BR0214703A - Derivados de aminoacetonitrila e seu uso para controlar parasitas - Google Patents

Derivados de aminoacetonitrila e seu uso para controlar parasitas

Info

Publication number
BR0214703A
BR0214703A BR0214703-3A BR0214703A BR0214703A BR 0214703 A BR0214703 A BR 0214703A BR 0214703 A BR0214703 A BR 0214703A BR 0214703 A BR0214703 A BR 0214703A
Authority
BR
Brazil
Prior art keywords
control parasites
amino acetonitrile
acetonitrile derivatives
parasites
derivatives
Prior art date
Application number
BR0214703-3A
Other languages
English (en)
Inventor
Pierre Ducray
Thomas Goebel
Original Assignee
Novartis Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Novartis Ag filed Critical Novartis Ag
Publication of BR0214703A publication Critical patent/BR0214703A/pt

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C255/00—Carboxylic acid nitriles
    • C07C255/01—Carboxylic acid nitriles having cyano groups bound to acyclic carbon atoms
    • C07C255/32—Carboxylic acid nitriles having cyano groups bound to acyclic carbon atoms having cyano groups bound to acyclic carbon atoms of a carbon skeleton containing at least one six-membered aromatic ring
    • C07C255/42—Carboxylic acid nitriles having cyano groups bound to acyclic carbon atoms having cyano groups bound to acyclic carbon atoms of a carbon skeleton containing at least one six-membered aromatic ring the carbon skeleton being further substituted by singly-bound nitrogen atoms, not being further bound to other hetero atoms
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N37/00—Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom having three bonds to hetero atoms with at the most two bonds to halogen, e.g. carboxylic acids
    • A01N37/34—Nitriles
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A61P33/10—Anthelmintics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A61P33/14—Ectoparasiticides, e.g. scabicides
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C255/00—Carboxylic acid nitriles
    • C07C255/01—Carboxylic acid nitriles having cyano groups bound to acyclic carbon atoms
    • C07C255/24—Carboxylic acid nitriles having cyano groups bound to acyclic carbon atoms containing cyano groups and singly-bound nitrogen atoms, not being further bound to other hetero atoms, bound to the same saturated acyclic carbon skeleton
    • C07C255/29—Carboxylic acid nitriles having cyano groups bound to acyclic carbon atoms containing cyano groups and singly-bound nitrogen atoms, not being further bound to other hetero atoms, bound to the same saturated acyclic carbon skeleton containing cyano groups and acylated amino groups bound to the carbon skeleton
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C2601/00—Systems containing only non-condensed rings
    • C07C2601/02—Systems containing only non-condensed rings with a three-membered ring

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Public Health (AREA)
  • Agronomy & Crop Science (AREA)
  • Environmental Sciences (AREA)
  • Plant Pathology (AREA)
  • Engineering & Computer Science (AREA)
  • Dentistry (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Pest Control & Pesticides (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Pyridine Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)

Abstract

"DERIVADOS DE AMINOACETONITRILA E SEU USO PARA CONTROLAR PARASITAS". A presente invenção refere-se a novos compostos da fórmula geral em que R~ 1~, R~ 2~, X, Ar~ 1~, e Ar~ 2~ são como definido na reivindicação 1, e em quaisquer enanciómeros destes. Os ingredientes ativos tem propriedades terapêuticas vantajosas. Elas são particularmente adequadas para controlar parasitas em animais homeotérmicos.
BR0214703-3A 2001-12-06 2002-12-05 Derivados de aminoacetonitrila e seu uso para controlar parasitas BR0214703A (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
CH22252001 2001-12-06
PCT/EP2002/013811 WO2003048112A1 (en) 2001-12-06 2002-12-05 Aminoacetonitrile derivatives and their use for controlling parasites

Publications (1)

Publication Number Publication Date
BR0214703A true BR0214703A (pt) 2004-08-31

Family

ID=4568089

Family Applications (1)

Application Number Title Priority Date Filing Date
BR0214703-3A BR0214703A (pt) 2001-12-06 2002-12-05 Derivados de aminoacetonitrila e seu uso para controlar parasitas

Country Status (15)

Country Link
US (2) US7091371B2 (pt)
EP (1) EP1456170A1 (pt)
JP (1) JP2005511685A (pt)
KR (1) KR100648117B1 (pt)
CN (2) CN1274672C (pt)
AR (1) AR037746A1 (pt)
AU (1) AU2002358620B2 (pt)
BR (1) BR0214703A (pt)
CA (1) CA2466570A1 (pt)
CO (1) CO5590952A2 (pt)
MX (1) MXPA04005455A (pt)
RU (1) RU2293725C2 (pt)
TW (1) TWI261053B (pt)
WO (1) WO2003048112A1 (pt)
ZA (1) ZA200403577B (pt)

Families Citing this family (15)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
RU2284990C2 (ru) * 2001-05-15 2006-10-10 Новартис Аг Производные бензамидоацетонитрила, способ их получения, содержащая их композиция для борьбы с нематодами и их применение
TW200400932A (en) * 2002-06-19 2004-01-16 Novartis Ag Organic compounds
GB0402677D0 (en) * 2003-11-06 2004-03-10 Novartis Ag Organic compounds
US20050158356A1 (en) * 2003-11-20 2005-07-21 Angiotech International Ag Implantable sensors and implantable pumps and anti-scarring agents
US8218748B2 (en) * 2006-07-24 2012-07-10 Hewlett-Packard Development Company, L.P. Telephone call chaining
PL3088384T3 (pl) 2007-05-15 2019-06-28 Merial, Inc. Związki aryloazol-2-ilo-cyjanoetyloaminowe, sposób ich wytwarzania oraz sposób ich stosowania
CA2741186C (en) * 2008-10-21 2016-07-19 Merial Limited Thioamide compounds, method of making and method of using thereof
CN102209758A (zh) * 2008-11-07 2011-10-05 亨斯迈石油化学有限责任公司 多氨基乙腈、其制备方法和用途
PL3050874T3 (pl) * 2008-11-14 2019-07-31 Merial Inc. Wzbogacone enancjomerycznie aryloazol-2-ilocyjanoetyloaminowe związki pasożytobójcze
MX345339B (es) * 2011-03-02 2017-01-25 Univ Tokyo Agente de control de endoparásitos.
MY157429A (en) 2011-06-24 2016-06-15 Amgen Inc Trpm8 antagonists and their use in treatments
JP2014517074A (ja) 2011-06-24 2014-07-17 アムジエン・インコーポレーテツド Ｔｒｐｍ８アンタゴニストおよび治療におけるそれらの使用
US8952009B2 (en) 2012-08-06 2015-02-10 Amgen Inc. Chroman derivatives as TRPM8 inhibitors
US8822689B2 (en) 2012-09-19 2014-09-02 Merial Limited Aryloazol-2-yl cyanoethylamino compounds, method of making and method of using thereof
CN110407681B (zh) * 2019-08-12 2023-05-02 海南大学 一种脱氢姜酮衍生物、其制备方法及应用

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3457294A (en) * 1966-04-22 1969-07-22 Abbott Lab N-(substituted-benzoyl) aminoaceto- and aminopropionitriles
US4515731A (en) * 1975-08-25 1985-05-07 Monsanto Company Asymmetric catalysis
US5959870A (en) 1998-02-20 1999-09-28 Gamma-Metrics Real-time optimization for mix beds
US6239077B1 (en) * 1998-05-01 2001-05-29 Nihon Nohyaku Co., Ltd. Aminoacetonitrile derivative agricultural and horticultural insecticide containing the same and use thereof
AR035523A1 (es) * 2000-12-20 2004-06-02 Novartis Ag Uso de compuestos de aminoacetonitrilo para combatir animales daninos endoparasitarios en animales utiles y domesticos de sangre caliente

Also Published As

Publication number Publication date
CN1293047C (zh) 2007-01-03
AU2002358620A1 (en) 2003-06-17
AU2002358620B2 (en) 2006-08-31
KR20050044719A (ko) 2005-05-12
CN1274672C (zh) 2006-09-13
CA2466570A1 (en) 2003-06-12
MXPA04005455A (es) 2005-04-19
TWI261053B (en) 2006-09-01
US7091371B2 (en) 2006-08-15
CN1668580A (zh) 2005-09-14
EP1456170A1 (en) 2004-09-15
US20060264653A1 (en) 2006-11-23
ZA200403577B (en) 2006-06-28
US20050033081A1 (en) 2005-02-10
CO5590952A2 (es) 2005-12-30
AR037746A1 (es) 2004-12-01
WO2003048112A1 (en) 2003-06-12
KR100648117B1 (ko) 2006-11-24
TW200300755A (en) 2003-06-16
CN1599716A (zh) 2005-03-23
JP2005511685A (ja) 2005-04-28
RU2004120790A (ru) 2005-05-27
RU2293725C2 (ru) 2007-02-20

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Legal Events

Date Code Title Description
B08F Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette]

Free format text: REFERENTE A 6A E 7A ANUIDADES.

B08K Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette]

Free format text: REFERENTE AO DESPACHO 8.6 PUBLICADO NA RPI 2064 DE 27/07/2010.