BG62792B1 - Изотиазолони - Google Patents
Изотиазолони Download PDFInfo
- Publication number
- BG62792B1 BG62792B1 BG102077A BG10207797A BG62792B1 BG 62792 B1 BG62792 B1 BG 62792B1 BG 102077 A BG102077 A BG 102077A BG 10207797 A BG10207797 A BG 10207797A BG 62792 B1 BG62792 B1 BG 62792B1
- Authority
- BG
- Bulgaria
- Prior art keywords
- compound
- oxo
- mmol
- methyl
- isothiazol
- Prior art date
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Classifications
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- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/425—Thiazoles
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D275/00—Heterocyclic compounds containing 1,2-thiazole or hydrogenated 1,2-thiazole rings
- C07D275/04—Heterocyclic compounds containing 1,2-thiazole or hydrogenated 1,2-thiazole rings condensed with carbocyclic rings or ring systems
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- A—HUMAN NECESSITIES
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- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
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- A—HUMAN NECESSITIES
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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- A—HUMAN NECESSITIES
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- A61P31/12—Antivirals
- A61P31/14—Antivirals for RNA viruses
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D275/00—Heterocyclic compounds containing 1,2-thiazole or hydrogenated 1,2-thiazole rings
- C07D275/04—Heterocyclic compounds containing 1,2-thiazole or hydrogenated 1,2-thiazole rings condensed with carbocyclic rings or ring systems
- C07D275/06—Heterocyclic compounds containing 1,2-thiazole or hydrogenated 1,2-thiazole rings condensed with carbocyclic rings or ring systems with hetero atoms directly attached to the ring sulfur atom
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
- C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
- C07D513/04—Ortho-condensed systems
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
- C07D513/12—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains three hetero rings
- C07D513/14—Ortho-condensed systems
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
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Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US08/456,149 US5620997A (en) | 1995-05-31 | 1995-05-31 | Isothiazolones |
| PCT/US1996/005821 WO1996038144A1 (en) | 1995-05-31 | 1996-04-26 | Isothiazolones |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| BG102077A BG102077A (en) | 1998-11-30 |
| BG62792B1 true BG62792B1 (bg) | 2000-08-31 |
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Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| BG102077A BG62792B1 (bg) | 1995-05-31 | 1997-11-27 | Изотиазолони |
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| Country | Link |
|---|---|
| US (4) | US5620997A (de) |
| EP (1) | EP0828488B1 (de) |
| JP (1) | JP2002502353A (de) |
| KR (2) | KR19990022132A (de) |
| CN (1) | CN1114402C (de) |
| AR (1) | AR002740A1 (de) |
| AT (1) | ATE232385T1 (de) |
| AU (1) | AU723233B2 (de) |
| BG (1) | BG62792B1 (de) |
| CA (1) | CA2218253A1 (de) |
| CO (1) | CO4700292A1 (de) |
| CZ (1) | CZ373997A3 (de) |
| DE (1) | DE69626203T2 (de) |
| DK (1) | DK0828488T3 (de) |
| EA (1) | EA000898B1 (de) |
| EE (1) | EE9700287A (de) |
| ES (1) | ES2192224T3 (de) |
| GE (1) | GEP20012375B (de) |
| GT (1) | GT199600026A (de) |
| HN (1) | HN1996000017A (de) |
| HR (1) | HRP960216B1 (de) |
| HU (1) | HUP9900917A3 (de) |
| IL (1) | IL117859A (de) |
| MX (1) | MX9707948A (de) |
| MY (1) | MY118452A (de) |
| NO (1) | NO975496L (de) |
| NZ (1) | NZ307023A (de) |
| OA (1) | OA10745A (de) |
| PE (1) | PE55097A1 (de) |
| PL (1) | PL323683A1 (de) |
| PT (1) | PT828488E (de) |
| SK (1) | SK162297A3 (de) |
| SV (2) | SV1996000026A (de) |
| TW (1) | TW418206B (de) |
| UY (1) | UY24244A1 (de) |
| WO (1) | WO1996038144A1 (de) |
| ZA (1) | ZA964441B (de) |
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| US5219875A (en) * | 1990-11-27 | 1993-06-15 | Rohm And Haas Company | Antimicrobial compositions comprising iodopropargyl butylcarbamate and 1,2-benzisothiazolin-3-one and methods of controlling microbes |
| NO304832B1 (no) * | 1992-05-27 | 1999-02-22 | Ube Industries | Aminokinolonderivater samt middel mot HIV |
| FR2695378B1 (fr) * | 1992-09-10 | 1994-12-02 | Aerospatiale | Dispositif à sangle pour le maintien temporaire d'objets ensemble. |
| RU2118322C1 (ru) * | 1993-07-05 | 1998-08-27 | Дюфар Интернэшнл Рисерч Б.В. | 2,3-дигидро-1,4-бензодиокси-5-ил-пиперазиновые производные или их соли |
-
1995
- 1995-05-31 US US08/456,149 patent/US5620997A/en not_active Expired - Fee Related
- 1995-12-15 TW TW084113376A patent/TW418206B/zh not_active IP Right Cessation
- 1995-12-15 CO CO95059308A patent/CO4700292A1/es unknown
-
1996
- 1996-04-09 IL IL11785996A patent/IL117859A/xx not_active IP Right Cessation
- 1996-04-19 SV SV1996000026A patent/SV1996000026A/es unknown
- 1996-04-26 EP EP96913177A patent/EP0828488B1/de not_active Expired - Lifetime
- 1996-04-26 WO PCT/US1996/005821 patent/WO1996038144A1/en not_active Ceased
- 1996-04-26 EA EA199700444A patent/EA000898B1/ru not_active IP Right Cessation
- 1996-04-26 PL PL96323683A patent/PL323683A1/xx unknown
- 1996-04-26 KR KR1019970708611A patent/KR19990022132A/ko not_active Abandoned
- 1996-04-26 EE EE9700287A patent/EE9700287A/xx unknown
- 1996-04-26 SK SK1622-97A patent/SK162297A3/sk unknown
- 1996-04-26 CZ CZ973739A patent/CZ373997A3/cs unknown
- 1996-04-26 DE DE69626203T patent/DE69626203T2/de not_active Expired - Fee Related
- 1996-04-26 AT AT96913177T patent/ATE232385T1/de not_active IP Right Cessation
- 1996-04-26 NZ NZ307023A patent/NZ307023A/en unknown
- 1996-04-26 CN CN96194276A patent/CN1114402C/zh not_active Expired - Fee Related
- 1996-04-26 MX MX9707948A patent/MX9707948A/es not_active IP Right Cessation
- 1996-04-26 AU AU55771/96A patent/AU723233B2/en not_active Ceased
- 1996-04-26 ES ES96913177T patent/ES2192224T3/es not_active Expired - Lifetime
- 1996-04-26 JP JP53647396A patent/JP2002502353A/ja not_active Abandoned
- 1996-04-26 KR KR10-2003-7011364A patent/KR20040004547A/ko not_active Ceased
- 1996-04-26 GE GEAP19964062A patent/GEP20012375B/en unknown
- 1996-04-26 PT PT96913177T patent/PT828488E/pt unknown
- 1996-04-26 CA CA002218253A patent/CA2218253A1/en not_active Abandoned
- 1996-04-26 DK DK96913177T patent/DK0828488T3/da active
- 1996-04-26 HU HU9900917A patent/HUP9900917A3/hu unknown
- 1996-05-07 US US08/646,188 patent/US5668162A/en not_active Expired - Fee Related
- 1996-05-08 HR HR960216A patent/HRP960216B1/xx not_active IP Right Cessation
- 1996-05-15 HN HN1996000017A patent/HN1996000017A/es unknown
- 1996-05-15 AR ARP960102576A patent/AR002740A1/es not_active Application Discontinuation
- 1996-05-24 GT GT199600026A patent/GT199600026A/es unknown
- 1996-05-24 SV SV1996000033A patent/SV1996000033A/es not_active Application Discontinuation
- 1996-05-29 MY MYPI96002063A patent/MY118452A/en unknown
- 1996-05-30 ZA ZA964441A patent/ZA964441B/xx unknown
- 1996-05-30 UY UY24244A patent/UY24244A1/es unknown
- 1996-05-30 PE PE1996000385A patent/PE55097A1/es not_active Application Discontinuation
- 1996-11-26 US US08/757,716 patent/US5733921A/en not_active Expired - Fee Related
-
1997
- 1997-06-26 US US08/882,846 patent/US6133270A/en not_active Expired - Fee Related
- 1997-11-12 OA OA70126A patent/OA10745A/en unknown
- 1997-11-27 BG BG102077A patent/BG62792B1/bg unknown
- 1997-11-28 NO NO975496A patent/NO975496L/no not_active Application Discontinuation
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