BRPI0509213A - método para previnir, reduzir ou minimizar a formação de impurezas de tioamida durante a tionação de um composto de carbonila, produto, e, uso de um agente extrator - Google Patents
método para previnir, reduzir ou minimizar a formação de impurezas de tioamida durante a tionação de um composto de carbonila, produto, e, uso de um agente extratorInfo
- Publication number
- BRPI0509213A BRPI0509213A BRPI0509213-2A BRPI0509213A BRPI0509213A BR PI0509213 A BRPI0509213 A BR PI0509213A BR PI0509213 A BRPI0509213 A BR PI0509213A BR PI0509213 A BRPI0509213 A BR PI0509213A
- Authority
- BR
- Brazil
- Prior art keywords
- formation
- minimizing
- preventing
- reducing
- product
- Prior art date
Links
- 230000015572 biosynthetic process Effects 0.000 title abstract 3
- 238000000034 method Methods 0.000 title abstract 3
- 150000001728 carbonyl compounds Chemical class 0.000 title abstract 2
- AEOCXXJPGCBFJA-UHFFFAOYSA-N ethionamide Chemical compound CCC1=CC(C(N)=S)=CC=N1 AEOCXXJPGCBFJA-UHFFFAOYSA-N 0.000 title abstract 2
- 238000007280 thionation reaction Methods 0.000 title abstract 2
- 239000012535 impurity Substances 0.000 title 1
- 150000001875 compounds Chemical class 0.000 abstract 1
- 125000002560 nitrile group Chemical group 0.000 abstract 1
- 150000003556 thioamides Chemical class 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
- C07D333/02—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings
- C07D333/04—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
- C07D333/26—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D333/38—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
- C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
- C07D403/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Plural Heterocyclic Compounds (AREA)
- Glass Compositions (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US56040304P | 2004-04-08 | 2004-04-08 | |
| PCT/US2005/013657 WO2005100347A1 (en) | 2004-04-08 | 2005-04-07 | Methods for minimizing thioamide impurities |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| BRPI0509213A true BRPI0509213A (pt) | 2007-08-28 |
Family
ID=34966434
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| BRPI0509213-2A BRPI0509213A (pt) | 2004-04-08 | 2005-04-07 | método para previnir, reduzir ou minimizar a formação de impurezas de tioamida durante a tionação de um composto de carbonila, produto, e, uso de um agente extrator |
Country Status (14)
| Country | Link |
|---|---|
| US (2) | US7314932B2 (de) |
| EP (1) | EP1732922B1 (de) |
| JP (1) | JP4950027B2 (de) |
| CN (1) | CN1938298B (de) |
| AT (1) | ATE409699T1 (de) |
| AU (1) | AU2005233648B2 (de) |
| BR (1) | BRPI0509213A (de) |
| CA (1) | CA2561313C (de) |
| DE (1) | DE602005010065D1 (de) |
| DK (1) | DK1732922T3 (de) |
| ES (1) | ES2313334T3 (de) |
| MX (1) | MXPA06011695A (de) |
| PL (1) | PL1732922T3 (de) |
| WO (1) | WO2005100347A1 (de) |
Families Citing this family (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| ATE409699T1 (de) | 2004-04-08 | 2008-10-15 | Wyeth Corp | Verfahren zur minimierung von thioamidverunreinigungen |
| CA2561014C (en) * | 2004-04-08 | 2013-09-10 | Wyeth | Thioamide derivatives as progesterone receptor modulators |
| EA201070715A1 (ru) * | 2007-12-20 | 2011-02-28 | Тева Вимен'С Хелс, Инк. | Режимы дозирования, фармацевтические композиции и упаковки для экстренной контрацепции |
Family Cites Families (17)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB8308064D0 (en) * | 1983-03-24 | 1983-05-05 | Beecham Group Plc | Active compounds |
| US4997950A (en) * | 1989-04-20 | 1991-03-05 | Richard Finbar Murphy | Novel C-terminal gastrin antagonists |
| JPH0834775A (ja) * | 1994-05-16 | 1996-02-06 | Sumitomo Chem Co Ltd | テトラゾール化合物の製造法 |
| US6407101B1 (en) * | 1999-05-04 | 2002-06-18 | American Home Products Corporation | Cyanopyrroles |
| US6417214B1 (en) * | 1999-05-04 | 2002-07-09 | Wyeth | 3,3-substituted indoline derivatives |
| BR0010216A (pt) * | 1999-05-04 | 2002-03-19 | American Home Prod | Derivados de tio-oxindol |
| US6391907B1 (en) * | 1999-05-04 | 2002-05-21 | American Home Products Corporation | Indoline derivatives |
| HUP0203332A3 (en) * | 1999-05-04 | 2004-12-28 | Wyeth Corp | Cyclothiocarbamate derivatives, their use as progesterone receptor modulators and pharmaceutical compositions containing them |
| US6509334B1 (en) * | 1999-05-04 | 2003-01-21 | American Home Products Corporation | Cyclocarbamate derivatives as progesterone receptor modulators |
| UA73119C2 (en) * | 2000-04-19 | 2005-06-15 | American Home Products Corpoir | Derivatives of cyclic thiocarbamates, pharmaceutical composition including noted derivatives of cyclic thiocarbamates and active ingredients of medicines as modulators of progesterone receptors |
| US7132445B2 (en) * | 2001-04-16 | 2006-11-07 | Schering Corporation | 3,4-Di-substituted cyclobutene-1,2-diones as CXC-chemokine receptor ligands |
| RU2005101624A (ru) * | 2002-06-25 | 2005-06-27 | Уайт (Us) | Применение производных тиооксиндола в терапии кожных нарушений |
| TW200407124A (en) * | 2002-06-25 | 2004-05-16 | Wyeth Corp | Use of thio-oxindole derivatives in treatment of hormone-related conditions |
| CN1665510A (zh) * | 2002-06-25 | 2005-09-07 | 惠氏公司 | 作为pr调节剂的环硫代氨基甲酸酯衍生物的衍生物和其用于治疗皮肤病的用途 |
| CN1662241A (zh) * | 2002-06-25 | 2005-08-31 | 惠氏公司 | 环硫代氨基甲酸酯衍生物在治疗与激素有关的病症中的用途 |
| ATE409699T1 (de) | 2004-04-08 | 2008-10-15 | Wyeth Corp | Verfahren zur minimierung von thioamidverunreinigungen |
| CA2561014C (en) * | 2004-04-08 | 2013-09-10 | Wyeth | Thioamide derivatives as progesterone receptor modulators |
-
2005
- 2005-04-07 AT AT05738187T patent/ATE409699T1/de not_active IP Right Cessation
- 2005-04-07 WO PCT/US2005/013657 patent/WO2005100347A1/en not_active Ceased
- 2005-04-07 DE DE602005010065T patent/DE602005010065D1/de not_active Expired - Lifetime
- 2005-04-07 PL PL05738187T patent/PL1732922T3/pl unknown
- 2005-04-07 AU AU2005233648A patent/AU2005233648B2/en not_active Ceased
- 2005-04-07 DK DK05738187T patent/DK1732922T3/da active
- 2005-04-07 CN CN2005800102930A patent/CN1938298B/zh not_active Expired - Fee Related
- 2005-04-07 ES ES05738187T patent/ES2313334T3/es not_active Expired - Lifetime
- 2005-04-07 CA CA2561313A patent/CA2561313C/en not_active Expired - Fee Related
- 2005-04-07 US US11/100,863 patent/US7314932B2/en not_active Expired - Fee Related
- 2005-04-07 MX MXPA06011695A patent/MXPA06011695A/es active IP Right Grant
- 2005-04-07 EP EP05738187A patent/EP1732922B1/de not_active Expired - Lifetime
- 2005-04-07 JP JP2007507577A patent/JP4950027B2/ja not_active Expired - Fee Related
- 2005-04-07 BR BRPI0509213-2A patent/BRPI0509213A/pt not_active IP Right Cessation
-
2007
- 2007-11-16 US US11/985,774 patent/US7572824B2/en not_active Expired - Fee Related
Also Published As
| Publication number | Publication date |
|---|---|
| AU2005233648B2 (en) | 2011-06-23 |
| MXPA06011695A (es) | 2006-12-14 |
| CA2561313A1 (en) | 2005-10-27 |
| EP1732922A1 (de) | 2006-12-20 |
| DE602005010065D1 (de) | 2008-11-13 |
| ES2313334T3 (es) | 2009-03-01 |
| PL1732922T3 (pl) | 2009-03-31 |
| CN1938298B (zh) | 2013-02-06 |
| CN1938298A (zh) | 2007-03-28 |
| US7314932B2 (en) | 2008-01-01 |
| CA2561313C (en) | 2012-12-04 |
| US20050228179A1 (en) | 2005-10-13 |
| ATE409699T1 (de) | 2008-10-15 |
| JP4950027B2 (ja) | 2012-06-13 |
| EP1732922B1 (de) | 2008-10-01 |
| WO2005100347A1 (en) | 2005-10-27 |
| US20080071083A1 (en) | 2008-03-20 |
| JP2007532581A (ja) | 2007-11-15 |
| DK1732922T3 (da) | 2009-01-12 |
| US7572824B2 (en) | 2009-08-11 |
| AU2005233648A1 (en) | 2005-10-27 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| B06F | Objections, documents and/or translations needed after an examination request according [chapter 6.6 patent gazette] | ||
| B25D | Requested change of name of applicant approved |
Owner name: WYETH LLC. (US) |
|
| B08F | Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette] |
Free format text: REFERENTE A 11A ANUIDADE. |
|
| B08K | Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette] |
Free format text: EM VIRTUDE DO ARQUIVAMENTO PUBLICADO NA RPI 2384 DE 13-09-2016 E CONSIDERANDO AUSENCIA DE MANIFESTACAO DENTRO DOS PRAZOS LEGAIS, INFORMO QUE CABE SER MANTIDO O ARQUIVAMENTO DO PEDIDO DE PATENTE, CONFORME O DISPOSTO NO ARTIGO 12, DA RESOLUCAO 113/2013. |