BR0307735A - Carboxamidas heteroaromáticas com ligação-n em ponte biciclìcas fundidas para o tratamento de doença - Google Patents

Carboxamidas heteroaromáticas com ligação-n em ponte biciclìcas fundidas para o tratamento de doença

Info

Publication number
BR0307735A
BR0307735A BR0307735-7A BR0307735A BR0307735A BR 0307735 A BR0307735 A BR 0307735A BR 0307735 A BR0307735 A BR 0307735A BR 0307735 A BR0307735 A BR 0307735A
Authority
BR
Brazil
Prior art keywords
fused bicyclic
disease treatment
bridged
heteroaromatic carboxamides
carboxamides
Prior art date
Application number
BR0307735-7A
Other languages
English (en)
Inventor
Bruce N Rogers
David W Piotrowski
Daniel P Walker
Eric Jon Jabobsen
Brad A Acker
Donn Gregory Wishka
Vincent Edward Groppi
Original Assignee
Upjohn Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Upjohn Co filed Critical Upjohn Co
Publication of BR0307735A publication Critical patent/BR0307735A/pt

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D519/00—Heterocyclic compounds containing more than one system of two or more relevant hetero rings condensed among themselves or condensed with a common carbocyclic ring system not provided for in groups C07D453/00 or C07D455/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
    • A61P25/16—Anti-Parkinson drugs
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/22—Anxiolytics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/24—Antidepressants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00—Drugs for disorders of the senses
    • A61P27/02—Ophthalmic agents
    • A61P27/06—Antiglaucoma agents or miotics

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Psychiatry (AREA)
  • Ophthalmology & Optometry (AREA)
  • Psychology (AREA)
  • Pain & Pain Management (AREA)
  • Hospice & Palliative Care (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)

Abstract

"CARBOXAMIDAS HETEROAROMáTICAS COM LIGAçãO-N EM PONTE BICICLìCAS FUNDIDAS PARA O TRATAMENTO DE DOENçA". A presente invenção refere-se a compostos de Fórmula I: Estes compostos podem estar na forma de sais ou composições farmacêuticos, podem estar na forma enantiomérica pura ou como misturas racêmicas, e são úteis em fármacos para o tratamento de condições ou doenças nas quais se sabe que o <244>7 está envolvido.
BR0307735-7A 2002-02-19 2003-02-14 Carboxamidas heteroaromáticas com ligação-n em ponte biciclìcas fundidas para o tratamento de doença BR0307735A (pt)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US35791702P 2002-02-19 2002-02-19
US42315702P 2002-11-01 2002-11-01
PCT/US2003/002687 WO2003070732A1 (en) 2002-02-19 2003-02-14 Fused bicyclic-n-bridged-heteroaromatic carboxamides for the treatment of disease

Publications (1)

Publication Number Publication Date
BR0307735A true BR0307735A (pt) 2005-01-25

Family

ID=27760475

Family Applications (1)

Application Number Title Priority Date Filing Date
BR0307735-7A BR0307735A (pt) 2002-02-19 2003-02-14 Carboxamidas heteroaromáticas com ligação-n em ponte biciclìcas fundidas para o tratamento de doença

Country Status (8)

Country Link
US (2) US6858613B2 (pt)
EP (1) EP1476449A1 (pt)
JP (1) JP2005523288A (pt)
AU (1) AU2003219690A1 (pt)
BR (1) BR0307735A (pt)
CA (1) CA2476681A1 (pt)
MX (1) MXPA04008038A (pt)
WO (1) WO2003070732A1 (pt)

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WO2003070732A1 (en) 2003-08-28
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AU2003219690A1 (en) 2003-09-09
MXPA04008038A (es) 2004-11-26
EP1476449A1 (en) 2004-11-17
US20030236264A1 (en) 2003-12-25
US20050215584A1 (en) 2005-09-29
US6858613B2 (en) 2005-02-22

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