BRPI0607461A2 - dispositivo para liberação de agonistas de trpv1 - Google Patents

dispositivo para liberação de agonistas de trpv1

Info

Publication number
BRPI0607461A2
BRPI0607461A2 BRPI0607461-8A BRPI0607461A BRPI0607461A2 BR PI0607461 A2 BRPI0607461 A2 BR PI0607461A2 BR PI0607461 A BRPI0607461 A BR PI0607461A BR PI0607461 A2 BRPI0607461 A2 BR PI0607461A2
Authority
BR
Brazil
Prior art keywords
trpv1 agonist
release device
agonist release
delivery devices
drug delivery
Prior art date
Application number
BRPI0607461-8A
Other languages
English (en)
Inventor
Naweed Muhammad
Gene Curtis Jamieson
Keith R Bley
Original Assignee
Neurogesx Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Neurogesx Inc filed Critical Neurogesx Inc
Publication of BRPI0607461A2 publication Critical patent/BRPI0607461A2/pt

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/16—Amides, e.g. hydroxamic acids
    • A61K31/165—Amides, e.g. hydroxamic acids having aromatic rings, e.g. colchicine, atenolol, progabide
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
    • A61K31/565—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/16—Amides, e.g. hydroxamic acids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K36/00—Medicinal preparations of undetermined constitution containing material from algae, lichens, fungi or plants, or derivatives thereof, e.g. traditional herbal medicines
    • A61K36/18—Magnoliophyta (angiosperms)
    • A61K36/185—Magnoliopsida (dicotyledons)
    • A61K36/81—Solanaceae (Potato family), e.g. tobacco, nightshade, tomato, belladonna, capsicum or jimsonweed
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/70—Web, sheet or filament bases ; Films; Fibres of the matrix type containing drug
    • A61K9/7023—Transdermal patches and similar drug-containing composite devices, e.g. cataplasms
    • A61K9/703—Transdermal patches and similar drug-containing composite devices, e.g. cataplasms characterised by shape or structure; Details concerning release liner or backing; Refillable patches; User-activated patches
    • A61K9/7084—Transdermal patches having a drug layer or reservoir, and one or more separate drug-free skin-adhesive layers, e.g. between drug reservoir and skin, or surrounding the drug reservoir; Liquid-filled reservoir patches
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Natural Medicines & Medicinal Plants (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Dermatology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Microbiology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Mycology (AREA)
  • Organic Chemistry (AREA)
  • Alternative & Traditional Medicine (AREA)
  • Biotechnology (AREA)
  • Botany (AREA)
  • Medical Informatics (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Medicinal Preparation (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Materials For Medical Uses (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)

Abstract

DISPOSITIVO PARA LIBERAçãO DE AGONISTAS DE TRPV1. São descritas aqui dispositivos de distribuição de fármaco incluindo uma camada de revestimento oclusivo e um depósito de fármaco contendo um agonista de TRPV1 e um solvente não-hidrofílico. O depósito de fármaco pode tomar várias formas, tal como uma matriz polimérica adesiva, reservatório de líquido ou gotículas de micro-reservatório. Métodos de fabricação e uso dos dispositivos de distribuição de fármaco também são descritos.
BRPI0607461-8A 2005-02-14 2006-02-14 dispositivo para liberação de agonistas de trpv1 BRPI0607461A2 (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US65292305P 2005-02-14 2005-02-14
PCT/US2006/005453 WO2006089012A2 (en) 2005-02-14 2006-02-14 Device for delivery of trpv1 agonists

Publications (1)

Publication Number Publication Date
BRPI0607461A2 true BRPI0607461A2 (pt) 2009-09-08

Family

ID=36917039

Family Applications (1)

Application Number Title Priority Date Filing Date
BRPI0607461-8A BRPI0607461A2 (pt) 2005-02-14 2006-02-14 dispositivo para liberação de agonistas de trpv1

Country Status (11)

Country Link
US (1) US20060204561A1 (pt)
EP (1) EP1858495A2 (pt)
JP (1) JP2008530139A (pt)
KR (1) KR20070121666A (pt)
CN (1) CN101189000A (pt)
AU (1) AU2006214289A1 (pt)
BR (1) BRPI0607461A2 (pt)
CA (1) CA2597651A1 (pt)
NO (1) NO20074680L (pt)
WO (1) WO2006089012A2 (pt)
ZA (1) ZA200707492B (pt)

Families Citing this family (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP1610742B1 (en) 2003-04-10 2015-01-21 Neurogesx, Inc. Uses and compositions for administration of capsaicin
EP1865933B1 (en) * 2005-03-30 2015-11-04 Vanderbilt Royalty Sub L.P. Low-concentration capsaicin patch and methods for treating neuropathic pain
US7943666B2 (en) * 2006-07-24 2011-05-17 Trinity Laboratories, Inc. Esters of capsaicin for treating pain
WO2009009651A1 (en) * 2007-07-10 2009-01-15 Agile Therapeutics, Inc. Dermal delivery device with ultrasonic weld
WO2009009649A1 (en) 2007-07-10 2009-01-15 Agile Therapeutics, Inc. Dermal delivery device with in situ seal
WO2009142993A1 (en) * 2008-05-21 2009-11-26 The Regents Of The University Of California Topical application of analgesic for pain relief
US9211274B2 (en) 2012-02-01 2015-12-15 Warsaw Orthopedic, Inc. TRPV1 compounds in a biodegradable polymer carrier
WO2015100118A1 (en) * 2013-12-24 2015-07-02 The Procter & Gamble Company Cosmetic compositions and methods providing enhanced penetration of skin care actives
US11607026B2 (en) 2014-05-30 2023-03-21 Johnson & Johnson Consumer Inc. Device for delivery of skin care composition
US20180296497A1 (en) * 2014-10-31 2018-10-18 Avent, Inc. Method and Articles for Inhibiting Bladder Contractions
US10549129B2 (en) 2016-06-24 2020-02-04 The Procter & Gamble Company Cosmetic compositions and methods providing enhanced penetration of skin care actives
JP6635881B2 (ja) * 2016-06-27 2020-01-29 ユニ・チャーム株式会社 温感シート
WO2022143640A1 (en) * 2020-12-30 2022-07-07 Elkem Silicones Shanghai Co., Ltd. A patch coated with a capsaicin-containing silicone gel
EP4046630A1 (en) * 2021-02-18 2022-08-24 LTS Lohmann Therapie-Systeme AG Tts-formulation with thc
CN115006374A (zh) * 2022-07-13 2022-09-06 广州文翰生物科技有限公司 香兰基丁醚在制备治疗头屑和体癣产品中的应用
JP2026508602A (ja) * 2023-03-15 2026-03-11 エルテーエス ローマン テラピー－ジステーメ アーゲー 皮膚刺激活性薬剤を含む医療用パッチ

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US4532139A (en) * 1983-07-14 1985-07-30 The Procter & Gamble Company Compounds and compositions useful for producing analgesia
US4564633A (en) * 1983-07-14 1986-01-14 The Procter & Gamble Company Compositions and methods useful for producing analgesia
US4493848A (en) * 1983-07-14 1985-01-15 The Procter & Gamble Company Compositions and methods useful for producing analgesia
US4544668A (en) * 1983-07-14 1985-10-01 The Procter & Gamble Company Compounds and compositions useful for producing analgesia
US4544669A (en) * 1983-07-14 1985-10-01 The Procter & Gamble Company Compounds and compositions useful for producing analgesia
US4599342A (en) * 1984-01-16 1986-07-08 The Procter & Gamble Company Pharmaceutical products providing enhanced analgesia
US4927687A (en) * 1984-10-01 1990-05-22 Biotek, Inc. Sustained release transdermal drug delivery composition
IE58110B1 (en) * 1984-10-30 1993-07-14 Elan Corp Plc Controlled release powder and process for its preparation
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WO1998055105A1 (en) * 1997-06-05 1998-12-10 Hemosphere, Inc. Fibrinogen-coated microspheres
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PT1094781E (pt) * 1998-07-07 2008-10-08 Transdermal Technologies Inc Composições para administração transdérmica rápida e não irritante de agentes farmacologicamente activos e métodos para formulação de tais composições e sua administração
JP3211027B2 (ja) * 1998-11-13 2001-09-25 丸石製薬株式会社 カプサイシン含有外用剤
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US20040126415A1 (en) * 2002-11-21 2004-07-01 Lu Guang Wei Dermal delivery of a water-soluble selective cyclooxygenase-2 inhibitor
EP1610742B1 (en) * 2003-04-10 2015-01-21 Neurogesx, Inc. Uses and compositions for administration of capsaicin
PT1613297E (pt) * 2003-04-14 2007-08-23 Lohmann Therapie Syst Lts Emplastro terapêutico com matriz de polissiloxano compreendendo capsaicina
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Also Published As

Publication number Publication date
WO2006089012A2 (en) 2006-08-24
EP1858495A2 (en) 2007-11-28
NO20074680L (no) 2007-11-13
WO2006089012A3 (en) 2007-05-18
CA2597651A1 (en) 2006-08-24
US20060204561A1 (en) 2006-09-14
JP2008530139A (ja) 2008-08-07
CN101189000A (zh) 2008-05-28
KR20070121666A (ko) 2007-12-27
AU2006214289A1 (en) 2006-08-24
ZA200707492B (en) 2009-02-25

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Legal Events

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B08L Patent application lapsed because of non payment of annual fee [chapter 8.12 patent gazette]

Free format text: REFERENTE AO NAO RECOLHIMENTO DAS 5A E 8A ANUIDADES.

B08H Application fees: decision cancelled [chapter 8.8 patent gazette]

Free format text: REFERENTE AO DESPACHO 8.12 NA RPI 2260 DE 29/04/2014

B08F Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette]

Free format text: REFERENTE A 8A ANUIDADE

B08K Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette]

Free format text: REFERENTE AO DESPACHO 8.6 PUBLICADO NA RPI 2268 DE 24/06/2014.