BRPI0613407A2 - Complexos contendo perfluoralquila, bem como composição farmacêutica, uso e processos de preparação dos mesmos - Google Patents

Complexos contendo perfluoralquila, bem como composição farmacêutica, uso e processos de preparação dos mesmos Download PDF

Info

Publication number: BRPI0613407A2
Authority: BR; Brazil
Prior art keywords: formula; groups; mmol; original document; document page
Prior art date: 2005-07-15

Application number

BRPI0613407-6A

Other languages

English (en)

Portuguese (pt)

Inventor

Heiko Schirmer

Hanns-Joachim Weinmann

Johannes Platzek

Ludwig Zorn

Bernd Misselwitz

Joerg Meding

Heribert Schmitt-Willich

Thomas Brumby

Original Assignee

Bayer Schering Pharma Ag

Epix Pharm Inc

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2005-07-15

Filing date

2006-07-11

Publication date

2011-01-11

2006-07-11 Application filed by Bayer Schering Pharma Ag, Epix Pharm Inc filed Critical Bayer Schering Pharma Ag

2011-01-11 Publication of BRPI0613407A2 publication Critical patent/BRPI0613407A2/pt

Links

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ORZHVTYKPFFVMG-UHFFFAOYSA-N xylenol orange Chemical compound OC(=O)CN(CC(O)=O)CC1=C(O)C(C)=CC(C2(C3=CC=CC=C3S(=O)(=O)O2)C=2C=C(CN(CC(O)=O)CC(O)=O)C(O)=C(C)C=2)=C1 ORZHVTYKPFFVMG-UHFFFAOYSA-N 0.000 description 1
CKLHRQNQYIJFFX-UHFFFAOYSA-K ytterbium(III) chloride Chemical compound [Cl-].[Cl-].[Cl-].[Yb+3] CKLHRQNQYIJFFX-UHFFFAOYSA-K 0.000 description 1
VWQVUPCCIRVNHF-UHFFFAOYSA-N yttrium atom Chemical compound [Y] VWQVUPCCIRVNHF-UHFFFAOYSA-N 0.000 description 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D257/00—Heterocyclic compounds containing rings having four nitrogen atoms as the only ring hetero atoms
- C07D257/02—Heterocyclic compounds containing rings having four nitrogen atoms as the only ring hetero atoms not condensed with other rings
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K49/00—Preparations for testing in vivo
- A61K49/06—Nuclear magnetic resonance [NMR] contrast preparations; Magnetic resonance imaging [MRI] contrast preparations
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

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Organic Chemistry (AREA)
Chemical & Material Sciences (AREA)
Health & Medical Sciences (AREA)
General Health & Medical Sciences (AREA)
Veterinary Medicine (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Public Health (AREA)
Animal Behavior & Ethology (AREA)
Life Sciences & Earth Sciences (AREA)
Pharmacology & Pharmacy (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Radiology & Medical Imaging (AREA)
Bioinformatics & Cheminformatics (AREA)
Engineering & Computer Science (AREA)
Epidemiology (AREA)
Medicines Containing Antibodies Or Antigens For Use As Internal Diagnostic Agents (AREA)
Steroid Compounds (AREA)
Saccharide Compounds (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)

BRPI0613407-6A 2005-07-15 2006-07-11 Complexos contendo perfluoralquila, bem como composição farmacêutica, uso e processos de preparação dos mesmos BRPI0613407A2 (pt)

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Application Number	Priority Date	Filing Date	Title
DE102005033902.6		2005-07-15
DE102005033902A DE102005033902B3 (de)	2005-07-15	2005-07-15	Perfluoralkylhaltige Komplexe, Verfahren zu deren Herstellung, sowie deren Verwendung und diese enthaltende pharmazeutische Mittel
PCT/EP2006/006777 WO2007009638A2 (de)	2005-07-15	2006-07-11	Perfluoralkylhaltige komplexe, verfahren zu deren herstellung sowie deren verwendung

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EP (1)	EP1904463A2 (de)
JP (1)	JP2009501174A (de)
KR (1)	KR20080043762A (de)
CN (1)	CN101223148A (de)
AR (1)	AR054865A1 (de)
AU (1)	AU2006272025A1 (de)
BR (1)	BRPI0613407A2 (de)
CA (1)	CA2615443A1 (de)
CR (1)	CR9645A (de)
DE (1)	DE102005033902B3 (de)
DO (1)	DOP2006000167A (de)
EC (1)	ECSP088100A (de)
GT (1)	GT200600313A (de)
IL (1)	IL187926A0 (de)
NO (1)	NO20080813L (de)
PE (1)	PE20070376A1 (de)
RU (1)	RU2008105356A (de)
TN (1)	TNSN08016A1 (de)
TW (1)	TW200706538A (de)
UY (1)	UY29664A1 (de)
WO (1)	WO2007009638A2 (de)
ZA (1)	ZA200801523B (de)

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DE102007015598A1 (de) *	2007-03-29	2008-10-02	Heinrich-Heine-Universität Düsseldorf	Verwendung von fluorhaltigen Verbindungen zu Diagnosezwecken mit Hilfe bildgebender Verfahren
JP5730581B2 (ja)	2008-01-08	2015-06-10	ランセウスメディカルイメージング，インコーポレイテッド	造影剤としてのｎ−アルコキシアミド抱合体
WO2021067738A1 (en) *	2019-10-04	2021-04-08	United States Government As Represented By The Department Of Veterans Affairs	Development of imaging and therapeutic glucose analogues for sodium dependent glucose transporters
EP4059925A1 (de)	2021-03-15	2022-09-21	Bayer Aktiengesellschaft	Neues kontrastmittel zur verwendung in der magnetresonanzbildgebung
CN114181164A (zh) *	2021-12-13	2022-03-15	武汉大学中南医院	基于Fe(Ⅱ)特异性MRI对比剂的合成方法及其应用
EP4335462A1 (de)	2022-09-09	2024-03-13	Bayer AG	Kontrastmittel zur verwendung in der diagnostischen bildgebung mittels computertomografie
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2005
- 2005-07-15 DE DE102005033902A patent/DE102005033902B3/de not_active Expired - Fee Related
2006
- 2006-07-11 KR KR1020087001084A patent/KR20080043762A/ko not_active Withdrawn
- 2006-07-11 EP EP06791535A patent/EP1904463A2/de not_active Withdrawn
- 2006-07-11 JP JP2008520780A patent/JP2009501174A/ja not_active Withdrawn
- 2006-07-11 CA CA002615443A patent/CA2615443A1/en not_active Abandoned
- 2006-07-11 CN CNA2006800258905A patent/CN101223148A/zh active Pending
- 2006-07-11 BR BRPI0613407-6A patent/BRPI0613407A2/pt not_active Application Discontinuation
- 2006-07-11 WO PCT/EP2006/006777 patent/WO2007009638A2/de not_active Ceased
- 2006-07-11 RU RU2008105356/04A patent/RU2008105356A/ru not_active Application Discontinuation
- 2006-07-11 UY UY29664A patent/UY29664A1/es not_active Application Discontinuation
- 2006-07-11 AU AU2006272025A patent/AU2006272025A1/en not_active Abandoned
- 2006-07-13 DO DO2006000167A patent/DOP2006000167A/es unknown
- 2006-07-14 AR ARP060103020A patent/AR054865A1/es unknown
- 2006-07-14 GT GT200600313A patent/GT200600313A/es unknown
- 2006-07-14 PE PE2006000844A patent/PE20070376A1/es not_active Application Discontinuation
- 2006-07-14 TW TW095125755A patent/TW200706538A/zh unknown
2007
- 2007-12-06 IL IL187926A patent/IL187926A0/en unknown
2008
- 2008-01-08 CR CR9645A patent/CR9645A/es unknown
- 2008-01-11 EC EC2008008100A patent/ECSP088100A/es unknown
- 2008-01-14 TN TNP2008000016A patent/TNSN08016A1/en unknown
- 2008-02-14 NO NO20080813A patent/NO20080813L/no not_active Application Discontinuation
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Also Published As

Publication number	Publication date
AU2006272025A1 (en)	2007-01-25
TW200706538A (en)	2007-02-16
WO2007009638A3 (de)	2007-04-26
DOP2006000167A (es)	2007-02-28
GT200600313A (es)	2007-04-23
EP1904463A2 (de)	2008-04-02
AR054865A1 (es)	2007-07-25
CR9645A (es)	2008-05-21
ZA200801523B (en)	2008-11-26
PE20070376A1 (es)	2007-04-20
KR20080043762A (ko)	2008-05-19
UY29664A1 (es)	2007-02-28
ECSP088100A (es)	2008-05-30
NO20080813L (no)	2008-04-09
TNSN08016A1 (en)	2009-07-14
JP2009501174A (ja)	2009-01-15
RU2008105356A (ru)	2009-08-20
CA2615443A1 (en)	2007-01-25
DE102005033902B3 (de)	2007-04-05
CN101223148A (zh)	2008-07-16
WO2007009638A2 (de)	2007-01-25
IL187926A0 (en)	2008-03-20

Legal Events

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2011-07-26	B11A	Dismissal acc. art.33 of ipl - examination not requested within 36 months of filing
2011-11-01	B11Y	Definitive dismissal - extension of time limit for request of examination expired [chapter 11.1.1 patent gazette]

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