BG98409A - 5-member heterocycles, method for their preparation and medicaments containing them - Google Patents
5-member heterocycles, method for their preparation and medicaments containing themInfo
- Publication number
- BG98409A BG98409A BG98409A BG9840994A BG98409A BG 98409 A BG98409 A BG 98409A BG 98409 A BG98409 A BG 98409A BG 9840994 A BG9840994 A BG 9840994A BG 98409 A BG98409 A BG 98409A
- Authority
- BG
- Bulgaria
- Prior art keywords
- preparation
- medicaments containing
- member heterocycles
- heterocycles
- medicaments
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P7/00—Drugs for disorders of the blood or the extracellular fluid
- A61P7/02—Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/10—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing aromatic rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
- C07D417/06—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
Landscapes
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- Veterinary Medicine (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Heart & Thoracic Surgery (AREA)
- Cardiology (AREA)
- Diabetes (AREA)
- Urology & Nephrology (AREA)
- Vascular Medicine (AREA)
- Hematology (AREA)
- Pulmonology (AREA)
- Epidemiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DE4302051A DE4302051A1 (en) | 1993-01-26 | 1993-01-26 | 5-membered heterocycles, process for their preparation and medicaments containing these compounds |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| BG98409A true BG98409A (en) | 1994-09-30 |
Family
ID=6478937
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| BG98409A BG98409A (en) | 1993-01-26 | 1994-01-24 | 5-member heterocycles, method for their preparation and medicaments containing them |
Country Status (18)
| Country | Link |
|---|---|
| EP (1) | EP0608858A1 (en) |
| JP (1) | JPH072851A (en) |
| KR (1) | KR940018382A (en) |
| CN (1) | CN1097753A (en) |
| AU (1) | AU5398494A (en) |
| BG (1) | BG98409A (en) |
| CA (1) | CA2114178A1 (en) |
| CZ (1) | CZ18194A3 (en) |
| DE (1) | DE4302051A1 (en) |
| FI (1) | FI940378A7 (en) |
| HU (1) | HU9400217D0 (en) |
| IL (1) | IL108436A0 (en) |
| NO (1) | NO940261L (en) |
| NZ (1) | NZ250762A (en) |
| PL (1) | PL302018A1 (en) |
| RU (1) | RU94002482A (en) |
| SK (1) | SK8394A3 (en) |
| ZA (1) | ZA94495B (en) |
Families Citing this family (50)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5849736A (en) * | 1993-11-24 | 1998-12-15 | The Dupont Merck Pharmaceutical Company | Isoxazoline and isoxazole fibrinogen receptor antagonists |
| ZA963391B (en) * | 1995-05-24 | 1997-10-29 | Du Pont Merck Pharma | Isoxazoline fibrinogen receptor antagonists. |
| EP0858457A1 (en) * | 1995-10-20 | 1998-08-19 | Dr. Karl Thomae GmbH | 5-membered heterocycles, pharmaceutical agents containing said compounds and the use thereof and methods of producing them |
| US6083986A (en) * | 1996-07-26 | 2000-07-04 | Icagen, Inc. | Potassium channel inhibitors |
| US6333337B1 (en) | 1998-01-27 | 2001-12-25 | Icagen, Inc. | Potassium channel inhibitors |
| WO2000001679A1 (en) * | 1998-07-01 | 2000-01-13 | Takeda Chemical Industries, Ltd. | Retinoid-associated receptor regulators |
| US7084279B1 (en) | 1999-02-11 | 2006-08-01 | Emisphere Technologies Inc. | Oxadiazole compounds and compositions for delivering active agents |
| ATE311373T1 (en) * | 1999-02-11 | 2005-12-15 | Emisphere Tech Inc | OXADIAZOLE COMPOUNDS AND COMPOSITIONS FOR DELIVERING ACTIVE INGREDIENTS |
| AU781365B2 (en) | 1999-12-21 | 2005-05-19 | Icagen, Inc. | Potassium channel inhibitors |
| AU2000223275A1 (en) * | 2000-02-08 | 2001-08-20 | Yamanouchi Pharmaceutical Co..Ltd. | Novel triazole derivatives |
| EP1293503A4 (en) * | 2000-05-19 | 2008-04-02 | Astellas Pharma Inc | Triazole derivatives |
| US6566380B2 (en) | 2000-07-25 | 2003-05-20 | Icagen, Inc. | Potassium channel inhibitors |
| US6620849B2 (en) | 2000-07-26 | 2003-09-16 | Icafen, Inc. | Potassium channel inhibitors |
| US6849634B2 (en) | 2000-12-21 | 2005-02-01 | Icagen | Potassium channel inhibitors |
| EP1405636A4 (en) * | 2001-06-26 | 2009-04-15 | Takeda Pharmaceutical | REGULATOR OF RECTINTOR FUNCTION RELATING TO RETINOIDS |
| US7390813B1 (en) | 2001-12-21 | 2008-06-24 | Xenon Pharmaceuticals Inc. | Pyridylpiperazines and aminonicotinamides and their use as therapeutic agents |
| US7087604B2 (en) | 2002-03-08 | 2006-08-08 | Bristol-Myers Squibb Company | Cyclic derivatives as modulators of chemokine receptor activity |
| ATE329909T1 (en) | 2002-11-27 | 2006-07-15 | Boehringer Ingelheim Pharma | 1,2,3-TRIAZOLAMIDE DERIVATIVES AS CYTOKIN INHIBITORS |
| US7078419B2 (en) | 2003-03-10 | 2006-07-18 | Boehringer Ingelheim Pharmaceuticals, Inc. | Cytokine inhibitors |
| NZ543102A (en) | 2003-04-24 | 2008-12-24 | Incyte Corp | Aza spiro alkane derivatives as inhibitors of metalloproteases |
| EP1648874B1 (en) | 2003-07-30 | 2011-10-05 | Xenon Pharmaceuticals Inc. | Piperazine derivatives and their use as therapeutic agents |
| DE602004031759D1 (en) | 2003-12-03 | 2011-04-21 | Boehringer Ingelheim Pharma | 1,2,3-TRIAZOLAMIDE DERIVATIVES AS INHIBITORS OF CYTOKINE PRODUCTION |
| DE602005014621D1 (en) | 2004-03-09 | 2009-07-09 | Boehringer Ingelheim Pharma | 3-A4-HETEROCYCLYL-1,2,3-TRIAZOL-1-YLÜ-N-ARYLBENZAMIDES AS INHIBITORS OF CYTOKIN PRODUCTION FOR THE TREATMENT OF CHRONIC INFLAMMATORY DISEASES |
| WO2005108387A2 (en) | 2004-05-03 | 2005-11-17 | Boehringer Ingelheim Pharmaceuticals, Inc. | Cytokine inhibitors |
| US7485657B2 (en) | 2004-05-12 | 2009-02-03 | Boehringer Ingelheim Pharmaceuticals, Inc. | Anti-cytokine heterocyclic compounds |
| EP2289510A1 (en) | 2004-09-20 | 2011-03-02 | Xenon Pharmaceuticals Inc. | Heterocyclic derivatives for the treatment of diseases mediated by stearoyl-coa desaturase enzymes |
| EP1807085B1 (en) | 2004-09-20 | 2013-08-21 | Xenon Pharmaceuticals Inc. | Heterocyclic derivatives and their use as stearoyl-coa desaturase inhibitors |
| CA2580857A1 (en) | 2004-09-20 | 2006-09-28 | Xenon Pharmaceuticals Inc. | Heterocyclic derivatives and their use as stearoyl-coa desaturase inhibitors |
| US7829712B2 (en) | 2004-09-20 | 2010-11-09 | Xenon Pharmaceuticals Inc. | Pyridazine derivatives for inhibiting human stearoyl-CoA-desaturase |
| AR051091A1 (en) | 2004-09-20 | 2006-12-20 | Xenon Pharmaceuticals Inc | HETEROCICLIC DERIVATIVES AND THEIR USE AS INHIBITORS OF ESTEAROIL-COA DESATURASA |
| CA2580762A1 (en) | 2004-09-20 | 2006-03-30 | Xenon Pharmaceuticals Inc. | Heterocyclic derivatives and their use as therapeutic agents |
| AU2005286648A1 (en) | 2004-09-20 | 2006-03-30 | Xenon Pharmaceuticals Inc. | Heterocyclic derivatives and their use as stearoyl-CoA desaturase inhibitors |
| US7531560B2 (en) | 2004-11-10 | 2009-05-12 | Boehringer Ingelheim Pharmaceuticals, Inc. | Anti-cytokine heterocyclic compounds |
| AP2007004047A0 (en) | 2005-01-20 | 2007-06-30 | Pfizer Ltd | Substituted triazole derivatives as oxtocin antagonists |
| AU2006343359A1 (en) | 2005-06-03 | 2007-11-15 | Xenon Pharmaceuticals Inc. | Aminothiazole derivatives as human stearoyl-coa desaturase inhibitors |
| TW200811164A (en) * | 2006-05-12 | 2008-03-01 | Jerini Ag | New heterocyclic compounds for the inhibition of integrins and use thereof |
| US7910108B2 (en) | 2006-06-05 | 2011-03-22 | Incyte Corporation | Sheddase inhibitors combined with CD30-binding immunotherapeutics for the treatment of CD30 positive diseases |
| TW200813018A (en) | 2006-06-09 | 2008-03-16 | Astrazeneca Ab | Novel compounds |
| JP2010501567A (en) | 2006-08-24 | 2010-01-21 | ノバルティス アクチエンゲゼルシャフト | 2- (pyrazin-2-yl) -thiazole and 2- (1H-pyrazole-3-) as stearoyl-CoA desaturase (SCD) inhibitors for the treatment of metabolic, cardiovascular and other disorders Yl) thiazole derivatives and related compounds |
| AU2007292155B2 (en) | 2006-09-05 | 2012-11-01 | Kyowa Kirin Co., Ltd. | Imidazole derivative |
| DK2142529T3 (en) | 2007-04-27 | 2014-02-10 | Purdue Pharma Lp | TRPV1 ANTAGONISTS AND APPLICATIONS THEREOF |
| US8119661B2 (en) | 2007-09-11 | 2012-02-21 | Astrazeneca Ab | Piperidine derivatives and their use as muscarinic receptor modulators |
| AU2011261375B2 (en) | 2010-06-04 | 2016-09-22 | Albany Molecular Research, Inc. | Glycine transporter-1 inhibitors, methods of making them, and uses thereof |
| HRP20170507T1 (en) | 2011-06-22 | 2017-06-02 | Purdue Pharma Lp | TRPV1 ANTAGONISTS INCLUDING DIHYDROXY SUBSTITUTES AND THEIR USE |
| WO2014122474A1 (en) | 2013-02-07 | 2014-08-14 | Takeda Pharmaceutical Company Limited | Piperidin-1 -yl and azepin-1 -yl carboxylates as muscarinic m4 receptor agonists |
| GB201810071D0 (en) * | 2018-06-19 | 2018-08-08 | Univ Oslo Hf | Compounds |
| US12030875B2 (en) | 2018-09-07 | 2024-07-09 | PIC Therapeutics, Inc. | EIF4E inhibitors and uses thereof |
| AU2021230289A1 (en) | 2020-03-03 | 2022-09-29 | PIC Therapeutics, Inc. | eIF4E inhibitors and uses thereof |
| US12157732B2 (en) | 2021-08-25 | 2024-12-03 | PIC Therapeutics, Inc. | eIF4E inhibitors and uses thereof |
| JP2024534127A (en) | 2021-08-25 | 2024-09-18 | ピク セラピューティクス， インコーポレイテッド | eIF4E inhibitors and uses thereof |
Family Cites Families (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| IL98757A (en) * | 1990-07-18 | 1997-01-10 | Novo Nordisk As | Piperidine derivatives their preparation and pharmaceutical compositions containing them |
| DE4124942A1 (en) * | 1991-07-27 | 1993-01-28 | Thomae Gmbh Dr K | 5-LOW HETEROCYCLES, METHOD FOR THE PRODUCTION THEREOF AND MEDICAMENTS CONTAINING SUCH COMPOUNDS |
-
1993
- 1993-01-26 DE DE4302051A patent/DE4302051A1/en not_active Withdrawn
-
1994
- 1994-01-24 BG BG98409A patent/BG98409A/en unknown
- 1994-01-24 SK SK83-94A patent/SK8394A3/en unknown
- 1994-01-25 RU RU94002482/04A patent/RU94002482A/en unknown
- 1994-01-25 ZA ZA94495A patent/ZA94495B/en unknown
- 1994-01-25 HU HU9400217A patent/HU9400217D0/en unknown
- 1994-01-25 NO NO940261A patent/NO940261L/en unknown
- 1994-01-25 CN CN94100575A patent/CN1097753A/en active Pending
- 1994-01-25 KR KR1019940001441A patent/KR940018382A/en not_active Withdrawn
- 1994-01-25 PL PL94302018A patent/PL302018A1/en unknown
- 1994-01-25 CA CA002114178A patent/CA2114178A1/en not_active Abandoned
- 1994-01-25 JP JP6006295A patent/JPH072851A/en active Pending
- 1994-01-26 FI FI940378A patent/FI940378A7/en not_active Application Discontinuation
- 1994-01-26 NZ NZ250762A patent/NZ250762A/en unknown
- 1994-01-26 CZ CZ94181A patent/CZ18194A3/en unknown
- 1994-01-26 IL IL10843694A patent/IL108436A0/en unknown
- 1994-01-26 EP EP94101125A patent/EP0608858A1/en not_active Withdrawn
- 1994-01-27 AU AU53984/94A patent/AU5398494A/en not_active Abandoned
Also Published As
| Publication number | Publication date |
|---|---|
| KR940018382A (en) | 1994-08-16 |
| NO940261L (en) | 1994-07-27 |
| FI940378A0 (en) | 1994-01-26 |
| SK8394A3 (en) | 1995-02-08 |
| FI940378L (en) | 1994-07-27 |
| DE4302051A1 (en) | 1994-07-28 |
| NZ250762A (en) | 1995-08-28 |
| RU94002482A (en) | 1996-08-27 |
| NO940261D0 (en) | 1994-01-25 |
| EP0608858A1 (en) | 1994-08-03 |
| ZA94495B (en) | 1995-07-25 |
| CA2114178A1 (en) | 1994-07-27 |
| HU9400217D0 (en) | 1994-05-30 |
| PL302018A1 (en) | 1994-08-08 |
| CZ18194A3 (en) | 1994-11-16 |
| CN1097753A (en) | 1995-01-25 |
| AU5398494A (en) | 1994-08-04 |
| JPH072851A (en) | 1995-01-06 |
| IL108436A0 (en) | 1994-04-12 |
| FI940378A7 (en) | 1994-07-27 |
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