BRPI0416882A - composto, composição farmacêutica, método de tratar um distúrbio, e, uso de um composto - Google Patents

composto, composição farmacêutica, método de tratar um distúrbio, e, uso de um composto

Info

Publication number
BRPI0416882A
BRPI0416882A BRPI0416882-8A BRPI0416882A BRPI0416882A BR PI0416882 A BRPI0416882 A BR PI0416882A BR PI0416882 A BRPI0416882 A BR PI0416882A BR PI0416882 A BRPI0416882 A BR PI0416882A
Authority
BR
Brazil
Prior art keywords
compound
pharmaceutical composition
formula
treating
disorder
Prior art date
Application number
BRPI0416882-8A
Other languages
English (en)
Inventor
Konstantinos Gavardinas
Jonathan Edward Green
Prabhakar Kondaji Jadhav
Donald P Matthews
Original Assignee
Lilly Co Eli
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Lilly Co Eli filed Critical Lilly Co Eli
Publication of BRPI0416882A publication Critical patent/BRPI0416882A/pt

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D235/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings
    • C07D235/02—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings condensed with carbocyclic rings or ring systems
    • C07D235/04—Benzimidazoles; Hydrogenated benzimidazoles
    • C07D235/24—Benzimidazoles; Hydrogenated benzimidazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached in position 2
    • C07D235/26—Oxygen atoms
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  • Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
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  • Chemical Kinetics & Catalysis (AREA)
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Abstract

"COMPOSTO, COMPOSIçãO FARMACêUTICA, E, USO DE UM COMPOSTO". A presente invenção proporciona um composto da fórmula (I): ou um sal farmaceuticamente aceitável do mesmo; composição farmacêutica compreendendo uma quantidade efetiva de um composto de Fórmula (I) em combinação com um veículo, diluente, ou excipiente vantajoso; e métodos para tratar distúrbios fisiológicos, particularmente doença cardíaca, hipertensão, artrite reumatóide ou inflamação, compreendendo administrar a um paciente que disto necessita uma quantidade efetiva de um composto de Fórmula (I).
BRPI0416882-8A 2003-12-19 2004-12-08 composto, composição farmacêutica, método de tratar um distúrbio, e, uso de um composto BRPI0416882A (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US53128303P 2003-12-19 2003-12-19
PCT/US2004/038233 WO2005066161A1 (en) 2003-12-19 2004-12-08 Tricyclic steroid hormone nuclear receptor modulators

Publications (1)

Publication Number Publication Date
BRPI0416882A true BRPI0416882A (pt) 2007-02-27

Family

ID=34748755

Family Applications (1)

Application Number Title Priority Date Filing Date
BRPI0416882-8A BRPI0416882A (pt) 2003-12-19 2004-12-08 composto, composição farmacêutica, método de tratar um distúrbio, e, uso de um composto

Country Status (21)

Country Link
US (1) US7803814B2 (pt)
EP (1) EP1697350B1 (pt)
JP (1) JP4846596B2 (pt)
CN (1) CN1918151A (pt)
AR (1) AR046951A1 (pt)
AT (1) ATE399163T1 (pt)
AU (1) AU2004312293A1 (pt)
BR (1) BRPI0416882A (pt)
CA (1) CA2549053C (pt)
CY (1) CY1108309T1 (pt)
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PT1697350E (pt) 2008-09-18
AU2004312293A1 (en) 2005-07-21
PL1697350T3 (pl) 2008-11-28
CN1918151A (zh) 2007-02-21
WO2005066161A1 (en) 2005-07-21
ES2308296T3 (es) 2008-12-01
CA2549053A1 (en) 2005-07-21
DK1697350T3 (da) 2008-10-13
NO20063329L (no) 2006-09-14
EP1697350A1 (en) 2006-09-06
CA2549053C (en) 2012-08-28
SI1697350T1 (sl) 2008-12-31
AR046951A1 (es) 2006-01-04
US20070037788A1 (en) 2007-02-15
DE602004014640D1 (de) 2008-08-07
EP1697350B1 (en) 2008-06-25
JP2007515431A (ja) 2007-06-14
MXPA06007055A (es) 2007-01-30
IL175996A0 (en) 2006-10-05
ATE399163T1 (de) 2008-07-15
CY1108309T1 (el) 2014-02-12
US7803814B2 (en) 2010-09-28
JP4846596B2 (ja) 2011-12-28

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