BRPI0501708A - dispositivo de liberação lenta por processo transdérmico de um medicamento contra o excesso de colesterol e método de produção de um dispositivo transdérmico - Google Patents
dispositivo de liberação lenta por processo transdérmico de um medicamento contra o excesso de colesterol e método de produção de um dispositivo transdérmicoInfo
- Publication number
- BRPI0501708A BRPI0501708A BRPI0501708A BRPI0501708A BR PI0501708 A BRPI0501708 A BR PI0501708A BR PI0501708 A BRPI0501708 A BR PI0501708A BR PI0501708 A BRPI0501708 A BR PI0501708A
- Authority
- BR
- Brazil
- Prior art keywords
- transdermal
- slow
- producing
- release device
- excess
- Prior art date
Links
- HVYWMOMLDIMFJA-DPAQBDIFSA-N cholesterol Chemical compound C1C=C2C[C@@H](O)CC[C@]2(C)[C@@H]2[C@@H]1[C@@H]1CC[C@H]([C@H](C)CCCC(C)C)[C@@]1(C)CC2 HVYWMOMLDIMFJA-DPAQBDIFSA-N 0.000 title abstract 6
- 235000012000 cholesterol Nutrition 0.000 title abstract 3
- 238000000034 method Methods 0.000 title abstract 2
- 239000003814 drug Substances 0.000 title 1
- 229940079593 drug Drugs 0.000 title 1
- 239000011159 matrix material Substances 0.000 abstract 2
- 229940121710 HMGCoA reductase inhibitor Drugs 0.000 abstract 1
- 238000004519 manufacturing process Methods 0.000 abstract 1
- 229940126601 medicinal product Drugs 0.000 abstract 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/70—Web, sheet or filament bases ; Films; Fibres of the matrix type containing drug
- A61K9/7023—Transdermal patches and similar drug-containing composite devices, e.g. cataplasms
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/185—Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
- A61K31/19—Carboxylic acids, e.g. valproic acid
- A61K31/20—Carboxylic acids, e.g. valproic acid having a carboxyl group bound to a chain of seven or more carbon atoms, e.g. stearic, palmitic, arachidic acids
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Dermatology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicinal Preparation (AREA)
Abstract
DIPOSITIVO DE LIBERAçãO LENTA POR PROCESSO TRANSDéRMICO DE UM MEDICAMENTO CONTRA O EXECESSO DE COLESTEROL E MéTODO DE PRODUçãO DE UM DISPOSITIVO TRANSDéRMICO,o qual é caracterizado por prever um dispositivo bi-laminar,leberação lenta transdérmica constituída de uma matriz macromolecular flexível (2) de uma espessura de 0,15 0, 6 cm e de uma superfície entre 10 e 100 cm quadrados e apresentando de um lado um revestimento posterior (1), permitindo uma redução considerável (mais de 15 vezes) das doses diárias a serem asministradas no tratamento do excesso de colesterol,a matriz macromolecular contendo e liberando de maneira contínua durante um período de 1 a 4 meses 0, 05 a 18% por dias de seu peso total em ómega 3 e/ou estatina,pela superfície em contato com a pele do paciente sem precisar aderir de forma fixa e permanente à pele do mesmo.
Priority Applications (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| BRPI0501708 BRPI0501708A (pt) | 2005-05-10 | 2005-05-10 | dispositivo de liberação lenta por processo transdérmico de um medicamento contra o excesso de colesterol e método de produção de um dispositivo transdérmico |
| PCT/BR2006/000090 WO2006119598A2 (en) | 2005-05-10 | 2006-05-10 | Transdermal device for the slow delivery of an omega-3-fatty acid, optionally in combination with a hmg coa reductase inhibitor |
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| BRPI0501708 BRPI0501708A (pt) | 2005-05-10 | 2005-05-10 | dispositivo de liberação lenta por processo transdérmico de um medicamento contra o excesso de colesterol e método de produção de um dispositivo transdérmico |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| BRPI0501708A true BRPI0501708A (pt) | 2007-05-02 |
Family
ID=37396906
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| BRPI0501708 BRPI0501708A (pt) | 2005-05-10 | 2005-05-10 | dispositivo de liberação lenta por processo transdérmico de um medicamento contra o excesso de colesterol e método de produção de um dispositivo transdérmico |
Country Status (2)
| Country | Link |
|---|---|
| BR (1) | BRPI0501708A (pt) |
| WO (1) | WO2006119598A2 (pt) |
Families Citing this family (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| FR2940116B1 (fr) | 2008-12-22 | 2012-07-06 | Philippe Perovitch | Formulation pour l'administration d'hypolipemiant par voie trans-muqueuse buccale |
| US9107983B2 (en) | 2010-10-27 | 2015-08-18 | Warsaw Orthopedic, Inc. | Osteoconductive matrices comprising statins |
| US8877221B2 (en) | 2010-10-27 | 2014-11-04 | Warsaw Orthopedic, Inc. | Osteoconductive matrices comprising calcium phosphate particles and statins and methods of using the same |
| WO2012170417A2 (en) | 2011-06-06 | 2012-12-13 | Warsaw Orthopedic, Inc. | Methods and compositions to enhance bone growth comprising a statin |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| FR2548021B1 (fr) * | 1983-06-29 | 1986-02-28 | Dick P R | Compositions pharmaceutiques dermiques a action prolongee et continue a base d'acides gras essentiels |
| JP4062639B2 (ja) * | 1996-12-23 | 2008-03-19 | 日本水産株式会社 | 皮膚外用剤 |
| DE10056010A1 (de) * | 2000-11-11 | 2002-05-16 | Beiersdorf Ag | Pflaster mit hautpflegenden Substanzen |
-
2005
- 2005-05-10 BR BRPI0501708 patent/BRPI0501708A/pt not_active Application Discontinuation
-
2006
- 2006-05-10 WO PCT/BR2006/000090 patent/WO2006119598A2/en not_active Ceased
Also Published As
| Publication number | Publication date |
|---|---|
| WO2006119598A3 (en) | 2007-03-01 |
| WO2006119598A2 (en) | 2006-11-16 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| B11A | Dismissal acc. art.33 of ipl - examination not requested within 36 months of filing | ||
| B11Y | Definitive dismissal acc. article 33 of ipl - extension of time limit for request of examination expired |