BRPI0413787A - delta 15-d-homoesteróides com efeito androgênico - Google Patents

delta 15-d-homoesteróides com efeito androgênico

Info

Publication number
BRPI0413787A
BRPI0413787A BRPI0413787-6A BRPI0413787A BRPI0413787A BR PI0413787 A BRPI0413787 A BR PI0413787A BR PI0413787 A BRPI0413787 A BR PI0413787A BR PI0413787 A BRPI0413787 A BR PI0413787A
Authority
BR
Brazil
Prior art keywords
steroids
homo
delta
androgenic effect
androgenic
Prior art date
Application number
BRPI0413787-6A
Other languages
English (en)
Inventor
Ralf Wyrwa
Sven Ring
Guenter Kaufmann
Walter Elger
Birgitt Schneider
Original Assignee
Schering Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from DE10339532A external-priority patent/DE10339532A1/de
Application filed by Schering Ag filed Critical Schering Ag
Publication of BRPI0413787A publication Critical patent/BRPI0413787A/pt

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J63/00—Steroids in which the cyclopenta(a)hydrophenanthrene skeleton has been modified by expansion of only one ring by one or two atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A61P15/08—Drugs for genital or sexual disorders; Contraceptives for gonadal disorders or for enhancing fertility, e.g. inducers of ovulation or of spermatogenesis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00—Drugs for disorders of the endocrine system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00—Drugs for disorders of the endocrine system
    • A61P5/24—Drugs for disorders of the endocrine system of the sex hormones
    • A61P5/26—Androgens
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00—Drugs for disorders of the endocrine system
    • A61P5/24—Drugs for disorders of the endocrine system of the sex hormones
    • A61P5/30—Oestrogens
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J75/00—Processes for the preparation of steroids in general

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Endocrinology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Diabetes (AREA)
  • Reproductive Health (AREA)
  • Gynecology & Obstetrics (AREA)
  • Pregnancy & Childbirth (AREA)
  • Epidemiology (AREA)
  • Steroid Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

"DELTA15-D-HOMOESTERóIDES COM EFEITO ANDROGêNICO". A invenção refere-se a <30>¬ 15¬-D-homoesteróides da fórmula geral (I), a métodos para a produção dos mesmos, e a composições farmacêuticas que contêm os referidos compostos. Os compostos da fórmula geral (I) da invenção estão dotados de atividade androgênica.
BRPI0413787-6A 2003-08-21 2004-08-19 delta 15-d-homoesteróides com efeito androgênico BRPI0413787A (pt)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US49666903P 2003-08-21 2003-08-21
DE10339532A DE10339532A1 (de) 2003-08-21 2003-08-21 Delta 15-D-Homosteroide mit androgener Wirkung
PCT/EP2004/009468 WO2005021573A1 (de) 2003-08-21 2004-08-19 Δ15-d-homosteroide mit androgener wirkung

Publications (1)

Publication Number Publication Date
BRPI0413787A true BRPI0413787A (pt) 2006-11-07

Family

ID=34276519

Family Applications (1)

Application Number Title Priority Date Filing Date
BRPI0413787-6A BRPI0413787A (pt) 2003-08-21 2004-08-19 delta 15-d-homoesteróides com efeito androgênico

Country Status (11)

Country Link
US (1) US7388003B2 (pt)
EP (1) EP1658306A1 (pt)
JP (1) JP2007502801A (pt)
KR (1) KR20060091295A (pt)
AU (1) AU2004268040A1 (pt)
BR (1) BRPI0413787A (pt)
CA (1) CA2534831A1 (pt)
EC (1) ECSP066441A (pt)
IL (1) IL173608A0 (pt)
MX (1) MXPA06002034A (pt)
WO (1) WO2005021573A1 (pt)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TW200745156A (en) * 2005-06-17 2007-12-16 Organon Nv Steroids having a mixed androgenic and progestagenic profile

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1054262A (pt) *
IL50854A (en) * 1975-11-11 1979-12-30 Sparamedica Ag D-homosteroids their manufacture and pharmaceutical compositions containing them
IL51468A (en) * 1976-02-23 1981-01-30 Sparamedica Ag 17 -hydroxy- -d-homosteroid derivatives,their preparation and pharmaceutical compositions containing them
NL7703448A (nl) * 1976-04-13 1977-10-17 Hoffmann La Roche Nieuwe d-homosteroiden.
DE10247399A1 (de) * 2002-10-08 2004-04-29 Schering Ag Pharmazeutische Zubereitungen, Verwendung dieser Zubereitung und Verfahren zur Erhöhung der Bioverfügbarkeit von peroral zu applizierenden Arzneistoffen

Also Published As

Publication number Publication date
KR20060091295A (ko) 2006-08-18
US7388003B2 (en) 2008-06-17
WO2005021573A1 (de) 2005-03-10
AU2004268040A1 (en) 2005-03-10
MXPA06002034A (es) 2006-05-17
IL173608A0 (en) 2006-07-05
JP2007502801A (ja) 2007-02-15
EP1658306A1 (de) 2006-05-24
ECSP066441A (es) 2006-09-18
CA2534831A1 (en) 2005-03-10
US20050131076A1 (en) 2005-06-16

Similar Documents

Publication Publication Date Title
BRPI0512938A (pt) derivados da quinazolinediona como inibidores parp
BR0315296A (pt) Derivados do ciclohexanol espirocìclicos
BRPI0507462A (pt) compostos de quinolina substituìdos
BR0312513A (pt) Derivados de glicosìdeo de tiofeno, processos para a produção dos mesmos, medicamentos que contêm esses compostos e uso dos mesmos
BR0308967A (pt) Derivados de quinolina e isoquinolina, um processo para a sua preparação e sua aplicação como inibidores de inflamação
BRPI0514841A (pt) inibidores de piridila da sinalização de hedgehog, processo de preparação dos mesmos e composição compreendendo os referidos inibidores
BRPI0720972B8 (pt) compostos análogos de ciclopamina e composições farmacêuticas compreendendo os referidos compostos
BRPI0408347B8 (pt) derivados de pirimidina, seu uso, e composição e combinação farmacêuticas
BR0010555A (pt) Inibidores de neuraminidases
BR0208338A (pt) Derivados de piridina
BR0312464A (pt) Inibidores de tirosina quinases
BRPI0510410A (pt) compostos orgánicos
BRPI0510273A (pt) derivados de tetraazabenzo[e]azuleno e análogos destes
SE0102616D0 (sv) Novel compounds
BRPI0108395B8 (pt) derivados de pirrolopirimidinona, processos de preparação e uso
BRPI0513184A (pt) derivados de 2-carbamida-4-feniltiazol, preparação dos mesmos e aplicação dos mesmos em terapia
BR0310077A (pt) Novos compostos e sua utilização
BRPI0510260A (pt) método para purificar um composto, e, kit farmacêutico
BRPI0509588A (pt) derivados e tetraidronaftiridina e um processo para preparação dos mesmos
BRPI0408353A (pt) composto, composição farmacêutica, métodos para o tratamento de neoplasias suscetìveis e para o tratamento de infecções virais, e, uso de um composto
BRPI0418255A (pt) derivados de piperazina e piperidina n-substituìdos
CR9182A (es) Derivado de quinolina, su uso, preparacion y medicamento que lo contiene
BRPI0513891A (pt) derivados de propenil piperazina substituìdos como novos inibidores de histona deacetilase
BRPI0411092A (pt) benzo[b]tiofenos substituìdos com 3-arilsulfanila e com 3-heteroarilsulfanila como agentes terapêuticos
BRPI0512677A2 (pt) derivados de quinazolina

Legal Events

Date Code Title Description
B08F Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette]

Free format text: REFERENTE A 5A,6A E 7A ANUIDADE(S)

B08K Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette]

Free format text: REFERENTE AO DESPACHO 8.6 PUBLICADO NA RPI 2129 DE 25/10/2011.