BRPI0417117A - temozolomida cristalizada, processo de preparação de temozolomida cristalizada, composição farmacêutica, método de produção de medicamento contendo temozolomida e método de tratamento de uma condição médica para a qual a termozolomida é benéfica - Google Patents
temozolomida cristalizada, processo de preparação de temozolomida cristalizada, composição farmacêutica, método de produção de medicamento contendo temozolomida e método de tratamento de uma condição médica para a qual a termozolomida é benéficaInfo
- Publication number
- BRPI0417117A BRPI0417117A BRPI0417117-9A BRPI0417117A BRPI0417117A BR PI0417117 A BRPI0417117 A BR PI0417117A BR PI0417117 A BRPI0417117 A BR PI0417117A BR PI0417117 A BRPI0417117 A BR PI0417117A
- Authority
- BR
- Brazil
- Prior art keywords
- temozolomide
- crystallized
- beneficial
- pharmaceutical composition
- preparation process
- Prior art date
Links
- BPEGJWRSRHCHSN-UHFFFAOYSA-N Temozolomide Chemical compound O=C1N(C)N=NC2=C(C(N)=O)N=CN21 BPEGJWRSRHCHSN-UHFFFAOYSA-N 0.000 title abstract 8
- 229960004964 temozolomide Drugs 0.000 title abstract 8
- 238000000034 method Methods 0.000 title abstract 4
- 238000002360 preparation method Methods 0.000 title abstract 3
- 230000009286 beneficial effect Effects 0.000 title abstract 2
- 239000003814 drug Substances 0.000 title abstract 2
- 239000008194 pharmaceutical composition Substances 0.000 title abstract 2
- 229940079593 drug Drugs 0.000 abstract 1
- 238000004519 manufacturing process Methods 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
"TEMOZOLOMIDA CRISTALIZADA, PROCESSO DE PREPARAçãO DE TEMOZOLOMIDA CRISTALIZADA, COMPOSIçãO FARMACêUTICA, MéTODO DE PRODUçãO DE MEDICAMENTO CONTENDO TEMOZOLOMIDA E MéTODO DE TRATAMENTO DE UMA CONDIçãO MéDICA PARA A QUAL A TEMOZOLOMIDA é BENéFICA". Prevê, novas formas cristalinas de Temozolomida, métodos de preparação das mesmas, medicamentos incluindo as novas formas cristalinas de Temozolomida, e usos das mesmas no tratamento de condições médicas.
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US53294403P | 2003-12-30 | 2003-12-30 | |
| PCT/IL2004/001189 WO2005063757A2 (en) | 2003-12-30 | 2004-12-30 | Novel crystalline forms of temozolomide |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| BRPI0417117A true BRPI0417117A (pt) | 2007-03-06 |
Family
ID=34738847
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| BRPI0417117-9A BRPI0417117A (pt) | 2003-12-30 | 2004-12-30 | temozolomida cristalizada, processo de preparação de temozolomida cristalizada, composição farmacêutica, método de produção de medicamento contendo temozolomida e método de tratamento de uma condição médica para a qual a termozolomida é benéfica |
Country Status (5)
| Country | Link |
|---|---|
| US (2) | US7615632B2 (pt) |
| EP (2) | EP1706407A2 (pt) |
| BR (1) | BRPI0417117A (pt) |
| CA (1) | CA2552095A1 (pt) |
| WO (1) | WO2005063757A2 (pt) |
Families Citing this family (9)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| BRPI0417117A (pt) * | 2003-12-30 | 2007-03-06 | Chemagis Ltd | temozolomida cristalizada, processo de preparação de temozolomida cristalizada, composição farmacêutica, método de produção de medicamento contendo temozolomida e método de tratamento de uma condição médica para a qual a termozolomida é benéfica |
| DE102006007309B4 (de) | 2005-02-17 | 2012-11-29 | Chemagis Ltd. | Verbessertes Verfahren zur Herstellung von Temozolomid |
| WO2008111092A1 (en) * | 2007-03-09 | 2008-09-18 | Fresenius Kabi Oncology Limited | Crystalline temozolomide monohydrate and process for preparation thereof |
| EP2509421B1 (en) | 2009-12-10 | 2020-02-05 | Cedars-Sinai Medical Center | Drug delivery of temozolomide for systemic based treatment of cancer |
| US9623041B2 (en) | 2010-12-30 | 2017-04-18 | Cedars-Sinai Medical Center | Polymalic acid-based nanobiopolymer compositions |
| CN102329319B (zh) * | 2011-07-19 | 2014-01-15 | 江苏奥赛康药业股份有限公司 | 替莫唑胺的晶型、其制备方法及其药用组合物 |
| ES2827312T3 (es) * | 2013-10-29 | 2021-05-20 | Jiangsu Tasly Diyi Pharmaceutical Co Ltd | Las formas cristalinas de temozolomida y el método para preparar las mismas |
| DK3613436T3 (da) | 2018-12-13 | 2021-06-21 | Orphelia Pharma | Oral suspension af temozolomid |
| CN116655640A (zh) * | 2023-05-31 | 2023-08-29 | 南通大学 | 替莫唑胺晶体及其制备方法 |
Family Cites Families (15)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4418208A (en) * | 1980-12-29 | 1983-11-29 | E. R. Squibb & Sons, Inc. | N-Substituted iminodiacetic acids |
| US5260291A (en) | 1981-08-24 | 1993-11-09 | Cancer Research Campaign Technology Limited | Tetrazine derivatives |
| OA07174A (fr) * | 1981-08-24 | 1984-04-30 | May & Baker Ltd | Nouvelles imidazotétrazionones, leur préparation et les médicaments qui les contiennent. |
| DE3568549D1 (en) * | 1984-09-06 | 1989-04-13 | Fujimori Kogyo Co Ltd | Laminated film for packaging |
| US4805001A (en) * | 1986-10-02 | 1989-02-14 | Sharp Kabushiki Kaisha | Magnification converting mechanism for a variable magnification copying apparatus |
| US4731053A (en) * | 1986-12-23 | 1988-03-15 | Merck & Co., Inc. | Container device for separately storing and mixing two ingredients |
| US6858631B1 (en) | 1999-11-29 | 2005-02-22 | Merck & Co., Inc. | Polymorphic, amorphous and hydrated forms of 5-chloro-3-(4-methanesulfonylphenyl)-6′-methyl-[2,3′]bipyridinyl |
| US20040223951A1 (en) | 2000-01-24 | 2004-11-11 | Schering Corporation | Combination therapy for cancer |
| US6346596B1 (en) * | 2000-07-14 | 2002-02-12 | Valspar Corporation | Gas barrier polymer composition |
| CA2434300A1 (en) | 2001-01-18 | 2002-07-25 | Schering Corporation | Synthesis of temozolomide and analogs |
| CA2434308C (en) | 2001-01-18 | 2010-09-21 | Schering Corporation | Synthesis of temozolomide and analogs |
| US20040226852A1 (en) * | 2003-02-19 | 2004-11-18 | Michael Pesachovich | Method of stabilizing azithromycin |
| US6874938B2 (en) * | 2002-04-22 | 2005-04-05 | S.C. Johnson Home Storage, Inc. | Jacketed reclosable container |
| BRPI0417117A (pt) | 2003-12-30 | 2007-03-06 | Chemagis Ltd | temozolomida cristalizada, processo de preparação de temozolomida cristalizada, composição farmacêutica, método de produção de medicamento contendo temozolomida e método de tratamento de uma condição médica para a qual a termozolomida é benéfica |
| DE102006007309B4 (de) * | 2005-02-17 | 2012-11-29 | Chemagis Ltd. | Verbessertes Verfahren zur Herstellung von Temozolomid |
-
2004
- 2004-12-30 BR BRPI0417117-9A patent/BRPI0417117A/pt not_active IP Right Cessation
- 2004-12-30 CA CA002552095A patent/CA2552095A1/en not_active Abandoned
- 2004-12-30 WO PCT/IL2004/001189 patent/WO2005063757A2/en not_active Ceased
- 2004-12-30 EP EP04806720A patent/EP1706407A2/en not_active Ceased
- 2004-12-30 US US11/024,443 patent/US7615632B2/en not_active Expired - Fee Related
- 2004-12-30 EP EP10177879A patent/EP2275425A1/en not_active Withdrawn
-
2009
- 2009-08-12 US US12/539,917 patent/US20100022609A1/en not_active Abandoned
Also Published As
| Publication number | Publication date |
|---|---|
| US20100022609A1 (en) | 2010-01-28 |
| WO2005063757A3 (en) | 2005-09-09 |
| EP1706407A2 (en) | 2006-10-04 |
| US20050187206A1 (en) | 2005-08-25 |
| CA2552095A1 (en) | 2005-07-14 |
| WO2005063757A2 (en) | 2005-07-14 |
| EP2275425A1 (en) | 2011-01-19 |
| US7615632B2 (en) | 2009-11-10 |
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| IL226313A0 (en) | A method for producing gamma-carboxylated human prothrombin, isolated prothrombin produced by such a method, a pharmaceutical preparation including it and its use as drugs and for the production of drugs for the treatment of blood coagulation | |
| BRPI0406592A (pt) | Usos de n-desmetilclozapina, métodos para o tratamento de psicose, de distúrbios afetivos, de demência, de dor neuropática e de glaucoma e composição farmacêutica | |
| YU35503A (sh) | Nove kompozicije lekova bazirane na solima tiotropijuma i solima salmeterola | |
| DE50102490D1 (de) | Verwendung von substituierten imidazo [1,2-a]pyridin-, -pyrimidin- und -pyrazin-3-yl-amin-derivaten zur herstellung von medikamenten zur nos-inhibierung | |
| HUP0301022A2 (hu) | Tiotropinium-bromid-monohidrát, eljárás előállítására és alkalmazása gyógyszerkészítmény előállítására | |
| BRPI0210941B8 (pt) | produto farmacêutico contendo combinações de oxazolidinonas substituídas, seu uso, seu processo de produção, e medicamento | |
| TW200501983A (en) | Uses of anti-insulin-like growth factor I receptor antibodies | |
| BRPI0413393A (pt) | fexofenadina, composição farmaceuticamente aceitável, método de tratamento antihistamìnico, composição, processo para preparar fexofenadina e uso de fexofenadina | |
| CY1108401T1 (el) | Παραγωγα πυρρολοϊμιδαζολης, η παρασκευη τους, φαρμακευτικες συνθεσεις που τα περιεχουν και η χρηση τους ως νοοτροπικων παραγοντων | |
| ATE353645T1 (de) | Verwendung von 2-oxo-1-pyrrolidin-derivaten zur herstellung eines arzneimittels zur behandlung von dyskinesia | |
| ATE526015T1 (de) | Arzneimittel sowie deren herstellung und verwendung bei der behandlung von schmerzhaften neuropathien | |
| RU2006143659A (ru) | Применение ребоксетина для лечения боли | |
| ATE311866T1 (de) | Verwendung von r-arylpropionsäuren zur herstellung von arzneimitteln zur behandlung von erkrankungen rheumatischer natur | |
| BR0116653A (pt) | Medicamento contendo uma poliamina como substância ativa | |
| UA89753C2 (ru) | Применение модафинила и антидепрессанта при лечении депрессии и для сокращения времени до начала действия антидепрессанта | |
| MX9304365A (es) | Una forma de dosis osmotica para administrar tandospirona. | |
| NZ594154A (en) | Transdermal administration of buprenorphine for preoperative treatment of post operative pain | |
| TW200505830A (en) | Cycloalkyl-substituted alkanoic acid derivatives, processes for their preparation and their use as pharmaceuticals | |
| DE602004016754D1 (de) | Kombinationstherapie gegen krebserkrankungen mit azd2171 und zd1839 | |
| WO2005063757A3 (en) | Novel crystalline forms of temozolomide | |
| EE200200549A (et) | Jagatud doosi teraapia veresooni kahjustava aktiivsusega | |
| RU2006126294A (ru) | Способ лечения больных с хроническими формами периодонтитов и периодонтитов в стадии обострения | |
| ATE462706T1 (de) | 7h-pyrroloä2,3-düpyrimidinderivate sowie deren therapeutisch annehmbare salze, pharmazeutische zubereitungen, die diese enthalten, und verfahren zur herstellung des wirkstoffs | |
| RU2853936C1 (ru) | Способ получения биологически активной композиции для общеукрепляющих ванн | |
| BRPI0417797A (pt) | soro sangüìneo biologicamente ativo, métodos para produzi-lo e seus usos |
Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| B06F | Objections, documents and/or translations needed after an examination request according [chapter 6.6 patent gazette] | ||
| B08L | Patent application lapsed because of non payment of annual fee [chapter 8.12 patent gazette] |
Free format text: REFERENTE AO NAO RECOLHIMENTO DAS 8A E 9A ANUIDADES. |
|
| B08I | Publication cancelled [chapter 8.9 patent gazette] |
Free format text: ANULADA A PUBLICACAO CODIGO 8.12 NA RPI NO 2259 DE 22/04/2014 POR TER SIDO INDEVIDA. |
|
| B08F | Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette] |
Free format text: REFERENTE AS 8A, 9A, 10A, 11A, 12A, 13A, 14A E 15A ANUIDADES. |
|
| B08K | Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette] |
Free format text: EM VIRTUDE DO ARQUIVAMENTO PUBLICADO NA RPI 2602 DE 17-11-2020 E CONSIDERANDO AUSENCIA DE MANIFESTACAO DENTRO DOS PRAZOS LEGAIS, INFORMO QUE CABE SER MANTIDO O ARQUIVAMENTO DO PEDIDO DE PATENTE, CONFORME O DISPOSTO NO ARTIGO 12, DA RESOLUCAO 113/2013. |