BRPI0507628A - composto ou sal farmaceuticamente aceitável do mesmo, método de tratamento de uma infecção viral em um ser humano, uso de um composto composição farmacêutica, e, processo para a preparação de um composto - Google Patents
composto ou sal farmaceuticamente aceitável do mesmo, método de tratamento de uma infecção viral em um ser humano, uso de um composto composição farmacêutica, e, processo para a preparação de um compostoInfo
- Publication number
- BRPI0507628A BRPI0507628A BRPI0507628-5A BRPI0507628A BRPI0507628A BR PI0507628 A BRPI0507628 A BR PI0507628A BR PI0507628 A BRPI0507628 A BR PI0507628A BR PI0507628 A BRPI0507628 A BR PI0507628A
- Authority
- BR
- Brazil
- Prior art keywords
- compound
- treating
- preparing
- human
- pharmaceutically acceptable
- Prior art date
Links
- 150000001875 compounds Chemical class 0.000 title abstract 7
- 208000036142 Viral infection Diseases 0.000 title abstract 2
- 238000004519 manufacturing process Methods 0.000 title abstract 2
- 238000000034 method Methods 0.000 title abstract 2
- 239000008194 pharmaceutical composition Substances 0.000 title abstract 2
- 150000003839 salts Chemical class 0.000 title abstract 2
- 230000009385 viral infection Effects 0.000 title abstract 2
- 208000030507 AIDS Diseases 0.000 abstract 1
- 208000031886 HIV Infections Diseases 0.000 abstract 1
- 208000037357 HIV infectious disease Diseases 0.000 abstract 1
- 208000033519 human immunodeficiency virus infectious disease Diseases 0.000 abstract 1
- 239000003112 inhibitor Substances 0.000 abstract 1
- 230000002401 inhibitory effect Effects 0.000 abstract 1
- 230000010076 replication Effects 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
- A61P31/14—Antivirals for RNA viruses
- A61P31/18—Antivirals for RNA viruses for HIV
Landscapes
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Virology (AREA)
- General Chemical & Material Sciences (AREA)
- Veterinary Medicine (AREA)
- Oncology (AREA)
- Communicable Diseases (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Health & Medical Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- AIDS & HIV (AREA)
- Tropical Medicine & Parasitology (AREA)
- Molecular Biology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Abstract
COMPOSTO OU UM SAL FARMACEUTICAMENTE ACEITáVEL DO MESMO, MéTODO DE TRATAMENTO DE UMA INFECçãO VIRAL EM UM SER HUMANO, USO DE UM COMPOSTO, COMPOSIçãO FARMACêUTICA, E, PROCESSO PARA A PREPARAçãO DE UM COMPOSTO A presente invenção apresenta compostos que são inibidores de integrase do HIV e, portanto, são úteis na inibição da replicação do HIV, na prevenção e/ou no tratamento de infecção por HIV, e no tratamento de AIDS e/ou ARC.
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US54367004P | 2004-02-11 | 2004-02-11 | |
| PCT/US2005/004085 WO2005077050A2 (en) | 2004-02-11 | 2005-02-10 | Hiv integrase inhibitors |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| BRPI0507628A true BRPI0507628A (pt) | 2007-07-03 |
Family
ID=34860447
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| BRPI0507628-5A BRPI0507628A (pt) | 2004-02-11 | 2005-02-10 | composto ou sal farmaceuticamente aceitável do mesmo, método de tratamento de uma infecção viral em um ser humano, uso de um composto composição farmacêutica, e, processo para a preparação de um composto |
Country Status (15)
| Country | Link |
|---|---|
| US (3) | US8691991B2 (pt) |
| EP (1) | EP1720856B1 (pt) |
| JP (1) | JP4859676B2 (pt) |
| KR (1) | KR20070002006A (pt) |
| CN (1) | CN1976915A (pt) |
| AU (1) | AU2005211733A1 (pt) |
| BR (1) | BRPI0507628A (pt) |
| CA (1) | CA2555176A1 (pt) |
| ES (1) | ES2433477T3 (pt) |
| IL (1) | IL177189A0 (pt) |
| MA (1) | MA28358A1 (pt) |
| MX (1) | MXPA06009132A (pt) |
| NO (1) | NO20063958L (pt) |
| RU (1) | RU2006128848A (pt) |
| WO (1) | WO2005077050A2 (pt) |
Families Citing this family (33)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP1720856B1 (en) | 2004-02-11 | 2013-08-14 | GlaxoSmithKline LLC | Hiv integrase inhibitors |
| PT1874117E (pt) | 2005-04-28 | 2013-10-17 | Shionogi & Co | Derivado policíclico de carbamoílpiridona possuindo actividade inibidora de hiv-integrasse |
| EP1910363A4 (en) * | 2005-08-04 | 2010-05-26 | Glaxosmithkline Llc | INHIBITORS OF HIV INTEGRASE |
| WO2007019130A2 (en) * | 2005-08-04 | 2007-02-15 | Smithkline Beecham Corporation | Hiv integrase inhibitors |
| JP2009503083A (ja) * | 2005-08-04 | 2009-01-29 | スミスクライン ビーチャム コーポレーション | Hivインテグラーゼ阻害薬 |
| US20080194523A1 (en) * | 2005-08-04 | 2008-08-14 | Smithkline Beecham Corporation | Hiv Integrase Inhibitors |
| AR059733A1 (es) * | 2006-03-07 | 2008-04-23 | Smithkline Beecham Corp | Compuesto derivado de glicina n- sustituida con heteroaromaticos bicicicos, composicion farmaceutica que lo comprende, uso para preparar un medicamento para tratar la anemia y proceso para su preparacion |
| MX2008014908A (es) | 2006-05-26 | 2009-05-13 | Toyama Chemical Co Ltd | Compuesto heterociclico nuevo o sal del mismo e intermedio del mismo. |
| EP1956016A1 (en) * | 2006-12-15 | 2008-08-13 | Bayer Schering Pharma Aktiengesellschaft | Bicyclic acyltryptophanols |
| EP2111399A2 (en) | 2006-12-18 | 2009-10-28 | Amgen Inc. | Naphthalenone compounds exhibiting prolyl hydroxylase inhibitory activity, compositions, and uses thereof |
| ES2393326T3 (es) | 2006-12-18 | 2012-12-20 | Amgen, Inc | Compuestos basados en azaquinolona que presentan actividad inhibidora de prolil hidroxilasas, composiciones y usos de los mismos |
| ES2446418T3 (es) | 2007-04-18 | 2014-03-07 | Amgen, Inc | Derivados de indanona que inhiben la prolil hidroxilasa |
| EP2142509B1 (en) | 2007-04-18 | 2013-12-04 | Amgen, Inc | Quinolones and azaquinolones that inhibit prolyl hydroxylase |
| AU2008241503A1 (en) * | 2007-04-18 | 2008-10-30 | Merck Sharp & Dohme Corp. | Novel 1,8-naphthyridine compounds |
| WO2008137084A2 (en) | 2007-05-04 | 2008-11-13 | Amgen Inc. | Diazaquinolones that inhibit prolyl hydroxylase activity |
| US8030346B2 (en) | 2007-05-04 | 2011-10-04 | Amgen Inc. | Heterocyclic quinolone derivatives that inhibit prolyl hydroxylase activity |
| WO2010011818A1 (en) * | 2008-07-25 | 2010-01-28 | Smithkline Beecham Corporation | Chemical compounds |
| WO2010011819A1 (en) * | 2008-07-25 | 2010-01-28 | Smithkline Beecham Corporation | Chemical compounds |
| US8283366B2 (en) | 2010-01-22 | 2012-10-09 | Ambrilia Biopharma, Inc. | Derivatives of pyridoxine for inhibiting HIV integrase |
| UA105556C2 (uk) * | 2010-01-27 | 2014-05-26 | Віів Гелскер Компані | Комбінація сполук, що містить інгібітори віл інтегрази з іншими терапевтичними агентами |
| US20110223131A1 (en) * | 2010-02-24 | 2011-09-15 | Gilead Sciences, Inc. | Antiviral compounds |
| NZ603332A (en) | 2010-04-02 | 2014-11-28 | Senomyx Inc | Sweet flavor modifier |
| KR20130065728A (ko) | 2010-10-14 | 2013-06-19 | 임뮤나르 에이비 | Ahr 활성화제로서의 1,2-디히드로-4-히드록시-2-옥소-퀴놀린-3-카르복사닐리드 |
| CA2819889C (en) | 2010-12-06 | 2020-12-15 | Confluence Life Sciences, Inc. | Substituted pyridinone-pyridinyl compounds |
| US9359300B2 (en) | 2010-12-06 | 2016-06-07 | Confluence Life Sciences, Inc. | Methyl/difluorophenyl-methoxy substituted pyridinone-pyridinyl compounds, methyl-pyridinyl-methoxy substituted pyridinone-pyridinyl compounds, and methyl-pyrimidinyl-methoxy substituted pyridinone-pyridinyl compounds |
| WO2012147763A1 (ja) | 2011-04-26 | 2012-11-01 | 塩野義製薬株式会社 | オキサジン誘導体およびそれを含有するbace1阻害剤 |
| EP2742026B1 (en) | 2011-08-12 | 2016-10-05 | Senomyx, Inc. | Sweet flavor modifier |
| CA2893843C (en) | 2012-12-21 | 2018-09-04 | Gilead Sciences, Inc. | Polycyclic-carbamoylpyridone compounds and their pharmaceutical use |
| CA2917344C (en) | 2013-06-07 | 2021-09-07 | Confluence Life Sciences, Inc. | Methyl/fluoro-pyridinyl-methoxy substituted pyridinone-pyridinyl compounds and fluoro-pyrimidinyl-methoxy substituted pyridinone-pyridinyl compounds |
| US11339128B2 (en) | 2014-11-07 | 2022-05-24 | Firmenich Incorporated | Substituted 4-amino-5-(cyclohexyloxy)quinoline-3-carboxylic acids as sweet flavor modifiers |
| CN105348282B (zh) * | 2015-12-02 | 2018-06-29 | 北京工业大学 | 一种hiv-1整合酶抑制剂化合物及其制备方法和应用 |
| BR112022019349A2 (pt) | 2020-03-27 | 2022-11-16 | Aclaris Therapeutics Inc | Forma cristalina, composição farmacêutica, comprimido e método para isolar um composto |
| US11116737B1 (en) | 2020-04-10 | 2021-09-14 | University Of Georgia Research Foundation, Inc. | Methods of using probenecid for treatment of coronavirus infections |
Family Cites Families (12)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| AU1532802A (en) | 2000-10-12 | 2002-04-22 | Merck & Co Inc | Aza- and polyaza-naphthalenyl-carboxamides useful as hiv integrase inhibitors |
| DE60124577T2 (de) | 2000-10-12 | 2007-09-27 | Merck & Co., Inc. | Aza- und polyaza-naphthalenylcarbonsäureamide als hiv-integrase-hemmer |
| WO2002036734A2 (en) | 2000-10-12 | 2002-05-10 | Merck & Co., Inc. | Aza-and polyaza-naphthalenyl ketones useful as hiv integrase inhibitors |
| ATE430745T1 (de) | 2000-10-12 | 2009-05-15 | Merck & Co Inc | Aza- und polyaza naphthalenyl karboxamide als inhibitoren der hiv-integrase |
| IL157638A0 (en) | 2001-03-01 | 2004-03-28 | Shionogi & Co | Nitrogen-containing heteroaryl compounds having hiv integrase inhibitory activity |
| ES2291642T3 (es) * | 2002-01-17 | 2008-03-01 | MERCK & CO., INC. | Hidroxinaftiridinoncarboxamidas utiles como inhibidores de la integrasa de vih. |
| DE60322920D1 (de) | 2002-08-13 | 2008-09-25 | Shionogi & Co | Heterocyclische verbindungen mit hiv-integrase-hemmender wirkung |
| EP1545538A2 (en) | 2002-08-29 | 2005-06-29 | Merck & Co., Inc. | N-biarylmethyl aminocycloalkanecarboxamide derivatives |
| TW200505902A (en) * | 2003-03-20 | 2005-02-16 | Schering Corp | Cannabinoid receptor ligands |
| WO2005023189A2 (en) | 2003-09-03 | 2005-03-17 | Pharmacia Corporation | Method of cox-2 selective inhibitor and nitric oxide-donating agent |
| WO2005028478A1 (en) | 2003-09-19 | 2005-03-31 | Gilead Sciences, Inc. | Aza-quinolinol phosphonate integrase inhibitor compounds |
| EP1720856B1 (en) | 2004-02-11 | 2013-08-14 | GlaxoSmithKline LLC | Hiv integrase inhibitors |
-
2005
- 2005-02-10 EP EP05726489.7A patent/EP1720856B1/en not_active Expired - Lifetime
- 2005-02-10 KR KR1020067018565A patent/KR20070002006A/ko not_active Withdrawn
- 2005-02-10 US US10/597,902 patent/US8691991B2/en active Active
- 2005-02-10 CN CNA2005800122898A patent/CN1976915A/zh active Pending
- 2005-02-10 AU AU2005211733A patent/AU2005211733A1/en not_active Abandoned
- 2005-02-10 CA CA002555176A patent/CA2555176A1/en not_active Abandoned
- 2005-02-10 RU RU2006128848/04A patent/RU2006128848A/ru not_active Application Discontinuation
- 2005-02-10 JP JP2006553204A patent/JP4859676B2/ja not_active Expired - Lifetime
- 2005-02-10 ES ES05726489T patent/ES2433477T3/es not_active Expired - Lifetime
- 2005-02-10 BR BRPI0507628-5A patent/BRPI0507628A/pt not_active Application Discontinuation
- 2005-02-10 MX MXPA06009132A patent/MXPA06009132A/es not_active Application Discontinuation
- 2005-02-10 WO PCT/US2005/004085 patent/WO2005077050A2/en not_active Ceased
-
2006
- 2006-08-01 IL IL177189A patent/IL177189A0/en unknown
- 2006-08-11 MA MA29263A patent/MA28358A1/fr unknown
- 2006-09-05 NO NO20063958A patent/NO20063958L/no not_active Application Discontinuation
-
2014
- 2014-02-21 US US14/186,084 patent/US20140256713A1/en not_active Abandoned
-
2015
- 2015-04-27 US US14/696,784 patent/US20150225399A1/en not_active Abandoned
Also Published As
| Publication number | Publication date |
|---|---|
| WO2005077050A3 (en) | 2006-11-23 |
| EP1720856A4 (en) | 2009-11-11 |
| JP2007523086A (ja) | 2007-08-16 |
| JP4859676B2 (ja) | 2012-01-25 |
| AU2005211733A1 (en) | 2005-08-25 |
| KR20070002006A (ko) | 2007-01-04 |
| NO20063958L (no) | 2006-09-22 |
| EP1720856B1 (en) | 2013-08-14 |
| ES2433477T3 (es) | 2013-12-11 |
| US20140256713A1 (en) | 2014-09-11 |
| CN1976915A (zh) | 2007-06-06 |
| MA28358A1 (fr) | 2006-12-01 |
| CA2555176A1 (en) | 2005-08-25 |
| US20150225399A1 (en) | 2015-08-13 |
| EP1720856A2 (en) | 2006-11-15 |
| WO2005077050A2 (en) | 2005-08-25 |
| US8691991B2 (en) | 2014-04-08 |
| IL177189A0 (en) | 2006-12-10 |
| US20070124152A1 (en) | 2007-05-31 |
| RU2006128848A (ru) | 2008-03-20 |
| MXPA06009132A (es) | 2007-03-26 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| B11A | Dismissal acc. art.33 of ipl - examination not requested within 36 months of filing | ||
| B11Y | Definitive dismissal - extension of time limit for request of examination expired [chapter 11.1.1 patent gazette] |