BR0311221A - Derivados de 1h-imidazo[4,5-c]quinolina no tratamento de doenças dependentes de proteìna cinase - Google Patents

Derivados de 1h-imidazo[4,5-c]quinolina no tratamento de doenças dependentes de proteìna cinase

Info

Publication number
BR0311221A
BR0311221A BR0311221-7A BR0311221A BR0311221A BR 0311221 A BR0311221 A BR 0311221A BR 0311221 A BR0311221 A BR 0311221A BR 0311221 A BR0311221 A BR 0311221A
Authority
BR
Brazil
Prior art keywords
treatment
protein kinase
kinase dependent
imidazo
dependent diseases
Prior art date
Application number
BR0311221-7A
Other languages
English (en)
Inventor
Carlos Garcia-Echeverria
Hans-Georg Capraro
Pascal Furet
Original Assignee
Novartis Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Novartis Ag filed Critical Novartis Ag
Publication of BR0311221A publication Critical patent/BR0311221A/pt

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00—Drugs for disorders of the urinary system
    • A61P13/08—Drugs for disorders of the urinary system of the prostate
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A61P17/06—Antipsoriatics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A61P35/02—Antineoplastic agents specific for leukemia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Hematology (AREA)
  • Oncology (AREA)
  • Dermatology (AREA)
  • Urology & Nephrology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Enzymes And Modification Thereof (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)

Abstract

"DERIVADOS DE 1H-IMIDAZO[4,5-C]QUINOLINA NO TRATAMENTO DE DOENçAS DEPENDENTES DE PROTEìNA CINASE". A presente invenção refere-se ao uso de imidazoquinolinas e seus sais no tratamento de doenças dependentes de proteína cinase e para a fabricação de preparações farmacêuticas para o tratamento das ditas doenças, imidazoquinolinas para o uso no tratamento de doenças dependentes de proteína cinase, um método de tratamento contra as ditas doenças, compreendendo administrar as imidazoloquinolinas a um animal de sangue quente, especialmente um ser humano, preparações farmacêuticas compreendendo uma imidazoquinolina, especialmente para o tratamento de uma doença dependente de proteína cinase, novas imidazoquinolinas e um processo para a preparação das novas imidazoquinolinas.
BR0311221-7A 2002-05-21 2003-05-20 Derivados de 1h-imidazo[4,5-c]quinolina no tratamento de doenças dependentes de proteìna cinase BR0311221A (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GBGB0211649.9A GB0211649D0 (en) 2002-05-21 2002-05-21 Organic compounds
PCT/EP2003/005291 WO2003097641A2 (en) 2002-05-21 2003-05-20 1h-imidazo[4,5-c] quinoline derivatives in the treatment of protein kinase dependent diseases

Publications (1)

Publication Number Publication Date
BR0311221A true BR0311221A (pt) 2005-03-01

Family

ID=9937093

Family Applications (1)

Application Number Title Priority Date Filing Date
BR0311221-7A BR0311221A (pt) 2002-05-21 2003-05-20 Derivados de 1h-imidazo[4,5-c]quinolina no tratamento de doenças dependentes de proteìna cinase

Country Status (15)

Country Link
US (1) US7998972B2 (pt)
EP (1) EP1509521B8 (pt)
JP (1) JP4707389B2 (pt)
CN (1) CN100475207C (pt)
AT (1) ATE405564T1 (pt)
AU (1) AU2003240680A1 (pt)
BR (1) BR0311221A (pt)
CA (1) CA2485012A1 (pt)
DE (1) DE60323090D1 (pt)
DK (1) DK1509521T3 (pt)
ES (1) ES2312783T3 (pt)
GB (1) GB0211649D0 (pt)
PT (1) PT1509521E (pt)
SI (1) SI1509521T1 (pt)
WO (1) WO2003097641A2 (pt)

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CA2485012A1 (en) 2003-11-27
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US7998972B2 (en) 2011-08-16
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