BR9507355A - Derivodos de 22-tiavitamina D3 - Google Patents

Derivodos de 22-tiavitamina D3

Info

Publication number: BR9507355A
Authority: BR; Brazil
Prior art keywords: hydroxy; represents hydrogen; thiavitamin; derivatives; vitamin
Prior art date: 1994-04-11

Application number

BR9507355A

Other languages

English (en)

Inventor

Noboru Kubodera

Akira Kawase

Original Assignee

Chugai Pharmaceutical Co Ltd

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1994-04-11

Filing date

1995-04-10

Publication date

1997-09-09

1995-04-10 Application filed by Chugai Pharmaceutical Co Ltd filed Critical Chugai Pharmaceutical Co Ltd

1997-09-09 Publication of BR9507355A publication Critical patent/BR9507355A/pt

Links

UFHFLCQGNIYNRP-UHFFFAOYSA-N Hydrogen Chemical compound [H][H] UFHFLCQGNIYNRP-UHFFFAOYSA-N 0.000 abstract 2
229910052739 hydrogen Inorganic materials 0.000 abstract 2
239000001257 hydrogen Substances 0.000 abstract 2
125000002887 hydroxy group Chemical group [H]O* 0.000 abstract 2
125000000008 (C1-C10) alkyl group Chemical group 0.000 abstract 1
150000001875 compounds Chemical class 0.000 abstract 1
230000000694 effects Effects 0.000 abstract 1
239000003966 growth inhibitor Substances 0.000 abstract 1
210000002510 keratinocyte Anatomy 0.000 abstract 1
230000003389 potentiating effect Effects 0.000 abstract 1
229910052717 sulfur Inorganic materials 0.000 abstract 1
125000004434 sulfur atom Chemical group 0.000 abstract 1
230000002194 synthesizing effect Effects 0.000 abstract 1
150000003710 vitamin D derivatives Chemical group 0.000 abstract 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J51/00—Normal steroids with unmodified cyclopenta(a)hydrophenanthrene skeleton not provided for in groups C07J1/00 - C07J43/00
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/59—Compounds containing 9, 10- seco- cyclopenta[a]hydrophenanthrene ring systems
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C401/00—Irradiation products of cholesterol or its derivatives; Vitamin D derivatives, 9,10-seco cyclopenta[a]phenanthrene or analogues obtained by chemical preparation without irradiation
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J31/00—Normal steroids containing one or more sulfur atoms not belonging to a hetero ring
- C07J31/006—Normal steroids containing one or more sulfur atoms not belonging to a hetero ring not covered by C07J31/003
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J71/00—Steroids in which the cyclopenta(a)hydrophenanthrene skeleton is condensed with a heterocyclic ring
- C07J71/0036—Nitrogen-containing hetero ring
- C07J71/0042—Nitrogen only
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J9/00—Normal steroids containing carbon, hydrogen, halogen or oxygen substituted in position 17 beta by a chain of more than two carbon atoms, e.g. cholane, cholestane, coprostane

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
General Health & Medical Sciences (AREA)
Epidemiology (AREA)
Pharmacology & Pharmacy (AREA)
Medicinal Chemistry (AREA)
Life Sciences & Earth Sciences (AREA)
Animal Behavior & Ethology (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Steroid Compounds (AREA)

BR9507355A 1994-04-11 1995-04-10 Derivodos de 22-tiavitamina D3 BR9507355A (pt)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
JP10736694		1994-04-11
PCT/JP1995/000699 WO1995027697A1 (en)	1994-04-11	1995-04-10	22-thiavitamin d3 derivative

Publications (1)

Publication Number	Publication Date
BR9507355A true BR9507355A (pt)	1997-09-09

Family

ID=14457272

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
BR9507355A BR9507355A (pt)	1994-04-11	1995-04-10	Derivodos de 22-tiavitamina D3

Country Status (14)

Country	Link
US (1)	US5824811A (pt)
EP (1)	EP0755922B1 (pt)
KR (1)	KR100244060B1 (pt)
CN (1)	CN1046502C (pt)
AT (1)	ATE195513T1 (pt)
AU (1)	AU2148295A (pt)
BR (1)	BR9507355A (pt)
DE (1)	DE69518410T2 (pt)
DK (1)	DK0755922T3 (pt)
ES (1)	ES2150560T3 (pt)
GR (1)	GR3034322T3 (pt)
PT (1)	PT755922E (pt)
RU (1)	RU2142941C1 (pt)
WO (1)	WO1995027697A1 (pt)

Families Citing this family (14)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
GB9226877D0 (en) *	1992-12-23	1993-02-17	Leo Pharm Prod Ltd	Chemical compounds
EP0870503B9 (en) *	1995-12-28	2006-06-28	Chugai Seiyaku Kabushiki Kaisha	use of vitamin D derivatives for the manufacture of a medicament for treating MALIGNANT TUMOR METASTASIS
US6869940B2 (en)	1995-12-28	2005-03-22	Chugai Seiyaku Kabushiki Kaisha	Malignant tumor metastasis inhibitors
KR20050123185A (ko)	1996-12-20	2005-12-29	쥬가이 세이야쿠 가부시키가이샤	16-엔-비타민 ｄ 유도체
US6184398B1 (en) *	1996-12-20	2001-02-06	Chugai Seiyaku Kabushiki Kaisha	16-ene-vitamin D derivatives
CA2289209C (en)	1997-05-16	2006-07-25	Women & Infants Hospital	Cyclic ether vitamin d3 compounds, 1.alpha. (oh) 3-epi-vitamin d3 compounds and uses thereof
ATE462689T1 (de) *	1999-08-27	2010-04-15	Hiroaki Takayama	Vitamin-d-derivate mit substituenten an der 2- alpha-position
GB2364231A (en) *	2000-04-05	2002-01-23	Bush Boake Allen Ltd	Flavouring agent
US6899911B2 (en) *	2000-04-05	2005-05-31	International Flavors & Fragrances, Inc.	Ethyl 4-(thioacetoxy)butyrate as a flavoring agent and methods for preparing and using same
US7074777B2 (en) *	2000-04-19	2006-07-11	Chugai Seiyaku Kabushiki Kaisha	Vitamin D derivatives
US7985744B2 (en) *	2000-06-15	2011-07-26	Chugai Seiyaku Kabushiki Kaisha	Vitamin D derivatives
EA201691980A1 (ru)	2009-01-27	2017-07-31	БЕРГ ЭлЭлСи	Способы уменьшения побочных эффектов, связанных с химиотерапией
CN102655869B (zh)	2009-08-14	2016-08-10	博格有限责任公司	用于治疗脱发的维生素d3及其类似物
WO2014194133A1 (en)	2013-05-29	2014-12-04	Berg Llc	Preventing or mitigating chemotherapy induced alopecia using vitamin d

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
CA1332841C (en) *	1984-11-27	1994-11-01	Noboru Kubodera	Vitamin d derivatives and process for producing the same
JPS61267550A (ja)	1984-12-28	1986-11-27	Chugai Pharmaceut Co Ltd	９，１０−セコ−５，７，１０（１９）−プレグナトリエン誘導体
JP3050564B2 (ja) *	1989-12-15	2000-06-12	中外製薬株式会社	新規な２２―オキサビタミンｄ誘導体
GB9007236D0 (en)	1990-03-30	1990-05-30	Leo Pharm Prod Ltd	Chemical compounds
JP2752506B2 (ja) *	1990-07-26	1998-05-18	株式会社クラレ	１α―ヒドロキシタキステロール誘導体の製造方法
DE4220757A1 (de) *	1992-06-24	1994-01-05	Schering Ag	Derivate in der Vitamin D-Reihe mit Modifikationen in der 20-Position, Verfahren zu ihrer Herstellung, Zwischenprodukte für dieses Verfahren, diese Derivate enthaltende pharmazeutische Präparate sowie deren Verwendung zur Herstellung von Arzneimitteln
GB9226877D0 (en) *	1992-12-23	1993-02-17	Leo Pharm Prod Ltd	Chemical compounds
JP4089473B2 (ja) *	2003-03-12	2008-05-28	株式会社ジェイテクト	ブラケット一体型リザーブタンク

1995
- 1995-04-10 DK DK95914550T patent/DK0755922T3/da active
- 1995-04-10 KR KR1019960705708A patent/KR100244060B1/ko not_active Expired - Fee Related
- 1995-04-10 DE DE69518410T patent/DE69518410T2/de not_active Expired - Lifetime
- 1995-04-10 RU RU96121801A patent/RU2142941C1/ru not_active IP Right Cessation
- 1995-04-10 US US08/718,499 patent/US5824811A/en not_active Expired - Lifetime
- 1995-04-10 ES ES95914550T patent/ES2150560T3/es not_active Expired - Lifetime
- 1995-04-10 EP EP95914550A patent/EP0755922B1/en not_active Expired - Lifetime
- 1995-04-10 AU AU21482/95A patent/AU2148295A/en not_active Abandoned
- 1995-04-10 AT AT95914550T patent/ATE195513T1/de not_active IP Right Cessation
- 1995-04-10 CN CN95193058A patent/CN1046502C/zh not_active Expired - Fee Related
- 1995-04-10 PT PT95914550T patent/PT755922E/pt unknown
- 1995-04-10 BR BR9507355A patent/BR9507355A/pt not_active IP Right Cessation
- 1995-04-10 WO PCT/JP1995/000699 patent/WO1995027697A1/ja not_active Ceased
2000
- 2000-09-01 GR GR20000402009T patent/GR3034322T3/el not_active IP Right Cessation

Also Published As

Publication number	Publication date
RU2142941C1 (ru)	1999-12-20
ES2150560T3 (es)	2000-12-01
ATE195513T1 (de)	2000-09-15
DE69518410D1 (de)	2000-09-21
DK0755922T3 (da)	2000-11-13
GR3034322T3 (en)	2000-12-29
DE69518410T2 (de)	2000-12-14
US5824811A (en)	1998-10-20
WO1995027697A1 (en)	1995-10-19
CN1148380A (zh)	1997-04-23
EP0755922A4 (en)	1997-07-02
CN1046502C (zh)	1999-11-17
PT755922E (pt)	2000-11-30
EP0755922A1 (en)	1997-01-29
EP0755922B1 (en)	2000-08-16
AU2148295A (en)	1995-10-30
KR100244060B1 (ko)	2000-02-01
KR970702245A (ko)	1997-05-13

Legal Events

Date	Code	Title	Description
2001-05-29	FB36	Technical and formal requirements: requirement - article 36 of industrial property law
2003-05-06	HJEG	Technical examination (opinion): technical examination (opinion) related to article 229 of industrial property law
2003-12-23	FF	Decision: intention to grant
2004-04-13	B16A	Patent or certificate of addition of invention granted [chapter 16.1 patent gazette]
2011-04-19	B24C	Patent annual fee: request for for restoration	Free format text: REFERENTE A 13A,14A,15 E 16A ANUIDADE(S).
2014-04-15	B24H	Lapse because of non-payment of annual fees (definitively: art 78 iv lpi)
2020-12-01	B24F	Patent annual fee: publication cancelled	Free format text: ANULADA A PUBLICACAO CODIGO 24.8 NA RPI NO 2258 DE 15/04/2014 POR TER SIDO INDEVIDA.
2020-12-22	B21F	Lapse acc. art. 78, item iv - on non-payment of the annual fees in time	Free format text: REFERENTE AS 13A, 14A, 15A E 16A ANUIDADES.
2021-04-13	B24J	Lapse because of non-payment of annual fees (definitively: art 78 iv lpi, resolution 113/2013 art. 12)	Free format text: EM VIRTUDE DA EXTINCAO PUBLICADA NA RPI 2607 DE 22-12-2020 E CONSIDERANDO AUSENCIA DE MANIFESTACAO DENTRO DOS PRAZOS LEGAIS, INFORMO QUE CABE SER MANTIDA A EXTINCAO DA PATENTE E SEUS CERTIFICADOS, CONFORME O DISPOSTO NO ARTIGO 12, DA RESOLUCAO 113/2013.

Publication	Publication Date	Title
BR9507355A (pt)	1997-09-09	Derivodos de 22-tiavitamina D3
NO992549L (no)	1999-07-26	Sukkerforbindelse, geleringsmiddel og fremgangsmåte for fremstilling derav
DK0826688T3 (da)	2001-10-22	Pentacykliske forbindelser
NZ218325A (en)	1989-07-27	Triazole derivatives and plant growth regulating agents
PT918776E (pt)	2004-07-30	Sintese total de acilfulvenos antitumorais
NO971384L (no)	1997-05-23	Pyrimidinylpyrazol-derivat
PT947504E (pt)	2003-12-31	Derivados de vitamina d 16-eno
IL134788A0 (en)	2001-04-30	A process for preparing 2-alkyl-3-aminothiophene derivatives
MX9604735A (es)	1998-01-31	Derivados de la 22-tiavitamina d3.
GR3033386T3 (en)	2000-09-29	Vitamin d derivative and process for producing the same.
DE69303847D1 (de)	1996-09-05	Indolderivate
AU2639999A (en)	1999-09-15	Intermediate compounds in the synthesis of the a ring moiety of 2-substituted vitamin d derivatives
BR9006967A (pt)	1991-12-17	Derivados de sulfamidos sulfonilureia e herbicidas
ATE206699T1 (de)	2001-10-15	Uch-15-verbindungen
ES2164258T3 (es)	2002-02-16	Procedimiento de preparacion de derivados de carbamoilmetilurea.
DK1137660T3 (da)	2003-02-03	22S-hydroxycholesta-8,14-dienderivater med meioseregulerende aktivitet