BRPI0414527A - tratamento de tumores estromáticos gastrointestinais com imatinib e midostaurina - Google Patents

tratamento de tumores estromáticos gastrointestinais com imatinib e midostaurina

Info

Publication number
BRPI0414527A
BRPI0414527A BRPI0414527-5A BRPI0414527A BRPI0414527A BR PI0414527 A BRPI0414527 A BR PI0414527A BR PI0414527 A BRPI0414527 A BR PI0414527A BR PI0414527 A BRPI0414527 A BR PI0414527A
Authority
BR
Brazil
Prior art keywords
imatinib
midostaurin
treatment
gastrointestinal stromal
stromal tumors
Prior art date
Application number
BRPI0414527-5A
Other languages
English (en)
Inventor
Sasa Dimitrijevic
Jonathan A Fletcher
Sandra Leta Silberman
Original Assignee
Novartis Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Novartis Ag filed Critical Novartis Ag
Publication of BRPI0414527A publication Critical patent/BRPI0414527A/pt

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/4965—Non-condensed pyrazines
    • A61K31/497—Non-condensed pyrazines containing further heterocyclic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/55—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
    • A61K31/553—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole having at least one nitrogen and one oxygen as ring hetero atoms, e.g. loxapine, staurosporine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical & Material Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Epidemiology (AREA)
  • Organic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines Containing Material From Animals Or Micro-Organisms (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)

Abstract

"TRATAMENTO DE TUMORES ESTROMáTICOS GASTROINTESTINAIS COM IMATINIB E MIDOSTAURINA". A presente invenção refere-se ao uso de uma combinação que compreende (a) imatinib ou um sal farmaceuticamente aceitável do mesmo e midostaurina ou um sal farmaceuticamente aceitável do mesmo para a preparação de um medicamento para o tratamento de tumores estromáticos gastrointestinais, como por exemplo tumores estromáticos gastrointestinais resistentes ao imatinib.
BRPI0414527-5A 2003-09-19 2004-09-17 tratamento de tumores estromáticos gastrointestinais com imatinib e midostaurina BRPI0414527A (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US50424503P 2003-09-19 2003-09-19
PCT/EP2004/010467 WO2005027971A1 (en) 2003-09-19 2004-09-17 Treatment of gastrointestinal stromal tumors with imatinib and midostaurin

Publications (1)

Publication Number Publication Date
BRPI0414527A true BRPI0414527A (pt) 2006-11-07

Family

ID=34375467

Family Applications (1)

Application Number Title Priority Date Filing Date
BRPI0414527-5A BRPI0414527A (pt) 2003-09-19 2004-09-17 tratamento de tumores estromáticos gastrointestinais com imatinib e midostaurina

Country Status (11)

Country Link
US (1) US20080096864A1 (pt)
EP (1) EP1667719B1 (pt)
JP (1) JP2007505859A (pt)
CN (1) CN100467064C (pt)
AT (1) ATE489109T1 (pt)
AU (1) AU2004273605B2 (pt)
BR (1) BRPI0414527A (pt)
CA (1) CA2538523A1 (pt)
DE (1) DE602004030265D1 (pt)
MX (1) MXPA06003056A (pt)
WO (1) WO2005027971A1 (pt)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
PT1686997E (pt) * 2003-11-18 2009-07-17 Novartis Ag Inibidores da forma mutante de kit
RU2410098C2 (ru) * 2004-08-31 2011-01-27 Новартис Аг Применение мидостаурина для лечения желудочно-кишечных стромальных опухолей
CN103638028A (zh) * 2005-05-02 2014-03-19 诺瓦提斯公司 嘧啶基氨基苯甲酰胺衍生物用于治疗全身性肥大细胞增多症的应用
BRPI0613863A2 (pt) 2005-07-20 2011-02-15 Peter Valent composições para tratamento de mastocitose sistêmica
WO2007054579A1 (en) * 2005-11-14 2007-05-18 Universität Zürich Staurosporine derivatives for use in alveolar rhabdomyosarcoma

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CO4940418A1 (es) * 1997-07-18 2000-07-24 Novartis Ag Modificacion de cristal de un derivado de n-fenil-2- pirimidinamina, procesos para su fabricacion y su uso
ITMI992711A1 (it) * 1999-12-27 2001-06-27 Novartis Ag Composti organici
SK287335B6 (sk) * 2000-10-27 2010-07-07 Novartis Ag Použitie 4-{(4-metylpiperazin-1-ylmetyl)-N-[4-metyl-3-(4-pyrid-3- yl)pyrimidin-2-ylamino]fenyl}-benzamidu na prípravu farmaceutických kompozícií na liečenie gastrointestinálnych strómových tumorov
AU2003214079B2 (en) * 2002-02-28 2007-05-31 Novartis Ag N-{5-[4-(4-methyl-piperazino-methyl)-benzoylamido]-2-methylphenyl}-4-(3-pyridyl)-2-pyrimidine-amine coated stents
ES2303585T3 (es) * 2002-04-10 2008-08-16 Virginia Commonwealth University Combinacion de glivec(sti571) con un inhibidor de quinasa dependiente de ciclina, especialmente flavopiridol en el tratamiento de cancer.

Also Published As

Publication number Publication date
AU2004273605A1 (en) 2005-03-31
CA2538523A1 (en) 2005-03-31
ATE489109T1 (de) 2010-12-15
EP1667719A1 (en) 2006-06-14
EP1667719B1 (en) 2010-11-24
CN100467064C (zh) 2009-03-11
AU2004273605B2 (en) 2008-07-31
JP2007505859A (ja) 2007-03-15
DE602004030265D1 (de) 2011-01-05
CN1852738A (zh) 2006-10-25
US20080096864A1 (en) 2008-04-24
WO2005027971A1 (en) 2005-03-31
MXPA06003056A (es) 2006-05-31

Similar Documents

Publication Publication Date Title
CL2009000349A1 (es) Compuestos derivados de 4,5-dihidro-oxazol-2-ilamina; procedimiento de preparacion; composicion farmaceutica; y su uso para el tratamiento de la enfermedad de alzheimer.
BRPI0007487B8 (pt) difenil-uréias substituídas com w-carbóxi-arilas como inibidores de raf cinase
BRPI0410418A (pt) fenil quinolinas e seu uso como moduladores do receptor de estrogênio
CL2004001069A1 (es) Compuestos derivados de 1-benzoil-isoquinolinas sustituidos; procedimiento de preparacion, composicion farmaceutica; y uso para el tratamiento o profilaxis de diabetes tipo ii.
BR0312573A (pt) Derivados de fenil-[4-(3-fenil-1h-pirazol-4-il)-pirimidin-2-il]-amina
CL2007001427A1 (es) Sal de maleato de 5-amino-3-(2',3'-di-o-acetil-beta-d-ribofuranosil)-3h-tiazolo[4,5-d]pirimidin-2-ona; procedimiento de preparacion; composicion farmaceutica que comprende a dicho compuesto; y uso del compuesto para el tratamiento de una infeccion po
BRPI0418099A (pt) compostos, composição farmacêutica, e uso de um composto
MX2009003958A (es) Nuevos derivados de 1,4-benzotiepina-1,1-dioxido sustituidos con radicales bencilo, metodo para su preparacion, productos farmaceuticos que comprenden estos compuestos y su uso.
CL2008001932A1 (es) Compuestos derivados de 6-cicloamino-3-(piridin-4-il)imidazo[1,2-b]piridazina, inhibidores de cq1epsilon y/o ck1delta; procedimiento de preparacion; composicion farmaceutica que los comprende; y uso en el tratamiento de desordenes del sueno, trastorno del ritmo circadiano, cancer y enfermedad de alzheimer.
UY28931A1 (es) Derivados de pirrolotriazina utiles para tratar trastornos hiper-proliferativos y enfermedades asociadas con angiogenesis
PT1696905E (pt) 2-aminotetralinas substituídas para o tratamento preventivo da doença de parkinson
SV1999000194A (es) Preparado farmaceuticio de moxifloxacina ref. lea 33327-sv
CL2007001205A1 (es) Compuestos derivados de n-fenil-3-tio-4-fenil-azetedin-2-ona; procedimiento de preparacion; composicion farmaceutica; combinacion; uso en el tratamiento de una condicion hiperlipidemica, ateroesclerosis, alzheimer y tumores asociados a colesterol
CL2008001820A1 (es) Compuestos derivados de aril-isoxasol-imidazol; procedimiento de preparacion; composicion farmaceutica que los contiene; y uso en la preparacion de medicamentos utiles en el tratamiento de trastornos cognitivos y enfermedades relacionadas con alzheimer.
BR0113590A (pt) 7-oxo-piridopirimidinas
CL2007003189A1 (es) Compuestos derivados de indol y benzofurano; composicion farmaceutica; y uso para el tratamiento o la prevencion de la enfermedad de alzheimer.
BR0213684A (pt) Uso de antagonistas do receptor de endotelina para o tratamento de doenças tumorìgenas
CL2008001719A1 (es) Compuestos derivados de [1,10]-fenantrolina; procedimiento de preparacion; composicion farmaceutica; y uso en el tratamiento de enfermedades neurodegenerativas o hematologicas.
GT200800066A (es) Derivados de 9-cloro-15-deoxiprostaglandina, procedimiento para su preparacion y su uso como medicamento.
BR0309878A (pt) Heterotriciclil-6-alquilideno-penemas como inibidores de beta-lactamase
GT200600106A (es) Agentes endoparasiticidas
CL2007003281A1 (es) Compuesto 1-(4-metilfenil)dihidro-1h-pirrolo[1,2-a]imidazol-2,5-(3h,6h)-diona; composicion farmaceutica; y uso para el tratamiento terapeutico o preventivo de la neurotoxicidad periferica inducida por quimioterapeuticos.
GB0606015D0 (en) therapeutic agents
CL2004001272A1 (es) Compuestos derivados de 3-(4-metoxi-7-morfolin-4-il-benzotiazol-2-il)-1,1-disustituido-urea; procedimiento de preparacion; composicion farmaceutica; y uso del compuesto en el tratamiento del compuesto en el tratamiento de enfermedades relacionadas co
DE602004030265D1 (de) Behandlung von gastrointestinalen stromatumoren mit imatinib und midostaurin

Legal Events

Date Code Title Description
B06F Objections, documents and/or translations needed after an examination request according [chapter 6.6 patent gazette]
B08F Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette]

Free format text: REFERENTE A 8A ANUIDADE.

B08K Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette]

Free format text: REFERENTE AO DESPACHO 8.6 PUBLICADO NA RPI 2167 DE 17/07/2012.