BRPI0620687A8 - Polimorfo cristalino, pseudomorfo em hemi-solvato, composto amorfo, mistura polimórfica, processo para a preparação de um polimorfo cristalino, processo para a preparação de um pseudomorfo de 5-amino-1-[2,6-dicloro-4-(trifluorometil)fenil] -4- [(trifluorometil) sulfinil] -1h- pirazol-3-carbonitrila, processo para a preparação da forma amorfa de 5-amino-1-[2,6-dicloro-4-(trifluorometil) fenil] -4- [trifluorometil) sulfinil] -1h-pirazol-3-carbonitrila, composição pesticida e método para o controle de pragas num local - Google Patents
Polimorfo cristalino, pseudomorfo em hemi-solvato, composto amorfo, mistura polimórfica, processo para a preparação de um polimorfo cristalino, processo para a preparação de um pseudomorfo de 5-amino-1-[2,6-dicloro-4-(trifluorometil)fenil] -4- [(trifluorometil) sulfinil] -1h- pirazol-3-carbonitrila, processo para a preparação da forma amorfa de 5-amino-1-[2,6-dicloro-4-(trifluorometil) fenil] -4- [trifluorometil) sulfinil] -1h-pirazol-3-carbonitrila, composição pesticida e método para o controle de pragas num localInfo
- Publication number
- BRPI0620687A8 BRPI0620687A8 BRPI0620687A BRPI0620687A BRPI0620687A8 BR PI0620687 A8 BRPI0620687 A8 BR PI0620687A8 BR PI0620687 A BRPI0620687 A BR PI0620687A BR PI0620687 A BRPI0620687 A BR PI0620687A BR PI0620687 A8 BRPI0620687 A8 BR PI0620687A8
- Authority
- BR
- Brazil
- Prior art keywords
- trifluoromethyl
- carbonitrile
- dichloro
- phenyl
- amino
- Prior art date
Links
- 238000000034 method Methods 0.000 title abstract 6
- 239000000203 mixture Substances 0.000 title abstract 5
- WZKSXHQDXQKIQJ-UHFFFAOYSA-N F[C](F)F Chemical class F[C](F)F WZKSXHQDXQKIQJ-UHFFFAOYSA-N 0.000 title abstract 4
- CIUQDSCDWFSTQR-UHFFFAOYSA-N [C]1=CC=CC=C1 Chemical compound [C]1=CC=CC=C1 CIUQDSCDWFSTQR-UHFFFAOYSA-N 0.000 title abstract 4
- 238000004519 manufacturing process Methods 0.000 title abstract 4
- 150000001875 compounds Chemical class 0.000 title abstract 2
- 239000000575 pesticide Substances 0.000 title abstract 2
- ZOCSXAVNDGMNBV-UHFFFAOYSA-N 5-amino-1-[2,6-dichloro-4-(trifluoromethyl)phenyl]-4-[(trifluoromethyl)sulfinyl]-1H-pyrazole-3-carbonitrile Chemical compound NC1=C(S(=O)C(F)(F)F)C(C#N)=NN1C1=C(Cl)C=C(C(F)(F)F)C=C1Cl ZOCSXAVNDGMNBV-UHFFFAOYSA-N 0.000 abstract 2
- 230000000361 pesticidal effect Effects 0.000 abstract 2
- 239000005899 Fipronil Substances 0.000 abstract 1
- 239000003795 chemical substances by application Substances 0.000 abstract 1
- 229940013764 fipronil Drugs 0.000 abstract 1
- 230000000749 insecticidal effect Effects 0.000 abstract 1
- 239000012453 solvate Substances 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
- C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D231/28—Two oxygen or sulfur atoms
-
- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
- A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
- A01N43/56—1,2-Diazoles; Hydrogenated 1,2-diazoles
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
- C07B2200/00—Indexing scheme relating to specific properties of organic compounds
- C07B2200/13—Crystalline forms, e.g. polymorphs
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- Dentistry (AREA)
- Pest Control & Pesticides (AREA)
- Plant Pathology (AREA)
- Health & Medical Sciences (AREA)
- Engineering & Computer Science (AREA)
- Agronomy & Crop Science (AREA)
- General Health & Medical Sciences (AREA)
- Wood Science & Technology (AREA)
- Zoology (AREA)
- Environmental Sciences (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
Abstract
POLIMORFO CRISTALINO, PSEUDOMORFO EM HEMI-SOLVATO, COMPOSTO AMORFO, MISTURA POLIMÓRFICA, PROCESSO PARA A PREPARAÇÃO DE UM POLIMORFO CRISTALINO, PROCESSO PARA A PREPARAÇÃO DE UM PSEUDOMORFO DE 5-AMINO-1- [2,6-DICLORO-4-(TRIFLUOROMETIL) FENIL] -4- [(TRIFLUOROMETIL) SULFINILI] -1H-PIRAZOL-3-CARBONITRILA, PROCESSO PARA A PREPARAÇÃO DA FORMA AMORFA DE 5-AMINO-1- [2,6-DICLORO-4-(TRIFLUOROMETIL) FENIL] -4- [(TRIFLUOROMETIL) SULFINIL] -1H-PIRAZOL-3-CARBONITRILA, COMPOSIÇÃO PESTICIDA E MÉTODO PARA O CONTROLE DE PRAGAS NUM LOCAL. A presente invenção refere-se a polimorfos cristalinos novos, pseudomorfos em solvato novos e à forma amorfa nova de 5-amino-1- [2,6-dicloro-4- (trifluorometil)fenil] -4- [(trifluorometil) sulfinil]-1H-pirazol-3-carbonitrila (fipronil). A presente invenção também provê métodos para preparar os polimorfos, pseudomorfos novos e a forma amorfa nova, bem como as composições inseticidas ou pesticidas compreendendo os mesmos, e métodos de uso dos mesmos como agente pesticida.
Applications Claiming Priority (5)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US75004605P | 2005-12-14 | 2005-12-14 | |
| US60/750,046 | 2005-12-14 | ||
| IL172585 | 2005-12-14 | ||
| IL172585A IL172585A0 (en) | 2005-12-14 | 2005-12-14 | Polymorphs of 5-amino-1-[2,6-dichloro-4- (trifluoromethyl)phenyl]-4-[(trifluoromethyl)sulfinyl]- 1h-pyrazole-3-carbonitrile |
| PCT/IL2006/001441 WO2007069254A2 (en) | 2005-12-14 | 2006-12-14 | POLYMORPHS AND AMORPHOUS FORMS OF 5-AMINO-l-[2,6- DICHLORO-4-(TRIFLUOROMETHYL)PHENYL]-4- [(TRIFLUOROMETHYL)SULFINYL]-IH-PYRAZOLE-3-CARBONITRILE |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| BRPI0620687A2 BRPI0620687A2 (pt) | 2011-11-22 |
| BRPI0620687A8 true BRPI0620687A8 (pt) | 2017-04-11 |
Family
ID=42331702
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| BRPI0620687A BRPI0620687A8 (pt) | 2005-12-14 | 2006-12-14 | Polimorfo cristalino, pseudomorfo em hemi-solvato, composto amorfo, mistura polimórfica, processo para a preparação de um polimorfo cristalino, processo para a preparação de um pseudomorfo de 5-amino-1-[2,6-dicloro-4-(trifluorometil)fenil] -4- [(trifluorometil) sulfinil] -1h- pirazol-3-carbonitrila, processo para a preparação da forma amorfa de 5-amino-1-[2,6-dicloro-4-(trifluorometil) fenil] -4- [trifluorometil) sulfinil] -1h-pirazol-3-carbonitrila, composição pesticida e método para o controle de pragas num local |
Country Status (4)
| Country | Link |
|---|---|
| KR (1) | KR20140096396A (pt) |
| BR (1) | BRPI0620687A8 (pt) |
| CA (2) | CA2808257A1 (pt) |
| IL (1) | IL172585A0 (pt) |
-
2005
- 2005-12-14 IL IL172585A patent/IL172585A0/en unknown
-
2006
- 2006-12-14 CA CA2808257A patent/CA2808257A1/en not_active Abandoned
- 2006-12-14 KR KR1020147019887A patent/KR20140096396A/ko not_active Ceased
- 2006-12-14 BR BRPI0620687A patent/BRPI0620687A8/pt not_active Application Discontinuation
- 2006-12-14 CA CA2808259A patent/CA2808259A1/en not_active Abandoned
Also Published As
| Publication number | Publication date |
|---|---|
| CA2808257A1 (en) | 2007-06-21 |
| CA2808259A1 (en) | 2007-06-21 |
| BRPI0620687A2 (pt) | 2011-11-22 |
| KR20140096396A (ko) | 2014-08-05 |
| IL172585A0 (en) | 2006-04-10 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| B25D | Requested change of name of applicant approved |
Owner name: ADAMA MAKHTESHIM LTD. (IL) |
|
| B07D | Technical examination (opinion) related to article 229 of industrial property law [chapter 7.4 patent gazette] | ||
| B06F | Objections, documents and/or translations needed after an examination request according [chapter 6.6 patent gazette] | ||
| B07G | Grant request does not fulfill article 229-c lpi (prior consent of anvisa) [chapter 7.7 patent gazette] |
Free format text: NOTIFICACAO DE DEVOLUCAO DO PEDIDO POR NAO SE ENQUADRAR NO ART. 229-C DA LPI. |
|
| B07A | Application suspended after technical examination (opinion) [chapter 7.1 patent gazette] | ||
| B09B | Patent application refused [chapter 9.2 patent gazette] | ||
| B12B | Appeal against refusal [chapter 12.2 patent gazette] |