BR9612187A - Nova sintese - Google Patents

Nova sintese

Info

Publication number: BR9612187A
Authority: BR; Brazil
Prior art keywords: new synthesis; synthesis; new
Prior art date: 1995-12-22

Application number

BR9612187A

Other languages

English (en)

Inventor

Joseph Sisko

Original Assignee

Smithkline Beecham Corp

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1995-12-22

Filing date

1996-12-20

Publication date

1999-07-13

1996-12-20 Application filed by Smithkline Beecham Corp filed Critical Smithkline Beecham Corp

1999-07-13 Publication of BR9612187A publication Critical patent/BR9612187A/pt

Links

230000015572 biosynthetic process Effects 0.000 title 1
238000003786 synthesis reaction Methods 0.000 title 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Plural Heterocyclic Compounds (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)
Epoxy Resins (AREA)

BR9612187A 1995-12-22 1996-12-20 Nova sintese BR9612187A (pt)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
US909895P	1995-12-22	1995-12-22
PCT/US1996/020599 WO1997023479A1 (en)	1995-12-22	1996-12-20	Novel synthesis

Publications (1)

Publication Number	Publication Date
BR9612187A true BR9612187A (pt)	1999-07-13

Family

ID=21735553

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
BR9612187A BR9612187A (pt)	1995-12-22	1996-12-20	Nova sintese

Country Status (18)

Country	Link
US (3)	US6100399A (pt)
EP (1)	EP1019393A4 (pt)
JP (1)	JP3245175B2 (pt)
KR (1)	KR19990076625A (pt)
CN (1)	CN1209128A (pt)
AR (3)	AR004405A1 (pt)
AU (1)	AU704500B2 (pt)
BR (1)	BR9612187A (pt)
CZ (1)	CZ198598A3 (pt)
HU (1)	HUP9902466A3 (pt)
IL (2)	IL124908A (pt)
NO (1)	NO982850D0 (pt)
NZ (1)	NZ326574A (pt)
PL (1)	PL327311A1 (pt)
TR (1)	TR199801121T2 (pt)
TW (1)	TW434236B (pt)
WO (1)	WO1997023479A1 (pt)
ZA (1)	ZA9610687B (pt)

Families Citing this family (38)

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ZA9711092B (en) *	1996-12-11	1999-07-22	Smithkline Beecham Corp	Novel compounds.
US6979686B1 (en)	2001-12-07	2005-12-27	Pharmacia Corporation	Substituted pyrazoles as p38 kinase inhibitors
EP1019394A1 (en)	1997-05-22	2000-07-19	G.D. Searle & Co.	PYRAZOLE DERIVATIVES AS p38 KINASE INHIBITORS
US6514977B1 (en)	1997-05-22	2003-02-04	G.D. Searle & Company	Substituted pyrazoles as p38 kinase inhibitors
AU7966198A (en)	1997-06-13	1998-12-30	Smithkline Beecham Corporation	Novel pyrazole and pyrazoline substituted compounds
EP0994870A4 (en)	1997-06-19	2002-10-23	Smithkline Beecham	NEW IMIDAZOLE COMPOUNDS SUBSTITUTED BY AN ARYLOXYREST
US6489325B1 (en)	1998-07-01	2002-12-03	Smithkline Beecham Corporation	Substituted imidazole compounds
US6562832B1 (en)	1997-07-02	2003-05-13	Smithkline Beecham Corporation	Substituted imidazole compounds
US7301021B2 (en)	1997-07-02	2007-11-27	Smithkline Beecham Corporation	Substituted imidazole compounds
CA2306077A1 (en)	1997-10-08	1999-04-15	Smithkline Beecham Corporation	Novel cycloalkenyl substituted compounds
AU1924699A (en)	1997-12-19	1999-07-12	Smithkline Beecham Corporation	Compounds of heteroaryl substituted imidazole, their pharmaceutical compositionsand uses
US6858617B2 (en)	1998-05-26	2005-02-22	Smithkline Beecham Corporation	Substituted imidazole compounds
CA2341370A1 (en) *	1998-08-20	2000-03-02	Smithkline Beecham Corporation	Novel substituted triazole compounds
DE69914357T2 (de)	1998-11-04	2004-11-11	Smithkline Beecham Corp.	Pyridin-4-yl oder pyrimidin-4-yl substituierte pyrazine
US6239279B1 (en) *	1998-12-16	2001-05-29	Smithkline Beecham Corporation	Synthesis for 4-aryl-5-pyrimidine imidazole substituted derivatives
US6857013B2 (en) *	1999-01-29	2005-02-15	Intermec Ip.Corp.	Remote anomaly diagnosis and reconfiguration of an automatic data collection device platform over a telecommunications network
US20050274801A1 (en) *	1999-01-29	2005-12-15	Intermec Ip Corp.	Method, apparatus and article for validating ADC devices, such as barcode, RFID and magnetic stripe readers
US7122666B2 (en)	1999-07-21	2006-10-17	Sankyo Company, Limited	Heteroaryl-substituted pyrrole derivatives, their preparation and their therapeutic uses
US6976062B1 (en) *	1999-09-22	2005-12-13	Intermec Ip Corp.	Automated software upgrade utility
US6759410B1 (en) *	1999-11-23	2004-07-06	Smithline Beecham Corporation	3,4-dihydro-(1H)-quinazolin-2-ones and their use as CSBP/p38 kinase inhibitors
ATE281439T1 (de)	1999-11-23	2004-11-15	Smithkline Beecham Corp	3,4-dihydro-(1h)chinazolin-2-on-verbindungen als csbp/p38-kinase-inhibitoren
JP2003514900A (ja)	1999-11-23	2003-04-22	スミスクライン・ビーチャム・コーポレイション	ＣＳＢＰ／ｐ３８キナーゼ阻害剤としての３，４−ジヒドロ−（１Ｈ）−キナゾリン−２−オン化合物
EP1233950B1 (en)	1999-11-23	2005-10-05	Smithkline Beecham Corporation	3,4-DIHYDRO-(1H)QUINAZOLIN-2-ONE COMPOUNDS AS CSBP/P39 kINASE INHIBITORS
RU2198170C2 (ru) *	1999-12-27	2003-02-10	Санкио Компани, Лимитед	Производные пиррола, фармацевтические композиции на их основе и способ лечения
US7235551B2 (en) *	2000-03-02	2007-06-26	Smithkline Beecham Corporation	1,5-disubstituted-3,4-dihydro-1h-pyrimido[4,5-d]pyrimidin-2-one compounds and their use in treating csbp/p38 kinase mediated diseases
CN100525768C (zh) *	2000-10-23	2009-08-12	史密丝克莱恩比彻姆公司	新化合物
ATE377598T1 (de)	2001-01-22	2007-11-15	Sankyo Co	Durch bicyclische aminogruppen substituierte verbindungen
WO2002094267A1 (en) *	2001-05-24	2002-11-28	Sankyo Company, Limited	Pharmaceutical composition for prevention or treatment of arthritis
AR039241A1 (es) *	2002-04-04	2005-02-16	Biogen Inc	Heteroarilos trisustituidos y metodos para su produccion y uso de los mismos
UA80295C2 (en) *	2002-09-06	2007-09-10	Biogen Inc	Pyrazolopyridines and using the same
CL2004000234A1 (es) *	2003-02-12	2005-04-15	Biogen Idec Inc	Compuestos derivados 3-(piridin-2-il)-4-heteroaril-pirazol sustituidos, antagonistas de aik5 y/o aik4; composicion farmaceutica y uso del compuesto en el tratamiento de desordenes fibroticos como esclerodermia, lupus nefritico, cicatrizacion de herid
MY145343A (en) *	2005-03-25	2012-01-31	Glaxo Group Ltd	Novel compounds
US20080096905A1 (en) *	2005-03-25	2008-04-24	Glaxo Group Limited	Process For Preparing Pyrido[2,3-D]Pyrimidin-7-One And 3,4-Dihydropyrimido{4,5-D}Pyrimidin-2(1H)-One Derivatives
US8944332B2 (en)	2006-08-04	2015-02-03	Intermec Ip Corp.	Testing automatic data collection devices, such as barcode, RFID and/or magnetic stripe readers
WO2019168874A1 (en)	2018-02-27	2019-09-06	The Research Foundation For The State University Of New York	Difluoromethoxylation and trifluoromethoxylation compositions and methods for synthesizing same

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US2748119A (en) *	1954-06-23	1956-05-29	Searle & Co	6-furyl and 6-thienyl derivatives of 4-trifluoromethyl-2-pyrimidinamines
US3557114A (en) *	1968-12-23	1971-01-19	Merck & Co Inc	1-substituted-3-(2-pyrimidinyl) imidazolium salts
US3707475A (en) *	1970-11-16	1972-12-26	Pfizer	Antiinflammatory imidazoles
US3929807A (en) *	1971-05-10	1975-12-30	Ciba Geigy Corp	2-Substituted-4(5)-(aryl)-5(4)-(2,3 or -4-pyridyl)-imidazoles
US3940486A (en) *	1971-05-10	1976-02-24	Ciba-Geigy Corporation	Imidazole derivatives in the treatment of pain
US4058614A (en) *	1973-12-04	1977-11-15	Merck & Co., Inc.	Substituted imidazole compounds and therapeutic compositions therewith
US4199592A (en) *	1978-08-29	1980-04-22	E. I. Du Pont De Nemours And Company	Antiinflammatory 4,5-diaryl-2-nitroimidazoles
GR75287B (pt) *	1980-07-25	1984-07-13	Ciba Geigy Ag
US4503065A (en) *	1982-08-03	1985-03-05	E. I. Du Pont De Nemours And Company	Antiinflammatory 4,5-diaryl 1-2-halo imidazoles
US4565875A (en) *	1984-06-27	1986-01-21	Fmc Corporation	Imidazole plant growth regulators
US4686231A (en) *	1985-12-12	1987-08-11	Smithkline Beckman Corporation	Inhibition of 5-lipoxygenase products
ES2087056T3 (es) *	1986-01-13	1996-07-16	American Cyanamid Co	2-pirimidinaminas sustituidas en las posiciones 4, 5 y 6.
IL83467A0 (en) *	1986-08-15	1988-01-31	Fujisawa Pharmaceutical Co	Imidazole derivatives,processes for their preparation and pharmaceutical compositions containing the same
GB8906965D0 (en) *	1989-03-28	1989-05-10	Schering Agrochemicals Ltd	Fungicides
US5312828A (en) *	1989-06-14	1994-05-17	Finkelstein Joseph A	Substituted imidazoles having angiotensin II receptor blocking activity
US5234917A (en) *	1989-12-29	1993-08-10	Finkelstein Joseph A	Substituted 5-(alkyl)carboxamide imidazoles
ZA919797B (en) *	1990-12-13	1992-10-28	Smithkline Beecham Corp	Bicyclo-5,6-dihydro-7h-pyrrolo-1,20-imidazol-7-ols and 7-ones
AU9137591A (en) *	1990-12-13	1992-07-08	Smithkline Beecham Corporation	Novel csaids
US5656644A (en) *	1994-07-20	1997-08-12	Smithkline Beecham Corporation	Pyridyl imidazoles
MX9300141A (es) *	1992-01-13	1994-07-29	Smithkline Beecham Corp	Compuestos de imidazol novedosos, procedimiento para su preparacion y composiciones farmaceuticas que lo contienen.
US5593992A (en) *	1993-07-16	1997-01-14	Smithkline Beecham Corporation	Compounds
US5670527A (en) *	1993-07-16	1997-09-23	Smithkline Beecham Corporation	Pyridyl imidazole compounds and compositions
US5593991A (en) *	1993-07-16	1997-01-14	Adams; Jerry L.	Imidazole compounds, use and process of making
IL110296A (en) *	1993-07-16	1999-12-31	Smithkline Beecham Corp	Imidazole compounds process for their preparation and pharmaceutical compositions containing them
PT672041E (pt) *	1993-10-01	2002-04-29	Novartis Ag	Derivados da piridina farmacologicamente activos e processos para a sua preparacao
US5543520A (en) *	1993-10-01	1996-08-06	Ciba-Geigy Corporation	Pyrimidine derivatives
WO1995009851A1 (en) *	1993-10-01	1995-04-13	Ciba-Geigy Ag	Pharmacologically active pyrimidineamine derivatives and processes for the preparation thereof
WO1995009847A1 (en) *	1993-10-01	1995-04-13	Ciba-Geigy Ag	Pyrimidineamine derivatives and processes for the preparation thereof
DE4337611A1 (de) *	1993-11-04	1995-05-11	Boehringer Ingelheim Kg	Neue Benzoylguanidine, ihre Herstellung und ihre Verwendung in Arzneimitteln
CZ219597A3 (cs) *	1995-01-12	1998-03-18	Smithkline Beecham Corporation	Nové sloučeniny
US5739143A (en) *	1995-06-07	1998-04-14	Smithkline Beecham Corporation	Imidazole compounds and compositions
IL118544A (en) *	1995-06-07	2001-08-08	Smithkline Beecham Corp	History of imidazole, the process for their preparation and the pharmaceutical preparations containing them
ZA9610687B (en) *	1995-12-22	1997-09-29	Smithkline Beecham Corp	Novel synthesis.
ZA97175B (en) *	1996-01-11	1997-11-04	Smithkline Beecham Corp	Novel substituted imidazole compounds.
PL187516B1 (pl) *	1996-01-11	2004-07-30	Smithkline Beecham Corp	Nowe podstawione pochodne imidazolu, sposób ich wytwarzania oraz kompozycja farmaceutyczna zawierająca te związki
EP0883402A4 (en) *	1996-01-11	1999-08-11	Smithkline Beecham Corp	NEW CYCLOALKYL-SUBSTITUTED IMIDAZOLES
AP9700912A0 (en) *	1996-01-11	1997-01-31	Smithkline Beecham Corp	Novel cycloalkyl substituted imidazoles
EP0889887A4 (en) *	1996-03-25	2003-06-11	Smithkline Beecham Corp	TREATMENT OF CENTRAL NERVOUS SYSTEM INJURIES
EP0889888A4 (en) *	1996-03-25	2003-01-08	Smithkline Beecham Corp	NEW TREATMENT OF LESIONS IN THE CENTRAL NERVOUS SYSTEM

1996
- 1996-12-19 ZA ZA9610687A patent/ZA9610687B/xx unknown
- 1996-12-20 AU AU14681/97A patent/AU704500B2/en not_active Ceased
- 1996-12-20 KR KR1019980704729A patent/KR19990076625A/ko not_active Ceased
- 1996-12-20 EP EP96945272A patent/EP1019393A4/en not_active Withdrawn
- 1996-12-20 BR BR9612187A patent/BR9612187A/pt not_active Application Discontinuation
- 1996-12-20 JP JP52385597A patent/JP3245175B2/ja not_active Expired - Fee Related
- 1996-12-20 NZ NZ326574A patent/NZ326574A/xx unknown
- 1996-12-20 CZ CZ981985A patent/CZ198598A3/cs unknown
- 1996-12-20 AR ARP960105842A patent/AR004405A1/es unknown
- 1996-12-20 CN CN96180018A patent/CN1209128A/zh active Pending
- 1996-12-20 PL PL96327311A patent/PL327311A1/xx unknown
- 1996-12-20 TR TR1998/01121T patent/TR199801121T2/xx unknown
- 1996-12-20 HU HU9902466A patent/HUP9902466A3/hu unknown
- 1996-12-20 US US09/091,799 patent/US6100399A/en not_active Expired - Fee Related
- 1996-12-20 IL IL12490896A patent/IL124908A/xx not_active IP Right Cessation
- 1996-12-20 WO PCT/US1996/020599 patent/WO1997023479A1/en not_active Ceased
- 1996-12-20 US US08/771,320 patent/US5917043A/en not_active Expired - Fee Related
- 1996-12-20 IL IL14351796A patent/IL143517A/xx not_active IP Right Cessation
1997
- 1997-08-22 TW TW086112050A patent/TW434236B/zh not_active IP Right Cessation
1998
- 1998-03-30 AR ARP980101440A patent/AR015579A1/es not_active Application Discontinuation
- 1998-03-30 AR ARP980101441A patent/AR012567A1/es not_active Application Discontinuation
- 1998-06-19 NO NO982850A patent/NO982850D0/no not_active Application Discontinuation
1999
- 1999-01-20 US US09/233,511 patent/US6255491B1/en not_active Expired - Fee Related

Also Published As

Publication number	Publication date
AR015579A1 (es)	2001-05-16
JP2000502683A (ja)	2000-03-07
AR004405A1 (es)	1998-11-04
HUP9902466A3 (en)	2002-11-28
HUP9902466A2 (hu)	2000-05-28
IL143517A (en)	2003-09-17
WO1997023479A1 (en)	1997-07-03
IL143517A0 (en)	2002-04-21
KR19990076625A (ko)	1999-10-15
AU1468197A (en)	1997-07-17
TR199801121T2 (xx)	1998-08-21
AU704500B2 (en)	1999-04-22
ZA9610687B (en)	1997-09-29
EP1019393A1 (en)	2000-07-19
NZ326574A (en)	2000-01-28
AR012567A1 (es)	2000-11-08
CZ198598A3 (cs)	1998-10-14
IL124908A0 (en)	1999-01-26
US6100399A (en)	2000-08-08
IL124908A (en)	2003-05-29
JP3245175B2 (ja)	2002-01-07
US5917043A (en)	1999-06-29
US6255491B1 (en)	2001-07-03
NO982850L (no)	1998-06-19
EP1019393A4 (en)	2000-07-19
NO982850D0 (no)	1998-06-19
CN1209128A (zh)	1999-02-24
PL327311A1 (en)	1998-12-07
TW434236B (en)	2001-05-16

Legal Events

Date	Code	Title	Description
2004-11-30	B07A	Application suspended after technical examination (opinion) [chapter 7.1 patent gazette]
2005-05-03	B09B	Patent application refused [chapter 9.2 patent gazette]

Publication	Publication Date	Title
BR9612187A (pt)	1999-07-13	Nova sintese
FI972970A0 (fi)	1997-07-11	Uusia yhdisteitä
DE69620399D1 (de)	2002-05-08	Sprachsynthese
FI20030162L (fi)	2003-02-03	Uusia yhdisteitä
ID16345A (id)	1997-09-25	Senyawa-senyawa heterosiklik
NO964922D0 (no)	1996-11-19	Dypvanns-stigerörssammenstilling
DK0791016T3 (da)	2000-10-09	Polymersyntese
EP0857067A4 (en)	2005-01-19	RADIATION PROTECTION SUBSTANCES
FI951018A0 (fi)	1995-03-06	Hoeghastighetsdataoeverfoering i mobiltelesystem
DE69630414D1 (de)	2003-11-27	5B4T-Kodierungsschema
NO974100D0 (no)	1997-09-05	Talesyntese
EE9800172A (et)	1998-12-15	Ühendid
NO974170D0 (no)	1997-09-09	Polyazacykloalkan-forbindelser
BR9610194A (pt)	1998-12-15	Aminouracilas substituídas
DE59600405D1 (de)	1998-09-10	Gehhilfe
KR970014750U (ko)	1997-04-28	저울
SE9503561D0 (sv)	1995-10-12	New Compounds
SE9502559D0 (sv)	1995-07-11	Novel compounds
FI951528A0 (fi)	1995-03-31	Tofttrappa; anordning foer stigning fraon vatten i baot
NO952168D0 (no)	1995-06-01	Musikkteknologi
NO951858D0 (no)	1995-05-11	Musikkteknologi
KR970008217U (ko)	1997-03-27	소리나는 블럭
ITMI950031A0 (it)	1995-01-10	Composti dibenzoalchilenici
BR1100842A (pt)	2000-04-18	Compostos
FI2050U1 (fi)	1995-08-03	Rullstol foer fastmontering i fordonsgolv