BRPI0519138A2 - mÉtodo para produÇço de um composto do sal (4,5- diidroisoxazol-3-il) tiocarboxamidina - Google Patents
mÉtodo para produÇço de um composto do sal (4,5- diidroisoxazol-3-il) tiocarboxamidinaInfo
- Publication number
- BRPI0519138A2 BRPI0519138A2 BRPI0519138-6A BRPI0519138A BRPI0519138A2 BR PI0519138 A2 BRPI0519138 A2 BR PI0519138A2 BR PI0519138 A BRPI0519138 A BR PI0519138A BR PI0519138 A2 BRPI0519138 A2 BR PI0519138A2
- Authority
- BR
- Brazil
- Prior art keywords
- compound
- dihydroisoxazol
- thiocarboxamidine
- halogen
- producing
- Prior art date
Links
- 150000001875 compounds Chemical class 0.000 title abstract 4
- 238000004519 manufacturing process Methods 0.000 title abstract 4
- 150000003839 salts Chemical class 0.000 title abstract 4
- -1 4,5-dihydroisoxazol-3-yl Chemical group 0.000 title abstract 3
- 239000002253 acid Chemical group 0.000 abstract 2
- 125000000217 alkyl group Chemical group 0.000 abstract 2
- 125000000753 cycloalkyl group Chemical group 0.000 abstract 2
- 229910052736 halogen Inorganic materials 0.000 abstract 2
- 125000005843 halogen group Chemical group 0.000 abstract 2
- 125000004435 hydrogen atom Chemical class [H]* 0.000 abstract 2
- UMGDCJDMYOKAJW-UHFFFAOYSA-N thiourea Chemical compound NC(N)=S UMGDCJDMYOKAJW-UHFFFAOYSA-N 0.000 abstract 2
- XSQUKJJJFZCRTK-UHFFFAOYSA-N Urea Natural products NC(N)=O XSQUKJJJFZCRTK-UHFFFAOYSA-N 0.000 abstract 1
- 125000000129 anionic group Chemical group 0.000 abstract 1
- 125000004429 atom Chemical group 0.000 abstract 1
- 125000004432 carbon atom Chemical group C* 0.000 abstract 1
- 229910052739 hydrogen Inorganic materials 0.000 abstract 1
- 239000001257 hydrogen Substances 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D261/00—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings
- C07D261/02—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings not condensed with other rings
- C07D261/06—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings not condensed with other rings having two or more double bonds between ring members or between ring members and non-ring members
- C07D261/10—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings not condensed with other rings having two or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D261/18—Carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D261/00—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings
- C07D261/20—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings condensed with carbocyclic rings or ring systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D261/00—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings
- C07D261/02—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings not condensed with other rings
- C07D261/04—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Abstract
MÉTODO PARA PRODUÇçO DE UM COMPOSTO DO SAL (4,5-DIIDROISOXAZOL-3-IL)TIOCARBOXAMIDINA. A presente invenção refere-se a um método para produzir um composto do sal (4,5 - diidroisoxazol - 3-il) tiocarboxamidina, de modo simples, com segurança e com bom rendimento, através do qual foram resolvidos os inconvenientes da técnica anterior. Um método para produzir um composto do sal (4,5 - diidroisoxa- zol - 3-il) tiocarboxamidina de acordo com a fórmula (2): em que cada um dos R¹ e R², que são independentes um do outro, é um átomo de hidrogênio, um grupo alquila ou um grupo cicloalquila, cada um dos Rü e R^ 4^, que são independentes um do outro, é um átomo de hidrogénio ou um grupo alquila, com a condição de que R¹ e R², ou R² e Rü, possam estar ligados para formar um grupo cicloalquila juntamente com os átomos de carbono aos quais estão ligados, e X² é um halogênio ou um resíduo aniônico derivado de um ácido, que compreende a reação de um composto 3 - halogeno - 4,5 - diidroisoxazol de acordo com a fórmula (1): em que R¹, R², Rü e R^ 4^ são tal como definidos acima, e X¹ é um halogênio, com a tiouréia em presença de um ácido.
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP2004367418 | 2004-12-20 | ||
| PCT/JP2005/023270 WO2006068092A1 (ja) | 2004-12-20 | 2005-12-19 | （４，５－ジヒドロイソオキサゾロ－３－イル）チオカルボキサミジン塩化合物の製造方法 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| BRPI0519138A2 true BRPI0519138A2 (pt) | 2008-12-23 |
| BRPI0519138B1 BRPI0519138B1 (pt) | 2016-05-10 |
Family
ID=36601692
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| BRPI0519138A BRPI0519138B1 (pt) | 2004-12-20 | 2005-12-19 | método para produção de um composto do sal (4,5- diidroisoxazol-3-il) tiocarboxamidina, e compostos do sal (4,5-diidroisoxazol-3-il)tiocarboxamidina |
Country Status (20)
| Country | Link |
|---|---|
| US (1) | US7714142B2 (pt) |
| EP (1) | EP1829868B1 (pt) |
| JP (1) | JP4927565B2 (pt) |
| KR (1) | KR101233037B1 (pt) |
| CN (1) | CN100588651C (pt) |
| AR (1) | AR052058A1 (pt) |
| AU (1) | AU2005320157B9 (pt) |
| BR (1) | BRPI0519138B1 (pt) |
| CA (1) | CA2586449C (pt) |
| CR (1) | CR9199A (pt) |
| ES (1) | ES2487896T3 (pt) |
| IL (1) | IL183700A0 (pt) |
| IN (1) | IN2007KO02166A (pt) |
| MX (1) | MX274842B (pt) |
| NZ (1) | NZ554870A (pt) |
| PL (1) | PL1829868T3 (pt) |
| RU (1) | RU2378261C2 (pt) |
| TW (1) | TW200633989A (pt) |
| UA (1) | UA86268C2 (pt) |
| WO (1) | WO2006068092A1 (pt) |
Families Citing this family (13)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2006037945A1 (en) | 2004-10-05 | 2006-04-13 | Syngenta Limited | Isoxazoline derivatives and their use as herbicides |
| GB0916267D0 (en) | 2009-09-16 | 2009-10-28 | Syngenta Ltd | Herbicidal compounds |
| CN102666502B (zh) | 2009-11-26 | 2015-01-07 | 巴斯夫欧洲公司 | 生产5,5-二取代的4,5-二氢异噁唑-3-硫基甲脒盐的方法 |
| CA2781409A1 (en) | 2009-11-26 | 2011-06-03 | Basf Se | Method for producing 5,5-disubstituted 2-isoxazolines |
| JP6664036B2 (ja) * | 2017-12-27 | 2020-03-13 | クミアイ化学工業株式会社 | チオカルボキサミジン塩化合物の製造方法 |
| EP4053125B1 (en) | 2019-10-31 | 2024-12-04 | Kumiai Chemical Industry Co., Ltd. | Process for the production of a pyroxasulfone herbicide |
| WO2021176456A1 (en) * | 2020-03-05 | 2021-09-10 | Adama Agan Ltd. | Process and intermediates for the preparation of pyroxasulfone |
| EP4177252A3 (en) | 2020-07-10 | 2023-08-09 | Adama Agan Ltd. | Process and intermediates for the preparation of pyroxasulfone, fenoxasulfone and various sulfone analogs of 5,5-dimethyl-4h-1,2-oxazole |
| CN112110912B (zh) * | 2020-07-31 | 2022-07-05 | 绍兴贝斯美化工股份有限公司 | 一种合成硫醚类中间体的方法 |
| CN114315747A (zh) * | 2020-09-30 | 2022-04-12 | 山东润博生物科技有限公司 | 一种5,5-二甲基异噁唑烷-3-硫酮的制备方法 |
| CN112645894B (zh) * | 2020-11-30 | 2022-04-15 | 江苏中旗科技股份有限公司 | 制备砜吡草唑中间体5,5-二甲基-4,5-二氢异恶唑-3-硫代甲脒盐酸盐的方法 |
| WO2023074828A1 (ja) | 2021-10-29 | 2023-05-04 | クミアイ化学工業株式会社 | ジスルフィド化合物、ポリスルフィド化合物及びその用途 |
| AR127776A1 (es) | 2021-11-28 | 2024-02-28 | Adama Agan Ltd | Composiciones de concentrado en suspensión de alta carga |
Family Cites Families (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| KR100602776B1 (ko) * | 1999-08-10 | 2006-07-20 | 구미아이 가가쿠 고교 가부시키가이샤 | 이소옥사졸린유도체 및 이것을 유효성분으로 하는 제초제 |
| JP4465133B2 (ja) * | 2001-02-08 | 2010-05-19 | クミアイ化学工業株式会社 | イソオキサゾリン誘導体及びこれを有効成分とする除草剤 |
| EP1405853B1 (en) * | 2001-06-21 | 2010-11-03 | Kumiai Chemical Industry Co., Ltd. | Isoxazoline derivatives and herbicides |
| AU2003252447B2 (en) * | 2002-08-01 | 2008-06-05 | Kumiai Chemical Industry Co., Ltd. | Pyrazole derivatives and process for the production thereof |
| JP2004224714A (ja) * | 2003-01-21 | 2004-08-12 | Ihara Chem Ind Co Ltd | イソオキサゾリジン−３−チオン誘導体の製造法 |
| JP4621939B2 (ja) * | 2004-03-31 | 2011-02-02 | イハラケミカル工業株式会社 | ５−ヒドロキシ−４−チオメチルピラゾール化合物の製造方法 |
| JP2007246396A (ja) * | 2004-04-28 | 2007-09-27 | Ihara Chem Ind Co Ltd | ５−ジフルオロメトキシ−４−チオメチルピラゾール化合物の製造方法 |
-
2005
- 2005-12-19 US US11/722,256 patent/US7714142B2/en active Active
- 2005-12-19 JP JP2006548975A patent/JP4927565B2/ja not_active Expired - Lifetime
- 2005-12-19 WO PCT/JP2005/023270 patent/WO2006068092A1/ja not_active Ceased
- 2005-12-19 BR BRPI0519138A patent/BRPI0519138B1/pt active IP Right Grant
- 2005-12-19 UA UAA200705075A patent/UA86268C2/uk unknown
- 2005-12-19 AR ARP050105332A patent/AR052058A1/es active IP Right Grant
- 2005-12-19 PL PL05816486T patent/PL1829868T3/pl unknown
- 2005-12-19 MX MX2007007407A patent/MX274842B/es active IP Right Grant
- 2005-12-19 CA CA2586449A patent/CA2586449C/en not_active Expired - Lifetime
- 2005-12-19 ES ES05816486.4T patent/ES2487896T3/es not_active Expired - Lifetime
- 2005-12-19 NZ NZ554870A patent/NZ554870A/en not_active IP Right Cessation
- 2005-12-19 CN CN200580043474.3A patent/CN100588651C/zh not_active Expired - Lifetime
- 2005-12-19 AU AU2005320157A patent/AU2005320157B9/en not_active Expired
- 2005-12-19 RU RU2007127663/04A patent/RU2378261C2/ru active
- 2005-12-19 KR KR1020077013289A patent/KR101233037B1/ko not_active Expired - Lifetime
- 2005-12-19 EP EP05816486.4A patent/EP1829868B1/en not_active Expired - Lifetime
- 2005-12-20 TW TW094145311A patent/TW200633989A/zh not_active IP Right Cessation
-
2007
- 2007-06-05 IL IL183700A patent/IL183700A0/en active IP Right Grant
- 2007-06-13 IN IN2166KO2007 patent/IN2007KO02166A/en unknown
- 2007-06-20 CR CR9199A patent/CR9199A/es unknown
Also Published As
| Publication number | Publication date |
|---|---|
| MX274842B (es) | 2010-03-30 |
| CR9199A (es) | 2007-10-03 |
| AR052058A1 (es) | 2007-02-28 |
| EP1829868A4 (en) | 2011-03-16 |
| KR101233037B1 (ko) | 2013-02-13 |
| TW200633989A (en) | 2006-10-01 |
| BRPI0519138B1 (pt) | 2016-05-10 |
| NZ554870A (en) | 2009-09-25 |
| UA86268C2 (uk) | 2009-04-10 |
| IL183700A0 (en) | 2007-09-20 |
| TWI353970B (pt) | 2011-12-11 |
| CA2586449A1 (en) | 2006-06-29 |
| MX2007007407A (es) | 2007-07-12 |
| CA2586449C (en) | 2012-04-24 |
| CN100588651C (zh) | 2010-02-10 |
| US20080275249A1 (en) | 2008-11-06 |
| AU2005320157A1 (en) | 2006-06-29 |
| KR20070089153A (ko) | 2007-08-30 |
| PL1829868T3 (pl) | 2015-03-31 |
| ES2487896T3 (es) | 2014-08-25 |
| EP1829868A1 (en) | 2007-09-05 |
| RU2007127663A (ru) | 2009-01-27 |
| IN2007KO02166A (pt) | 2007-08-17 |
| RU2378261C2 (ru) | 2010-01-10 |
| US7714142B2 (en) | 2010-05-11 |
| JP4927565B2 (ja) | 2012-05-09 |
| CN101080397A (zh) | 2007-11-28 |
| JPWO2006068092A1 (ja) | 2008-06-12 |
| AU2005320157B9 (en) | 2011-07-21 |
| WO2006068092A1 (ja) | 2006-06-29 |
| EP1829868B1 (en) | 2014-07-23 |
| AU2005320157B2 (en) | 2011-04-28 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| B06A | Patent application procedure suspended [chapter 6.1 patent gazette] | ||
| B07A | Application suspended after technical examination (opinion) [chapter 7.1 patent gazette] | ||
| B09A | Decision: intention to grant [chapter 9.1 patent gazette] | ||
| B16A | Patent or certificate of addition of invention granted [chapter 16.1 patent gazette] |
Free format text: PRAZO DE VALIDADE: 10 (DEZ) ANOS CONTADOS A PARTIR DE 10/05/2016, OBSERVADAS AS CONDICOES LEGAIS. |
|
| B25A | Requested transfer of rights approved |