BRPI0417117A - temozolomida cristalizada, processo de preparação de temozolomida cristalizada, composição farmacêutica, método de produção de medicamento contendo temozolomida e método de tratamento de uma condição médica para a qual a termozolomida é benéfica - Google Patents

temozolomida cristalizada, processo de preparação de temozolomida cristalizada, composição farmacêutica, método de produção de medicamento contendo temozolomida e método de tratamento de uma condição médica para a qual a termozolomida é benéfica

Info

Publication number
BRPI0417117A
BRPI0417117A BRPI0417117-9A BRPI0417117A BRPI0417117A BR PI0417117 A BRPI0417117 A BR PI0417117A BR PI0417117 A BRPI0417117 A BR PI0417117A BR PI0417117 A BRPI0417117 A BR PI0417117A
Authority
BR
Brazil
Prior art keywords
temozolomide
crystallized
beneficial
pharmaceutical composition
preparation process
Prior art date
Application number
BRPI0417117-9A
Other languages
English (en)
Inventor
Itai Adin
Carmen Iustain
Original Assignee
Chemagis Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Chemagis Ltd filed Critical Chemagis Ltd
Publication of BRPI0417117A publication Critical patent/BRPI0417117A/pt

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

"TEMOZOLOMIDA CRISTALIZADA, PROCESSO DE PREPARAçãO DE TEMOZOLOMIDA CRISTALIZADA, COMPOSIçãO FARMACêUTICA, MéTODO DE PRODUçãO DE MEDICAMENTO CONTENDO TEMOZOLOMIDA E MéTODO DE TRATAMENTO DE UMA CONDIçãO MéDICA PARA A QUAL A TEMOZOLOMIDA é BENéFICA". Prevê, novas formas cristalinas de Temozolomida, métodos de preparação das mesmas, medicamentos incluindo as novas formas cristalinas de Temozolomida, e usos das mesmas no tratamento de condições médicas.
BRPI0417117-9A 2003-12-30 2004-12-30 temozolomida cristalizada, processo de preparação de temozolomida cristalizada, composição farmacêutica, método de produção de medicamento contendo temozolomida e método de tratamento de uma condição médica para a qual a termozolomida é benéfica BRPI0417117A (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US53294403P 2003-12-30 2003-12-30
PCT/IL2004/001189 WO2005063757A2 (en) 2003-12-30 2004-12-30 Novel crystalline forms of temozolomide

Publications (1)

Publication Number Publication Date
BRPI0417117A true BRPI0417117A (pt) 2007-03-06

Family

ID=34738847

Family Applications (1)

Application Number Title Priority Date Filing Date
BRPI0417117-9A BRPI0417117A (pt) 2003-12-30 2004-12-30 temozolomida cristalizada, processo de preparação de temozolomida cristalizada, composição farmacêutica, método de produção de medicamento contendo temozolomida e método de tratamento de uma condição médica para a qual a termozolomida é benéfica

Country Status (5)

Country Link
US (2) US7615632B2 (pt)
EP (2) EP1706407A2 (pt)
BR (1) BRPI0417117A (pt)
CA (1) CA2552095A1 (pt)
WO (1) WO2005063757A2 (pt)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
BRPI0417117A (pt) * 2003-12-30 2007-03-06 Chemagis Ltd temozolomida cristalizada, processo de preparação de temozolomida cristalizada, composição farmacêutica, método de produção de medicamento contendo temozolomida e método de tratamento de uma condição médica para a qual a termozolomida é benéfica
DE102006007309B4 (de) 2005-02-17 2012-11-29 Chemagis Ltd. Verbessertes Verfahren zur Herstellung von Temozolomid
WO2008111092A1 (en) * 2007-03-09 2008-09-18 Fresenius Kabi Oncology Limited Crystalline temozolomide monohydrate and process for preparation thereof
EP2509421B1 (en) 2009-12-10 2020-02-05 Cedars-Sinai Medical Center Drug delivery of temozolomide for systemic based treatment of cancer
US9623041B2 (en) 2010-12-30 2017-04-18 Cedars-Sinai Medical Center Polymalic acid-based nanobiopolymer compositions
CN102329319B (zh) * 2011-07-19 2014-01-15 江苏奥赛康药业股份有限公司 替莫唑胺的晶型、其制备方法及其药用组合物
ES2827312T3 (es) * 2013-10-29 2021-05-20 Jiangsu Tasly Diyi Pharmaceutical Co Ltd Las formas cristalinas de temozolomida y el método para preparar las mismas
DK3613436T3 (da) 2018-12-13 2021-06-21 Orphelia Pharma Oral suspension af temozolomid
CN116655640A (zh) * 2023-05-31 2023-08-29 南通大学 替莫唑胺晶体及其制备方法

Family Cites Families (15)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4418208A (en) * 1980-12-29 1983-11-29 E. R. Squibb & Sons, Inc. N-Substituted iminodiacetic acids
US5260291A (en) 1981-08-24 1993-11-09 Cancer Research Campaign Technology Limited Tetrazine derivatives
OA07174A (fr) * 1981-08-24 1984-04-30 May & Baker Ltd Nouvelles imidazotétrazionones, leur préparation et les médicaments qui les contiennent.
DE3568549D1 (en) * 1984-09-06 1989-04-13 Fujimori Kogyo Co Ltd Laminated film for packaging
US4805001A (en) * 1986-10-02 1989-02-14 Sharp Kabushiki Kaisha Magnification converting mechanism for a variable magnification copying apparatus
US4731053A (en) * 1986-12-23 1988-03-15 Merck & Co., Inc. Container device for separately storing and mixing two ingredients
US6858631B1 (en) 1999-11-29 2005-02-22 Merck & Co., Inc. Polymorphic, amorphous and hydrated forms of 5-chloro-3-(4-methanesulfonylphenyl)-6′-methyl-[2,3′]bipyridinyl
US20040223951A1 (en) 2000-01-24 2004-11-11 Schering Corporation Combination therapy for cancer
US6346596B1 (en) * 2000-07-14 2002-02-12 Valspar Corporation Gas barrier polymer composition
CA2434300A1 (en) 2001-01-18 2002-07-25 Schering Corporation Synthesis of temozolomide and analogs
CA2434308C (en) 2001-01-18 2010-09-21 Schering Corporation Synthesis of temozolomide and analogs
US20040226852A1 (en) * 2003-02-19 2004-11-18 Michael Pesachovich Method of stabilizing azithromycin
US6874938B2 (en) * 2002-04-22 2005-04-05 S.C. Johnson Home Storage, Inc. Jacketed reclosable container
BRPI0417117A (pt) 2003-12-30 2007-03-06 Chemagis Ltd temozolomida cristalizada, processo de preparação de temozolomida cristalizada, composição farmacêutica, método de produção de medicamento contendo temozolomida e método de tratamento de uma condição médica para a qual a termozolomida é benéfica
DE102006007309B4 (de) * 2005-02-17 2012-11-29 Chemagis Ltd. Verbessertes Verfahren zur Herstellung von Temozolomid

Also Published As

Publication number Publication date
US20100022609A1 (en) 2010-01-28
WO2005063757A3 (en) 2005-09-09
EP1706407A2 (en) 2006-10-04
US20050187206A1 (en) 2005-08-25
CA2552095A1 (en) 2005-07-14
WO2005063757A2 (en) 2005-07-14
EP2275425A1 (en) 2011-01-19
US7615632B2 (en) 2009-11-10

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Legal Events

Date Code Title Description
B06F Objections, documents and/or translations needed after an examination request according [chapter 6.6 patent gazette]
B08L Patent application lapsed because of non payment of annual fee [chapter 8.12 patent gazette]

Free format text: REFERENTE AO NAO RECOLHIMENTO DAS 8A E 9A ANUIDADES.

B08I Publication cancelled [chapter 8.9 patent gazette]

Free format text: ANULADA A PUBLICACAO CODIGO 8.12 NA RPI NO 2259 DE 22/04/2014 POR TER SIDO INDEVIDA.

B08F Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette]

Free format text: REFERENTE AS 8A, 9A, 10A, 11A, 12A, 13A, 14A E 15A ANUIDADES.

B08K Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette]

Free format text: EM VIRTUDE DO ARQUIVAMENTO PUBLICADO NA RPI 2602 DE 17-11-2020 E CONSIDERANDO AUSENCIA DE MANIFESTACAO DENTRO DOS PRAZOS LEGAIS, INFORMO QUE CABE SER MANTIDO O ARQUIVAMENTO DO PEDIDO DE PATENTE, CONFORME O DISPOSTO NO ARTIGO 12, DA RESOLUCAO 113/2013.