BRPI0509074A - composições farmacêuticas compreendendo agonistas do receptor da tiróide - Google Patents

composições farmacêuticas compreendendo agonistas do receptor da tiróide

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Publication number
BRPI0509074A
BRPI0509074A BRPI0509074-1A BRPI0509074A BRPI0509074A BR PI0509074 A BRPI0509074 A BR PI0509074A BR PI0509074 A BRPI0509074 A BR PI0509074A BR PI0509074 A BRPI0509074 A BR PI0509074A
Authority
BR
Brazil
Prior art keywords
thyroid receptor
pharmaceutical compositions
receptor agonists
amide
salt
Prior art date
Application number
BRPI0509074-1A
Other languages
English (en)
Inventor
Anna Maria Garcia Collazo
Thomas Anders Wilson Ericsson
Neeraj Garg
Anton Joakim Loefstedt
Thomas Fredrik Hansson
Original Assignee
Karobio Ab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Karobio Ab filed Critical Karobio Ab
Publication of BRPI0509074A publication Critical patent/BRPI0509074A/pt

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    • C07C311/01—Sulfonamides having sulfur atoms of sulfonamide groups bound to acyclic carbon atoms
    • C07C311/02—Sulfonamides having sulfur atoms of sulfonamide groups bound to acyclic carbon atoms of an acyclic saturated carbon skeleton
    • C07C311/08—Sulfonamides having sulfur atoms of sulfonamide groups bound to acyclic carbon atoms of an acyclic saturated carbon skeleton having the nitrogen atom of at least one of the sulfonamide groups bound to a carbon atom of a six-membered aromatic ring
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Abstract

COMPOSIçõES FARMACêUTICAS COMPREENDENDO AGONISTAS DO RECEPTOR DA TIRóIDE. A invenção fornece compostos de fórmula (I) ou um éster, amida, solvado ou sal farmaceuticamente aceitável disso, incluindo um sal de tal éster ou amida, e um solvato de tal éster, amida ou sal. A invenção também fornece o emprego de tais compostos no tratamento ou profixia de uma condição mediada por um receptor de tiróide. em que R¬ 1¬, R¬ 2¬, n Y Y', R¬ 3¬, R¬ 4¬, W e R¬ 5¬ são como definidos no relatório.
BRPI0509074-1A 2004-03-22 2005-03-22 composições farmacêuticas compreendendo agonistas do receptor da tiróide BRPI0509074A (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GBGB0406378.0A GB0406378D0 (en) 2004-03-22 2004-03-22 Novel pharmaceutical compositions
PCT/EP2005/003030 WO2005092316A1 (en) 2004-03-22 2005-03-22 Novel pharmaceutical compositions comprising agonists of the thyroid receptor

Publications (1)

Publication Number Publication Date
BRPI0509074A true BRPI0509074A (pt) 2007-08-21

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ID=32118142

Family Applications (1)

Application Number Title Priority Date Filing Date
BRPI0509074-1A BRPI0509074A (pt) 2004-03-22 2005-03-22 composições farmacêuticas compreendendo agonistas do receptor da tiróide

Country Status (12)

Country Link
US (1) US20080004251A1 (pt)
EP (1) EP1732532A1 (pt)
JP (1) JP2007529566A (pt)
KR (1) KR20060130728A (pt)
CN (1) CN1933826A (pt)
AU (1) AU2005226914A1 (pt)
BR (1) BRPI0509074A (pt)
CA (1) CA2560526A1 (pt)
GB (1) GB0406378D0 (pt)
IL (1) IL177665A0 (pt)
NO (1) NO20064705L (pt)
WO (1) WO2005092316A1 (pt)

Families Citing this family (22)

* Cited by examiner, † Cited by third party
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EP1688138A4 (en) * 2003-11-26 2008-01-16 Takeda Pharmaceutical RECEPTOR FUNCTIONAL REGULATING MEANS
FR2872159B1 (fr) * 2004-06-28 2007-10-05 Merck Sante Soc Par Actions Si Nouveaux derives acides carboxyliques phenyliques et leur utilisation dans le traitement du diabete
GB0519294D0 (en) * 2005-09-21 2005-11-02 Karobio Ab Compounds
BRPI0715160A2 (pt) 2006-08-08 2013-06-11 Sanofi Aventis imidazolidina-2,4-dionas substituÍdas por arilamimoaril-alquil-, processo para preparÁ-las, medicamentos compeendendo estes compostos, e seu uso
WO2010003624A2 (en) 2008-07-09 2010-01-14 Sanofi-Aventis Heterocyclic compounds, processes for their preparation, medicaments comprising these compounds, and the use thereof
WO2010068601A1 (en) 2008-12-08 2010-06-17 Sanofi-Aventis A crystalline heteroaromatic fluoroglycoside hydrate, processes for making, methods of use and pharmaceutical compositions thereof
DK2470552T3 (en) 2009-08-26 2014-02-17 Sanofi Sa NOVEL, CRYSTALLINE, heteroaromatic FLUORGLYCOSIDHYDRATER, MEDICINES COVERING THESE COMPOUNDS AND THEIR USE
AU2011296737A1 (en) 2010-08-31 2013-04-11 Snu R&Db Foundation Use of the fetal reprogramming of a PPAR delta agonist
WO2012120056A1 (de) 2011-03-08 2012-09-13 Sanofi Tetrasubstituierte oxathiazinderivate, verfahren zu deren herstellung, ihre verwendung als medikament sowie sie enthaltendes arzneimittel und deren verwendung
WO2012120054A1 (de) 2011-03-08 2012-09-13 Sanofi Di- und trisubstituierte oxathiazinderivate, verfahren zu deren herstellung, ihre verwendung als medikament sowie sie enthaltendes arzneimittel und deren verwendung
US8809325B2 (en) 2011-03-08 2014-08-19 Sanofi Benzyl-oxathiazine derivatives substituted with adamantane and noradamantane, medicaments containing said compounds and use thereof
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JP2007529566A (ja) 2007-10-25
AU2005226914A1 (en) 2005-10-06
US20080004251A1 (en) 2008-01-03
CN1933826A (zh) 2007-03-21
CA2560526A1 (en) 2005-10-06
EP1732532A1 (en) 2006-12-20
NO20064705L (no) 2006-12-19

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