BRPI0712332A2 - composto e derivados farmaceuticamente aceitáveis dos mesmos, composição farmacêutica, método de antagonização de um receptor dp-2, e, uso de um composto - Google Patents

composto e derivados farmaceuticamente aceitáveis dos mesmos, composição farmacêutica, método de antagonização de um receptor dp-2, e, uso de um composto Download PDF

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Publication number
BRPI0712332A2
BRPI0712332A2 BRPI0712332-9A BRPI0712332A BRPI0712332A2 BR PI0712332 A2 BRPI0712332 A2 BR PI0712332A2 BR PI0712332 A BRPI0712332 A BR PI0712332A BR PI0712332 A2 BRPI0712332 A2 BR PI0712332A2
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BR
Brazil
Prior art keywords
phenyl
piperidin
acetic acid
compound
fluorophenylsulfonyl
Prior art date
Application number
BRPI0712332-9A
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English (en)
Portuguese (pt)
Inventor
Thomas Dudler
Francine Farouz
Kerry Fowler
Nataly Hawthorn
Danwen Huang
Jin Bohan
Musong Kim
Andrew Lover
Joshua Odingo
Amy Oliver
Mark Reed
Fuqiang Ruan
Eugene Thorsett
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Icos Corp
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Publication date
Application filed by Icos Corp filed Critical Icos Corp
Publication of BRPI0712332A2 publication Critical patent/BRPI0712332A2/pt

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    • C07D267/02—Seven-membered rings
    • C07D267/08—Seven-membered rings having the hetero atoms in positions 1 and 4
    • C07D267/12—Seven-membered rings having the hetero atoms in positions 1 and 4 condensed with carbocyclic rings or ring systems
    • C07D267/14—Seven-membered rings having the hetero atoms in positions 1 and 4 condensed with carbocyclic rings or ring systems condensed with one six-membered ring
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  • Animal Behavior & Ethology (AREA)
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  • Rheumatology (AREA)
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  • Obesity (AREA)
  • Pulmonology (AREA)
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  • Child & Adolescent Psychology (AREA)
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BRPI0712332-9A 2006-06-09 2007-06-08 composto e derivados farmaceuticamente aceitáveis dos mesmos, composição farmacêutica, método de antagonização de um receptor dp-2, e, uso de um composto BRPI0712332A2 (pt)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US81239906P 2006-06-09 2006-06-09
US60/812399 2006-06-09
PCT/US2007/070805 WO2007146838A2 (en) 2006-06-09 2007-06-08 Substituted phenyl acetic acids as dp-2 antagonists

Publications (1)

Publication Number Publication Date
BRPI0712332A2 true BRPI0712332A2 (pt) 2012-12-18

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BRPI0712332-9A BRPI0712332A2 (pt) 2006-06-09 2007-06-08 composto e derivados farmaceuticamente aceitáveis dos mesmos, composição farmacêutica, método de antagonização de um receptor dp-2, e, uso de um composto

Country Status (10)

Country Link
EP (1) EP2044017A2 (no)
JP (1) JP2009539881A (no)
CN (1) CN101490001A (no)
AU (1) AU2007257841A1 (no)
BR (1) BRPI0712332A2 (no)
CA (1) CA2654927A1 (no)
EA (2) EA200802417A1 (no)
MX (1) MX2008015638A (no)
NO (1) NO20090139L (no)
WO (1) WO2007146838A2 (no)

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DE102007034620A1 (de) * 2007-07-25 2009-01-29 Boehringer Ingelheim Pharma Gmbh & Co. Kg Neue B1-Antagonisten
KR101618068B1 (ko) 2007-10-19 2016-05-04 얀센 파마슈티카 엔.브이. γ-세크레타아제의 탄소 결합된 조절제
WO2009052126A1 (en) * 2007-10-19 2009-04-23 Janssen Pharmaceutica, N.V. PIPERIDINYL AND PIPERAZINYL MODULATORS OF γ-SECRETASE
CN101903335A (zh) 2007-10-19 2010-12-01 詹森药业有限公司 连接有胺的γ-分泌酶调节剂
KR20120046762A (ko) * 2009-07-31 2012-05-10 판미라 파마슈티칼스, 엘엘씨 Ｄｐ2 수용체 길항제의 피부 제형
EP2521713A4 (en) * 2010-01-06 2013-10-02 Panmira Pharmaceuticals Llc ANTAGONIST OF DP2 AND ITS USES
CN102958914B (zh) 2010-07-05 2015-05-27 埃科特莱茵药品有限公司 1-苯基取代的杂环衍生物及其作为前列腺素d2受体调节剂的用途
EP2457900A1 (en) 2010-11-25 2012-05-30 Almirall, S.A. New pyrazole derivatives having CRTh2 antagonistic behaviour
EP2487159A1 (en) * 2011-02-11 2012-08-15 MSD Oss B.V. RorgammaT inhibitors
CN103547580B (zh) 2011-03-22 2016-12-07 阿迪维纳斯疗法有限公司 取代的稠合三环化合物、其组合物及医药用途
EP3812387A1 (en) 2011-07-21 2021-04-28 Sumitomo Dainippon Pharma Oncology, Inc. Heterocyclic protein kinase inhibitors
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CA2654927A1 (en) 2007-12-21
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