 | 2013-02-20 | エフ.ホフマン−ラ ロシュ アーゲー | 医薬化合物 |
| CL2007001167A1 (es) | 2006-04-26 | 2008-01-25 | Genentech Inc | Compuestos derivados de pirimidina condensada, inhibidores de p13-quinasa; procesos para preparar los compuestos; composicion farmaceutica que los comprende; uso de los compuestos en la preparacion de medicamentos; proceso para preparar la composicion farmaceutica; y kit que incluye a la composicionfarmaceutica. |
| ES2571028T3 (es) | 2006-12-07 | 2016-05-23 | Genentech Inc | Compuestos inhibidores de fosfoinositida 3-cinasa y métodos de uso |
| JP5284977B2 (ja) | 2006-12-07 | 2013-09-11 | エフ・ホフマン−ラ・ロシュ・アクチェンゲゼルシャフト | ホスホイノシチド3−キナーゼ阻害剤化合物及び使用方法 |
| ES2399774T3 (es) | 2007-09-24 | 2013-04-03 | Genentech, Inc. | Compuestos de tiazolopirimidina inhibidores de PI3K y métodos de uso |
| BRPI0817781A2 (pt) * | 2007-10-19 | 2019-09-24 | Boehringer Ingelheim Int | piperazino-diidroteinopirimidinas substituídas com heterociclo |
| CN101909631B (zh) * | 2007-10-25 | 2012-09-12 | 健泰科生物技术公司 | 制备噻吩并嘧啶化合物的方法 |
| GB0721095D0 (en) | 2007-10-26 | 2007-12-05 | Piramed Ltd | Pharmaceutical compounds |
| EP2405916B1 (fr) | 2009-03-12 | 2018-02-07 | Genentech, Inc. | Combinaison de composés inhibiteurs de la phosphoinositide 3-kinase et d'agents chimiothérapeutiques pour le traitement de tumeurs malignes hématopoïétiques |
| CA2772371A1 (fr) * | 2009-05-27 | 2010-12-02 | F. Hoffmann-La Roche Ag | Composes bicycliques indole-pyrimidine inhibiteurs de pi3k selectifs pour p110 delta et leurs procedes d'utilisation |
| EP2435438A1 (fr) | 2009-05-27 | 2012-04-04 | Genentech, Inc. | Composés pyrimidines bicycliques inhibiteurs de pi3k sélectifs pour p110 delta, et procédés d'utilisation |
| JP2013528787A (ja) | 2010-04-16 | 2013-07-11 | ジェネンテック, インコーポレイテッド | Pi3k/aktキナーゼ経路インヒビターの効果の予測バイオマーカーとしてのfox03a |
| WO2012088254A1 (fr) | 2010-12-22 | 2012-06-28 | Genentech, Inc. | Polythérapie par inducteur et inhibiteur d'autophagie pour le traitement de néoplasmes |
| CA2901126C (fr) | 2013-02-25 | 2022-01-25 | Genentech, Inc. | Procedes et compositions pour detecter et traiter un mutant d'akt resistant aux medicaments |
| GB201410816D0 (en) * | 2014-06-17 | 2014-07-30 | Ucb Biopharma Sprl And Katholieke Universiteit Leuven | Therapeutic agents |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3259623A (en) * | 1963-06-14 | 1966-07-05 | Olin Mathieson | Process for preparing 2-(secondary amino)-halogenopyrimidines |
| DE1470356A1 (de) * | 1964-01-15 | 1970-04-30 | Thomae Gmbh Dr K | Neue Thieno[3,2-d]pyrimidine und Verfahren zu ihrer Herstellung |
| US3210368A (en) * | 1964-09-29 | 1965-10-05 | Ciba Geigy Corp | Certain 2-amino-4-aryl-5-n, n-disubstituted amino-lower alkyl-thiazole compounds |
-
1972
- 1972-04-28 RO RO7200070735A patent/RO62428A/fr unknown
- 1972-05-02 ES ES402302A patent/ES402302A1/es not_active Expired
- 1972-05-02 HU HUTO875A patent/HU163960B/hu unknown
- 1972-05-03 US US249782A patent/US3888851A/en not_active Expired - Lifetime
- 1972-05-03 IL IL39341A patent/IL39341A/xx unknown
- 1972-05-03 PL PL1972155128A patent/PL82381B1/pl unknown
- 1972-05-03 BG BG020371A patent/BG20593A3/xx unknown
- 1972-05-03 DK DK219672AA patent/DK129844B/da unknown
- 1972-05-03 AU AU41815/72A patent/AU4181572A/en not_active Expired
- 1972-05-03 DD DD162711A patent/DD97656A5/xx unknown
- 1972-05-03 GB GB2058472A patent/GB1393161A/en not_active Expired
- 1972-05-03 AT AT382972A patent/AT318619B/de not_active IP Right Cessation
- 1972-05-04 BE BE783044A patent/BE783044A/fr unknown
- 1972-05-04 FR FR7215929A patent/FR2135294B1/fr not_active Expired
- 1972-05-04 NL NL7206041A patent/NL7206041A/xx unknown
Also Published As
| Publication number | Publication date |
|---|---|
| IL39341A (en) | 1975-08-31 |
| AT318619B (de) | 1974-11-11 |
| FR2135294A1 (fr) | 1972-12-15 |
| DD97656A5 (fr) | 1973-05-12 |
| PL82381B1 (fr) | 1975-10-31 |
| NL7206041A (fr) | 1972-11-07 |
| AU4181572A (en) | 1973-11-08 |
| HU163960B (fr) | 1973-11-28 |
| FR2135294B1 (fr) | 1975-10-17 |
| ES402302A1 (es) | 1975-04-01 |
| DK129844C (fr) | 1975-05-12 |
| US3888851A (en) | 1975-06-10 |
| GB1393161A (en) | 1975-05-07 |
| DK129844B (da) | 1974-11-25 |
| IL39341A0 (en) | 1972-07-26 |
| RO62428A (fr) | 1978-01-15 |
| BG20593A3 (bg) | 1975-12-05 |
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