BG60459B1 - МЕТОД ЗА ПОЛУЧАВАНЕ НА β-КАРБОНИЛ-КАРБОКСИАМИДИ НА 1,3-ТИАЗО- ЛИДИНИ - Google Patents

МЕТОД ЗА ПОЛУЧАВАНЕ НА β-КАРБОНИЛ-КАРБОКСИАМИДИ НА 1,3-ТИАЗО- ЛИДИНИ Download PDF

Info

Publication number
BG60459B1
BG60459B1 BG92842A BG9284290A BG60459B1 BG 60459 B1 BG60459 B1 BG 60459B1 BG 92842 A BG92842 A BG 92842A BG 9284290 A BG9284290 A BG 9284290A BG 60459 B1 BG60459 B1 BG 60459B1
Authority
BG
Bulgaria
Prior art keywords
formula
thiazolidine
group
compounds
compound
Prior art date
Application number
BG92842A
Other languages
Bulgarian (bg)
English (en)
Other versions
BG92842A (bg
Inventor
Carmelo A Gandolfi
Domenico Roberto Di
Silvano Spinelli
Licia Gallico
Bruno Lumachi
Sergio Tognella
Original Assignee
Boehringer Mannheim Italia
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Boehringer Mannheim Italia filed Critical Boehringer Mannheim Italia
Publication of BG92842A publication Critical patent/BG92842A/bg
Publication of BG60459B1 publication Critical patent/BG60459B1/bg

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/14—Antitussive agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
    • C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
    • C07D277/04—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having no double bonds between ring members or between ring members and non-ring members

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pulmonology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Macromolecular Compounds Obtained By Forming Nitrogen-Containing Linkages In General (AREA)
  • Electric Double-Layer Capacitors Or The Like (AREA)
  • Carbon And Carbon Compounds (AREA)
BG92842A 1988-03-17 1990-09-14 МЕТОД ЗА ПОЛУЧАВАНЕ НА β-КАРБОНИЛ-КАРБОКСИАМИДИ НА 1,3-ТИАЗО- ЛИДИНИ BG60459B1 (bg)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
IT8819813A IT1216119B (it) 1988-03-17 1988-03-17 Beta_carbonil_carbossiamidi di 1,3_tiazolidine.
PCT/EP1989/000205 WO1989008648A1 (en) 1988-03-17 1989-03-02 beta-CARBONYL-CARBOXYAMIDES OF 1,3-THIAZOLIDINES

Publications (2)

Publication Number Publication Date
BG92842A BG92842A (bg) 1993-12-24
BG60459B1 true BG60459B1 (bg) 1995-04-28

Family

ID=11161493

Family Applications (1)

Application Number Title Priority Date Filing Date
BG92842A BG60459B1 (bg) 1988-03-17 1990-09-14 МЕТОД ЗА ПОЛУЧАВАНЕ НА β-КАРБОНИЛ-КАРБОКСИАМИДИ НА 1,3-ТИАЗО- ЛИДИНИ

Country Status (19)

Country Link
US (1) US5206254A (de)
EP (2) EP0407403A1 (de)
JP (1) JPH0688987B2 (de)
KR (1) KR960011381B1 (de)
AT (1) ATE95814T1 (de)
AU (1) AU624124B2 (de)
BG (1) BG60459B1 (de)
CA (1) CA1325632C (de)
DE (1) DE68909815T2 (de)
DK (1) DK168486B1 (de)
ES (1) ES2059595T3 (de)
FI (1) FI95247C (de)
HU (1) HU205920B (de)
IT (1) IT1216119B (de)
NO (1) NO179370C (de)
RO (1) RO107656B1 (de)
RU (1) RU1833378C (de)
WO (1) WO1989008648A1 (de)
ZA (1) ZA892014B (de)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IT1245712B (it) * 1991-04-09 1994-10-14 Boehringer Mannheim Italia Ammine eterocicliche utili terapia dell'asma e dell'infiammazione delle vie aeree
IT1270594B (it) * 1994-07-07 1997-05-07 Recordati Chem Pharm Composizione farmaceutica a rilascio controllato di moguisteina in sospensione liquida
US6586466B2 (en) 1995-10-30 2003-07-01 Smithkline Beecham Corporation Carbohydrazide-protease inhibitors
US5773455A (en) * 1996-06-28 1998-06-30 Biomeasure, Incorporated Inhibitors of prenyl transferases
US6083964A (en) * 1998-02-18 2000-07-04 K And K Biosciences, Inc. Optical resolution of racemic aminoalkylpyridine anticonvulsants and (+) aminoalkylpyridine enantiomers as highly potent orally effective anticonvulsant drugs and excitatory amino acid antagonists
AU1738800A (en) 1998-11-23 2000-06-13 Bonnie Davis Dosage formulations for acetylcholinesterase inhibitors
CN1319955C (zh) * 2003-06-10 2007-06-06 浙江海正药业股份有限公司 莫吉斯坦晶型
WO2008144956A1 (en) * 2007-05-28 2008-12-04 Tianjin Institute Of Pharmaceutical Research New ambroxol compounds, their preparation processes and uses
EP2070915A1 (de) * 2007-12-03 2009-06-17 A.M.S.A. ANONIMA MATERIE SINTETICHE E AFFINI S.p.A. Neues Verfahren zur Synthese von Moguistein
CN102653527A (zh) * 2011-12-22 2012-09-05 东莞达信生物技术有限公司 一种莫吉司坦合成工艺

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
HU195492B (en) * 1984-07-27 1988-05-30 Boehringer Biochemia Srl Process for producing 2-substituted thiazolidine derivatives with antitussive and mucus regulating action and pharmaceuticals comprising these compounds as active ingredient
GB2164333B (en) * 1984-07-27 1988-11-16 Boehringer Biochemia Srl Antitussive and mucus regulating 2-substituted thiazolidines
IT1201489B (it) * 1985-11-13 1989-02-02 Chiesi Farma Spa Derivati di tiazolidina,loro procedimento di preparazione e formulazioni farmaceutiche
IT1228251B (it) * 1987-07-02 1991-06-05 Boehringer Biochemia Srl Amidi di amino-tioacetali ciclici, procedimento per la loro preparazione e composizioni farmaceutiche che li contengono

Also Published As

Publication number Publication date
ATE95814T1 (de) 1993-10-15
FI904512A0 (fi) 1990-09-13
KR960011381B1 (ko) 1996-08-22
DK221490A (da) 1990-09-14
AU624124B2 (en) 1992-06-04
IT8819813A0 (it) 1988-03-17
FI95247C (fi) 1996-01-10
NO179370C (no) 1996-09-25
NO179370B (no) 1996-06-17
EP0407403A1 (de) 1991-01-16
JPH03504123A (ja) 1991-09-12
HU205920B (en) 1992-07-28
EP0333080B1 (de) 1993-10-13
RO107656B1 (ro) 1993-12-30
US5206254A (en) 1993-04-27
ZA892014B (en) 1989-11-29
DE68909815D1 (de) 1993-11-18
KR900700470A (ko) 1990-08-13
IT1216119B (it) 1990-02-22
JPH0688987B2 (ja) 1994-11-09
EP0333080A1 (de) 1989-09-20
NO904031L (no) 1990-11-16
FI95247B (fi) 1995-09-29
AU3189289A (en) 1989-10-05
WO1989008648A1 (en) 1989-09-21
DK168486B1 (da) 1994-04-05
DE68909815T2 (de) 1994-03-24
CA1325632C (en) 1993-12-28
HU891559D0 (en) 1991-06-28
DK221490D0 (da) 1990-09-14
BG92842A (bg) 1993-12-24
HUT56355A (en) 1991-08-28
RU1833378C (en) 1993-08-07
ES2059595T3 (es) 1994-11-16
NO904031D0 (no) 1990-09-14

Similar Documents

Publication Publication Date Title
DK169337B1 (da) Xanthinforbindelser, farmaceutisk præparat indeholdende disse, xanthinforbindelser til anvendelse som et farmaceutisk middel samt fremgangsmåde til fremstilling af forbindelserne
JP4259615B2 (ja) 薬物常用および特にアルコール中毒の治寮へのγ―ヒドロキシ酪酸アミドの使用
AU4780699A (en) Farnesyl protein transferase inhibitors for treating arthropathies
CZ281669B6 (cs) Nové dihydroisochinolinové deriváty
EA021755B1 (ru) ПИРАЗИНОВЫЕ ПРОИЗВОДНЫЕ В КАЧЕСТВЕ ENaC БЛОКАТОРОВ
EP0633882A1 (de) 4-(4'piperidinyl oder 3'-pyrrolidinyl) substituierte imidazole als h3-rezeptor-antagonisten und ihre therapeutische verwendung
WO1995011894A1 (en) Histamine h3-receptor antagonists and therapeutic uses thereof
NL2013012B1 (en) Compounds for the treatment of chronic obstructive airway diseases.
KR960011381B1 (ko) 1, 3-티아졸라딘의 β-카르보닐-카르복시아미드
CN109790170B (zh) Gaba(a)受体调节剂和控制哮喘中气道高反应性和炎症的方法
JP7050336B2 (ja) 重水素化化合物及びその医薬的用途
JP2006506402A (ja) 四級アンモニウム化合物およびその抗ムスカリン薬としての使用
AU599981B2 (en) Novel pharmaceutical compositions comprising and use of cis- 6-(4-acetanilido)-8,9-dimethoxy-2-methyl-1,2,3,4,4a,-10b- hexanhydro-benzo{c}{1,6}naphthyridine
HK32694A (en) Beta-carbonyl-carboxyamides of 1,3-thiazolidines
JP2021515811A (ja) ３”，５”−ジアルコシベンゾイル−３’−アミノ−３’−デオキシアデノシン−５’−三リン酸及びその医薬用途
CA3111275A1 (en) Methods and compositions for treatment of asthma or parkinson's disease
WO2025104491A1 (en) Indole derivatives as serotonergic agents useful for the treatment of disorders related thereto
JPH0625117A (ja) （ｓ）−２−アミノ−２−（３，４−ジクロロベンジル）−１−プロパノールから誘導される新規なエナンチオマー
JP2005047900A (ja) 経肺投与用医薬組成物