BRPI0412721A - processo para preparar bromidrato de eletriptano alfa-polimórfico - Google Patents

processo para preparar bromidrato de eletriptano alfa-polimórfico

Info

Publication number
BRPI0412721A
BRPI0412721A BRPI0412721-8A BRPI0412721A BRPI0412721A BR PI0412721 A BRPI0412721 A BR PI0412721A BR PI0412721 A BRPI0412721 A BR PI0412721A BR PI0412721 A BRPI0412721 A BR PI0412721A
Authority
BR
Brazil
Prior art keywords
electriptan
hydrobromide
polymorphic
preparing alpha
preparing
Prior art date
Application number
BRPI0412721-8A
Other languages
English (en)
Inventor
Patrick Joseph Furlong
Cornelius Joseph Kelly
Ronald James Ogilvie
Vincent Ryan
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=27772518&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=BRPI0412721(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Pfizer filed Critical Pfizer
Publication of BRPI0412721A publication Critical patent/BRPI0412721A/pt

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/06—Antimigraine agents

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Neurosurgery (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Neurology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pain & Pain Management (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Biomedical Technology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Indole Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Electrolytic Production Of Non-Metals, Compounds, Apparatuses Therefor (AREA)

Abstract

"PROCESSO PARA PREPARAR BROMIDRATO DE ELETRIPTANO ALFA-POLIMóRFICO". A presente invenção apresenta um processo melhorado para o preparo de bromidrato de eletriptano apolimórfico.
BRPI0412721-8A 2003-07-23 2004-07-12 processo para preparar bromidrato de eletriptano alfa-polimórfico BRPI0412721A (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GBGB0317229.3A GB0317229D0 (en) 2003-07-23 2003-07-23 Improved process
PCT/IB2004/002322 WO2005007649A1 (en) 2003-07-23 2004-07-12 Improved process for preparing alpha-polymorphic eletriptan hydrobromide

Publications (1)

Publication Number Publication Date
BRPI0412721A true BRPI0412721A (pt) 2006-09-26

Family

ID=27772518

Family Applications (1)

Application Number Title Priority Date Filing Date
BRPI0412721-8A BRPI0412721A (pt) 2003-07-23 2004-07-12 processo para preparar bromidrato de eletriptano alfa-polimórfico

Country Status (25)

Country Link
EP (1) EP1660485B1 (pt)
JP (1) JP2006528172A (pt)
KR (1) KR100694962B1 (pt)
CN (1) CN100430388C (pt)
AR (1) AR046509A1 (pt)
AT (1) ATE349442T1 (pt)
AU (1) AU2004256994A1 (pt)
BR (1) BRPI0412721A (pt)
CA (1) CA2532111A1 (pt)
CO (1) CO5650232A2 (pt)
CY (1) CY1105980T1 (pt)
DE (1) DE602004003966T2 (pt)
DK (1) DK1660485T3 (pt)
ES (1) ES2274473T3 (pt)
GB (1) GB0317229D0 (pt)
IL (1) IL172765A0 (pt)
MX (1) MXPA06000793A (pt)
NO (1) NO20056238L (pt)
NZ (1) NZ544305A (pt)
PL (1) PL1660485T3 (pt)
PT (1) PT1660485E (pt)
RU (1) RU2320655C2 (pt)
TW (1) TWI291956B (pt)
WO (1) WO2005007649A1 (pt)
ZA (1) ZA200600607B (pt)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP1663978B1 (en) 2003-07-23 2007-11-28 Bayer Pharmaceuticals Corporation Fluoro substituted omega-carboxyaryl diphenyl urea for the treatment and prevention of diseases and conditions
JP5214124B2 (ja) 2006-08-17 2013-06-19 三星電子株式会社 通信システム、通信装置、尤度計算方法、及びプログラム
US20090299077A1 (en) * 2008-05-22 2009-12-03 Vinod Kumar Kansal Salts of (R)-5-(2phenylsulphonylethenyl)-3-(N-methylpyrrolidin-2-ylmethyl)-1H-indole, 5-bromo-3-[(R)-1-methyl-pyrrolidin-2-ylmethyl]-1H-indole and of eletriptan
WO2010116386A2 (en) * 2009-04-08 2010-10-14 Biophore India Pharmaceuticals Pvt. Ltd. Novel polymorph of eletriptan hydrobromide and process for the preparation thereof
IT1393700B1 (it) * 2009-04-22 2012-05-08 F S I Fabbrica Italiana Sint Sintesi di 3-{[(2r)-1-metilpirrolidin-2-il]metil}-5-[2-(fenilsulfonil)etil]-1h-indolo
WO2011004391A2 (en) * 2009-06-25 2011-01-13 Matrix Laboratories Ltd An improved process for the preparation of eletriptan and its salt thereof
US8754239B2 (en) 2010-01-19 2014-06-17 Sms Pharmaceuticals Limited Process for preparing eletriptan hydrobromide having α-form
WO2012004811A1 (en) * 2010-07-06 2012-01-12 Ind-Swift Laboratories Limited Process for the preparation of 5-substsituted indole derivative
CN102786514B (zh) * 2012-07-26 2014-01-29 武汉人福医药集团股份有限公司 依来曲普坦的制备方法
CN104341397A (zh) * 2013-07-31 2015-02-11 上海威智医药科技有限公司 具晶型的依来曲普坦自由碱及其制法和应用

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TW288010B (pt) * 1992-03-05 1996-10-11 Pfizer
FR2701026B1 (fr) * 1993-02-02 1995-03-31 Adir Nouveaux dérivés de l'indole, de l'indazole et du benzisoxazole, leur procédé de préparation et les compositions pharmaceutiques qui les contiennent.
WO1996004842A1 (en) * 1994-08-12 1996-02-22 Thomas Donald D Ii Miniaturized blood pressure monitor kit
GB9417310D0 (en) * 1994-08-27 1994-10-19 Pfizer Ltd Therapeutic agents
GB9825988D0 (en) * 1998-11-27 1999-01-20 Pfizer Ltd Indole derivatives
GB0031094D0 (en) * 2000-12-20 2001-01-31 Pfizer Ltd New Process

Also Published As

Publication number Publication date
MXPA06000793A (es) 2006-04-07
EP1660485A1 (en) 2006-05-31
CO5650232A2 (es) 2006-06-30
KR20060030118A (ko) 2006-04-07
GB0317229D0 (en) 2003-08-27
DE602004003966T2 (de) 2007-05-24
CA2532111A1 (en) 2005-01-27
PT1660485E (pt) 2007-01-31
RU2006101689A (ru) 2006-06-27
WO2005007649A1 (en) 2005-01-27
IL172765A0 (en) 2006-04-10
CN100430388C (zh) 2008-11-05
RU2320655C2 (ru) 2008-03-27
TW200510388A (en) 2005-03-16
TWI291956B (en) 2008-01-01
DE602004003966D1 (de) 2007-02-08
CN1823060A (zh) 2006-08-23
DK1660485T3 (da) 2007-03-19
NZ544305A (en) 2008-09-26
KR100694962B1 (ko) 2007-03-14
ATE349442T1 (de) 2007-01-15
ZA200600607B (en) 2007-05-30
ES2274473T3 (es) 2007-05-16
AR046509A1 (es) 2005-12-14
EP1660485B1 (en) 2006-12-27
JP2006528172A (ja) 2006-12-14
PL1660485T3 (pl) 2007-04-30
CY1105980T1 (el) 2011-04-06
AU2004256994A1 (en) 2005-01-27
NO20056238L (no) 2006-04-05

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Legal Events

Date Code Title Description
B08F Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette]

Free format text: REFERENTE AS 6A E 7A ANUIDADES.

B08K Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette]

Free format text: REFERENTE AO DESPACHO 8.6 PUBLICADO NA RPI 2159 DE 22/05/2012.