DK1137660T3 - 22S-hydroxycholesta-8,14-dienderivater med meioseregulerende aktivitet - Google Patents

22S-hydroxycholesta-8,14-dienderivater med meioseregulerende aktivitet

Info

Publication number: DK1137660T3
Authority: DK; Denmark
Prior art keywords: hydroxycholesta; alkyl; hydrogen; meios; diene derivatives
Prior art date: 1998-12-11

Application number

DK99929207T

Other languages

English (en)

Inventor

Dirk Leysen

Der Louw Jaap Van

Robert Gerard Jules Ma Hanssen

Anja Wiersma

Original Assignee

Akzo Nobel Nv

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1998-12-11

Filing date

1999-06-10

Publication date

2003-02-03

1998-12-11 Priority claimed from PCT/EP1998/008130 external-priority patent/WO1999032506A1/en

1999-06-10 Application filed by Akzo Nobel Nv filed Critical Akzo Nobel Nv

2003-02-03 Application granted granted Critical

2003-02-03 Publication of DK1137660T3 publication Critical patent/DK1137660T3/da

Links

230000001105 regulatory effect Effects 0.000 title 1
229910052739 hydrogen Inorganic materials 0.000 abstract 5
239000001257 hydrogen Substances 0.000 abstract 5
UFHFLCQGNIYNRP-UHFFFAOYSA-N Hydrogen Chemical compound [H][H] UFHFLCQGNIYNRP-UHFFFAOYSA-N 0.000 abstract 4
125000000217 alkyl group Chemical group 0.000 abstract 4
125000002252 acyl group Chemical group 0.000 abstract 2
125000004432 carbon atom Chemical group C* 0.000 abstract 2
229910052736 halogen Inorganic materials 0.000 abstract 2
150000002367 halogens Chemical class 0.000 abstract 2
230000003213 activating effect Effects 0.000 abstract 1
125000003545 alkoxy group Chemical group 0.000 abstract 1
150000001875 compounds Chemical class 0.000 abstract 1
230000035558 fertility Effects 0.000 abstract 1
150000002431 hydrogen Chemical class 0.000 abstract 1
125000002887 hydroxy group Chemical group [H]O* 0.000 abstract 1
230000021121 meiosis Effects 0.000 abstract 1
150000003839 salts Chemical class 0.000 abstract 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J9/00—Normal steroids containing carbon, hydrogen, halogen or oxygen substituted in position 17 beta by a chain of more than two carbon atoms, e.g. cholane, cholestane, coprostane
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A61P15/08—Drugs for genital or sexual disorders; Contraceptives for gonadal disorders or for enhancing fertility, e.g. inducers of ovulation or of spermatogenesis
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A61P15/16—Masculine contraceptives
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A61P15/18—Feminine contraceptives

Landscapes

Health & Medical Sciences (AREA)
Organic Chemistry (AREA)
Chemical & Material Sciences (AREA)
General Health & Medical Sciences (AREA)
Reproductive Health (AREA)
Life Sciences & Earth Sciences (AREA)
Endocrinology (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Animal Behavior & Ethology (AREA)
Bioinformatics & Cheminformatics (AREA)
Pharmacology & Pharmacy (AREA)
Engineering & Computer Science (AREA)
Chemical Kinetics & Catalysis (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
Gynecology & Obstetrics (AREA)
Pregnancy & Childbirth (AREA)
Steroid Compounds (AREA)
Saccharide Compounds (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)

DK99929207T 1998-12-11 1999-06-10 22S-hydroxycholesta-8,14-dienderivater med meioseregulerende aktivitet DK1137660T3 (da)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
PCT/EP1998/008130 WO1999032506A1 (en)	1997-12-18	1998-12-11	17β-ARYL (ARYLMETHYL) OXY(THIO)ALKYL -ANDROSTANE DERIVATIVES
PCT/EP1999/004099 WO2000035938A1 (en)	1998-12-11	1999-06-10	22s-hydroxycholesta-8, 14-diene derivatives with meiosis regulating activity

Publications (1)

Publication Number	Publication Date
DK1137660T3 true DK1137660T3 (da)	2003-02-03

Family

ID=8167154

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
DK99929207T DK1137660T3 (da)	1998-12-11	1999-06-10	22S-hydroxycholesta-8,14-dienderivater med meioseregulerende aktivitet

Country Status (10)

Country	Link
US (1)	US6528501B1 (da)
EP (1)	EP1137660B1 (da)
JP (1)	JP2002532511A (da)
AT (1)	ATE225366T1 (da)
AU (1)	AU759344B2 (da)
CA (1)	CA2352337A1 (da)
DE (1)	DE69903346T2 (da)
DK (1)	DK1137660T3 (da)
ES (1)	ES2185360T3 (da)
WO (1)	WO2000035938A1 (da)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
EP1212345B1 (en) *	1999-04-06	2003-08-06	Akzo Nobel N.V.	Orally active 7-alpha-alkyl androgens

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US5716777A (en) *	1994-06-23	1998-02-10	Novo Nordisk A/S	Regulation of meiosis using sterols
HUP9800731A3 (en) *	1995-03-06	2000-03-28	Novo Nordisk As	Stimulation of meiosis
CA2224866A1 (en)	1995-06-23	1997-01-09	Novo Nordisk A/S	Meiosis regulating compounds
JP2001506656A (ja) *	1996-12-20	2001-05-22	ノボノルディスクアクティーゼルスカブ	減数分裂調節化合物
JP2001526293A (ja)	1997-12-18	2001-12-18	アクゾ・ノベル・エヌ・ベー	１７β−アリール（アリールメチル）オキシ（チオ）アルキル−アンドロスタン誘導体

1999
- 1999-06-10 US US09/857,731 patent/US6528501B1/en not_active Expired - Fee Related
- 1999-06-10 ES ES99929207T patent/ES2185360T3/es not_active Expired - Lifetime
- 1999-06-10 JP JP2000588196A patent/JP2002532511A/ja active Pending
- 1999-06-10 DK DK99929207T patent/DK1137660T3/da active
- 1999-06-10 WO PCT/EP1999/004099 patent/WO2000035938A1/en not_active Ceased
- 1999-06-10 CA CA002352337A patent/CA2352337A1/en not_active Abandoned
- 1999-06-10 EP EP99929207A patent/EP1137660B1/en not_active Expired - Lifetime
- 1999-06-10 AU AU46100/99A patent/AU759344B2/en not_active Ceased
- 1999-06-10 DE DE69903346T patent/DE69903346T2/de not_active Expired - Fee Related
- 1999-06-10 AT AT99929207T patent/ATE225366T1/de not_active IP Right Cessation

Also Published As

Publication number	Publication date
DE69903346T2 (de)	2003-01-30
ES2185360T3 (es)	2003-04-16
EP1137660B1 (en)	2002-10-02
EP1137660A1 (en)	2001-10-04
AU759344B2 (en)	2003-04-10
JP2002532511A (ja)	2002-10-02
DE69903346D1 (de)	2002-11-07
AU4610099A (en)	2000-07-03
CA2352337A1 (en)	2000-06-22
ATE225366T1 (de)	2002-10-15
US6528501B1 (en)	2003-03-04
WO2000035938A1 (en)	2000-06-22

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