BR0308403A - Método para tratamento de um distúrbio do olho de um paciente humano ou veterinário, e, uso de um composto - Google Patents

Método para tratamento de um distúrbio do olho de um paciente humano ou veterinário, e, uso de um composto

Info

Publication number
BR0308403A
BR0308403A BR0308403-5A BR0308403A BR0308403A BR 0308403 A BR0308403 A BR 0308403A BR 0308403 A BR0308403 A BR 0308403A BR 0308403 A BR0308403 A BR 0308403A
Authority
BR
Brazil
Prior art keywords
corneal
eye
urea
compound
guanidinium
Prior art date
Application number
BR0308403-5A
Other languages
English (en)
Inventor
Vicken Karageozian
David Castillejos
John Park
Gabriel Arthuro Carpio Aragon
Jose Luis Gutierres Flores
Original Assignee
Vitreo Retinal Technologies In
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Vitreo Retinal Technologies In filed Critical Vitreo Retinal Technologies In
Publication of BR0308403A publication Critical patent/BR0308403A/pt

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/16Amides, e.g. hydroxamic acids
    • A61K31/17Amides, e.g. hydroxamic acids having the group >N—C(O)—N< or >N—C(S)—N<, e.g. urea, thiourea, carmustine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/513Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim having oxo groups directly attached to the heterocyclic ring, e.g. cytosine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
    • A61K31/52Purines, e.g. adenine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/70Carbohydrates; Sugars; Derivatives thereof
    • A61K31/7042Compounds having saccharide radicals and heterocyclic rings
    • A61K31/7052Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides
    • A61K31/706Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides containing six-membered rings with nitrogen as a ring hetero atom
    • A61K31/7064Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides containing six-membered rings with nitrogen as a ring hetero atom containing condensed or non-condensed pyrimidines
    • A61K31/7076Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides containing six-membered rings with nitrogen as a ring hetero atom containing condensed or non-condensed pyrimidines containing purines, e.g. adenosine, adenylic acid
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00Drugs for disorders of the senses
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00Drugs for disorders of the senses
    • A61P27/02Ophthalmic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00Drugs for disorders of the senses
    • A61P27/02Ophthalmic agents
    • A61P27/06Antiglaucoma agents or miotics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00Drugs for disorders of the senses
    • A61P27/02Ophthalmic agents
    • A61P27/10Ophthalmic agents for accommodation disorders, e.g. myopia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Epidemiology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Ophthalmology & Optometry (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Molecular Biology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicinal Preparation (AREA)

Abstract

"MéTODO PARA TRATAMENTO DE UM DISTúRBIO DO OLHO DE UM PACIENTE HUMANO OU VETERINáRIO, E, USO DE UM COMPOSTO". Métodos e preparações para tratamento de distúrbios do olho e/ou dissolução de proteoglicanos da córnea, cicatrização organizada do estroma corneal, amolecimento da córnea para correção refrativa não cirúrgica da vista, remoção de névoa e opacificação corneal, inibição de fibroblastos e prevenção de fibrose corneal e formação de cicatrizes, tratamento de pterígios, tratamentos de neovascularização corneal e neovascularização da íris. São admistradas ao olho, em montantes terapeuticamente eficazes, preparações contendo a) uréia, b) derivados de uréia (por exemplo, hidroxiuréia, tiouréia), c) antimetabólitos, e) uréia, derivados de uréia, proteínas não enzimáticas, nucleosídeos, nucleotídeos e seus derivados (por exemplo, adenina, adenosina, citosina, citadina, guanina, guanitadina, guanidínio, cloreto de guanidínio, sais de guanidínio, timidina, timitadina, uradina, uracila, cisteína), ácido tióctico reduzido, ácido úrico, acetil salicilato de cálcio, sulfato de amónio, álcool isopropílico, etanol, polietileno glicol, polipropileno glicol ou outro composto capaz de causar dissolução não enzimática dos proteoglicanos da córnea ou f) quaisquer das combinações possíveis dos mesmos.
BR0308403-5A 2002-03-14 2003-03-14 Método para tratamento de um distúrbio do olho de um paciente humano ou veterinário, e, uso de um composto BR0308403A (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US36397902P 2002-03-14 2002-03-14
PCT/US2003/007700 WO2003077898A1 (en) 2002-03-14 2003-03-14 Agents for corneal or intrastromal administration to treat or prevent disorders of the eye

Publications (1)

Publication Number Publication Date
BR0308403A true BR0308403A (pt) 2005-01-18

Family

ID=28041849

Family Applications (1)

Application Number Title Priority Date Filing Date
BR0308403-5A BR0308403A (pt) 2002-03-14 2003-03-14 Método para tratamento de um distúrbio do olho de um paciente humano ou veterinário, e, uso de um composto

Country Status (10)

Country Link
EP (1) EP1482922A4 (pt)
JP (1) JP2005522464A (pt)
KR (1) KR20040094793A (pt)
CN (1) CN1642536A (pt)
AU (2) AU2003213858A1 (pt)
BR (1) BR0308403A (pt)
CA (1) CA2478965A1 (pt)
MX (1) MXPA04008776A (pt)
RU (1) RU2363459C2 (pt)
WO (1) WO2003077898A1 (pt)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US20030199574A1 (en) 2000-03-02 2003-10-23 Vitreo-Retinal Technologies, Inc. Treatment of ophthalmic disorders using urea and urea derivatives
CN101231121B (zh) * 2007-01-24 2012-06-13 泰州乐金电子冷机有限公司 冰箱用托盘拉出装置
CN102859344A (zh) * 2010-03-12 2013-01-02 独立行政法人理化学研究所 用于生物材料的澄清试剂和其用途
RU2442609C1 (ru) * 2010-11-12 2012-02-20 Озеров Александр Александрович Средство для ухода за мягкими и жесткими контактными линзами
EP2711682B1 (en) 2011-05-20 2019-07-10 Riken Clarifying reagent for biological materials and use thereof
WO2015022883A1 (ja) 2013-08-14 2015-02-19 独立行政法人理化学研究所 光透過性に優れた生物材料を調製するための組成物およびその利用
DE102013110608A1 (de) * 2013-09-26 2015-03-26 Florian Lang Substanz zur Hemmung von Gewebskalzifizierung, Gewebsfibrosierung und altersassoziierten Erkrankungen
CN110237238A (zh) * 2019-08-02 2019-09-17 山东省眼科研究所 Manf在促进角膜损伤修复中的应用
US12350250B2 (en) 2022-04-01 2025-07-08 The Regent Of The University Of Colorado, A Body Corporate Aggrelytes for treating ocular conditions

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
RU2094031C1 (ru) * 1992-04-09 1997-10-27 Малое государственное предприятие "Научно-экспериментальное производство" Способ профилактики новообразованных сосудов роговицы после сквозной и послойной кератопластики
US5470881A (en) * 1993-09-09 1995-11-28 West Virginia University Research Corporation Urea ophthalmic ointment and solution
RU2082434C1 (ru) * 1994-12-19 1997-06-27 Уфимский научно-исследовательский институт глазных болезней Глазная мазь
ATE396734T1 (de) * 1999-03-02 2008-06-15 Vitreo Retinal Technologies In Mittel für intravitreale verabreichung zur behandlung oder vorbeugung von augenerkrankungen
ATE428412T1 (de) * 2002-02-13 2009-05-15 Vitreo Retinal Technologies In Behandlung von augenkrankheiten mit harnstoff und harnstoffderivaten

Also Published As

Publication number Publication date
AU2009201897A1 (en) 2009-06-04
AU2009201897B2 (en) 2011-09-15
EP1482922A1 (en) 2004-12-08
WO2003077898A1 (en) 2003-09-25
RU2363459C2 (ru) 2009-08-10
EP1482922A4 (en) 2005-06-08
RU2004129761A (ru) 2005-06-10
CN1642536A (zh) 2005-07-20
AU2003213858A1 (en) 2003-09-29
JP2005522464A (ja) 2005-07-28
CA2478965A1 (en) 2003-09-25
MXPA04008776A (es) 2005-04-19
KR20040094793A (ko) 2004-11-10

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Legal Events

Date Code Title Description
B06F Objections, documents and/or translations needed after an examination request according [chapter 6.6 patent gazette]
B15K Others concerning applications: alteration of classification

Free format text: PARA INT.CL: A61K 31/17, A61P 27/02, A61P 41/00

Ipc: A61K 31/17 (2011.01), A61P 27/02 (2011.01), A61P 4

B07D Technical examination (opinion) related to article 229 of industrial property law [chapter 7.4 patent gazette]
B07E Notification of approval relating to section 229 industrial property law [chapter 7.5 patent gazette]

Free format text: NOTIFICACAO DE ANUENCIA RELACIONADA COM O ART 229 DA LPI

B07A Application suspended after technical examination (opinion) [chapter 7.1 patent gazette]
B09B Patent application refused [chapter 9.2 patent gazette]
B09B Patent application refused [chapter 9.2 patent gazette]