BRPI0516905A - processo para a preparação de um derivado n-[2-(2-piridinil)etil]carboxamida e compostos - Google Patents

processo para a preparação de um derivado n-[2-(2-piridinil)etil]carboxamida e compostos

Info

Publication number
BRPI0516905A
BRPI0516905A BRPI0516905-4A BRPI0516905A BRPI0516905A BR PI0516905 A BRPI0516905 A BR PI0516905A BR PI0516905 A BRPI0516905 A BR PI0516905A BR PI0516905 A BRPI0516905 A BR PI0516905A
Authority
BR
Brazil
Prior art keywords
pyridinyl
ethyl
preparation
compounds
carboxamide derivative
Prior art date
Application number
BRPI0516905-4A
Other languages
English (en)
Inventor
Frederic Lhermitte
Pierre-Yves Coqueron
Philippe Desbordes
Thomas Himmler
Original Assignee
Bayer Cropscience Sa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bayer Cropscience Sa filed Critical Bayer Cropscience Sa
Publication of BRPI0516905A publication Critical patent/BRPI0516905A/pt
Publication of BRPI0516905B1 publication Critical patent/BRPI0516905B1/pt

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/24—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with substituted hydrocarbon radicals attached to ring carbon atoms
    • C07D213/54—Radicals substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
    • C07D213/56—Amides
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C233/00—Carboxylic acid amides
    • C07C233/64—Carboxylic acid amides having carbon atoms of carboxamide groups bound to carbon atoms of six-membered aromatic rings
    • C07C233/67—Carboxylic acid amides having carbon atoms of carboxamide groups bound to carbon atoms of six-membered aromatic rings having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a hydrocarbon radical substituted by singly-bound oxygen atoms
    • C07C233/68—Carboxylic acid amides having carbon atoms of carboxamide groups bound to carbon atoms of six-membered aromatic rings having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a hydrocarbon radical substituted by singly-bound oxygen atoms with the substituted hydrocarbon radical bound to the nitrogen atom of the carboxamide group by an acyclic carbon atom
    • C07C233/69—Carboxylic acid amides having carbon atoms of carboxamide groups bound to carbon atoms of six-membered aromatic rings having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a hydrocarbon radical substituted by singly-bound oxygen atoms with the substituted hydrocarbon radical bound to the nitrogen atom of the carboxamide group by an acyclic carbon atom of an acyclic saturated carbon skeleton
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/61—Halogen atoms or nitro radicals

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pyridine Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)

Abstract

PROCESSO PARA A PREPARAçãO DE UM DERIVADO N-¢2-(2-PIRIDINIL)ETIL!CARBOXAMIDA E COMPOSTOS. Processo para a preparação e um derivado N-¢2-(2-piridinil)etil!carboxamida de fórmula geral (1) ou um sal deste. Intermediário de fórmula geral (II). Intermediário de fórmula geral (III).
BRPI0516905A 2004-12-21 2005-12-19 processo para a preparação de um derivado n-[2-(2-piridinil)etil]carboxamida e compostos BRPI0516905B1 (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP04356203 2004-12-21
PCT/EP2005/056895 WO2006067103A2 (en) 2004-12-21 2005-12-19 Process for the preparation of a 2-pyridylethylcarboxamide derivative

Publications (2)

Publication Number Publication Date
BRPI0516905A true BRPI0516905A (pt) 2008-09-23
BRPI0516905B1 BRPI0516905B1 (pt) 2016-09-20

Family

ID=34931762

Family Applications (1)

Application Number Title Priority Date Filing Date
BRPI0516905A BRPI0516905B1 (pt) 2004-12-21 2005-12-19 processo para a preparação de um derivado n-[2-(2-piridinil)etil]carboxamida e compostos

Country Status (13)

Country Link
US (2) US7790901B2 (pt)
EP (1) EP1831169B1 (pt)
JP (2) JP4869251B2 (pt)
KR (1) KR101312816B1 (pt)
CN (1) CN101080391B (pt)
AT (1) ATE553083T1 (pt)
BR (1) BRPI0516905B1 (pt)
DK (1) DK1831169T3 (pt)
ES (1) ES2383903T3 (pt)
IL (2) IL183662A (pt)
MX (1) MX2007007105A (pt)
TW (2) TWI379826B (pt)
WO (1) WO2006067103A2 (pt)

Families Citing this family (27)

* Cited by examiner, † Cited by third party
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EP2606727A1 (en) 2011-12-21 2013-06-26 Bayer CropScience AG Compounds with nematicidal activity
EP2606728A1 (en) 2011-12-21 2013-06-26 Bayer CropScience AG Compounds with nematicidal activity
EP2773203A1 (en) 2011-11-02 2014-09-10 Bayer Intellectual Property GmbH Compounds with nematicidal activity
KR20140088532A (ko) 2011-11-02 2014-07-10 바이엘 인텔렉쳐 프로퍼티 게엠베하 살선충 활성을 갖는 화합물
EP2589292A1 (en) 2011-11-02 2013-05-08 Bayer CropScience AG Compounds with nematicidal activity
EP2589294A1 (en) 2011-11-02 2013-05-08 Bayer CropScience AG Compounds with nematicidal activity
UA115666C2 (uk) 2012-07-12 2017-12-11 Ніссан Кемікал Індастріз, Лтд. Заміщена оксимом амідна сполука і засіб для боротьби зі шкідниками
CN103535353A (zh) * 2012-07-13 2014-01-29 陕西美邦农药有限公司 一种高效杀菌组合物
CN103535354A (zh) * 2012-07-13 2014-01-29 陕西美邦农药有限公司 一种高效杀菌组合物
CN103535355A (zh) * 2012-07-13 2014-01-29 陕西美邦农药有限公司 一种高效杀菌组合物
CN103535362A (zh) * 2012-07-13 2014-01-29 陕西美邦农药有限公司 一种高效杀菌组合物
UY35772A (es) 2013-10-14 2015-05-29 Bayer Cropscience Ag Nuevos compuestos plaguicidas
US10167250B2 (en) * 2014-06-16 2019-01-01 Srf Limited Process for the preparation of 2-(trihalomethyl) benzamide
KR101719565B1 (ko) * 2014-10-02 2017-03-24 한국화학연구원 광산화환원 촉매와 CF3SO2Cl을 사용한 알켄 화합물의 클로로트리플루오로메틸레이션 방법
KR102522231B1 (ko) * 2016-12-21 2023-04-14 바이엘 크롭사이언스 악티엔게젤샤프트 2-피리딜에틸카복사미드 유도체의 제조 방법
WO2020020897A1 (en) * 2018-07-26 2020-01-30 Bayer Aktiengesellschaft Crystalline form of fluopyram
CN108822024B (zh) * 2018-08-28 2021-03-09 陕西恒润化学工业有限公司 一种氟吡菌酰胺及其合成方法
CN108752268A (zh) * 2018-08-28 2018-11-06 陕西恒润化学工业有限公司 一种2-（3-氯-5-三氟甲基吡啶）-丙二酸二甲酯及其合成方法
CN110437138B (zh) * 2019-08-12 2021-03-02 大连九信精细化工有限公司 一种氟吡菌酰胺的改进合成工艺
CN112979539B (zh) * 2021-05-17 2021-07-20 湖南速博生物技术有限公司 一种氟吡菌酰胺中间体的合成方法
CN113429338B (zh) * 2021-05-20 2023-05-02 陕西泰合利华工业有限公司 一种合成氟吡菌酰胺的方法
CN117440848A (zh) * 2021-06-11 2024-01-23 C·R·巴德股份有限公司 间歇导管和方法
CN113620867B (zh) * 2021-09-03 2023-06-16 内蒙古蓝科生物科技有限公司 一种氟吡菌酰胺的合成方法
CN114195667A (zh) * 2021-11-30 2022-03-18 江西永通科技股份有限公司 一种邻三氟甲基苯甲酰胺的合成方法
CN117003691B (zh) * 2023-06-27 2026-04-14 一帆生物科技(上海)有限公司 一种制备氟吡菌酰胺的方法
CN116874415A (zh) * 2023-07-14 2023-10-13 利民化学有限责任公司 一种氟吡菌酰胺的新晶型及其制备方法
CN120247782B (zh) * 2025-06-04 2025-08-19 北京颖泰嘉和生物科技股份有限公司 氟吡菌酰胺类化合物及其制备方法

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DE1034644B (de) * 1956-09-26 1958-07-24 Bayer Ag Verfahren zur Herstellung von Acylaminomethyl-Verbindungen
JPS5363337A (en) * 1976-11-12 1978-06-06 Nippon Kayaku Co Ltd Benzamide derivs, process for their preparation and herbicides contg.the same as active constituents
EP0061836B1 (en) * 1981-03-19 1986-12-30 Imperial Chemical Industries Plc Amide derivatives, processes for preparing them, their use as fungicides and pesticidal compositions containing them
DE4138026A1 (de) * 1991-11-19 1993-06-03 Bayer Ag Substituierte pyridin-4-carbonsaeureamide
AU7278500A (en) * 1999-08-18 2001-03-13 Aventis Cropscience Gmbh Fungicides
JP2001213869A (ja) * 2000-01-28 2001-08-07 Nippon Bayer Agrochem Co Ltd イソチアゾールカルボン酸誘導体および病害防除剤
US20060009461A1 (en) * 2002-05-23 2006-01-12 Bhatia Pramila A Acetamides and benzamides that are useful in treating sexual dysfunction
US20030232836A1 (en) * 2002-05-23 2003-12-18 Stewart Andrew O. Acetamides and benzamides that are useful in treating sexual dysfunction
WO2003099266A2 (en) * 2002-05-23 2003-12-04 Abbott Laboratories Acetamides and benzamides that are useful in treating sexual dysfunction
US20040029887A1 (en) * 2002-05-23 2004-02-12 Bhatia Pramila A. Acetamides and benzamides that are useful in treating sexual dysfunction
AU2003266316B2 (en) * 2002-08-12 2007-10-25 Bayer S.A.S. Novel 2-pyridylethylbenzamide derivative
EP1500651A1 (en) * 2003-07-25 2005-01-26 Bayer CropScience S.A. N-[2-(2-Pyridinyl)ethyl]benzamide compounds and their use as fungicides
TWI368482B (en) * 2003-12-19 2012-07-21 Bayer Sas New 2-pyridinylethylbenzamide derivatives
EP1548007A1 (en) * 2003-12-19 2005-06-29 Bayer CropScience S.A. 2-Pyridinylethylcarboxamide derivatives and their use as fungicides
EP1574511A1 (en) * 2004-03-03 2005-09-14 Bayer CropScience S.A. 2-Pyridinylethylcarboxamide derivatives and their use as fungicides

Also Published As

Publication number Publication date
TWI370121B (en) 2012-08-11
TW200637822A (en) 2006-11-01
KR101312816B1 (ko) 2013-09-27
WO2006067103A2 (en) 2006-06-29
US7790901B2 (en) 2010-09-07
IL217962A0 (en) 2012-03-29
IL183662A (en) 2012-06-28
EP1831169A2 (en) 2007-09-12
TW201215594A (en) 2012-04-16
WO2006067103A3 (en) 2006-11-16
JP5559745B2 (ja) 2014-07-23
KR20070087668A (ko) 2007-08-28
ATE553083T1 (de) 2012-04-15
US20080086008A1 (en) 2008-04-10
ES2383903T3 (es) 2012-06-27
CN101080391A (zh) 2007-11-28
EP1831169B1 (en) 2012-04-11
JP2008524307A (ja) 2008-07-10
US8865908B2 (en) 2014-10-21
IL183662A0 (en) 2007-09-20
BRPI0516905B1 (pt) 2016-09-20
TWI379826B (en) 2012-12-21
MX2007007105A (es) 2007-08-08
US20100292485A1 (en) 2010-11-18
IL217962A (en) 2015-02-26
JP4869251B2 (ja) 2012-02-08
JP2011236216A (ja) 2011-11-24
CN101080391B (zh) 2010-09-22
DK1831169T3 (da) 2012-07-09

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Legal Events

Date Code Title Description
B06F Objections, documents and/or translations needed after an examination request according [chapter 6.6 patent gazette]
B25A Requested transfer of rights approved

Owner name: BAYER SAS (FR)

B06A Patent application procedure suspended [chapter 6.1 patent gazette]
B25C Requirement related to requested transfer of rights

Owner name: BAYER SAS (FR)

Free format text: A FIM DE ATENDER A(S) TRANSFERENCIA(S), REQUERIDA(S) ATRAVES DA PETICAO NO 860150256045, DE 03/11/2015, E NECESSARIO REAPRESENTAR O DOCUMENTO DE CESSAO COM A ASSINATURA DE CEDENTE E CESSIONARIO NOTARIZADAS E LEGALIZADAS.

B09A Decision: intention to grant [chapter 9.1 patent gazette]
B16A Patent or certificate of addition of invention granted [chapter 16.1 patent gazette]

Free format text: PRAZO DE VALIDADE: 10 (DEZ) ANOS CONTADOS A PARTIR DE 20/09/2016, OBSERVADAS AS CONDICOES LEGAIS.

B25A Requested transfer of rights approved
B25G Requested change of headquarter approved
B25A Requested transfer of rights approved