ATE553083T1 - Verfahren zur herstellung eines 2- pyridylethylcarbonsäureamidderivats - Google Patents

Verfahren zur herstellung eines 2- pyridylethylcarbonsäureamidderivats

Info

Publication number
ATE553083T1
ATE553083T1 AT05823830T AT05823830T ATE553083T1 AT E553083 T1 ATE553083 T1 AT E553083T1 AT 05823830 T AT05823830 T AT 05823830T AT 05823830 T AT05823830 T AT 05823830T AT E553083 T1 ATE553083 T1 AT E553083T1
Authority
AT
Austria
Prior art keywords
pyridylethylcarboxylic
producing
amide derivative
general formula
derivative
Prior art date
Application number
AT05823830T
Other languages
English (en)
Inventor
Frederic Lhermitte
Pierre-Yves Coqueron
Philippe Desbordes
Thomas Himmler
Original Assignee
Bayer Cropscience Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bayer Cropscience Ag filed Critical Bayer Cropscience Ag
Application granted granted Critical
Publication of ATE553083T1 publication Critical patent/ATE553083T1/de

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/24—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with substituted hydrocarbon radicals attached to ring carbon atoms
    • C07D213/54—Radicals substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
    • C07D213/56—Amides
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C233/00—Carboxylic acid amides
    • C07C233/64—Carboxylic acid amides having carbon atoms of carboxamide groups bound to carbon atoms of six-membered aromatic rings
    • C07C233/67—Carboxylic acid amides having carbon atoms of carboxamide groups bound to carbon atoms of six-membered aromatic rings having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a hydrocarbon radical substituted by singly-bound oxygen atoms
    • C07C233/68—Carboxylic acid amides having carbon atoms of carboxamide groups bound to carbon atoms of six-membered aromatic rings having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a hydrocarbon radical substituted by singly-bound oxygen atoms with the substituted hydrocarbon radical bound to the nitrogen atom of the carboxamide group by an acyclic carbon atom
    • C07C233/69—Carboxylic acid amides having carbon atoms of carboxamide groups bound to carbon atoms of six-membered aromatic rings having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a hydrocarbon radical substituted by singly-bound oxygen atoms with the substituted hydrocarbon radical bound to the nitrogen atom of the carboxamide group by an acyclic carbon atom of an acyclic saturated carbon skeleton
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/61—Halogen atoms or nitro radicals

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pyridine Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
AT05823830T 2004-12-21 2005-12-19 Verfahren zur herstellung eines 2- pyridylethylcarbonsäureamidderivats ATE553083T1 (de)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP04356203 2004-12-21
PCT/EP2005/056895 WO2006067103A2 (en) 2004-12-21 2005-12-19 Process for the preparation of a 2-pyridylethylcarboxamide derivative

Publications (1)

Publication Number Publication Date
ATE553083T1 true ATE553083T1 (de) 2012-04-15

Family

ID=34931762

Family Applications (1)

Application Number Title Priority Date Filing Date
AT05823830T ATE553083T1 (de) 2004-12-21 2005-12-19 Verfahren zur herstellung eines 2- pyridylethylcarbonsäureamidderivats

Country Status (13)

Country Link
US (2) US7790901B2 (de)
EP (1) EP1831169B1 (de)
JP (2) JP4869251B2 (de)
KR (1) KR101312816B1 (de)
CN (1) CN101080391B (de)
AT (1) ATE553083T1 (de)
BR (1) BRPI0516905B1 (de)
DK (1) DK1831169T3 (de)
ES (1) ES2383903T3 (de)
IL (2) IL183662A (de)
MX (1) MX2007007105A (de)
TW (2) TWI370121B (de)
WO (1) WO2006067103A2 (de)

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* Cited by examiner, † Cited by third party
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EP2606727A1 (de) 2011-12-21 2013-06-26 Bayer CropScience AG Verbindungen mit nematizider Aktivität
EP2606728A1 (de) 2011-12-21 2013-06-26 Bayer CropScience AG Verbindungen mit nematizider Aktivität
EP2589294A1 (de) 2011-11-02 2013-05-08 Bayer CropScience AG Verbindungen mit nematizider Aktivität
CN104023540A (zh) 2011-11-02 2014-09-03 拜耳知识产权有限责任公司 具有杀线虫活性的化合物
EP2589292A1 (de) 2011-11-02 2013-05-08 Bayer CropScience AG Verbindungen mit nematizider Aktivität
PE20141996A1 (es) 2011-11-02 2014-11-28 Bayer Ip Gmbh Compuestos con actividad nematicida
PT2873658T (pt) 2012-07-12 2018-12-05 Nissan Chemical Corp Composto de amida substituída com oxima e agente de controlo de pragas
CN103535362A (zh) * 2012-07-13 2014-01-29 陕西美邦农药有限公司 一种高效杀菌组合物
CN103535355A (zh) * 2012-07-13 2014-01-29 陕西美邦农药有限公司 一种高效杀菌组合物
CN103535354A (zh) * 2012-07-13 2014-01-29 陕西美邦农药有限公司 一种高效杀菌组合物
CN103535353A (zh) * 2012-07-13 2014-01-29 陕西美邦农药有限公司 一种高效杀菌组合物
UY35772A (es) 2013-10-14 2015-05-29 Bayer Cropscience Ag Nuevos compuestos plaguicidas
EP3154933B1 (de) * 2014-06-16 2019-03-27 Srf Limited Verfahren zur herstellung von 2-(trihalomethyl)benzamid
KR101719565B1 (ko) * 2014-10-02 2017-03-24 한국화학연구원 광산화환원 촉매와 CF3SO2Cl을 사용한 알켄 화합물의 클로로트리플루오로메틸레이션 방법
KR102522231B1 (ko) * 2016-12-21 2023-04-14 바이엘 크롭사이언스 악티엔게젤샤프트 2-피리딜에틸카복사미드 유도체의 제조 방법
JP2021532138A (ja) * 2018-07-26 2021-11-25 バイエル、アクチエンゲゼルシャフトBayer Aktiengesellschaft フルオピラムの結晶形
CN108752268A (zh) * 2018-08-28 2018-11-06 陕西恒润化学工业有限公司 一种2-（3-氯-5-三氟甲基吡啶）-丙二酸二甲酯及其合成方法
CN108822024B (zh) * 2018-08-28 2021-03-09 陕西恒润化学工业有限公司 一种氟吡菌酰胺及其合成方法
CN110437138B (zh) * 2019-08-12 2021-03-02 大连九信精细化工有限公司 一种氟吡菌酰胺的改进合成工艺
CN112979539B (zh) * 2021-05-17 2021-07-20 湖南速博生物技术有限公司 一种氟吡菌酰胺中间体的合成方法
CN113429338B (zh) * 2021-05-20 2023-05-02 陕西泰合利华工业有限公司 一种合成氟吡菌酰胺的方法
CN113620867B (zh) * 2021-09-03 2023-06-16 内蒙古蓝科生物科技有限公司 一种氟吡菌酰胺的合成方法
CN114195667A (zh) * 2021-11-30 2022-03-18 江西永通科技股份有限公司 一种邻三氟甲基苯甲酰胺的合成方法
CN117003691A (zh) * 2023-06-27 2023-11-07 上海农帆生物科技有限公司 一种制备氟吡菌酰胺的方法
CN116874415A (zh) * 2023-07-14 2023-10-13 利民化学有限责任公司 一种氟吡菌酰胺的新晶型及其制备方法
CN120247782B (zh) * 2025-06-04 2025-08-19 北京颖泰嘉和生物科技股份有限公司 氟吡菌酰胺类化合物及其制备方法

Family Cites Families (15)

* Cited by examiner, † Cited by third party
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DE1034644B (de) * 1956-09-26 1958-07-24 Bayer Ag Verfahren zur Herstellung von Acylaminomethyl-Verbindungen
JPS5363337A (en) * 1976-11-12 1978-06-06 Nippon Kayaku Co Ltd Benzamide derivs, process for their preparation and herbicides contg.the same as active constituents
EP0061836B1 (de) * 1981-03-19 1986-12-30 Imperial Chemical Industries Plc Amidderivate, Verfahren zu ihrer Herstellung, ihre Verwendung als Fungizide und Pestizide, die sie enthalten
DE4138026A1 (de) * 1991-11-19 1993-06-03 Bayer Ag Substituierte pyridin-4-carbonsaeureamide
PT1204323E (pt) 1999-08-18 2004-11-30 Aventis Cropscience Gmbh Fungicidas
JP2001213869A (ja) * 2000-01-28 2001-08-07 Nippon Bayer Agrochem Co Ltd イソチアゾールカルボン酸誘導体および病害防除剤
WO2003099266A2 (en) * 2002-05-23 2003-12-04 Abbott Laboratories Acetamides and benzamides that are useful in treating sexual dysfunction
US20040029887A1 (en) * 2002-05-23 2004-02-12 Bhatia Pramila A. Acetamides and benzamides that are useful in treating sexual dysfunction
US20030232836A1 (en) * 2002-05-23 2003-12-18 Stewart Andrew O. Acetamides and benzamides that are useful in treating sexual dysfunction
US20060009461A1 (en) * 2002-05-23 2006-01-12 Bhatia Pramila A Acetamides and benzamides that are useful in treating sexual dysfunction
RU2316548C2 (ru) * 2002-08-12 2008-02-10 Байер Кропсайенс С.А. Новое производное 2-пиридилэтилбензамида, способ его получения, фунгицидная композиция, способ профилактического или лечебного подавления фитопатогенных грибков
EP1500651A1 (de) * 2003-07-25 2005-01-26 Bayer CropScience S.A. N-[2-(2-Pyridinyl)ethyl]benzamidverbindungen und ihre Verwendung als Fungizide
EP1548007A1 (de) * 2003-12-19 2005-06-29 Bayer CropScience S.A. 2-Pyridinylethylcarbonsäureamidderivate und ihre Verwendung als Fungizide
TWI368482B (en) * 2003-12-19 2012-07-21 Bayer Sas New 2-pyridinylethylbenzamide derivatives
EP1574511A1 (de) * 2004-03-03 2005-09-14 Bayer CropScience S.A. 2-Pyridinylethylcarboxamid-Derivate und ihre Verwendung als Fungizide

Also Published As

Publication number Publication date
JP4869251B2 (ja) 2012-02-08
ES2383903T3 (es) 2012-06-27
EP1831169B1 (de) 2012-04-11
TW200637822A (en) 2006-11-01
CN101080391A (zh) 2007-11-28
IL217962A (en) 2015-02-26
EP1831169A2 (de) 2007-09-12
TWI370121B (en) 2012-08-11
BRPI0516905A (pt) 2008-09-23
US20100292485A1 (en) 2010-11-18
KR20070087668A (ko) 2007-08-28
DK1831169T3 (da) 2012-07-09
US8865908B2 (en) 2014-10-21
KR101312816B1 (ko) 2013-09-27
JP2008524307A (ja) 2008-07-10
US7790901B2 (en) 2010-09-07
JP5559745B2 (ja) 2014-07-23
WO2006067103A3 (en) 2006-11-16
IL217962A0 (en) 2012-03-29
WO2006067103A2 (en) 2006-06-29
IL183662A0 (en) 2007-09-20
JP2011236216A (ja) 2011-11-24
CN101080391B (zh) 2010-09-22
BRPI0516905B1 (pt) 2016-09-20
TWI379826B (en) 2012-12-21
TW201215594A (en) 2012-04-16
IL183662A (en) 2012-06-28
MX2007007105A (es) 2007-08-08
US20080086008A1 (en) 2008-04-10

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