BRPI0717939A2 - Aminometil-4-imidazóis - Google Patents

Aminometil-4-imidazóis

Info

Publication number: BRPI0717939A2
Authority: BR; Brazil
Prior art keywords: immidazois; aminometil
Prior art date: 2006-10-19

Application number

BRPI0717939-1A2A

Other languages

English (en)

Inventor

Guido Galley

Annick Goergler

Katrin Groebke Zbinden

Roger Norcross

Henri Stalder

Original Assignee

Hoffmann La Roche

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2006-10-19

Filing date

2007-10-09

Publication date

2013-12-03

Family has litigation

First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=38876376&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=BRPI0717939(A2) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.

2007-10-09 Application filed by Hoffmann La Roche filed Critical Hoffmann La Roche

2013-12-03 Publication of BRPI0717939A2 publication Critical patent/BRPI0717939A2/pt

Links

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
- C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
- C07D233/64—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with substituted hydrocarbon radicals attached to ring carbon atoms, e.g. histidine
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/4164—1,3-Diazoles
- A61K31/4178—1,3-Diazoles not condensed 1,3-diazoles and containing further heterocyclic rings, e.g. pilocarpine, nitrofurantoin
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/06—Antimigraine agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/08—Antiepileptics; Anticonvulsants
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
- A61P25/16—Anti-Parkinson drugs
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/20—Hypnotics; Sedatives
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/22—Anxiolytics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/04—Anorexiants; Antiobesity agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/06—Antihyperlipidemics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
- A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/12—Antihypertensives

Landscapes

Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Engineering & Computer Science (AREA)
Bioinformatics & Cheminformatics (AREA)
Medicinal Chemistry (AREA)
Pharmacology & Pharmacy (AREA)
Life Sciences & Earth Sciences (AREA)
Animal Behavior & Ethology (AREA)
General Health & Medical Sciences (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
General Chemical & Material Sciences (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Chemical Kinetics & Catalysis (AREA)
Neurology (AREA)
Neurosurgery (AREA)
Biomedical Technology (AREA)
Diabetes (AREA)
Obesity (AREA)
Psychiatry (AREA)
Hematology (AREA)
Pain & Pain Management (AREA)
Cardiology (AREA)
Heart & Thoracic Surgery (AREA)
Endocrinology (AREA)
Emergency Medicine (AREA)
Urology & Nephrology (AREA)
Child & Adolescent Psychology (AREA)
Vascular Medicine (AREA)
Anesthesiology (AREA)
Addiction (AREA)
Psychology (AREA)
Hospice & Palliative Care (AREA)
Epidemiology (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Plural Heterocyclic Compounds (AREA)

BRPI0717939-1A2A 2006-10-19 2007-10-09 Aminometil-4-imidazóis BRPI0717939A2 (pt)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
EP06122586		2006-10-19
PCT/EP2007/060666 WO2008046757A1 (en)	2006-10-19	2007-10-09	Aminomethyl-4-imidazoles

Publications (1)

Publication Number	Publication Date
BRPI0717939A2 true BRPI0717939A2 (pt)	2013-12-03

Family

ID=38876376

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
BRPI0717939-1A2A BRPI0717939A2 (pt)	2006-10-19	2007-10-09	Aminometil-4-imidazóis

Country Status (20)

Country	Link
US (1)	US8586617B2 (pt)
EP (1)	EP2076497B1 (pt)
JP (2)	JP5335681B2 (pt)
KR (1)	KR101176699B1 (pt)
CN (1)	CN101528710B (pt)
AR (1)	AR063327A1 (pt)
AT (1)	ATE546437T1 (pt)
AU (1)	AU2007312390B2 (pt)
BR (1)	BRPI0717939A2 (pt)
CA (1)	CA2666762C (pt)
CL (1)	CL2007002971A1 (pt)
ES (1)	ES2381589T3 (pt)
IL (1)	IL197877A (pt)
MX (1)	MX2009003801A (pt)
NO (1)	NO20091478L (pt)
PE (1)	PE20080889A1 (pt)
RU (1)	RU2009112496A (pt)
TW (1)	TW200833685A (pt)
WO (1)	WO2008046757A1 (pt)
ZA (1)	ZA200902278B (pt)

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RU2439062C2 (ru) *	2006-10-19	2012-01-10	Ф.Хоффманн-Ля Рош Аг	Производные имидазолона и имидазолидинона как 11в-hsd1 ингибиторы при диабете
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2007
- 2007-10-09 AU AU2007312390A patent/AU2007312390B2/en not_active Ceased
- 2007-10-09 CA CA2666762A patent/CA2666762C/en not_active Expired - Fee Related
- 2007-10-09 RU RU2009112496/04A patent/RU2009112496A/ru not_active Application Discontinuation
- 2007-10-09 KR KR1020097007948A patent/KR101176699B1/ko not_active Expired - Fee Related
- 2007-10-09 AT AT07821039T patent/ATE546437T1/de active
- 2007-10-09 CN CN2007800388091A patent/CN101528710B/zh not_active Expired - Fee Related
- 2007-10-09 JP JP2009532767A patent/JP5335681B2/ja not_active Expired - Fee Related
- 2007-10-09 MX MX2009003801A patent/MX2009003801A/es active IP Right Grant
- 2007-10-09 WO PCT/EP2007/060666 patent/WO2008046757A1/en not_active Ceased
- 2007-10-09 BR BRPI0717939-1A2A patent/BRPI0717939A2/pt not_active IP Right Cessation
- 2007-10-09 ES ES07821039T patent/ES2381589T3/es active Active
- 2007-10-09 EP EP07821039A patent/EP2076497B1/en not_active Not-in-force
- 2007-10-15 US US11/872,203 patent/US8586617B2/en not_active Expired - Fee Related
- 2007-10-17 AR ARP070104590A patent/AR063327A1/es unknown
- 2007-10-17 PE PE2007001403A patent/PE20080889A1/es not_active Application Discontinuation
- 2007-10-17 CL CL200702971A patent/CL2007002971A1/es unknown
- 2007-10-17 TW TW096138932A patent/TW200833685A/zh unknown
2009
- 2009-03-26 IL IL197877A patent/IL197877A/en not_active IP Right Cessation
- 2009-04-01 ZA ZA200902278A patent/ZA200902278B/xx unknown
- 2009-04-17 NO NO20091478A patent/NO20091478L/no not_active Application Discontinuation
2013
- 2013-05-02 JP JP2013096834A patent/JP5567177B2/ja not_active Expired - Fee Related

Also Published As

Publication number	Publication date
JP5567177B2 (ja)	2014-08-06
JP5335681B2 (ja)	2013-11-06
ATE546437T1 (de)	2012-03-15
AR063327A1 (es)	2009-01-21
MX2009003801A (es)	2009-04-22
TW200833685A (en)	2008-08-16
WO2008046757A1 (en)	2008-04-24
IL197877A0 (en)	2009-12-24
CL2007002971A1 (es)	2008-05-30
ZA200902278B (en)	2010-03-31
ES2381589T3 (es)	2012-05-29
CA2666762C (en)	2014-12-30
US20080119535A1 (en)	2008-05-22
CA2666762A1 (en)	2008-04-24
AU2007312390A1 (en)	2008-04-24
AU2007312390B2 (en)	2013-03-28
JP2013173779A (ja)	2013-09-05
JP2010506875A (ja)	2010-03-04
CN101528710A (zh)	2009-09-09
NO20091478L (no)	2009-05-05
RU2009112496A (ru)	2010-11-27
EP2076497A1 (en)	2009-07-08
KR101176699B1 (ko)	2012-08-23
KR20090055035A (ko)	2009-06-01
IL197877A (en)	2015-07-30
US8586617B2 (en)	2013-11-19
EP2076497B1 (en)	2012-02-22
CN101528710B (zh)	2012-11-07
PE20080889A1 (es)	2008-06-27

Legal Events

Date	Code	Title	Description
2017-08-08	B08F	Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette]
2017-11-28	B08K	Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette]

Publication	Publication Date	Title
DE602007008423D1 (de)	2010-09-23	Flüssigkeitshärtung
DE602007009267D1 (de)	2010-10-28	Reifenaufblasverfahren
AT504580A3 (de)	2008-07-15	Scan-einrichtung
ATE546437T1 (de)	2012-03-15	Aminomethyl-4-imidazole
DE502007000218D1 (de)	2008-12-18	nsetzungen
FI20061014A0 (fi)	2006-11-17	Diffuusiopinnoitusmenetelmä
DE112007003147A5 (de)	2009-09-24	Rohr-Biegevorrichtung
DE602007012951D1 (de)	2011-04-21	Verbundschraubenausräumtür
DE502007005975D1 (de)	2011-01-27	Wischblatt
NO20065996L (no)	2008-06-23	SmartPacker
FI20060691A0 (fi)	2006-07-19	Laitekotelointi
ITPD20060387A1 (it)	2008-04-20	Espositore
DE112007001125A5 (de)	2009-02-05	Käfigmutter
NO20065028L (no)	2008-05-05	Limkobling
NO20060756L (no)	2007-08-17	Transportsystem
SE0700923L (sv)	2008-05-10	Halogenhårtork
FR2896376B1 (fr)	2010-03-26	Desherbeuse-emietteuse
FI7243U1 (fi)	2006-10-18	Hiirenpyydys
ES1064558Y (es)	2007-07-01	Salva-tendedero
FI7353U1 (fi)	2007-01-12	Riipukeläpivienti
FI7437U1 (fi)	2007-03-09	Katafalkki
FI7103U1 (fi)	2006-06-08	Pyrstömormuska
FI7355U1 (fi)	2007-01-12	Esiintymislava
FI7169U1 (fi)	2006-07-28	Paalileikkuri
DE602006013403D1 (de)	2010-05-20	Flüssigkeitsinjector