BRPI0416108A - formulação de substáncia ativa sólida - Google Patents

formulação de substáncia ativa sólida

Info

Publication number
BRPI0416108A
BRPI0416108A BRPI0416108-4A BRPI0416108A BRPI0416108A BR PI0416108 A BRPI0416108 A BR PI0416108A BR PI0416108 A BRPI0416108 A BR PI0416108A BR PI0416108 A BRPI0416108 A BR PI0416108A
Authority
BR
Brazil
Prior art keywords
active substance
solid active
substance formulation
active
active substances
Prior art date
Application number
BRPI0416108-4A
Other languages
English (en)
Inventor
Axel Eble
Udo Reckmann
Peter Baur
Karl Reizlein
Original Assignee
Bayer Technology Services Gmbh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bayer Technology Services Gmbh filed Critical Bayer Technology Services Gmbh
Publication of BRPI0416108A publication Critical patent/BRPI0416108A/pt

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/50—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
    • A61K9/51—Nanocapsules; Nanoparticles
    • A61K9/5107—Excipients; Inactive ingredients
    • A61K9/513—Organic macromolecular compounds; Dendrimers
    • A61K9/5138—Organic macromolecular compounds; Dendrimers obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone, poly(meth)acrylates
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N25/00—Biocides, pest repellants or attractants, or plant growth regulators, characterised by their forms, or by their non-active ingredients or by their methods of application, e.g. seed treatment or sequential application; Substances for reducing the noxious effect of the active ingredients to organisms other than pests
    • A01N25/08—Biocides, pest repellants or attractants, or plant growth regulators, characterised by their forms, or by their non-active ingredients or by their methods of application, e.g. seed treatment or sequential application; Substances for reducing the noxious effect of the active ingredients to organisms other than pests containing solids as carriers or diluents
    • A01N25/10—Macromolecular compounds
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N25/00—Biocides, pest repellants or attractants, or plant growth regulators, characterised by their forms, or by their non-active ingredients or by their methods of application, e.g. seed treatment or sequential application; Substances for reducing the noxious effect of the active ingredients to organisms other than pests
    • A01N25/12—Powders or granules
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N41/00—Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a sulfur atom bound to a hetero atom
    • A01N41/02—Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a sulfur atom bound to a hetero atom containing a sulfur-to-oxygen double bond
    • A01N41/10—Sulfones; Sulfoxides
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/64—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with three nitrogen atoms as the only ring hetero atoms
    • A01N43/647—Triazoles; Hydrogenated triazoles
    • A01N43/653—1,2,4-Triazoles; Hydrogenated 1,2,4-triazoles
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/72—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms as ring hetero atoms
    • A01N43/88—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms as ring hetero atoms six-membered rings with three ring hetero atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
    • A61K9/1682—Processes
    • A61K9/1694—Processes resulting in granules or microspheres of the matrix type containing more than 5% of excipient
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/50—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
    • A61K9/51—Nanocapsules; Nanoparticles
    • A61K9/5192—Processes

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • General Health & Medical Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Wood Science & Technology (AREA)
  • Dentistry (AREA)
  • Plant Pathology (AREA)
  • Pest Control & Pesticides (AREA)
  • Chemical & Material Sciences (AREA)
  • Agronomy & Crop Science (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Epidemiology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • Physics & Mathematics (AREA)
  • Optics & Photonics (AREA)
  • Nanotechnology (AREA)
  • Biomedical Technology (AREA)
  • Toxicology (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Medicinal Preparation (AREA)

Abstract

"FORMULAçãO DE SUBSTáNCIA ATIVA SóLIDA". A presente invenção refere-se a novas substâncias ativas sólidas, contendo formulações de substâncias ativas, agentes de dispersão, bem como polímeros, que juntos aceitam uma mistura de partículas finas, principalmente amorfa, um processo para a sua produção e seu uso para a aplicação das substâncias ativas biologicamente ativas obtidas.
BRPI0416108-4A 2003-10-31 2004-10-19 formulação de substáncia ativa sólida BRPI0416108A (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE10351087A DE10351087A1 (de) 2003-10-31 2003-10-31 Feste Wirkstoff-Formulierung
PCT/EP2004/011807 WO2005044221A2 (de) 2003-10-31 2004-10-19 Feste wirkstoff-formulierung

Publications (1)

Publication Number Publication Date
BRPI0416108A true BRPI0416108A (pt) 2007-01-02

Family

ID=34485186

Family Applications (1)

Application Number Title Priority Date Filing Date
BRPI0416108-4A BRPI0416108A (pt) 2003-10-31 2004-10-19 formulação de substáncia ativa sólida

Country Status (7)

Country Link
US (1) US20070081947A1 (pt)
EP (1) EP1682101A2 (pt)
JP (1) JP2007509870A (pt)
BR (1) BRPI0416108A (pt)
CA (1) CA2544257A1 (pt)
DE (1) DE10351087A1 (pt)
WO (1) WO2005044221A2 (pt)

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PT1380209E (pt) * 2001-04-17 2012-09-27 Nihon Nohyaku Co Ltd Composição de agente de controlo de pragas e método de utilização da mesma
IL160858A (en) * 2004-03-14 2015-09-24 Adama Makhteshim Ltd Nano-pesticide pesticide preparation and process for preparation
US8916550B2 (en) 2005-05-09 2014-12-23 Hydra Biosciences, Inc. Compounds for modulating TRPV3 function
EP2392328A1 (en) 2005-05-09 2011-12-07 Hydra Biosciences, Inc. Compounds for modulating TRPV3 Function
DE102005026755A1 (de) * 2005-06-09 2006-12-14 Basf Ag Herstellung von festen Lösungen schwerlöslicher Wirkstoffe durch Kurzzeitüberhitzung und schnelle Trocknung
EP1942728A1 (de) * 2005-10-27 2008-07-16 Basf Se Agrochemische nanopartikuläre wirkstoffformulierungen
EP1942727A1 (de) * 2005-10-27 2008-07-16 Basf Se Nanopartikuläre wirkstoffformulierungen
CN102977011A (zh) * 2005-11-23 2013-03-20 马克特辛姆化学工厂有限公司 制备吡啶胺及其新型多晶形物的方法
GB0613925D0 (en) * 2006-07-13 2006-08-23 Unilever Plc Improvements relating to nanodispersions
WO2008033564A1 (en) 2006-09-15 2008-03-20 Hydra Biosciences Inc. Compounds for modulating trpv3 function
EP2063970A1 (en) * 2006-09-19 2009-06-03 FUJIFILM Manufacturing Europe B.V. Preparation of fine particles
IL181125A0 (en) * 2007-02-01 2007-07-04 Maktheshim Chemical Works Ltd Polymorphs of 3-(e)-2-{2-[6-(2-
GB0714223D0 (en) * 2007-07-20 2007-08-29 Fujifilm Mfg Europe Bv Preparation of fine particles
DE102007048705A1 (de) * 2007-10-11 2009-04-16 Bayer Healthcare Ag Amorphe Formulierung
DE102007050335A1 (de) * 2007-10-18 2009-04-23 Bayer Technology Services Gmbh Anordnung und Verfahren zur Bereitstellung eines vorzugsweise zeitlich veränderlichen Flüssigkeitsgemisches
AR071339A1 (es) * 2008-02-05 2010-06-16 Arysta Lifescience North Ameri Formulacion solida de compuesto activo de baja fusion
JP5551371B2 (ja) * 2008-03-24 2014-07-16 石原産業株式会社 有害生物防除用固形組成物
JP5701207B2 (ja) * 2008-06-17 2015-04-15 マクテシム・ケミカル・ワークス・リミテツド プロチオコナゾールの結晶の修飾
CN102657198B (zh) * 2012-05-08 2014-03-19 陕西上格之路生物科学有限公司 一种含苯肽胺酸的杀菌增产组合物
WO2014016370A1 (en) * 2012-07-27 2014-01-30 Ratiopharm Gmbh Amorphous aleglitazar
US20150196708A1 (en) * 2012-08-17 2015-07-16 The Regents Of The University Of California Systems, methods and compositions for improved treatment of acidosis
GB2506426B (en) * 2012-09-28 2016-03-23 Agform Ltd Composition
ES2927760T3 (es) * 2013-10-18 2022-11-10 Blanchette Rockefeller Neurosciences Inst Esteres halogenados de ácidos grasos insaturados ciclopropanados para su utilización en el tratamiento de las enfermedades neurodegenerativas
BR112016018564B1 (pt) * 2014-02-14 2021-08-31 Nanjing Scienx Biological Technology Co. Ltd Formulações ecologicamente favoráveis de benzoato de emamectina e métodos para preparação das mesmas
WO2016063157A1 (en) * 2014-10-23 2016-04-28 Bend Research Inc. Spray nozzle and process for making nanoparticles
CA2962719A1 (en) 2014-10-31 2016-05-06 Bend Research Inc. Process for forming active domains dispersed in a matrix
US11197475B2 (en) 2015-01-20 2021-12-14 Everris International B.V. Synergistic granular herbicidal compositions
EP3258781B1 (en) 2015-02-20 2022-04-06 Basf Se Agrochemical granules made of polyalkoxylate, dispersant, sugar, and polyvinylpyrrolidone
EP4574822A3 (en) 2020-01-29 2025-08-27 Kamari Pharma Ltd. Compounds and compositions for use in treating skin disorders
JP2023151957A (ja) * 2022-04-01 2023-10-16 理研ビタミン株式会社 薬物含有粒子の製造方法
CN115676871B (zh) * 2022-11-04 2023-12-05 安徽铜冠产业技术研究院有限责任公司 一种纳米氧化铜粉体的制备工艺
US11905251B1 (en) * 2023-08-29 2024-02-20 King Faisal University 1-cyclopropyl-6-fluoro-7-(4-(2-hydroxy-3-(naphthalen-2-yloxy)propylpiperazin-1-yl)-4-oxo-1,4-dihydroquinoline-3-carboxylic acid as an eco-friendly insecticidal agent against Spodoptera littoralis (boisd.)

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Also Published As

Publication number Publication date
CA2544257A1 (en) 2005-05-19
WO2005044221A2 (de) 2005-05-19
WO2005044221A3 (de) 2006-04-06
JP2007509870A (ja) 2007-04-19
US20070081947A1 (en) 2007-04-12
EP1682101A2 (de) 2006-07-26
DE10351087A1 (de) 2005-05-25

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Legal Events

Date Code Title Description
B06F Objections, documents and/or translations needed after an examination request according [chapter 6.6 patent gazette]
B25A Requested transfer of rights approved

Owner name: BAYER INTELLECTUAL PROPERTY GMBH (DE)

B08F Application fees: application dismissed [chapter 8.6 patent gazette]

Free format text: REFERENTE A 10A ANUIDADE.

B08K Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette]

Free format text: REFERENTE AO DESPACHO 8.6 PUBLICADO NA RPI 2276 DE 19/08/2014.